G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Lodoxamide tromethamine
CAS:63610-09-3
Lodoxamide tromethamine is a mast cell stabilizer with anti-allergic properties and can be used in …
Formula:
C19H28ClN5O12
Purity:
99.58%
Color and Shape:
Solid
Molecular weight:
553.91
Ref: TM-T15772
| 5mg | 47.00 € | ||
| 10mg | 60.00 € | ||
| 25mg | 94.00 € | ||
| 50mg | 111.00 € | ||
| 100mg | 187.00 € | ||
| 200mg | 279.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Friday 2 May 2025
Ciproxifan
CAS:184025-18-1
Ciproxifan (FUB-359) is a highly effective and specific histamin H3-receptor antagonist (IC50: 9.2 nM).
Formula:
C16H18N2O2
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
270.33
Ref: TM-T6164
| 1mg | 44.00 € | ||
| 2mg | 55.00 € | ||
| 5mg | 81.00 € | ||
| 10mg | 111.00 € | ||
| 25mg | 225.00 € | ||
| 50mg | 401.00 € |
Estimated delivery in United States, on Friday 2 May 2025
Palosuran
CAS:540769-28-6
Palosuran (ACT-058362) (ACT-058362) is a new potent and specific antagonist of the human UT receptor.
Formula:
C25H30N4O2
Purity:
98.46%
Color and Shape:
Solid
Molecular weight:
418.53
Ref: TM-T2058
| 2mg | 47.00 € | ||
| 5mg | 74.00 € | ||
| 10mg | 107.00 € | ||
| 25mg | 235.00 € | ||
| 50mg | 393.00 € | ||
| 100mg | 645.00 € | ||
| 200mg | 898.00 € | ||
| 1mL*10mM (DMSO) | 202.00 € |
Estimated delivery in United States, on Friday 2 May 2025
NDT 9513727
CAS:439571-48-9
Complement C5a receptor (C5aR) antagonist
Formula:
C36H35N3O4
Purity:
Min. 95%
Molecular weight:
573.68 g/mol
Ref: 3D-BN162458
| 1mg | 219.00 € | ||
| 2mg | 350.00 € | ||
| 5mg | 511.00 € | ||
| 10mg | 766.00 € | ||
| 25mg | 1,309.00 € |
Estimated delivery in United States, on Friday 9 May 2025
LY 344864
CAS:186544-26-3
LY 344864, a specifc receptor agonist, is an affinity of 6 nM (Ki) at the …
Formula:
C21H22FN3O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
351.42
Ref: TM-T2344
| 2mg | 40.00 € | ||
| 5mg | 60.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 166.00 € | ||
| 50mg | 296.00 € | ||
| 100mg | 527.00 € | ||
| 1mL*10mM (DMSO) | 66.00 € |
Estimated delivery in United States, on Friday 9 May 2025
Clovoxamine
CAS:54739-19-4
Clovoxamine fumarate (DU 23811 fumarate) is a 5-HT reuptake, serotonin and norepinephrine inhibitor with antidepressant …
Formula:
C14H21ClN2O2
Purity:
98.88% - 99.16%
Color and Shape:
Solid
Molecular weight:
284.78
Ref: TM-T27047
| 1mg | 279.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € |
Estimated delivery in United States, on Friday 16 May 2025
GS-9667
CAS:618380-90-8
GS-9667, a selective and partial agonist of the A(1) adenosine receptor (AR), represents an effective …
Formula:
C21H24FN5O4S
Purity:
99.76% - 99.76%
Color and Shape:
Solid
Molecular weight:
461.51
Ref: TM-T27439
| 1mg | 111.00 € | ||
| 5mg | 274.00 € | ||
| 10mg | 376.00 € | ||
| 25mg | 620.00 € | ||
| 50mg | 847.00 € | ||
| 100mg | 1,169.00 € |
Estimated delivery in United States, on Friday 16 May 2025
RG 7152
CAS:107813-63-8
RG 7152 is a leukotriene D4 antagonist with anti-asthmatic properties and can be used in …
Formula:
C20H19N5O2
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
361.4
Ref: TM-T28529
| 1mg | 279.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € |
Estimated delivery in United States, on Friday 16 May 2025
ML-335
CAS:1069498-96-9
ML-335, a μ-δ targeted agonist and MOR/DOR ligand, may lead to isomer-biased drugs with pain-relief …
Formula:
C25H32N2O3
Purity:
98.52%
Color and Shape:
Solid
Molecular weight:
408.53
Ref: TM-T23002
| 2mg | 40.00 € | ||
| 5mg | 62.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 170.00 € | ||
| 50mg | 264.00 € | ||
| 100mg | 380.00 € | ||
| 200mg | 540.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Friday 16 May 2025
KI-7
CAS:1489263-00-4
KI-7 is an adenosine A2B receptor positive allosteric modulator.
Formula:
C23H18N2O2
Purity:
98.03%
Color and Shape:
Solid
Molecular weight:
354.4
Ref: TM-T9238
| 2mg | 38.00 € | ||
| 5mg | 58.00 € | ||
| 10mg | 90.00 € | ||
| 25mg | 182.00 € | ||
| 50mg | 279.00 € | ||
| 100mg | 420.00 € | ||
| 200mg | 592.00 € | ||
| 1mL*10mM (DMSO) | 65.00 € |
Estimated delivery in United States, on Friday 16 May 2025
NRA-0160
CAS:204718-47-8
NRA-0160 is a selective antagonist of dopamine D4 receptor(Ki of 0.48 nM)
Formula:
C24H23F2N3OS
Purity:
98%
Color and Shape:
Solid
Molecular weight:
439.52
Ref: TM-T12252
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Friday 16 May 2025
CJ 033466
CAS:519148-48-2
CJ 033466 is a selective partial agonist of 5-HT4 receptor (EC50 = 9 nM) with …
Formula:
C19H28ClN5O
Purity:
98.41%
Color and Shape:
Solid
Molecular weight:
377.91
Ref: TM-T22671
| 1mg | 48.00 € | ||
| 5mg | 101.00 € | ||
| 10mg | 170.00 € | ||
| 25mg | 270.00 € | ||
| 50mg | 386.00 € | ||
| 100mg | 520.00 € | ||
| 1mL*10mM (DMSO) | 158.00 € |
Estimated delivery in United States, on Friday 16 May 2025
Eplivanserin
CAS:130579-75-8
Eplivanserin (SR-46349) is an effective and selective antagonist of 5-HT2A receptor with a Kd of …
Formula:
C19H21FN2O2
Purity:
97.04%
Color and Shape:
Solid
Molecular weight:
328.38
Ref: TM-T11217
| 1mg | 185.00 € | ||
| 5mg | 415.00 € | ||
| 10mg | 613.00 € | ||
| 25mg | 938.00 € | ||
| 50mg | 1,311.00 € | ||
| 1mL*10mM (DMSO) | 420.00 € |
Estimated delivery in United States, on Friday 16 May 2025
NUCC-390
CAS:1060524-97-1
NUCC-390, a novel small-molecule CXCR4 receptor agonist, selectively induces CXCR4 receptor internalization while acting antagonistically …
Formula:
C23H33N5O
Purity:
98.18%
Color and Shape:
Solid
Molecular weight:
395.54
Ref: TM-T12269
| 1mg | 148.00 € | ||
| 5mg | 303.00 € | ||
| 10mg | 474.00 € | ||
| 25mg | 772.00 € | ||
| 50mg | 1,074.00 € | ||
| 100mg | 1,444.00 € | ||
| 500mg | 2,822.00 € | ||
| 1mL*10mM (DMSO) | 359.00 € |
Estimated delivery in United States, on Friday 16 May 2025
Nedocromil
CAS:69049-73-6
Nedocromil (FPL 59002) inhibits the action or formation of multiple mediators. Which including histamine, leukotriene …
Formula:
C19H17NO7
Purity:
95.00%
Color and Shape:
Solid
Molecular weight:
371.34
Ref: TM-T16280
| 5mg | 70.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 202.00 € | ||
| 50mg | 329.00 € | ||
| 100mg | 520.00 € |
Estimated delivery in United States, on Friday 16 May 2025
AT-121
CAS:2099681-31-7
AT-121 is a dual μ-opioid and neuropeptide receptor partial agonist (Kis 16.49 and 3.67 nM, …
Formula:
C24H38N4O3S
Purity:
97% - 97.95%
Color and Shape:
Solid
Molecular weight:
462.65
Ref: TM-T37610
| 1mg | 333.00 € | ||
| 5mg | 787.00 € | ||
| 10mg | 1,074.00 € | ||
| 25mg | 1,510.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € | ||
| 500mg | 4,655.00 € |
Estimated delivery in United States, on Friday 16 May 2025
DOV-216,303 Free Base
CAS:66504-40-3
DOV-216,303 inhibits serotonin, norepinephrine, dopamine reuptake (IC50s: 14, 20, 78 nM) with antidepressant properties.
Formula:
C11H11Cl2N
Purity:
96.7%
Color and Shape:
Solid
Molecular weight:
228.12
Ref: TM-T11087
| 2mg | 46.00 € | ||
| 5mg | 66.00 € | ||
| 10mg | 97.00 € | ||
| 25mg | 159.00 € | ||
| 50mg | 226.00 € | ||
| 100mg | 339.00 € | ||
| 1mL*10mM (DMSO) | 67.00 € |
Estimated delivery in United States, on Friday 16 May 2025
Seridopidine
CAS:883631-51-4
Seridopidine (ACR343) is a modulator of dopaminergic activity that is used as an oral therapy …
Formula:
C14H20FNO2S
Purity:
99.11%
Color and Shape:
Solid
Molecular weight:
285.38
Ref: TM-T34616
| 1mg | 139.00 € | ||
| 5mg | 333.00 € | ||
| 10mg | 504.00 € | ||
| 25mg | 817.00 € | ||
| 50mg | 1,121.00 € | ||
| 100mg | 1,510.00 € | ||
| 500mg | 3,030.00 € |
Estimated delivery in United States, on Friday 16 May 2025
Piclozotan
CAS:182415-09-4
Piclozotan (anhydrous), a 5-HT1A receptor agonist, demonstrated significant neuroprotective activity in a transient middle cerebral …
Formula:
C23H24ClN3O2
Purity:
99%
Color and Shape:
Solid
Molecular weight:
409.91
Ref: TM-T28414
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Friday 16 May 2025
MK-0686
CAS:578727-68-1
MK-0686 is an orally available bradykinin B1 receptor antagonist with potential anti-inflammatory activity.
Formula:
C22H19ClF4N2O4
Purity:
99.56%
Color and Shape:
Liquid
Molecular weight:
486.84
Ref: TM-T33421
| 1mg | 182.00 € | ||
| 5mg | 447.00 € | ||
| 10mg | 655.00 € | ||
| 25mg | 1,026.00 € | ||
| 50mg | 1,388.00 € | ||
| 100mg | 1,863.00 € | ||
| 500mg | 3,734.00 € |
Estimated delivery in United States, on Friday 16 May 2025
