G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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5-HT3 antagonist 2
CAS:128199-93-9
5-HT3 antagonist 2 is an antagonist of 5-HT3 receptor.
Formula:
C18H21N3O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
295.38
Ref: TM-T12988
| 25mg | 1,410.00 € | ||
| 50mg | 1,852.00 € | ||
| 100mg | 2,338.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
GPR40/FFAR1 modulator 1
CAS:874755-26-7
GPR40/FFAR1 modulator 1 is a Gq-coupled free fatty acid receptor 1 (GPR40/FFAR1) agonist and allosteric …
Formula:
C21H19N5O3
Purity:
99.72%
Color and Shape:
Solid
Molecular weight:
389.41
Ref: TM-T11458
| 1ml | 51.00 € | ||
| 10mg | 51.00 € | ||
| 25mg | 84.00 € | ||
| 50mg | 124.00 € | ||
| 100mg | 182.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Burixafor hydrobromide
CAS:1191450-19-7
Burixafor hydrobromide is an oral CXCR4 blocker with anti-angiogenic properties, potentially treating choroid neovascularization.
Formula:
C27H52BrN8O3P
Purity:
98%
Color and Shape:
Solid
Molecular weight:
647.644
Ref: TM-T10635
| 25mg | To inquire | ||
| 50mg | To inquire | ||
| 100mg | To inquire |
Estimated delivery in United States, on Monday 25 Nov 2024
TC LPA5 4
CAS:1393814-38-4
TC LPA5 4 is a LPA5 receptor antagonist.
Formula:
C23H23ClN2O3
Purity:
99.05%
Color and Shape:
Solid
Molecular weight:
410.89
Ref: TM-T23438
| 1mg | 58.00 € | ||
| 5mg | 124.00 € | ||
| 10mg | 183.00 € | ||
| 25mg | 425.00 € | ||
| 50mg | 625.00 € | ||
| 100mg | 891.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
GPR35 agonist 3
CAS:123021-85-2
GPR35 agonist 3 is a synthetic GPR35 agonist used in the study of cancer, type …
Formula:
C12H9NO5S
Purity:
98.79%
Color and Shape:
Solid
Molecular weight:
279.27
Ref: TM-T72755
| 1mg | 49.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 151.00 € | ||
| 25mg | 301.00 € | ||
| 50mg | 482.00 € | ||
| 100mg | 771.00 € | ||
| 500mg | 1,539.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Calhex 231 hydrochloride
CAS:2387505-78-2
Calhex 231 hydrochloride, a CaSR antagonist, may treat diabetic cardiomyopathy; IC50 is 0.39 μM in …
Formula:
C25H28Cl2N2O
Color and Shape:
Solid
Molecular weight:
443.41
Ref: TM-T10666
| 2mg | 95.00 € | ||
| 5mg | 144.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Octimibate
CAS:89838-96-0
Octimibate: non-prostaglandin antiplatelet, treats cardiovascular disease, aids atherosclerosis/thrombosis research.
Formula:
C29H30N2O3
Purity:
99.49%
Color and Shape:
Solid
Molecular weight:
454.56
Ref: TM-T24567
| 1mg | 138.00 € | ||
| 5mg | 335.00 € | ||
| 10mg | 492.00 € | ||
| 25mg | 798.00 € | ||
| 50mg | 1,096.00 € | ||
| 100mg | 1,483.00 € | ||
| 500mg | 2,960.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
CB1R Allosteric modulator 3
CAS:2633686-36-7
CB1R Allosteric modulator 3 is a CB1R modulator.CB1R Allosteric modulator 3 inhibits cAMP, and can …
Formula:
C22H17ClN2O2
Purity:
98.18%
Color and Shape:
Solid
Molecular weight:
376.84
Ref: TM-T61562
| 1mg | 42.00 € | ||
| 2mg | 55.00 € | ||
| 5mg | 89.00 € | ||
| 10mg | 136.00 € | ||
| 25mg | 220.00 € | ||
| 50mg | 328.00 € | ||
| 100mg | 486.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
SK1-IN-1
CAS:1218816-71-7
SK1-IN-1 is a SPHK1 inhibitor (IC50: 58 nM), with potential anticancer activity, and can be …
Formula:
C22H30N4O3
Purity:
98.72%
Color and Shape:
Solid
Molecular weight:
398.5
Ref: TM-T12927
| 1mg | 197.00 € | ||
| 1ml | 278.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
CB1R antagonist 1
CAS:334668-69-8
CB1R antagonist 1 is a potent CB1R antagonist that can be used to study diseases …
Formula:
C18H23F3N2O3S
Purity:
99.65%
Color and Shape:
Solid
Molecular weight:
404.45
Ref: TM-T61989
| 5mg | 73.00 € | ||
| 10mg | 114.00 € | ||
| 25mg | 184.00 € | ||
| 50mg | 273.00 € | ||
| 100mg | 407.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
GALNON
CAS:475115-35-6
Galnon is a galanin receptor agonist, improves intrinsic cortical bone tissue properties
Formula:
C40H46N4O6
Purity:
98%
Color and Shape:
Solid
Molecular weight:
678.82
Ref: TM-T8456
| 25mg | 759.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
CP-866087
CAS:519052-04-1
CP-866087 is a novel, potent and selective mu-opioid receptor antagonist for the study of female …
Formula:
C24H28N2O2
Purity:
100% - 99.44%
Color and Shape:
Soild
Molecular weight:
376.49
Ref: TM-T31081
| 1mg | 707.00 € | ||
| 5mg | 1,486.00 € | ||
| 25mg | 1,976.00 € | ||
| 50mg | 2,412.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
PRX-08066 Maleic acid
CAS:866206-55-5
PRX-08066 Maleic acid is a selective 5-HT2B receptor antagonist with IC50 of 3.4 nM, prevents …
Formula:
C19H17ClFN5S·C4H4O4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
517.96
Ref: TM-T6959
| 1ml | 400.00 € | ||
| 5mg | 169.00 € | ||
| 10mg | 229.00 € | ||
| 25mg | 411.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
I942
CAS:868145-09-9
I942 is a novel, selective ACyclic nucleotide (NCN) EPAC1 agonist that activates exchange proteins to …
Formula:
C20H19NO4S
Purity:
99.75%
Color and Shape:
Solid
Molecular weight:
369.43
Ref: TM-T24154
| 1mg | 93.00 € | ||
| 5mg | 223.00 € | ||
| 10mg | 362.00 € | ||
| 25mg | 593.00 € | ||
| 50mg | 820.00 € | ||
| 100mg | 1,105.00 € | ||
| 500mg | 2,256.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
NNC 92-1687
CAS:22903-37-3
NNC 92-1687 is a selective glucagon receptor antagonist that can be used to study type …
Formula:
C15H12N2O3S
Purity:
98.93% - 99.72%
Color and Shape:
Solid
Molecular weight:
300.33
Ref: TM-T28182
| 1mg | 376.00 € | ||
| 5mg | 905.00 € | ||
| 10mg | 1,117.00 € | ||
| 25mg | 1,496.00 € | ||
| 50mg | 1,839.00 € | ||
| 100mg | 2,321.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
GPR84 antagonist 8
CAS:1445846-30-9
GPR84 antagonist 8 is a selective GPR84 antagonist.
Formula:
C23H23N3O5
Color and Shape:
Solid
Molecular weight:
421.45
Ref: TM-T11462
| 25mg | 4,212.00 € | ||
| 50mg | 5,896.00 € | ||
| 100mg | 8,259.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
MG 1
CAS:148274-76-4
MG 1 is a potent alpha-1 adrenergic receptor antagonist.
Formula:
C17H25N3O2
Purity:
100% - 99.73%
Color and Shape:
Solid
Molecular weight:
303.4
Ref: TM-T12030
| 1mg | 650.00 € | ||
| 5mg | 1,671.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
BAY-1316957
CAS:1613264-40-6
BAY-1316957 is a highly potent and selective EP4 receptor antagonist. With an IC50 of 15.3 …
Formula:
C27H27N3O3
Color and Shape:
Solid
Molecular weight:
441.52
Ref: TM-T14500
| 50mg | 739.00 € | ||
| 100mg | 1,198.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Licogliflozin
CAS:1291094-73-9
Licogliflozin (LIK066) is an inhibitor of sodium-glucose cotransporter (SGLT1 and SGLT2).
Formula:
C23H28O7
Purity:
98%
Color and Shape:
Solid
Molecular weight:
416.46
Ref: TM-T15752
| 25mg | 800.00 € | ||
| 50mg | 1,049.00 € | ||
| 100mg | 1,741.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
L-692429
CAS:145455-23-8
L-692429 (MK-0751) is a GHS agonist with high affinity for G protein-coupled receptors and can …
Formula:
C29H31N7O2
Purity:
98.64% - 99.90%
Color and Shape:
Solid
Molecular weight:
509.614
Ref: TM-T11798
| 1mg | 152.00 € | ||
| 1ml | 420.00 € | ||
| 5mg | 371.00 € | ||
| 10mg | 546.00 € | ||
| 25mg | 890.00 € | ||
| 50mg | 1,208.00 € | ||
| 100mg | 1,623.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
