G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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ST3932
CAS:1246018-21-2
ST3932 is a ST1535 metabolite, is a adenosine A2A receptor antagonist(Kis of 8 nM and …
Formula:
C12H16N8O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
288.31
Ref: TM-T13008
| 25mg | 1,549.00 € | ||
| 50mg | 2,038.00 € | ||
| 100mg | 2,617.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
PRX933 hydrochloride
CAS:639029-42-8
PRX933 hydrochloride (GW876167 hydrochloride) is an agonist of 5-HT2C receptor and can be used in …
Formula:
C16H22ClN5O2
Purity:
97.99% - 99.72%
Color and Shape:
Solid
Molecular weight:
351.84
Ref: TM-T12565
| 1mg | 349.00 € | ||
| 5mg | 556.00 € | ||
| 10mg | 886.00 € | ||
| 25mg | 1,309.00 € | ||
| 50mg | 1,773.00 € | ||
| 100mg | 2,377.00 € | ||
| 1mL*10mM (DMSO) | 649.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Adenosine antagonist-1
CAS:431040-19-6
Adenosine antagonist-1 acts as an adenosine A3 receptor (AA3R) antagonist.
Formula:
C18H13N7S
Purity:
100% - 97%
Color and Shape:
Solid
Molecular weight:
359.41
Ref: TM-T10248
| 1mg | 232.00 € | ||
| 5mg | 585.00 € | ||
| 10mg | 831.00 € | ||
| 25mg | 1,205.00 € | ||
| 50mg | 1,523.00 € | ||
| 100mg | 1,850.00 € | ||
| 200mg | 2,606.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Masilukast
CAS:136564-68-6
Masilukast(MCC-847) is an oral leukotriene D4 (LTD4) receptor antagonist for the study of diseases associated …
Formula:
C31H32F3N3O5S
Purity:
99.00% - 99.53%
Color and Shape:
Solid
Molecular weight:
615.66
Ref: TM-T27979
| 1mg | 489.00 € | ||
| 5mg | 1,095.00 € | ||
| 10mg | 1,476.00 € | ||
| 25mg | 2,183.00 € | ||
| 50mg | 2,965.00 € | ||
| 100mg | 3,971.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Palonosetron
CAS:135729-61-2
Palonosetron, a 5-HT3 antagonist with Ki of 0.17 nM, is used in the prevention and …
Formula:
C19H24N2O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
296.41
Ref: TM-T22393
| 25mg | 1,406.00 € | ||
| 50mg | 1,852.00 € | ||
| 100mg | 2,338.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
CRTh2 antagonist 1
CAS:1379445-54-1
CRTh2 antagonist 1 is a CRTh2 antagonist (IC50: 89 nM).
Formula:
C23H25N3O5S
Purity:
97.39%
Color and Shape:
Solid
Molecular weight:
455.53
Ref: TM-T10084
| 1mg | 113.00 € | ||
| 5mg | 249.00 € | ||
| 10mg | 366.00 € | ||
| 25mg | 550.00 € | ||
| 50mg | 769.00 € | ||
| 100mg | 1,049.00 € | ||
| 500mg | 2,098.00 € | ||
| 1mL*10mM (DMSO) | 281.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Burixafor hydrobromide
CAS:1191450-19-7
Burixafor hydrobromide is an oral CXCR4 blocker with anti-angiogenic properties, potentially treating choroid neovascularization.
Formula:
C27H52BrN8O3P
Purity:
98%
Color and Shape:
Solid
Molecular weight:
647.644
Ref: TM-T10635
| 25mg | To inquire | ||
| 50mg | To inquire | ||
| 100mg | To inquire |
Estimated delivery in United States, on Monday 27 Jan 2025
TC LPA5 4
CAS:1393814-38-4
TC LPA5 4 is a LPA5 receptor antagonist.
Formula:
C23H23ClN2O3
Purity:
99.05%
Color and Shape:
Solid
Molecular weight:
410.89
Ref: TM-T23438
| 1mg | 58.00 € | ||
| 5mg | 124.00 € | ||
| 10mg | 183.00 € | ||
| 25mg | 425.00 € | ||
| 50mg | 625.00 € | ||
| 100mg | 891.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
GPR35 agonist 3
CAS:123021-85-2
GPR35 agonist 3 is a synthetic GPR35 agonist used in the study of cancer, type …
Formula:
C12H9NO5S
Purity:
98.79%
Color and Shape:
Liquid
Molecular weight:
279.27
Ref: TM-T72755
| 1mg | 49.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 151.00 € | ||
| 25mg | 301.00 € | ||
| 50mg | 482.00 € | ||
| 100mg | 771.00 € | ||
| 500mg | 1,539.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Iferanserin
CAS:58754-46-4
Iferanserin (S-MPEC) is a selective antagonist of the 5-HT receptor (serotonin receptor) with an affinity …
Formula:
C23H28N2O
Color and Shape:
Solid
Molecular weight:
348.48
Ref: TM-T15552
| 25mg | 1,299.00 € | ||
| 50mg | 1,704.00 € | ||
| 100mg | 2,340.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
H4R antagonist 1
CAS:1429375-54-1
H4R antagonist 1: selective histamine H4R inhibitor, IC50 27 nM, no affinity for H1R, H2R, …
Formula:
C11H11BrN8
Color and Shape:
Solid
Molecular weight:
335.16
Ref: TM-T11532
| 25mg | 1,410.00 € | ||
| 50mg | 1,854.00 € | ||
| 100mg | 2,340.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
CB1R Allosteric modulator 3
CAS:2633686-36-7
CB1R Allosteric modulator 3 is a CB1R modulator.CB1R Allosteric modulator 3 inhibits cAMP, and can …
Formula:
C22H17ClN2O2
Purity:
98.18%
Color and Shape:
Liquid
Molecular weight:
376.84
Ref: TM-T61562
| 1mg | 42.00 € | ||
| 2mg | 55.00 € | ||
| 5mg | 89.00 € | ||
| 10mg | 136.00 € | ||
| 25mg | 220.00 € | ||
| 50mg | 328.00 € | ||
| 100mg | 486.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
CB1R antagonist 1
CAS:334668-69-8
CB1R antagonist 1 is a potent CB1R antagonist that can be used to study diseases …
Formula:
C18H23F3N2O3S
Purity:
99.65%
Color and Shape:
Liquid
Molecular weight:
404.45
Ref: TM-T61989
| 5mg | 73.00 € | ||
| 10mg | 114.00 € | ||
| 25mg | 184.00 € | ||
| 50mg | 273.00 € | ||
| 100mg | 407.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
GALNON
CAS:475115-35-6
Galnon is a galanin receptor agonist, improves intrinsic cortical bone tissue properties
Formula:
C40H46N4O6
Purity:
98%
Color and Shape:
Solid
Molecular weight:
678.82
Ref: TM-T8456
| 25mg | 759.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Deramciclane
CAS:120444-71-5
Deramciclane has high affinity for 5-HT2A and 5-HT2C receptors.
Formula:
C20H31NO
Color and Shape:
Solid
Molecular weight:
301.47
Ref: TM-T10996
| 25mg | 1,002.00 € | ||
| 50mg | 1,320.00 € | ||
| 100mg | 1,863.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
CP-866087
CAS:519052-04-1
CP-866087 is a novel, potent and selective mu-opioid receptor antagonist for the study of female …
Formula:
C24H28N2O2
Purity:
100% - 99.44%
Color and Shape:
Soild
Molecular weight:
376.49
Ref: TM-T31081
| 1mg | 707.00 € | ||
| 5mg | 1,486.00 € | ||
| 25mg | 1,976.00 € | ||
| 50mg | 2,412.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
PRX-08066 Maleic acid
CAS:866206-55-5
PRX-08066 Maleic acid is a selective 5-HT2B receptor antagonist with IC50 of 3.4 nM, prevents …
Formula:
C19H17ClFN5S·C4H4O4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
517.96
Ref: TM-T6959
| 5mg | 169.00 € | ||
| 10mg | 229.00 € | ||
| 25mg | 411.00 € | ||
| 1mL*10mM (DMSO) | 400.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Tedatioxetine hydrobromide
CAS:960151-65-9
Tedatioxetine hydrobromide (Lu AA 24530 hydrobromide) is a serotonin-norepinephrine-dopamine reuptake inhibitor and 5-HT2A receptor antagonist.
Formula:
C18H22BrNS
Purity:
99.50%
Color and Shape:
Solid
Molecular weight:
364.34
Ref: TM-T13110
| 1mg | 132.00 € | ||
| 5mg | 318.00 € | ||
| 10mg | 507.00 € | ||
| 25mg | 1,062.00 € | ||
| 50mg | 1,694.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
A-65186
CAS:119295-94-2
A-65186 is a CCK antagonist used in the study of inflammation and gastrointestinal tract injury.
Formula:
C25H35N3O4
Purity:
98.37% - 99.94%
Color and Shape:
Solid
Molecular weight:
441.56
Ref: TM-T26483
| 1mg | 277.00 € | ||
| 5mg | 682.00 € | ||
| 10mg | 932.00 € | ||
| 25mg | 1,435.00 € | ||
| 50mg | 1,869.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
(±)-Tazifylline
CAS:79712-55-3
(±)-Tazifylline is a selective and long-acting antagonist of histamine H1 receptor.
Formula:
C23H32N6O3S
Purity:
98.97%
Color and Shape:
Solid
Molecular weight:
472.6
Ref: TM-T10000
| 1mg | 146.00 € | ||
| 5mg | 278.00 € | ||
| 10mg | 403.00 € | ||
| 25mg | 631.00 € | ||
| 50mg | 849.00 € | ||
| 100mg | 1,098.00 € | ||
| 1mL*10mM (DMSO) | 368.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
