G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Donitriptan
CAS:170912-52-4
Donitriptan is a 5-HT receptor agonist with pKis of 9.4 and 9.3 for 5-HT1B and …
Formula:
C23H25N5O2
Purity:
98.34%
Color and Shape:
Solid
Molecular weight:
403.48
Ref: TM-T11075
| 1mg | 55.00 € | ||
| 1ml | 130.00 € | ||
| 2mg | 80.00 € | ||
| 5mg | 118.00 € | ||
| 10mg | 184.00 € | ||
| 25mg | 425.00 € | ||
| 50mg | 627.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
ML230
CAS:1776055-05-0
ML230 is a selective ATP-binding cassette (ABC) transporter ABCG2 inhibitor.
Formula:
C25H21N5O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
439.47
Ref: TM-T16107
| 5mg | 844.00 € | ||
| 10mg | 1,499.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Radioprotectin-1
CAS:1622006-09-0
Radioprotectin-1 is a selective agonist of LPA2 with EC50 of 25 nM for murine LPA2 …
Formula:
C23H19ClN2O6S
Purity:
98.75% - 99.43%
Color and Shape:
Solid
Molecular weight:
486.92
Ref: TM-T12684
| 1mg | 118.00 € | ||
| 1ml | 309.00 € | ||
| 5mg | 276.00 € | ||
| 10mg | 422.00 € | ||
| 25mg | 693.00 € | ||
| 50mg | 915.00 € | ||
| 100mg | 1,261.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
GR 46611
CAS:185259-85-2
GR 46611 is a selective 5-HT1B and 5-HT1D receptor agonist and can be used in …
Formula:
C23H27N3O2
Purity:
99.9%
Color and Shape:
Solid
Molecular weight:
377.48
Ref: TM-T22808
| 1mg | 52.00 € | ||
| 5mg | 91.00 € | ||
| 10mg | 132.00 € | ||
| 25mg | 259.00 € | ||
| 50mg | 412.00 € | ||
| 100mg | 600.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Lavoltidine
CAS:76956-02-0
Lavoltidine, an irreversible oral H2-receptor antagonist, reduces stomach acid and increases gastrin.
Formula:
C19H29N5O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
359.47
Ref: TM-T15722
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
OPC-14523 hydrochloride
CAS:145969-31-9
OPC-14523 hydrochloride, an oral sigma/5-HT1A agonist, shows potent antidepressant activity with strong receptor affinity.
Formula:
C23H29Cl2N3O2
Purity:
99.70%
Color and Shape:
Solid
Molecular weight:
450.4
Ref: TM-T62711
| 1ml | 942.00 € | ||
| 5mg | 889.00 € | ||
| 10mg | 1,181.00 € | ||
| 25mg | 1,483.00 € | ||
| 50mg | 1,814.00 € | ||
| 100mg | 2,290.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Ecopipam
CAS:112108-01-7
Ecopipam: orally active, selective dopamine D1/D5 antagonist (Ki: 1.2 nM/2.0 nM). 40x more selective over …
Formula:
C19H20ClNO
Purity:
98.5%
Color and Shape:
Solid
Molecular weight:
313.82
Ref: TM-T31602
| 1mg | 182.00 € | ||
| 2mg | 273.00 € | ||
| 5mg | 417.00 € | ||
| 10mg | 612.00 € | ||
| 25mg | 917.00 € | ||
| 50mg | 1,282.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Rec 15/2615 dihydrochloride
CAS:173059-17-1
Rec 15/2615 dihydrochloride is an antagonist of α1B-adrenergic receptor.
Formula:
C26H35Cl2N5O5
Purity:
98.97% - 99.81%
Color and Shape:
Solid
Molecular weight:
568.49
Ref: TM-T23230
| 1mg | 82.00 € | ||
| 5mg | 172.00 € | ||
| 10mg | 254.00 € | ||
| 25mg | 419.00 € | ||
| 50mg | 589.00 € | ||
| 100mg | 796.00 € | ||
| 500mg | To inquire |
Estimated delivery in United States, on Monday 25 Nov 2024
Litoxetine
CAS:86811-09-8
Litoxetine: a selective 5-HT inhibitor & 5-HT3 antagonist, used as an antidepressant with antiemetic effects, …
Formula:
C16H19NO
Purity:
99.12%
Color and Shape:
Solid
Molecular weight:
241.33
Ref: TM-T67956
| 1mg | 95.00 € | ||
| 1ml | 187.00 € | ||
| 5mg | 214.00 € | ||
| 10mg | 319.00 € | ||
| 25mg | 547.00 € | ||
| 50mg | 782.00 € | ||
| 100mg | 1,077.00 € | ||
| 500mg | 2,168.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Felypressin acetate
CAS:914453-97-7
Felypressin acetate (PLV-2) is an agonist of vasopressin 1 and acts on all arginine vasopressin …
Formula:
C48H69N13O13S2
Purity:
97.06%
Color and Shape:
Solid
Molecular weight:
1100.27
Ref: TM-T2568L
| 5mg | 46.00 € | ||
| 10mg | 69.00 € | ||
| 25mg | 123.00 € | ||
| 50mg | 183.00 € | ||
| 100mg | 291.00 € | ||
| 200mg | 435.00 € | ||
| 500mg | 700.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Remogliflozin etabonate
CAS:442201-24-3
Remogliflozin etabonate is a prodrug SGLT2 inhibitor; Ki for hSGLT2: 1.95μM, rSGLT2: 2.14μM, rSGLT1: 8.57μM, …
Formula:
C26H38N2O9
Purity:
99%
Color and Shape:
Solid
Molecular weight:
522.59
Ref: TM-T34286
| 1mg | 37.00 € | ||
| 1ml | 91.00 € | ||
| 2mg | 51.00 € | ||
| 5mg | 89.00 € | ||
| 10mg | 144.00 € | ||
| 25mg | 263.00 € | ||
| 50mg | 404.00 € | ||
| 100mg | 562.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Tecalcet Hydrochloride
CAS:177172-49-5
Tecalcet Hydrochloride, an allosteric CaSR modulator, enhances extracellular Ca2+ sensitivity.
Formula:
C18H23Cl2NO
Purity:
99.44%
Color and Shape:
Solid
Molecular weight:
340.29
Ref: TM-T13918
| 1ml | 51.00 € | ||
| 2mg | 35.00 € | ||
| 5mg | 49.00 € | ||
| 10mg | 74.00 € | ||
| 25mg | 151.00 € | ||
| 50mg | 238.00 € | ||
| 100mg | 347.00 € | ||
| 200mg | To inquire |
Estimated delivery in United States, on Monday 25 Nov 2024
Rolapitant
CAS:552292-08-7
Rolapitant Hydrochloride is an oral NK1-receptor blocker that prevents nausea and has a fast onset …
Formula:
C25H26F6N2O2
Purity:
98.34%
Color and Shape:
Solid
Molecular weight:
500.48
Ref: TM-T3716
| 1mg | 51.00 € | ||
| 1ml | 91.00 € | ||
| 2mg | 65.00 € | ||
| 5mg | 92.00 € | ||
| 10mg | 121.00 € | ||
| 25mg | 184.00 € | ||
| 50mg | 305.00 € | ||
| 100mg | 456.00 € | ||
| 500mg | 1,013.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Lintopride
CAS:107429-63-0
Lintopride is an antagonist of 5HT4. It has moderate 5HT3 antagonist properties.
Formula:
C14H19ClN4O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
310.78
Ref: TM-T15760
| 25mg | 1,410.00 € | ||
| 50mg | 1,838.00 € | ||
| 100mg | 2,322.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Lusaperidone
CAS:214548-46-6
Kaerophyllin ( (-)-Kaerophylin) inhibits hepatic stellate cell activation and inhibits HSC activation to protect against …
Formula:
C22H21N3O2
Purity:
99.64%
Color and Shape:
Solid
Molecular weight:
359.42
Ref: TM-T11894
| 1mg | 131.00 € | ||
| 5mg | 305.00 € | ||
| 10mg | 491.00 € | ||
| 25mg | 1,012.00 € | ||
| 50mg | 1,718.00 € | ||
| 100mg | 2,524.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
ENMD-1068 HCl
CAS:789488-77-3
ENMD-1068 HCl (ENMD 1068) is a PAR-2 antagonist. ENMD-1068 HCl inhibits the development of endometriosis …
Formula:
C15H29N3O2
Purity:
95.79%
Color and Shape:
Solid
Molecular weight:
283.41
Ref: TM-T27267
| 1ml | 55.00 € | ||
| 10mg | 54.00 € | ||
| 25mg | 94.00 € | ||
| 50mg | 132.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
(R)-ZINC-3573
CAS:2089389-15-9
ZINC-3573: Potent, selective MRGPRX2 activator; triggers mast cell degranulation and calcium release.
Formula:
C18H21N5
Purity:
100%
Color and Shape:
Solid
Molecular weight:
307.39
Ref: TM-T29221
| 1ml | 77.00 € | ||
| 2mg | 46.00 € | ||
| 5mg | 69.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 212.00 € | ||
| 50mg | 319.00 € | ||
| 100mg | 462.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
PPTN
CAS:1160271-30-6
PPTN is a high-affinity, competitive and highly selective antagonist of P2Y14 receptor(KB value of 434 …
Formula:
C29H24F3NO2
Purity:
100%
Color and Shape:
Solid
Molecular weight:
475.5
Ref: TM-T12530
| 1mg | 113.00 € | ||
| 5mg | 250.00 € | ||
| 10mg | 367.00 € | ||
| 25mg | 550.00 € | ||
| 50mg | 775.00 € | ||
| 100mg | 1,040.00 € | ||
| 500mg | 2,098.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Zatosetron maleate
CAS:123482-23-5
Zatosetron maleate(LY 277359 maleate) is a potent and selective serotonin 5HT3 receptor antagonist for the …
Formula:
C23H29ClN2O6
Purity:
99.41%
Color and Shape:
Solid
Molecular weight:
464.94
Ref: TM-T17285
| 1mg | 650.00 € | ||
| 5mg | 1,671.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Taprenepag isopropyl
CAS:1005549-94-9
Taprenepag isopropyl is a highly selective agonist of the EP2 receptor.
Formula:
C27H28N4O5S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
520.6
Ref: TM-T16988
| 2mg | 52.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
