G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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JNJ-39220675
CAS:959740-39-7
JNJ-39220675, a selective histamine H3 receptor antagonist, reduces the abuse-related effects of alcohol in rats.
Formula:
C21H24FN3O2
Purity:
97.95% - 99.78%
Color and Shape:
Solid
Molecular weight:
369.43
Ref: TM-T27678
| 1mg | 274.00 € | ||
| 5mg | 673.00 € | ||
| 10mg | 920.00 € | ||
| 25mg | 1,417.00 € | ||
| 50mg | 1,846.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Roxindole
CAS:112192-04-8
Roxindole: dopamine agonist, serotonin reuptake inhibitor, 5-HT1A agonist, developed for schizophrenia.
Formula:
C23H26N2O
Purity:
99.08% - 99.18%
Color and Shape:
Solid
Molecular weight:
346.47
Ref: TM-T26126
| 1mg | 274.00 € | ||
| 5mg | 673.00 € | ||
| 10mg | 920.00 € | ||
| 25mg | 1,417.00 € | ||
| 50mg | 1,852.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Iodophenpropit dihydrobromide
CAS:145196-87-8
Iodophenpropit dihydrobromide: selective histamine H3 antagonist, reversible binding, high affinity (KD: 0.32 nM).
Formula:
C15H20BrIN4S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
495.22
Ref: TM-T15590
| 5mg | 279.00 € | ||
| 10mg | 418.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
ANR 94
CAS:634924-89-3
ANR94 is a potent hAA2AR antagonist (Ki 46 nM) with potential for Parkinson's research.
Formula:
C9H13N5O
Purity:
98.21%
Color and Shape:
Solid
Molecular weight:
207.23
Ref: TM-T22031
| 2mg | 41.00 € | ||
| 5mg | 62.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 182.00 € | ||
| 50mg | 318.00 € | ||
| 100mg | 449.00 € | ||
| 200mg | 631.00 € | ||
| 1mL*10mM (DMSO) | 61.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Arbutamine
CAS:128470-16-6
Arbutamine (GP 21213) is a β-adrenoceptor agonist with alpha-1-sympathomimetic activity that can be used to …
Formula:
C18H23NO4
Purity:
95.06%
Color and Shape:
Solid
Molecular weight:
317.38
Ref: TM-T10364
| 1mg | 378.00 € | ||
| 5mg | 905.00 € | ||
| 10mg | 1,122.00 € | ||
| 25mg | 1,502.00 € | ||
| 50mg | 1,846.00 € | ||
| 100mg | 2,331.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
PGD2-IN-1
CAS:885066-67-1
PGD2-IN-1 (PGD2-inhibitor) is an effective DP receptor antagonist (IC50:0.3 nM), a compound that can inhibit …
Formula:
C23H23Cl2N3O3
Purity:
99%
Color and Shape:
Solid
Molecular weight:
460.35
Ref: TM-T4624
| 1mg | 69.00 € | ||
| 5mg | 156.00 € | ||
| 10mg | 255.00 € | ||
| 25mg | 428.00 € | ||
| 50mg | 631.00 € | ||
| 100mg | 895.00 € | ||
| 500mg | 1,791.00 € | ||
| 1mL*10mM (DMSO) | 167.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
L-168049
CAS:191034-25-0
L-168049: Human glucagon receptor antagonist, IC50 - 3.7 nM human, 63 nM murine, 60 nM …
Formula:
C24H20BrClN2O
Purity:
100%
Color and Shape:
Solid
Molecular weight:
467.79
Ref: TM-T22893
| 1mg | 52.00 € | ||
| 5mg | 110.00 € | ||
| 10mg | 176.00 € | ||
| 25mg | 369.00 € | ||
| 50mg | 551.00 € | ||
| 100mg | 783.00 € | ||
| 500mg | 1,613.00 € | ||
| 1mL*10mM (DMSO) | 123.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Quinupramine
CAS:31721-17-2
Quinupramine: an oral antidepressant targeting the serotonin system; penetrates CNS; doesn’t affect β-adrenergic system.
Formula:
C21H24N2
Purity:
99.76%
Color and Shape:
Liquid
Molecular weight:
304.43
Ref: TM-T60707
| 1mg | 431.00 € | ||
| 5mg | 998.00 € | ||
| 25mg | 1,985.00 € | ||
| 50mg | 2,591.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
E-3620
CAS:151213-86-4
E-3620 is a potent antagonist of the 5-HT3 receptor and can be used to study …
Formula:
C20H27Cl2N3O2
Purity:
98.88% - 98.88%
Color and Shape:
Liquid
Molecular weight:
412.35
Ref: TM-T62107
| 1mg | 183.00 € | ||
| 5mg | To inquire |
Estimated delivery in United States, on Monday 27 Jan 2025
SCH 546738
CAS:906805-42-3
SCH 546738 is an orally available, selective and potent CXCR3 antagonist that attenuates the development …
Formula:
C23H31Cl2N7O
Purity:
98.67%
Color and Shape:
Solid
Molecular weight:
492.45
Ref: TM-T16863
| 2mg | 215.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Parogrelil Free Base
CAS:139145-27-0
Parogrelil Free Base is a phosphodiesterase inhibitor, improves claudication-limited exercise performance in patients with peripheral …
Formula:
C19H18BrClN4O2
Purity:
98.48% - 99%
Color and Shape:
Liquid
Molecular weight:
449.73
Ref: TM-T70793
| 1mg | 274.00 € | ||
| 5mg | 673.00 € | ||
| 10mg | 920.00 € | ||
| 25mg | 1,417.00 € | ||
| 50mg | 1,846.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
S 14506 hydrochloride
CAS:286369-38-8
S 14506 hydrochloride is a 5-HT1A receptor full agonist.
Formula:
C24H27ClFN3O2
Purity:
99.5%
Color and Shape:
Solid
Molecular weight:
443.94
Ref: TM-T23285
| 1mg | 45.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 140.00 € | ||
| 25mg | 272.00 € | ||
| 50mg | 416.00 € | ||
| 100mg | 628.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Pitolisant
CAS:362665-56-3
Pitolisant is a potent and selective nonimidazole inverse agonist that acts on the recombinant human …
Formula:
C17H26ClNO
Purity:
99.84%
Color and Shape:
Liquid
Molecular weight:
295.85
Ref: TM-T60636
| 5mg | 47.00 € | ||
| 10mg | 69.00 € | ||
| 25mg | 119.00 € | ||
| 50mg | 185.00 € | ||
| 100mg | 306.00 € | ||
| 500mg | 734.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Neldazosin
CAS:109713-79-3
Neldazosin is used as a potent α1-adrenoceptor antagonist.
Formula:
C18H25N5O4
Purity:
100% - 99.87%
Color and Shape:
Liquid
Molecular weight:
375.42
Ref: TM-T61535
| 1mg | 196.00 € | ||
| 5mg | 496.00 € | ||
| 10mg | 711.00 € | ||
| 25mg | 1,096.00 € | ||
| 50mg | 1,476.00 € | ||
| 100mg | 2,004.00 € | ||
| 500mg | 3,999.00 € | ||
| 1mL*10mM (DMSO) | 520.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
ADR-851 free base
CAS:138559-56-5
ADR-851 free base is an antagonist of the HT3 receptor.
Formula:
C14H18ClN3O2
Purity:
97.88% - 98.32%
Color and Shape:
Solid
Molecular weight:
295.77
Ref: TM-T23642
| 1mg | 274.00 € | ||
| 5mg | 673.00 € | ||
| 10mg | 920.00 € | ||
| 25mg | 1,417.00 € | ||
| 50mg | 1,846.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Crinecerfont
CAS:752253-39-7
Crinecerfont (SSR-125543) is a CRF1 antagonist, useful in congenital adrenal hyperplasia research.
Formula:
C27H28ClFN2OS
Purity:
98.01% - 99.10%
Color and Shape:
Solid
Molecular weight:
483.04
Ref: TM-T31095
| 1mg | 113.00 € | ||
| 2mg | 169.00 € | ||
| 5mg | 250.00 € | ||
| 10mg | 367.00 € | ||
| 25mg | 550.00 € | ||
| 50mg | 775.00 € | ||
| 100mg | 1,040.00 € | ||
| 500mg | 2,098.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Tildacerfont
CAS:1014983-00-6
Tildacerfont inhibits CRF1, lowers ACTH/adrenal androgens, and aids in congenital adrenal hyperplasia research.
Formula:
C20H26ClN5OS
Purity:
100.00%
Color and Shape:
Solid
Molecular weight:
419.97
Ref: TM-T26278
| 5mg | 35.00 € | ||
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 27 Jan 2025
CMF019
CAS:1586787-08-7
CMF019 is a potent agonist of the Apelin receptor (APJ) with G protein bias. CMF019 …
Formula:
C25H33N3O3S
Purity:
98.54%
Color and Shape:
Solid
Molecular weight:
455.61
Ref: TM-T10843
| 1mg | 118.00 € | ||
| 5mg | 241.00 € | ||
| 10mg | 407.00 € | ||
| 25mg | 663.00 € | ||
| 50mg | 919.00 € | ||
| 100mg | 1,226.00 € | ||
| 1mL*10mM (DMSO) | 244.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
SB-209670
CAS:157659-79-5
SB-209670 is a selective endothelin receptor antagonist that inhibits the activity of ET(B) receptors in …
Formula:
C29H28O9
Purity:
97.39% - 99.24%
Color and Shape:
Solid
Molecular weight:
520.53
Ref: TM-T34541
| 1mg | 325.00 € | ||
| 5mg | 769.00 € | ||
| 10mg | 1,054.00 € | ||
| 25mg | 1,476.00 € | ||
| 50mg | 1,846.00 € | ||
| 100mg | 2,320.00 € | ||
| 500mg | 4,577.00 € | ||
| 1mL*10mM (DMSO) | 791.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Nemazoline Free Base
CAS:130759-56-7
Nemazoline Free Base: a long-lasting nasal decongestant, better than oxymetazoline, with no systemic effects or …
Formula:
C10H11Cl2N3
Purity:
99.03% - 99.18%
Color and Shape:
Liquid
Molecular weight:
244.12
Ref: TM-T71012
| 1mg | 274.00 € | ||
| 5mg | 673.00 € | ||
| 10mg | 920.00 € | ||
| 25mg | 1,417.00 € | ||
| 50mg | 1,846.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
