G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
Read more
L-694,247
CAS:137403-12-4
L-694,247 is a 5-HT receptor agonist with affinity for 5-HT1D, 5-HT1A, 5-HT1B, 5-HT1C, and 5-HT1E …
Formula:
C20H21N5O3S
Purity:
98%
Color and Shape:
White Solid
Molecular weight:
411.48
Ref: TM-T19701
| 1mg | 83.00 € | ||
| 5mg | 264.00 € | ||
| 10mg | 451.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
RS 67333 hydrochloride
CAS:168986-60-5
RS 67333 hydrochloride is a selective 5-HT4R partial agonist (pKi=8.7) with neuroprotective properties for Alzheimer's …
Formula:
C19H30Cl2N2O2
Purity:
98.78%
Color and Shape:
Solid
Molecular weight:
389.36
Ref: TM-T23265
| 1ml | 52.00 € | ||
| 5mg | 50.00 € | ||
| 10mg | 79.00 € | ||
| 25mg | 166.00 € | ||
| 50mg | 252.00 € | ||
| 100mg | 369.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Org-12962
CAS:132834-56-1
Org-12962: 5-HT2C agonist (pEC50: 7.01), anti-panic in rats, affects 5-HT2A/B (pEC50: 6.38/6.28).
Formula:
C10H11ClF3N3
Purity:
98.34%
Color and Shape:
Solid
Molecular weight:
265.66
Ref: TM-T16401
| 1ml | 52.00 € | ||
| 5mg | 47.00 € | ||
| 10mg | 61.00 € | ||
| 25mg | 90.00 € | ||
| 50mg | 109.00 € | ||
| 100mg | 156.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Endomorphin 1 acetate
CAS:1276123-71-7
Endomorphin 1 acetate is a μ-opioid receptor agonist with antinociceptive and analgesic effects and can …
Formula:
C36H42N6O7
Color and Shape:
Solid
Molecular weight:
670.75
Ref: TM-T72423
| 2mg | 58.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
GPR35 agonist 2
CAS:494191-73-0
GPR35 agonist 2 (TC-G 1001) is a potent GPR35 agonist.The EC50 values of GPR35 agonist …
Formula:
C17H11FN2O3S
Purity:
98% - 98.40%
Color and Shape:
Solid
Molecular weight:
342.34
Ref: TM-T23434
| 1mg | 52.00 € | ||
| 1ml | 114.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 171.00 € | ||
| 25mg | 369.00 € | ||
| 50mg | 547.00 € | ||
| 100mg | 786.00 € | ||
| 500mg | 1,606.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
6-Chloromelatonin
CAS:63762-74-3
6-Chloromelatonin: potent, stable melatonin agonist; binds MT2 receptors (pKi=9.77); could help research sleep disorders.
Formula:
C13H15ClN2O2
Purity:
97.90% - 99.36%
Color and Shape:
Solid
Molecular weight:
266.72
Ref: TM-T22530
| 1mg | 325.00 € | ||
| 5mg | 774.00 € | ||
| 10mg | 1,050.00 € | ||
| 25mg | 1,477.00 € | ||
| 50mg | 1,839.00 € | ||
| 100mg | 2,322.00 € | ||
| 500mg | 4,551.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
ABT-080
CAS:189498-57-5
ABT-080 (VML 530), a leukotriene synthesis inhibitor, is used potentially for treatment of asthma.
Formula:
C37H31N2NaO4
Purity:
98.15%
Color and Shape:
Solid
Molecular weight:
590.64
Ref: TM-T26524
| 1ml | 51.00 € | ||
| 5mg | 34.00 € | ||
| 10mg | 52.00 € | ||
| 25mg | 82.00 € | ||
| 50mg | 109.00 € | ||
| 100mg | 163.00 € | ||
| 200mg | 237.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Torbafylline
CAS:105102-21-4
Torbafylline is a xanthine-based PDE inhibitor reducing protein breakdown via PDE4/cAMP/EPAC/PI3K/Akt in rats with burns, …
Formula:
C16H26N4O4
Purity:
98% - 99%
Color and Shape:
Soild
Molecular weight:
338.4
Ref: TM-T67965
| 1mg | 125.00 € | ||
| 1ml | 312.00 € | ||
| 5mg | 299.00 € | ||
| 10mg | 448.00 € | ||
| 25mg | 730.00 € | ||
| 50mg | 1,003.00 € | ||
| 100mg | 1,374.00 € | ||
| 500mg | 2,747.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Viloxazine
CAS:46817-91-8
Viloxazine (Viloxazin) (Viloxazin) is a dual-action compound that functions as a norepinephrine reuptake inhibitor and …
Formula:
C13H19NO3
Purity:
99.8%
Color and Shape:
Solid
Molecular weight:
237.29
Ref: TM-T60325
| 1mg | 181.00 € | ||
| 5mg | 409.00 € | ||
| 10mg | 602.00 € | ||
| 25mg | 922.00 € | ||
| 50mg | 1,299.00 € | ||
| 100mg | 1,743.00 € | ||
| 500mg | 3,477.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
GW438014A
CAS:469861-49-2
GW438014A is a potent, selective antagonist of the NPY-Y5 receptor, effectively inhibiting food consumption and …
Formula:
C23H23N3O4S
Purity:
100%
Color and Shape:
Solid
Molecular weight:
437.51
Ref: TM-T24121
| 1mg | 40.00 € | ||
| 5mg | 86.00 € | ||
| 10mg | 123.00 € | ||
| 25mg | 245.00 € | ||
| 50mg | 384.00 € | ||
| 100mg | 548.00 € | ||
| 500mg | 1,179.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Itasetron
CAS:123258-84-4
Itasetron, a 5-HT3 antagonist, prevents memory loss in rats and has antiemetic effects in cancer …
Formula:
C16H20N4O2
Purity:
100% - 99.63%
Color and Shape:
Solid
Molecular weight:
300.36
Ref: TM-T24184
| 1mg | 326.00 € | ||
| 5mg | 769.00 € | ||
| 10mg | 1,050.00 € | ||
| 25mg | 1,486.00 € | ||
| 50mg | 1,838.00 € | ||
| 100mg | 2,322.00 € | ||
| 500mg | 4,547.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
JNJ-20788560
CAS:825649-28-3
JNJ-20788560 is a delta opioid receptor (DOR) agonist with analgesic activity. It is more selective …
Formula:
C25H28N2O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
388.5
Ref: TM-T27667
| 1mg | 327.00 € | ||
| 1ml | 554.00 € | ||
| 5mg | 769.00 € | ||
| 10mg | 1,049.00 € | ||
| 25mg | 1,477.00 € | ||
| 50mg | 1,838.00 € | ||
| 100mg | 2,320.00 € | ||
| 500mg | 4,549.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
SLP9101555
SLP9101555 is a potent and selective sphingosine kinase 2 (SphK2) inhibitor with a Ki of …
Formula:
C16H22BrClN2
Purity:
99%
Color and Shape:
Solid
Molecular weight:
357.72
Ref: TM-T63047
| 1mg | 326.00 € | ||
| 1ml | 657.00 € | ||
| 5mg | 774.00 € | ||
| 10mg | 1,056.00 € | ||
| 25mg | 1,477.00 € | ||
| 50mg | 1,838.00 € | ||
| 100mg | 2,336.00 € | ||
| 500mg | 4,568.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
OPC-51803
CAS:192514-54-8
OPC-51803 is an orally available nonapeptidylpressor (AVP) V(2) receptor selective agonist for the treatment of …
Formula:
C26H32ClN3O2
Purity:
100% - 100%
Color and Shape:
Solid
Molecular weight:
454
Ref: TM-T28257
| 1mg | 325.00 € | ||
| 5mg | 769.00 € | ||
| 10mg | 1,053.00 € | ||
| 25mg | 1,477.00 € | ||
| 50mg | 1,839.00 € | ||
| 100mg | 2,321.00 € | ||
| 500mg | 4,568.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
PF-03654746 Tosylate
CAS:1039399-17-1
PF-03654746 Tosylate is selective antagonist of histamine H3 receptor with high brain penetration.
Formula:
C25H32F2N2O4S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
494.6
Ref: TM-T12416
| 25mg | 854.00 € | ||
| 50mg | 1,096.00 € | ||
| 100mg | 1,668.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Sinitrodil
CAS:143248-63-9
Sinitrodil (ITF-296) is a guanylate cyclase stimulant that may be used in the treatment of …
Formula:
C10H10N2O5
Purity:
99%
Color and Shape:
Solid
Molecular weight:
238.2
Ref: TM-T34648
| 1mg | 137.00 € | ||
| 1ml | 400.00 € | ||
| 5mg | 327.00 € | ||
| 10mg | 492.00 € | ||
| 25mg | 798.00 € | ||
| 50mg | 1,095.00 € | ||
| 100mg | 1,477.00 € | ||
| 500mg | 2,980.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
ML-335
CAS:1069498-96-9
ML-335, a μ-δ targeted agonist and MOR/DOR ligand, may lead to isomer-biased drugs with pain-relief …
Formula:
C25H32N2O3
Purity:
98.52%
Color and Shape:
Solid
Molecular weight:
408.53
Ref: TM-T23002
| 1mg | 46.00 € | ||
| 1ml | 55.00 € | ||
| 5mg | 90.00 € | ||
| 10mg | 144.00 € | ||
| 25mg | 269.00 € | ||
| 50mg | 430.00 € | ||
| 100mg | 621.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
AT-121
CAS:2099681-31-7
AT-121 is a dual μ-opioid and neuropeptide receptor partial agonist (Kis 16.49 and 3.67 nM, …
Formula:
C24H38N4O3S
Purity:
97% - 97.95%
Color and Shape:
Solid
Molecular weight:
462.65
Ref: TM-T37610
| 1mg | 325.00 € | ||
| 5mg | 769.00 € | ||
| 10mg | 1,049.00 € | ||
| 25mg | 1,483.00 € | ||
| 50mg | 1,850.00 € | ||
| 100mg | 2,321.00 € | ||
| 500mg | 4,577.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Seridopidine
CAS:883631-51-4
Seridopidine (ACR343) is a modulator of dopaminergic activity that is used as an oral therapy …
Formula:
C14H20FNO2S
Purity:
99.11%
Color and Shape:
Solid
Molecular weight:
285.38
Ref: TM-T34616
| 1mg | 137.00 € | ||
| 5mg | 327.00 € | ||
| 10mg | 493.00 € | ||
| 25mg | 797.00 € | ||
| 50mg | 1,103.00 € | ||
| 100mg | 1,477.00 € | ||
| 500mg | 2,962.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
TASP0390325
CAS:1642187-96-9
TASP0390325, a potent and orally active V1B receptor antagonist, has antidepressant and anxiolytic activities in …
Formula:
C25H30Cl2FN5O4
Purity:
98.62%
Color and Shape:
Solid
Molecular weight:
554.44
Ref: TM-T28926
| 1mg | 57.00 € | ||
| 5mg | 121.00 € | ||
| 10mg | 187.00 € | ||
| 25mg | 430.00 € | ||
| 50mg | 743.00 € | ||
| 100mg | 1,208.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
