G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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D-Kynurenine
CAS:13441-51-5
D-Kynurenine, ZINC901103, metabolizes from D-tryptophan, activates AhR, changes epithelium to mesenchyme, and tests for D-amino …
Formula:
C10H12N2O3
Purity:
97.08%
Color and Shape:
Solid
Molecular weight:
208.21
Ref: TM-T10938
| 25mg | 52.00 € | ||
| 50mg | 89.00 € | ||
| 100mg | 130.00 € | ||
| 200mg | 185.00 € |
Estimated delivery in United States, on Tuesday 8 Apr 2025
XL413
CAS:1169558-38-6
XL-413 is an oral CDC7 kinase inhibitor, potentially blocking DNA replication, mitosis, and cancer cell …
Formula:
C14H12ClN3O2
Purity:
100% - 99.38%
Color and Shape:
Solid
Molecular weight:
289.72
Ref: TM-T3352
| 1mg | 52.00 € | ||
| 5mg | 116.00 € | ||
| 10mg | 160.00 € | ||
| 25mg | 283.00 € | ||
| 50mg | 472.00 € | ||
| 100mg | 658.00 € |
Estimated delivery in United States, on Tuesday 8 Apr 2025
MK-5046
CAS:1022152-70-0
MK-5046 is a novel BRS-3 agonist, binding to BRS-3 with high affinity (mouse Ki = …
Formula:
C20H18F6N4O
Purity:
98.56%
Color and Shape:
Solid
Molecular weight:
444.37
Ref: TM-T2126
| 1mg | 84.00 € | ||
| 5mg | 170.00 € | ||
| 10mg | 251.00 € |
Estimated delivery in United States, on Tuesday 8 Apr 2025
Palosuran
CAS:540769-28-6
Palosuran (ACT-058362) (ACT-058362) is a new potent and specific antagonist of the human UT receptor.
Formula:
C25H30N4O2
Purity:
98.46%
Color and Shape:
Solid
Molecular weight:
418.53
Ref: TM-T2058
| 2mg | 47.00 € | ||
| 5mg | 74.00 € | ||
| 10mg | 107.00 € | ||
| 25mg | 235.00 € | ||
| 50mg | 393.00 € | ||
| 100mg | 645.00 € | ||
| 200mg | 898.00 € | ||
| 1mL*10mM (DMSO) | 202.00 € |
Estimated delivery in United States, on Tuesday 8 Apr 2025
Pardoprunox
CAS:269718-84-5
Pardoprunox (SLV-308) is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist …
Formula:
C12H15N3O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
233.27
Ref: TM-T1769
| 25mg | 842.00 € |
Estimated delivery in United States, on Tuesday 8 Apr 2025
NDT 9513727
CAS:439571-48-9
Complement C5a receptor (C5aR) antagonist
Formula:
C36H35N3O4
Purity:
Min. 95%
Molecular weight:
573.68 g/mol
Ref: 3D-BN162458
| 1mg | 230.00 € | ||
| 2mg | 345.00 € | ||
| 5mg | 538.00 € | ||
| 10mg | 805.00 € | ||
| 25mg | 1,377.00 € |
Estimated delivery in United States, on Tuesday 15 Apr 2025
LY 344864
CAS:186544-26-3
LY 344864, a specifc receptor agonist, is an affinity of 6 nM (Ki) at the …
Formula:
C21H22FN3O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
351.42
Ref: TM-T2344
| 2mg | 40.00 € | ||
| 5mg | 60.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 166.00 € | ||
| 50mg | 296.00 € | ||
| 100mg | 527.00 € | ||
| 1mL*10mM (DMSO) | 66.00 € |
Estimated delivery in United States, on Tuesday 15 Apr 2025
Xamoterol hemifumarate
CAS:73210-73-8
Xamoterol hemifumarate is a potent and selective β1-adrenoceptor agonist.Xamoterol hemifumarate is a potential compound for …
Formula:
C36H54N6O14
Purity:
99.79%
Color and Shape:
White Solid
Molecular weight:
794.37
Ref: TM-T23536
| 1mg | 49.00 € | ||
| 5mg | 97.00 € | ||
| 10mg | 156.00 € | ||
| 25mg | 311.00 € | ||
| 50mg | 512.00 € | ||
| 100mg | 817.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Radioprotectin-1
CAS:1622006-09-0
Radioprotectin-1 is a selective agonist of LPA2 with EC50 of 25 nM for murine LPA2 …
Formula:
C23H19ClN2O6S
Purity:
98.75% - 99.43%
Color and Shape:
Solid
Molecular weight:
486.92
Ref: TM-T12684
| 1mg | 81.00 € | ||
| 5mg | 170.00 € | ||
| 10mg | 259.00 € | ||
| 25mg | 425.00 € | ||
| 50mg | 562.00 € | ||
| 100mg | 775.00 € | ||
| 1mL*10mM (DMSO) | 187.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
(R)-ZINC-3573
CAS:2089389-15-9
ZINC-3573: Potent, selective MRGPRX2 activator; triggers mast cell degranulation and calcium release.
Formula:
C18H21N5
Purity:
100%
Color and Shape:
Solid
Molecular weight:
307.39
Ref: TM-T29221
| 2mg | 47.00 € | ||
| 5mg | 70.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 216.00 € | ||
| 50mg | 325.00 € | ||
| 100mg | 472.00 € | ||
| 1mL*10mM (DMSO) | 77.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Lesopitron dihydrochloride
CAS:132449-89-9
Lesopitron dihydrochloride with IC50 of 125 nM in rat hippocampal membranes, is a full and …
Formula:
C15H23Cl3N6
Purity:
98%
Color and Shape:
Solid
Molecular weight:
393.74
Ref: TM-T11839
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Elinogrel
CAS:936500-94-6
Elinogrel (PRT060128) is a competitive and reversible antagonist of platelet P2Y12 with IC50 of 20 …
Formula:
C20H15ClFN5O5S2
Purity:
97.09%
Color and Shape:
Solid
Molecular weight:
523.95
Ref: TM-T11177
| 1mg | 56.00 € | ||
| 5mg | 104.00 € | ||
| 10mg | 160.00 € | ||
| 25mg | 274.00 € | ||
| 50mg | 393.00 € | ||
| 100mg | 550.00 € | ||
| 200mg | 785.00 € | ||
| 1mL*10mM (DMSO) | 120.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Ecopipam
CAS:112108-01-7
Ecopipam: orally active, selective dopamine D1/D5 antagonist (Ki: 1.2 nM/2.0 nM). 40x more selective over …
Formula:
C19H20ClNO
Purity:
98.5%
Color and Shape:
Solid
Molecular weight:
313.82
Ref: TM-T31602
| 1mg | 185.00 € | ||
| 2mg | 279.00 € | ||
| 5mg | 424.00 € | ||
| 10mg | 627.00 € | ||
| 25mg | 938.00 € | ||
| 50mg | 1,311.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Rec 15/2615 dihydrochloride
CAS:173059-17-1
Rec 15/2615 dihydrochloride is an antagonist of α1B-adrenergic receptor.
Formula:
C26H35Cl2N5O5
Purity:
98.97% - 99.81%
Color and Shape:
Solid
Molecular weight:
568.49
Ref: TM-T23230
| 1mg | 50.00 € | ||
| 5mg | 105.00 € | ||
| 10mg | 160.00 € | ||
| 25mg | 255.00 € | ||
| 50mg | 359.00 € | ||
| 100mg | 485.00 € | ||
| 200mg | 657.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
ASP-4058
CAS:952565-91-2
ASP-4058: Safe, oral S1P1/S1P5 agonist; improves autoimmune encephalomyelitis in mice.
Formula:
C19H12F6N4O2
Purity:
99.5% - 99.51%
Color and Shape:
Solid
Molecular weight:
442.31
Ref: TM-T10385
| 1mg | 99.00 € | ||
| 5mg | 235.00 € | ||
| 10mg | 376.00 € | ||
| 25mg | 680.00 € | ||
| 50mg | 932.00 € | ||
| 100mg | 1,311.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
2-Arachidonoylglycerol
CAS:53847-30-6
In the central nervous system, 2-Arachidonoylglycerol is a second endogenous cannabinoid ligand
Formula:
C23H38O4
Purity:
95%
Color and Shape:
Liquid
Molecular weight:
378.55
Ref: TM-T14011
| 1mg (26.4mM*100μL in Acetonitrile) | 116.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
GR 46611
CAS:185259-85-2
GR 46611 is a selective 5-HT1B and 5-HT1D receptor agonist and can be used in …
Formula:
C23H27N3O2
Purity:
99.9%
Color and Shape:
Solid
Molecular weight:
377.48
Ref: TM-T22808
| 1mg | 52.00 € | ||
| 5mg | 92.00 € | ||
| 10mg | 135.00 € | ||
| 25mg | 264.00 € | ||
| 50mg | 420.00 € | ||
| 100mg | 613.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Felypressin acetate
CAS:914453-97-7
Felypressin acetate (PLV-2) is an agonist of vasopressin 1 and acts on all arginine vasopressin …
Formula:
C48H69N13O13S2
Purity:
97.06%
Color and Shape:
Solid
Molecular weight:
1100.27
Ref: TM-T2568L
| 5mg | 47.00 € | ||
| 10mg | 70.00 € | ||
| 25mg | 126.00 € | ||
| 50mg | 187.00 € | ||
| 100mg | 298.00 € | ||
| 200mg | 444.00 € | ||
| 500mg | 715.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Remogliflozin etabonate
CAS:442201-24-3
Remogliflozin etabonate is a prodrug SGLT2 inhibitor; Ki for hSGLT2: 1.95μM, rSGLT2: 2.14μM, rSGLT1: 8.57μM, …
Formula:
C26H38N2O9
Purity:
99%
Color and Shape:
Solid
Molecular weight:
522.59
Ref: TM-T34286
| 2mg | 35.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 164.00 € | ||
| 50mg | 245.00 € | ||
| 100mg | 340.00 € | ||
| 200mg | 472.00 € | ||
| 1mL*10mM (DMSO) | 62.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Litoxetine
CAS:86811-09-8
Litoxetine: a selective 5-HT inhibitor & 5-HT3 antagonist, used as an antidepressant with antiemetic effects, …
Formula:
C16H19NO
Purity:
99.12%
Color and Shape:
Liquid
Molecular weight:
241.33
Ref: TM-T67956
| 1mg | 97.00 € | ||
| 5mg | 217.00 € | ||
| 10mg | 325.00 € | ||
| 25mg | 557.00 € | ||
| 50mg | 797.00 € | ||
| 100mg | 1,103.00 € | ||
| 500mg | 2,205.00 € | ||
| 1mL*10mM (DMSO) | 188.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
