G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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ANR 94
CAS:634924-89-3
ANR94 is a potent hAA2AR antagonist (Ki 46 nM) with potential for Parkinson's research.
Formula:
C9H13N5O
Purity:
98.21%
Color and Shape:
Solid
Molecular weight:
207.23
Ref: TM-T22031
| 2mg | 42.00 € | ||
| 5mg | 64.00 € | ||
| 10mg | 97.00 € | ||
| 25mg | 188.00 € | ||
| 50mg | 329.00 € | ||
| 100mg | 465.00 € | ||
| 200mg | 655.00 € | ||
| 1mL*10mM (DMSO) | 63.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Arbutamine
CAS:128470-16-6
Arbutamine (GP 21213) is a β-adrenoceptor agonist with alpha-1-sympathomimetic activity that can be used to …
Formula:
C18H23NO4
Purity:
95.06%
Color and Shape:
Solid
Molecular weight:
317.38
Ref: TM-T10364
| 1mg | 378.00 € | ||
| 5mg | 922.00 € | ||
| 10mg | 1,121.00 € | ||
| 500µg | 255.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
PGD2-IN-1
CAS:885066-67-1
PGD2-IN-1 (PGD2-inhibitor) is an effective DP receptor antagonist (IC50:0.3 nM), a compound that can inhibit …
Formula:
C23H23Cl2N3O3
Purity:
99%
Color and Shape:
Solid
Molecular weight:
460.35
Ref: TM-T4624
| 1mg | 70.00 € | ||
| 5mg | 159.00 € | ||
| 10mg | 259.00 € | ||
| 25mg | 437.00 € | ||
| 50mg | 643.00 € | ||
| 100mg | 914.00 € | ||
| 500mg | 1,833.00 € | ||
| 1mL*10mM (DMSO) | 168.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
L-168049
CAS:191034-25-0
L-168049: Human glucagon receptor antagonist, IC50 - 3.7 nM human, 63 nM murine, 60 nM …
Formula:
C24H20BrClN2O
Purity:
100%
Color and Shape:
Solid
Molecular weight:
467.79
Ref: TM-T22893
| 1mg | 52.00 € | ||
| 5mg | 111.00 € | ||
| 10mg | 180.00 € | ||
| 25mg | 378.00 € | ||
| 50mg | 560.00 € | ||
| 100mg | 800.00 € | ||
| 500mg | 1,644.00 € | ||
| 1mL*10mM (DMSO) | 123.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Quinupramine
CAS:31721-17-2
Quinupramine: an oral antidepressant targeting the serotonin system; penetrates CNS; doesn’t affect β-adrenergic system.
Formula:
C21H24N2
Purity:
99.76%
Color and Shape:
Liquid
Molecular weight:
304.43
Ref: TM-T60707
| 1mg | 439.00 € | ||
| 5mg | 1,017.00 € | ||
| 25mg | 2,023.00 € | ||
| 50mg | 2,642.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
E-3620
CAS:151213-86-4
E-3620 is a potent antagonist of the 5-HT3 receptor and can be used to study …
Formula:
C20H27Cl2N3O2
Purity:
98.88% - 98.88%
Color and Shape:
Liquid
Molecular weight:
412.35
Ref: TM-T62107
| 1mg | 187.00 € | ||
| 5mg | To inquire |
Estimated delivery in United States, on Tuesday 22 Apr 2025
AM-4668
CAS:1011531-27-3
AM-4668: Type 2 diabetes GPR40 agonist with EC50s of 3.6 nM (IP3 assay) and 36 …
Formula:
C24H19F3N2O4S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
488.48
Ref: TM-T14202
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Parogrelil Free Base
CAS:139145-27-0
Parogrelil Free Base is a phosphodiesterase inhibitor, improves claudication-limited exercise performance in patients with peripheral …
Formula:
C19H18BrClN4O2
Purity:
98.48% - 99%
Color and Shape:
Liquid
Molecular weight:
449.73
Ref: TM-T70793
| 1mg | 279.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Neldazosin
CAS:109713-79-3
Neldazosin is used as a potent α1-adrenoceptor antagonist.
Formula:
C18H25N5O4
Purity:
100% - 99.87%
Color and Shape:
Liquid
Molecular weight:
375.42
Ref: TM-T61535
| 1mg | 200.00 € | ||
| 5mg | 504.00 € | ||
| 10mg | 727.00 € | ||
| 25mg | 1,121.00 € | ||
| 50mg | 1,510.00 € | ||
| 100mg | 2,043.00 € | ||
| 500mg | 4,075.00 € | ||
| 1mL*10mM (DMSO) | 525.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Pitolisant
CAS:362665-56-3
Pitolisant is a potent and selective nonimidazole inverse agonist that acts on the recombinant human …
Formula:
C17H26ClNO
Purity:
99.84%
Color and Shape:
Liquid
Molecular weight:
295.85
Ref: TM-T60636
| 5mg | 48.00 € | ||
| 10mg | 70.00 € | ||
| 25mg | 120.00 € | ||
| 50mg | 188.00 € | ||
| 100mg | 311.00 € | ||
| 500mg | 747.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
ADR-851 free base
CAS:138559-56-5
ADR-851 free base is an antagonist of the HT3 receptor.
Formula:
C14H18ClN3O2
Purity:
97.88% - 98.32%
Color and Shape:
Solid
Molecular weight:
295.77
Ref: TM-T23642
| 1mg | 279.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
SB-277011 dihydrochloride
CAS:1226917-67-4
SB-277011 dihydrochloride: potent, selective D3 antagonist; orally bioavailable; crosses blood-brain barrier; pKi 8.0 for D3 …
Formula:
C28H32Cl2N4O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
511.49
Ref: TM-T12861L
| 1mg | 108.00 € | ||
| 5mg | 280.00 € | ||
| 10mg | 459.00 € | ||
| 25mg | 1,008.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
SB-209670
CAS:157659-79-5
SB-209670 is a selective endothelin receptor antagonist that inhibits the activity of ET(B) receptors in …
Formula:
C29H28O9
Purity:
97.39% - 99.24%
Color and Shape:
Solid
Molecular weight:
520.53
Ref: TM-T34541
| 1mg | 333.00 € | ||
| 5mg | 787.00 € | ||
| 10mg | 1,074.00 € | ||
| 25mg | 1,510.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € | ||
| 500mg | 4,655.00 € | ||
| 1mL*10mM (DMSO) | 797.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
EMDT
CAS:263744-72-5
EMDT oxalate is a selective 5-HT6 agonist, and has antidepressant effects.
Formula:
C15H22N2O
Purity:
98.33% - 98.46%
Color and Shape:
Solid
Molecular weight:
246.35
Ref: TM-T11183
| 1mg | 92.00 € | ||
| 2mg | 125.00 € | ||
| 5mg | 170.00 € | ||
| 10mg | 213.00 € | ||
| 25mg | 474.00 € | ||
| 50mg | 688.00 € | ||
| 100mg | 938.00 € | ||
| 500mg | 1,882.00 € | ||
| 1mL*10mM (DMSO) | 170.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
SB 611812
CAS:345892-71-9
SB 611812 is an antagonist of urotensin-II (UT) and can be used in studies about …
Formula:
C17H16Cl3F3N2O3S
Purity:
99.34%
Color and Shape:
Solid
Molecular weight:
491.74
Ref: TM-T23323
| 2mg | 37.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 183.00 € | ||
| 50mg | 266.00 € | ||
| 100mg | 373.00 € | ||
| 1mL*10mM (DMSO) | 65.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Nemazoline Free Base
CAS:130759-56-7
Nemazoline Free Base: a long-lasting nasal decongestant, better than oxymetazoline, with no systemic effects or …
Formula:
C10H11Cl2N3
Purity:
99.03% - 99.18%
Color and Shape:
Liquid
Molecular weight:
244.12
Ref: TM-T71012
| 1mg | 279.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Flumexadol
CAS:30914-89-7
Flumexadol is a selective 5-HT2C receptor agonist with an affinity (Ki) of 25 nM for …
Formula:
C11H12F3NO
Purity:
98%
Color and Shape:
Solid
Molecular weight:
231.21
Ref: TM-T11302
| 50mg | To inquire | ||
| 100mg | To inquire |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Ticalopride
CAS:202590-69-0
Ticalopride: 5-HT3 agonist for digestive, orofacial, ENT disorders, and bulimia, GERD, IBS research.
Formula:
C14H20ClN3O3
Purity:
100%
Color and Shape:
Liquid
Molecular weight:
313.78
Ref: TM-T69984
| 1mg | 93.00 € | ||
| 5mg | 200.00 € | ||
| 10mg | 294.00 € | ||
| 25mg | 557.00 € | ||
| 50mg | 742.00 € | ||
| 100mg | 1,035.00 € | ||
| 500mg | 2,072.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
4-PPBP maleate
CAS:201216-39-9
4-PPBP maleate: potent σ1 agonist, selective NR1a/2B NMDA antagonist, neuroprotective.
Formula:
C25H31NO4
Purity:
99.54%
Color and Shape:
Solid
Molecular weight:
409.52
Ref: TM-T22513
| 5mg | 48.00 € | ||
| 10mg | 74.00 € | ||
| 25mg | 135.00 € | ||
| 50mg | 210.00 € | ||
| 100mg | 313.00 € | ||
| 200mg | 442.00 € | ||
| 1mL*10mM (DMSO) | 56.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
8-OH-Dpat
CAS:78950-78-4
8-OH-Dpat (8-Hydroxy-DPAT) is a serotonin 1A-receptor agonist that is used experimentally to test the effects …
Formula:
C16H25NO
Purity:
98%
Color and Shape:
Solid
Molecular weight:
247.38
Ref: TM-T4305
| 5mg | 418.00 € | ||
| 10mg | 672.00 € | ||
| 25mg | 1,024.00 € | ||
| 50mg | 1,538.00 € | ||
| 100mg | 2,307.00 € | ||
| 1mL*10mM (DMSO) | 454.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
