G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Immethridine dihydrobromide
CAS:699020-93-4
Immethridine dihydrobromide is a histamine H3 receptor agonist.
Formula:
C9H11Br2N3
Purity:
97.49% - 98.16%
Color and Shape:
Solid
Molecular weight:
321.01
Ref: TM-T22864
| 1mg | 63.00 € | ||
| 5mg | 183.00 € | ||
| 10mg | 245.00 € | ||
| 25mg | 549.00 € | ||
| 50mg | 915.00 € | ||
| 100mg | 1,258.00 € | ||
| 500mg | 2,497.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Soquinolol
CAS:61563-18-6
Soquinolol (Soquinolol mucate) is a beta-adrenergic receptor antagonist with weak local anesthetic activity.Soquinolol has good …
Formula:
C17H26N2O3
Purity:
98% - 98.49%
Color and Shape:
Solid
Molecular weight:
306.4
Ref: TM-T28829
| 1mg | 141.00 € | ||
| 5mg | 325.00 € | ||
| 10mg | 492.00 € | ||
| 25mg | 803.00 € | ||
| 50mg | 1,095.00 € | ||
| 100mg | 1,483.00 € | ||
| 500mg | 2,974.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Neldazosin
CAS:109713-79-3
Neldazosin is used as a potent α1-adrenoceptor antagonist.
Formula:
C18H25N5O4
Purity:
100% - 99.87%
Color and Shape:
Solid
Molecular weight:
375.42
Ref: TM-T61535
| 1mg | 196.00 € | ||
| 5mg | 496.00 € | ||
| 10mg | 711.00 € | ||
| 25mg | 1,096.00 € | ||
| 50mg | 1,476.00 € | ||
| 100mg | 2,004.00 € | ||
| 500mg | 3,999.00 € | ||
| 1mL*10mM (DMSO) | 520.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Cinitapride Hydrogen Tartrate
CAS:1207859-16-2
Cinitapride Hydrogen Tartrate is a gastroprokinetic agent that acts as an antagonist of the 5-HT2 …
Formula:
C25H36N4O10
Purity:
98%
Color and Shape:
Solid
Molecular weight:
552.581
Ref: TM-T22294
| 25mg | 1,410.00 € | ||
| 50mg | 1,852.00 € | ||
| 100mg | 2,338.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
CV-6209
CAS:100488-87-7
CV-6209 is a potent antagonist of the platelet-activating factor (PAF) receptor.
Formula:
C34H60ClN3O6
Purity:
100% - 100%
Color and Shape:
Solid
Molecular weight:
642.31
Ref: TM-T27102
| 1mg | 125.00 € | ||
| 5mg | 529.00 € | ||
| 10mg | 830.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
SB-209670
CAS:157659-79-5
SB-209670 is a selective endothelin receptor antagonist that inhibits the activity of ET(B) receptors in …
Formula:
C29H28O9
Purity:
97.39% - 99.24%
Color and Shape:
Solid
Molecular weight:
520.53
Ref: TM-T34541
| 1mg | 325.00 € | ||
| 5mg | 769.00 € | ||
| 10mg | 1,054.00 € | ||
| 25mg | 1,476.00 € | ||
| 50mg | 1,846.00 € | ||
| 100mg | 2,320.00 € | ||
| 500mg | 4,577.00 € | ||
| 1mL*10mM (DMSO) | 791.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
SB 611812
CAS:345892-71-9
SB 611812 is an antagonist of urotensin-II (UT) and can be used in studies about …
Formula:
C17H16Cl3F3N2O3S
Purity:
99.34%
Color and Shape:
Solid
Molecular weight:
491.74
Ref: TM-T23323
| 1mg | 45.00 € | ||
| 5mg | 89.00 € | ||
| 10mg | 143.00 € | ||
| 25mg | 300.00 € | ||
| 50mg | 434.00 € | ||
| 100mg | 609.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Molindone
CAS:7416-34-4
Molindone: antipsychotic for schizophrenia; blocks dopamine, often paired with serotonin; dosage affects error/response rates.
Formula:
C16H24N2O2
Purity:
98% - 99.37%
Color and Shape:
Off-White Solid
Molecular weight:
276.37
Ref: TM-T21432
| 1mg | 325.00 € | ||
| 5mg | 769.00 € | ||
| 10mg | 1,054.00 € | ||
| 25mg | 1,477.00 € | ||
| 50mg | 1,846.00 € | ||
| 100mg | 2,331.00 € | ||
| 500mg | 4,547.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
4-PPBP maleate
CAS:201216-39-9
4-PPBP maleate: potent σ1 agonist, selective NR1a/2B NMDA antagonist, neuroprotective.
Formula:
C25H31NO4
Purity:
99.54%
Color and Shape:
Solid
Molecular weight:
409.52
Ref: TM-T22513
| 5mg | 73.00 € | ||
| 10mg | 109.00 € | ||
| 25mg | 212.00 € | ||
| 50mg | 343.00 € | ||
| 100mg | 510.00 € | ||
| 500mg | 1,093.00 € | ||
| 1mL*10mM (DMSO) | 93.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
8-OH-Dpat
CAS:78950-78-4
8-OH-Dpat (8-Hydroxy-DPAT) is a serotonin 1A-receptor agonist that is used experimentally to test the effects …
Formula:
C16H25NO
Purity:
98%
Color and Shape:
Solid
Molecular weight:
247.38
Ref: TM-T4305
| 5mg | 46.00 € | ||
| 10mg | 59.00 € | ||
| 25mg | 109.00 € | ||
| 50mg | 172.00 € | ||
| 100mg | 252.00 € | ||
| 1mL*10mM (DMSO) | 53.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Fallypride
CAS:166173-78-0
Fallypride is a potent and selective dopamine D2/D3 receptor antagonist.
Formula:
C20H29FN2O3
Purity:
100% - 99.17%
Color and Shape:
Liquid
Molecular weight:
364.45
Ref: TM-T70302
| 1mg | 355.00 € | ||
| 5mg | 831.00 € | ||
| 10mg | 1,023.00 € | ||
| 25mg | 1,623.00 € | ||
| 50mg | 2,033.00 € | ||
| 100mg | 2,611.00 € | ||
| 1mL*10mM (DMSO) | 668.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
CGP 35949
CAS:111130-13-3
CGP 35949 is an LTD4 antagonist with phospholipase inhibitory activity.
Formula:
C23H25ClN5NaO5
Purity:
98.89%
Color and Shape:
Solid
Molecular weight:
509.92
Ref: TM-T30828
| 1mg | 113.00 € | ||
| 2mg | 169.00 € | ||
| 5mg | 249.00 € | ||
| 10mg | 367.00 € | ||
| 25mg | 550.00 € | ||
| 50mg | 769.00 € | ||
| 100mg | 1,049.00 € | ||
| 500mg | 2,108.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Pridefine
CAS:5370-41-2
Pridefine: antidepressant, balances serotonin, dopamine, norepinephrine reuptake, weakly releases them.
Formula:
C19H21N
Purity:
99.05% - 99.23%
Color and Shape:
Solid
Molecular weight:
263.38
Ref: TM-T24661
| 1mg | 274.00 € | ||
| 5mg | 673.00 € | ||
| 10mg | 920.00 € | ||
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
U 99194 maleate
CAS:234757-41-6
U 99194 maleate (U-99194A maleate) is a D3 antagonist and increases social behaviors of isolation-induced …
Formula:
C21H31NO6
Purity:
99.45%
Color and Shape:
Solid
Molecular weight:
393.47
Ref: TM-T23483
| 1mg | 91.00 € | ||
| 2mg | 121.00 € | ||
| 5mg | 177.00 € | ||
| 10mg | 212.00 € | ||
| 25mg | 467.00 € | ||
| 50mg | 678.00 € | ||
| 100mg | 926.00 € | ||
| 200mg | 724.00 € | ||
| 500mg | 1,846.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
SB 699551 dihydrochloride
CAS:864741-95-7
SB 699551 dihydrochloride is a 5-ht5a receptor antagonist.
Formula:
C34H47Cl2N3O
Purity:
96.53%
Color and Shape:
Solid
Molecular weight:
584.66
Ref: TM-T23325
| 1mg | 51.00 € | ||
| 5mg | 107.00 € | ||
| 10mg | 173.00 € | ||
| 25mg | 306.00 € | ||
| 50mg | 440.00 € | ||
| 100mg | 603.00 € | ||
| 1mL*10mM (DMSO) | 145.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
F13714 fumarate
CAS:208109-39-1
F13714 fumarate is a 5-HT1A receptor-biased agonist.
Formula:
C25H29ClF2N4O5
Color and Shape:
Solid
Molecular weight:
538.97
Ref: TM-T37622
| 1mg | 55.00 € | ||
| 5mg | 116.00 € | ||
| 10mg | 181.00 € | ||
| 25mg | 376.00 € | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 14 Jan 2025
AS-35
CAS:108427-72-1
AS-35, an oral selective leukotriene antagonist, counters ileum contractions with IC50: 8 nM (LTC4), 4 …
Formula:
C21H20N6O4
Purity:
98.68%
Color and Shape:
Solid
Molecular weight:
420.42
Ref: TM-T14326
| 1mg | 273.00 € | ||
| 2mg | 406.00 € | ||
| 5mg | 672.00 € | ||
| 10mg | 919.00 € | ||
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Falintolol
CAS:90581-63-8
Falintolol is a novel beta-adrenergic antagonist with antihypertensive effects and can be used to study …
Formula:
C12H24N2O2
Purity:
100% - 100%
Color and Shape:
Liquid
Molecular weight:
228.33
Ref: TM-T68402
| 1mg | 277.00 € | ||
| 5mg | 682.00 € | ||
| 10mg | 932.00 € | ||
| 25mg | 1,351.00 € | ||
| 50mg | 1,823.00 € | ||
| 100mg | 2,462.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
BMS 182874
CAS:153042-42-3
BMS 182874: Oral ETA antagonist, IC50=0.150 μM, Ki=0.055 μM, lowers hypertension in rats.
Formula:
C17H19N3O3S
Purity:
98.38%
Color and Shape:
Solid
Molecular weight:
345.42
Ref: TM-T26841
| 1mg | 73.00 € | ||
| 5mg | 157.00 € | ||
| 10mg | 244.00 € | ||
| 25mg | 422.00 € | ||
| 50mg | 601.00 € | ||
| 100mg | 827.00 € | ||
| 500mg | 1,687.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
SF-22
CAS:824981-55-7
SF-22 is a Y2R antagonist with potential anti-inflammatory activity that can be used to study …
Formula:
C28H26N2O3S
Purity:
99.09%
Color and Shape:
Liquid
Molecular weight:
470.58
Ref: TM-T71749
| 1mg | 36.00 € | ||
| 5mg | 74.00 € | ||
| 10mg | 111.00 € | ||
| 25mg | 233.00 € | ||
| 50mg | 374.00 € | ||
| 100mg | 594.00 € | ||
| 500mg | 1,217.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
