G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Octimibate
CAS:89838-96-0
Octimibate: non-prostaglandin antiplatelet, treats cardiovascular disease, aids atherosclerosis/thrombosis research.
Formula:
C29H30N2O3
Purity:
99.49%
Color and Shape:
Solid
Molecular weight:
454.56
Ref: TM-T24567
| 1mg | 138.00 € | ||
| 5mg | 335.00 € | ||
| 10mg | 492.00 € | ||
| 25mg | 798.00 € | ||
| 50mg | 1,096.00 € | ||
| 100mg | 1,483.00 € | ||
| 500mg | 2,960.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
I942
CAS:868145-09-9
I942 is a novel, selective ACyclic nucleotide (NCN) EPAC1 agonist that activates exchange proteins to …
Formula:
C20H19NO4S
Purity:
99.75%
Color and Shape:
Solid
Molecular weight:
369.43
Ref: TM-T24154
| 1mg | 93.00 € | ||
| 5mg | 223.00 € | ||
| 10mg | 362.00 € | ||
| 25mg | 593.00 € | ||
| 50mg | 820.00 € | ||
| 100mg | 1,105.00 € | ||
| 500mg | 2,256.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
NNC 92-1687
CAS:22903-37-3
NNC 92-1687 is a selective glucagon receptor antagonist that can be used to study type …
Formula:
C15H12N2O3S
Purity:
100% - 99.72%
Color and Shape:
Solid
Molecular weight:
300.33
Ref: TM-T28182
| 1mg | 376.00 € | ||
| 5mg | 905.00 € | ||
| 10mg | 1,117.00 € | ||
| 25mg | 1,496.00 € | ||
| 50mg | 1,839.00 € | ||
| 100mg | 2,321.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Cyamemazine
CAS:3546-03-0
Cyamemazine is an antipsychotic compound with sedative and anxiolytic activity.Cyamemazine is a 5-HT3, 5-HT2A, and …
Formula:
C19H21N3S
Purity:
97.01%
Color and Shape:
Solid
Molecular weight:
323.46
Ref: TM-T15026
| 1mg | 36.00 € | ||
| 5mg | 69.00 € | ||
| 10mg | 103.00 € | ||
| 25mg | 208.00 € | ||
| 50mg | 353.00 € | ||
| 100mg | 603.00 € | ||
| 1mL*10mM (DMSO) | 77.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
MG 1
CAS:148274-76-4
MG 1 is a potent alpha-1 adrenergic receptor antagonist.
Formula:
C17H25N3O2
Purity:
100% - 99.73%
Color and Shape:
Solid
Molecular weight:
303.4
Ref: TM-T12030
| 1mg | 650.00 € | ||
| 5mg | 1,671.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
hGPR91 antagonist 3
CAS:1314796-31-0
hGPR91 antagonist 3 is an hGPR91 antagonist. hGPR91 antagonist 3 can be used to study …
Formula:
C23H18F4N4O2
Purity:
98.82% - 98.82%
Color and Shape:
Liquid
Molecular weight:
458.41
Ref: TM-T62858
| 1mg | 147.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
SRT3190
CAS:1204707-73-2
SRT3190 is an antagonist of CXCR2.
Formula:
C18H23F2N5O4S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
475.53
Ref: TM-T16933
| 2mg | 137.00 € | ||
| 5mg | 231.00 € | ||
| 25mg | 619.00 € | ||
| 50mg | 821.00 € | ||
| 100mg | 1,213.00 € | ||
| 1mL*10mM (DMSO) | 402.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
CB1 agonist 1
CAS:851212-80-1
CB1 agonist 1 is a potent CB1 agonist with a pIC50 value of 5.7 for …
Formula:
C24H24N2O5S
Purity:
98.56%
Color and Shape:
Liquid
Molecular weight:
452.52
Ref: TM-T62761
| 5mg | 74.00 € | ||
| 10mg | 106.00 € | ||
| 25mg | 214.00 € | ||
| 50mg | 349.00 € | ||
| 100mg | 559.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
LY-2624803
CAS:879409-35-5
LY-2624803 is a 5-HT2A receptor antagonist and histamine receptor inverse agonist that can be used …
Formula:
C22H25N3O3
Purity:
100% - 99.87%
Color and Shape:
Solid
Molecular weight:
379.45
Ref: TM-T24421
| 1mg | 138.00 € | ||
| 5mg | 335.00 € | ||
| 10mg | 496.00 € | ||
| 25mg | 803.00 € | ||
| 50mg | 1,099.00 € | ||
| 100mg | 1,486.00 € | ||
| 500mg | 2,980.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Regrelor disodium
CAS:676251-22-2
Regrelor disodium (INS 50589) is a p2y12 receptor antagonist that prevents thrombosis, effectively inhibits vascular …
Formula:
C22H23N6Na2O8P
Purity:
100%
Color and Shape:
Solid
Molecular weight:
576.41
Ref: TM-T34280
| 1mg | 182.00 € | ||
| 5mg | 400.00 € | ||
| 10mg | 591.00 € | ||
| 25mg | 916.00 € | ||
| 50mg | 1,263.00 € | ||
| 100mg | 1,705.00 € | ||
| 500mg | 3,438.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Fezagepras sodium
CAS:1254472-97-3
Fezagepras sodium (Setogepram sodium salt) is an orally active GPR40 agonist and is an antagonist …
Formula:
C13H17NaO2
Purity:
99.59%
Color and Shape:
Solid
Molecular weight:
228.26
Ref: TM-T12375
| 1mg | 42.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 138.00 € | ||
| 25mg | 250.00 € | ||
| 50mg | 366.00 € | ||
| 100mg | 532.00 € | ||
| 500mg | 1,070.00 € | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Calhex 231 hydrochloride
CAS:2387505-78-2
Calhex 231 hydrochloride, a CaSR antagonist, may treat diabetic cardiomyopathy; IC50 is 0.39 μM in …
Formula:
C25H28Cl2N2O
Color and Shape:
Solid
Molecular weight:
443.41
Ref: TM-T10666
| 2mg | 95.00 € | ||
| 5mg | 144.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
ADL-5747
CAS:850176-30-6
ADL-5747 (ADL-5747 (free base)) (free base) is a delta opioid receptor agonist used in the …
Formula:
C24H28N2O3
Purity:
100% - 99.44%
Color and Shape:
Solid
Molecular weight:
392.49
Ref: TM-T29663
| 1mg | 138.00 € | ||
| 5mg | 335.00 € | ||
| 10mg | 495.00 € | ||
| 25mg | 798.00 € | ||
| 50mg | 1,100.00 € | ||
| 100mg | 1,483.00 € | ||
| 500mg | 2,971.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
NE-100 hydrochloride
CAS:149409-57-4
NE-100 hydrochloride (NE-100 HCl) is a potent and selective antagonist of σ1 (IC50 = 4.16 …
Formula:
C23H34ClNO2
Purity:
98.85%
Color and Shape:
Solid
Molecular weight:
391.98
Ref: TM-T20797
| 1mg | 45.00 € | ||
| 2mg | 57.00 € | ||
| 5mg | 91.00 € | ||
| 10mg | 134.00 € | ||
| 25mg | 217.00 € | ||
| 50mg | 323.00 € | ||
| 100mg | 479.00 € | ||
| 200mg | 688.00 € | ||
| 500mg | 1,019.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Kira8 Hydrochloride
CAS:2250019-92-0
Kira8 Hydrochloride is a mono-selective IRE1α inhibitor that allosterically attenuates IRE1α RNase activity with an …
Formula:
C31H30Cl2N6O3S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
637.58
Ref: TM-T11762
| 5mg | 752.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Naphazoline
CAS:835-31-4
Naphazoline (Naphcon-a) is a sympathomimetic compound with marked alpha adrenergic activity.
Formula:
C14H14N2
Purity:
99.25%
Color and Shape:
White Crystalline Powder Solid
Molecular weight:
210.27
Ref: TM-T21445
| 5mg | 54.00 € | ||
| 10mg | 76.00 € | ||
| 25mg | 110.00 € | ||
| 50mg | 162.00 € | ||
| 100mg | 231.00 € | ||
| 500mg | 497.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
AZ-1355
CAS:75451-07-9
AZ-1355 is a novel dibenzoxepine derivative with lipid-lowering properties.
Formula:
C17H17NO4
Purity:
100%
Color and Shape:
Solid
Molecular weight:
299.32
Ref: TM-T13563
| 1mg | 168.00 € | ||
| 5mg | 411.00 € | ||
| 10mg | 554.00 € | ||
| 25mg | 836.00 € | ||
| 50mg | 1,143.00 € | ||
| 100mg | 1,490.00 € | ||
| 200mg | 2,042.00 € | ||
| 1mL*10mM (DMSO) | 371.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
SK1-IN-1
CAS:1218816-71-7
SK1-IN-1 is a SPHK1 inhibitor (IC50: 58 nM), with potential anticancer activity, and can be …
Formula:
C22H30N4O3
Purity:
98.72%
Color and Shape:
Solid
Molecular weight:
398.5
Ref: TM-T12927
| 1mg | 197.00 € | ||
| 1mL*10mM (DMSO) | 278.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
RS 67333 hydrochloride
CAS:168986-60-5
RS 67333 hydrochloride is a selective 5-HT4R partial agonist (pKi=8.7) with neuroprotective properties for Alzheimer's …
Formula:
C19H30Cl2N2O2
Purity:
98.78%
Color and Shape:
Solid
Molecular weight:
389.36
Ref: TM-T23265
| 5mg | 50.00 € | ||
| 10mg | 79.00 € | ||
| 25mg | 166.00 € | ||
| 50mg | 252.00 € | ||
| 100mg | 369.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Org-12962
CAS:132834-56-1
Org-12962: 5-HT2C agonist (pEC50: 7.01), anti-panic in rats, affects 5-HT2A/B (pEC50: 6.38/6.28).
Formula:
C10H11ClF3N3
Purity:
98.34%
Color and Shape:
Solid
Molecular weight:
265.66
Ref: TM-T16401
| 5mg | 47.00 € | ||
| 10mg | 61.00 € | ||
| 25mg | 90.00 € | ||
| 50mg | 109.00 € | ||
| 100mg | 156.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
