G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Ordopidine
CAS:871351-60-9
Ordopidine (ACR325) is a dopaminergic stabilizer that suppresses psychostimulant-induced hyperactivity disorder and stimulates behavior during …
Formula:
C14H20FNO2S
Purity:
99.52%
Color and Shape:
Solid
Molecular weight:
285.38
Ref: TM-T33816
| 1mg | 137.00 € | ||
| 5mg | 327.00 € | ||
| 10mg | 493.00 € | ||
| 25mg | 798.00 € | ||
| 50mg | 1,100.00 € | ||
| 100mg | 1,483.00 € | ||
| 500mg | 2,980.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Quinpirole Hydrochloride
CAS:85798-08-9
Quinpirole Hydrochloride (LY 171555), as an agonist with high affinity for dopamine receptor D2/D3, has …
Formula:
C13H22ClN3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
255.79
Ref: TM-T12606
| 1mg | 101.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
PNU-177864
CAS:250266-51-4
PNU-177864 is a selective dopamine D3 receptor antagonist.
Formula:
C18H21F3N2O3S
Purity:
99.82%
Color and Shape:
Solid
Molecular weight:
402.43
Ref: TM-T23167
| 1mg | 63.00 € | ||
| 2mg | 95.00 € | ||
| 5mg | 121.00 € | ||
| 10mg | 151.00 € | ||
| 25mg | 330.00 € | ||
| 50mg | 462.00 € | ||
| 100mg | 638.00 € | ||
| 500mg | 1,291.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
JP1302
CAS:80259-18-3
JP1302: α2C adrenoceptor antagonist, Kb 16 nM, Ki 28 nM, antidepressant, FACT disruptor, studies: neuropsychiatric, …
Formula:
C24H24N4
Purity:
99.48%
Color and Shape:
Solid
Molecular weight:
368.47
Ref: TM-T22882
| 1mg | 45.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 128.00 € | ||
| 25mg | 234.00 € | ||
| 50mg | 406.00 € | ||
| 100mg | 604.00 € | ||
| 500mg | 1,287.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Imetit dihydrobromide
CAS:32385-58-3
Imetit dihydrobromide is a high affinity and effective agonist of histamine H3 and H4 receptors …
Formula:
C6H12Br2N4S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
332.06
Ref: TM-T15565
| 50mg | To inquire | ||
| 100mg | To inquire |
Estimated delivery in United States, on Monday 25 Nov 2024
AZD8797
CAS:911715-90-7
AZD8797 (KAND567) is a CX3CR1 antagonist with potential protective effects against neuronal damage and prevents …
Formula:
C19H25N5OS2
Purity:
98.73% - 99.68%
Color and Shape:
Solid
Molecular weight:
403.56
Ref: TM-T14384
| 1mg | 91.00 € | ||
| 1ml | 216.00 € | ||
| 5mg | 184.00 € | ||
| 10mg | 346.00 € | ||
| 25mg | 733.00 € | ||
| 50mg | 918.00 € | ||
| 100mg | 1,329.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Lorglumide sodium salt
CAS:1021868-76-7
Lorglumide sodium salt (CR-1409 sodium salt) is an antagonist of cholecystokinin receptors (CCK).
Formula:
C22H31Cl2N2NaO4
Purity:
99.32%
Color and Shape:
Solid
Molecular weight:
481.39
Ref: TM-T11868
| 1ml | 36.00 € | ||
| 5mg | 34.00 € | ||
| 10mg | 50.00 € | ||
| 25mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 25 Nov 2024
Safotibant
CAS:633698-99-4
Safotibant (LF-22-0542) is a bradykinin B1 receptor antagonist with anti-inflammatory and analgesic activity for the …
Formula:
C25H34N4O5S
Purity:
99% - 99.53%
Color and Shape:
Solid
Molecular weight:
502.63
Ref: TM-T34485
| 1mg | 141.00 € | ||
| 5mg | 326.00 € | ||
| 10mg | 492.00 € | ||
| 25mg | 803.00 € | ||
| 50mg | 1,103.00 € | ||
| 100mg | 1,476.00 € | ||
| 500mg | 2,974.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Taprizosin
CAS:210538-44-6
Taprizosin(UK-338003) is a selective and orally active α1-adrenoceptor antagonist for vasodilatation in the treatment of …
Formula:
C25H26N6O4S
Purity:
97.01% - 99.11%
Color and Shape:
Solid
Molecular weight:
506.58
Ref: TM-T28922
| 1mg | 355.00 € | ||
| 5mg | 832.00 € | ||
| 10mg | 1,169.00 € | ||
| 25mg | 1,787.00 € | ||
| 50mg | 2,410.00 € | ||
| 100mg | 3,176.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Aplindore Fumarate
CAS:189681-71-8
Aplindore Fumarate (DAB-452), a selective dopamine D2/D3 partial agonist, is used in Parkinson's and schizophrenia …
Formula:
C22H22N2O7
Purity:
100%
Color and Shape:
Solid
Molecular weight:
426.42
Ref: TM-T30098
| 1mg | 274.00 € | ||
| 5mg | 681.00 € | ||
| 10mg | 920.00 € | ||
| 25mg | 1,421.00 € | ||
| 50mg | 1,839.00 € | ||
| 100mg | 2,601.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
VA-K-14 hydrochloride
CAS:1171341-19-7
VA-K-14 hydrochloride(VAK14 HCl) is a selective thyrotropin receptor (TSHR) antagonist (IC50= 12.3 μM) that inhibits …
Formula:
C18H16ClN3S
Purity:
98.01%
Color and Shape:
Solid
Molecular weight:
341.86
Ref: TM-T29087
| 1mg | 58.00 € | ||
| 5mg | 122.00 € | ||
| 10mg | 182.00 € | ||
| 25mg | 368.00 € | ||
| 50mg | 599.00 € | ||
| 100mg | 916.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
MK-0686
CAS:1159193-97-1
MK-0686 is an orally available bradykinin B1 receptor antagonist with potential anti-inflammatory activity.
Formula:
C22H19ClF4N2O4
Purity:
99.56%
Color and Shape:
Solid
Molecular weight:
486.84
Ref: TM-T33421
| 1mg | 178.00 € | ||
| 5mg | 437.00 € | ||
| 10mg | 644.00 € | ||
| 25mg | 1,003.00 € | ||
| 50mg | 1,364.00 € | ||
| 100mg | 1,819.00 € | ||
| 500mg | 3,650.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
SKF83959
CAS:80751-85-5
SKF83959: dopamine D1 partial agonist, Ki: D1(1.18 nM), D5(7.56 nM), D2(920 nM), D3(399 nM); improves …
Formula:
C18H20ClNO2
Purity:
98.45%
Color and Shape:
Solid
Molecular weight:
317.81
Ref: TM-T60835
| 1mg | 52.00 € | ||
| 1ml | 113.00 € | ||
| 5mg | 102.00 € | ||
| 10mg | 166.00 € | ||
| 25mg | 353.00 € | ||
| 50mg | 522.00 € | ||
| 100mg | 741.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Piclozotan
CAS:182415-09-4
Piclozotan (anhydrous), a 5-HT1A receptor agonist, demonstrated significant neuroprotective activity in a transient middle cerebral …
Formula:
C23H24ClN3O2
Purity:
99%
Color and Shape:
Solid
Molecular weight:
409.91
Ref: TM-T28414
| 25mg | 1,410.00 € | ||
| 50mg | 1,838.00 € | ||
| 100mg | 2,320.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
DOV-216,303 Free Base
CAS:66504-40-3
DOV-216,303 inhibits serotonin, norepinephrine, dopamine reuptake (IC50s: 14, 20, 78 nM) with antidepressant properties.
Formula:
C11H11Cl2N
Purity:
96.7%
Color and Shape:
Solid
Molecular weight:
228.12
Ref: TM-T11087
| 1ml | 67.00 € | ||
| 2mg | 45.00 € | ||
| 5mg | 65.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 156.00 € | ||
| 50mg | 221.00 € | ||
| 100mg | 332.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
NUCC-390
CAS:1060524-97-1
NUCC-390, a novel small-molecule CXCR4 receptor agonist, selectively induces CXCR4 receptor internalization while acting antagonistically …
Formula:
C23H33N5O
Purity:
98.18%
Color and Shape:
Solid
Molecular weight:
395.54
Ref: TM-T12269
| 1mg | 146.00 € | ||
| 1ml | 356.00 € | ||
| 5mg | 298.00 € | ||
| 10mg | 465.00 € | ||
| 25mg | 759.00 € | ||
| 50mg | 1,054.00 € | ||
| 100mg | 1,412.00 € | ||
| 500mg | 2,759.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Eplivanserin
CAS:130579-75-8
Eplivanserin (SR-46349) is an effective and selective antagonist of 5-HT2A receptor with a Kd of …
Formula:
C19H21FN2O2
Purity:
97.04%
Color and Shape:
Solid
Molecular weight:
328.38
Ref: TM-T11217
| 1mg | 182.00 € | ||
| 1ml | 419.00 € | ||
| 5mg | 406.00 € | ||
| 10mg | 600.00 € | ||
| 25mg | 917.00 € | ||
| 50mg | 1,281.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
CJ 033466
CAS:519148-48-2
CJ 033466 is a selective partial agonist of 5-HT4 receptor (EC50 = 9 nM) with …
Formula:
C19H28ClN5O
Purity:
98.41%
Color and Shape:
Solid
Molecular weight:
377.91
Ref: TM-T22671
| 1mg | 74.00 € | ||
| 1ml | 253.00 € | ||
| 5mg | 166.00 € | ||
| 10mg | 277.00 € | ||
| 25mg | 441.00 € | ||
| 50mg | 630.00 € | ||
| 100mg | 847.00 € | ||
| 500mg | To inquire |
Estimated delivery in United States, on Monday 25 Nov 2024
NRA-0160
CAS:204718-47-8
NRA-0160 is a selective antagonist of dopamine D4 receptor(Ki of 0.48 nM)
Formula:
C24H23F2N3OS
Purity:
98%
Color and Shape:
Solid
Molecular weight:
439.52
Ref: TM-T12252
| 25mg | 1,410.00 € | ||
| 50mg | 1,852.00 € | ||
| 100mg | 2,338.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
KI-7
CAS:1489263-00-4
KI-7 is an adenosine A2B receptor positive allosteric modulator.
Formula:
C23H18N2O2
Purity:
98.03%
Color and Shape:
Solid
Molecular weight:
354.4
Ref: TM-T9238
| 1mg | 45.00 € | ||
| 1ml | 96.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 147.00 € | ||
| 25mg | 296.00 € | ||
| 50mg | 456.00 € | ||
| 100mg | 690.00 € | ||
| 500mg | 1,427.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
