G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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JTE-907
CAS:282089-49-0
JTE-907 is a CB2 receptor inverse agonist with high selectivity and oral activity.JTE-907 exhibits anti-inflammatory …
Formula:
C24H26N2O6
Purity:
100%
Color and Shape:
Solid
Molecular weight:
438.47
Ref: TM-T19705
| 1mg | 55.00 € | ||
| 5mg | 123.00 € | ||
| 10mg | 183.00 € | ||
| 25mg | 323.00 € | ||
| 50mg | 482.00 € | ||
| 100mg | 688.00 € | ||
| 1mL*10mM (DMSO) | 150.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
CAY10595
CAS:916047-16-0
CAY10595 is an antagonist of the CRTh2 (DP2) receptor with a Ki of 10 nM.
Formula:
C20H13Cl2FN2O5
Purity:
100% - 99.71%
Color and Shape:
Solid
Molecular weight:
451.23
Ref: TM-T10691
| 1mg | 50.00 € | ||
| 5mg | 185.00 € | ||
| 10mg | 324.00 € | ||
| 25mg | 429.00 € | ||
| 50mg | 641.00 € | ||
| 100mg | 864.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Landipirdine
CAS:1000308-25-7
Landipirdine (RO-5025181) is a selective 5-HT6R antagonist for the study of central nervous system disorders …
Formula:
C18H19FN2O3S
Purity:
97.50% - 99.33%
Color and Shape:
Solid
Molecular weight:
362.42
Ref: TM-T27795
| 1mg | 227.00 € | ||
| 5mg | 541.00 € | ||
| 10mg | 726.00 € | ||
| 25mg | 1,172.00 € | ||
| 50mg | 1,493.00 € | ||
| 100mg | 2,124.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
T-0509
CAS:96843-99-1
T-0509 is a selective beta 1 receptor agonist that increases inotropy in canine ventricular muscle …
Formula:
C18H23NO5
Purity:
97.46% - 98.21%
Color and Shape:
Solid
Molecular weight:
333.38
Ref: TM-T28895
| 1mg | 327.00 € | ||
| 5mg | 769.00 € | ||
| 10mg | 1,056.00 € | ||
| 25mg | 1,477.00 € | ||
| 50mg | 1,839.00 € | ||
| 100mg | 2,331.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Iodophenpropit dihydrobromide
CAS:145196-87-8
Iodophenpropit dihydrobromide: selective histamine H3 antagonist, reversible binding, high affinity (KD: 0.32 nM).
Formula:
C15H20BrIN4S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
495.22
Ref: TM-T15590
| 5mg | 279.00 € | ||
| 10mg | 418.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
ENMD-1068 HCl
CAS:789488-77-3
ENMD-1068 HCl (ENMD 1068) is a PAR-2 antagonist. ENMD-1068 HCl inhibits the development of endometriosis …
Formula:
C15H29N3O2
Purity:
95.79%
Color and Shape:
Solid
Molecular weight:
283.41
Ref: TM-T27267
| 10mg | 54.00 € | ||
| 25mg | 94.00 € | ||
| 50mg | 132.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
BTB09089
CAS:245728-44-3
BTB09089 (GPR65 agonist ) is a T cell death-associated gene 8 (TDAG8/GPR65)-specific agonist.BTB09089 induces TDAG8 …
Formula:
C14H12Cl2N4OS2
Purity:
100%
Color and Shape:
Soild
Molecular weight:
387.31
Ref: TM-T67892
| 1mg | 71.00 € | ||
| 5mg | 122.00 € | ||
| 10mg | 184.00 € | ||
| 25mg | 336.00 € | ||
| 50mg | 510.00 € | ||
| 100mg | 733.00 € | ||
| 500mg | 1,514.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
ADRA1D receptor antagonist 1 HCl
CAS:1191908-14-1
ADRA1D receptor antagonist 1 HCl is a selective α1D adrenergic receptor antagonist (Ki: 1.6 nM) …
Formula:
C15H14Cl2N4O
Purity:
98.13%
Color and Shape:
Solid
Molecular weight:
337.2
Ref: TM-T10250
| 1mg | 185.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
OPC-14523 hydrochloride
CAS:145969-31-9
OPC-14523 hydrochloride, an oral sigma/5-HT1A agonist, shows potent antidepressant activity with strong receptor affinity.
Formula:
C23H29Cl2N3O2
Purity:
99.70%
Color and Shape:
Solid
Molecular weight:
450.4
Ref: TM-T62711
| 5mg | 889.00 € | ||
| 10mg | 1,181.00 € | ||
| 25mg | 1,483.00 € | ||
| 50mg | 1,814.00 € | ||
| 100mg | 2,290.00 € | ||
| 1mL*10mM (DMSO) | 942.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
S 14506 hydrochloride
CAS:286369-38-8
S 14506 hydrochloride is a 5-HT1A receptor full agonist.
Formula:
C24H27ClFN3O2
Purity:
99.5%
Color and Shape:
Solid
Molecular weight:
443.94
Ref: TM-T23285
| 1mg | 45.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 140.00 € | ||
| 25mg | 272.00 € | ||
| 50mg | 416.00 € | ||
| 100mg | 628.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
ReN-1869
CAS:170149-99-2
ReN-1869 is a novel selective histamine H(1) receptor antagonist with anti-neurogenic pain and anti-inflammatory activity …
Formula:
C24H27NO2
Purity:
99.87% - 99.89%
Color and Shape:
Solid
Molecular weight:
361.48
Ref: TM-T28516
| 1mg | 201.00 € | ||
| 5mg | 502.00 € | ||
| 10mg | 725.00 € | ||
| 25mg | 1,117.00 € | ||
| 50mg | 1,852.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
SLM6031434 HCl
CAS:1897379-34-8
SLM6031434 HCl (SLM-6031434 HCl) is a SphK2 inhibitor that reduces LPS-induced TNF伪 and IL-1尾 production.
Formula:
C22H31ClF3N5O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
489.96
Ref: TM-T28806
| 1mg | 126.00 € | ||
| 5mg | 397.00 € | ||
| 10mg | 546.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
CMF019
CAS:1586787-08-7
CMF019 is a potent agonist of the Apelin receptor (APJ) with G protein bias. CMF019 …
Formula:
C25H33N3O3S
Purity:
98.54%
Color and Shape:
Solid
Molecular weight:
455.61
Ref: TM-T10843
| 1mg | 118.00 € | ||
| 5mg | 241.00 € | ||
| 10mg | 407.00 € | ||
| 25mg | 663.00 € | ||
| 50mg | 919.00 € | ||
| 100mg | 1,226.00 € | ||
| 1mL*10mM (DMSO) | 244.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Lusaperidone
CAS:214548-46-6
Kaerophyllin ( (-)-Kaerophylin) inhibits hepatic stellate cell activation and inhibits HSC activation to protect against …
Formula:
C22H21N3O2
Purity:
99.64%
Color and Shape:
Solid
Molecular weight:
359.42
Ref: TM-T11894
| 1mg | 131.00 € | ||
| 5mg | 305.00 € | ||
| 10mg | 491.00 € | ||
| 25mg | 1,012.00 € | ||
| 50mg | 1,718.00 € | ||
| 100mg | 2,524.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
p-MPPF dihydrochloride
CAS:223699-41-0
p-MPPF dihydrochloride is a 5-HT antagonist that can be used to study neurological diseases.
Formula:
C25H29Cl2FN4O2
Purity:
99.78%
Color and Shape:
Solid
Molecular weight:
507.43
Ref: TM-T69750
| 1mg | 266.00 € | ||
| 5mg | 655.00 € | ||
| 10mg | 896.00 € | ||
| 25mg | 1,437.00 € | ||
| 50mg | 1,872.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Lintopride
CAS:107429-63-0
Lintopride is an antagonist of 5HT4. It has moderate 5HT3 antagonist properties.
Formula:
C14H19ClN4O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
310.78
Ref: TM-T15760
| 25mg | 1,410.00 € | ||
| 50mg | 1,838.00 € | ||
| 100mg | 2,322.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
RG 7152
CAS:107813-63-8
RG 7152 is a leukotriene D4 antagonist with anti-asthmatic properties and can be used in …
Formula:
C20H19N5O2
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
361.4
Ref: TM-T28529
| 1mg | 277.00 € | ||
| 5mg | 681.00 € | ||
| 10mg | 931.00 € | ||
| 25mg | 1,434.00 € | ||
| 50mg | 1,867.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
P2Y2R/GPR17 antagonist 1
CAS:2395016-49-4
P2Y2R/GPR17 antagonist 1 (Compound 14m) is a dual P2Y2R (IC50: 3.17 μM) and GPR17 (IC50: …
Formula:
C19H13ClN2O6S
Purity:
98.21%
Color and Shape:
Liquid
Molecular weight:
432.83
Ref: TM-T62420
| 5mg | 37.00 € | ||
| 10mg | 52.00 € | ||
| 25mg | 87.00 € | ||
| 50mg | 161.00 € | ||
| 100mg | 334.00 € | ||
| 200mg | To inquire | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
GS-9667
CAS:618380-90-8
GS-9667, a selective and partial agonist of the A(1) adenosine receptor (AR), represents an effective …
Formula:
C21H24FN5O4S
Purity:
99.76% - 99.76%
Color and Shape:
Solid
Molecular weight:
461.51
Ref: TM-T27439
| 1mg | 107.00 € | ||
| 5mg | 265.00 € | ||
| 10mg | 363.00 € | ||
| 25mg | 598.00 € | ||
| 50mg | 817.00 € | ||
| 100mg | 1,126.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Lecozotan HCl
CAS:433282-68-9
Lecozotan HCl is a selective 5-HT antagonist boosting glutamate and acetylcholine release without causing 5-HT(1A) …
Formula:
C28H30ClN5O3
Purity:
99.47%
Color and Shape:
Solid
Molecular weight:
520.02
Ref: TM-T27806
| 1mg | 156.00 € | ||
| 5mg | 363.00 € | ||
| 10mg | 552.00 € | ||
| 25mg | 875.00 € | ||
| 50mg | 1,189.00 € | ||
| 100mg | 1,616.00 € | ||
| 500mg | 3,211.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
