G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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AB21 HCl
AB21 HCl: σ1 receptor antagonist, Ki 13 nM; less potent at σ2 (102 nM). Reduces …
Formula:
C23H29ClN2O
Purity:
99.89%
Color and Shape:
Liquid
Molecular weight:
384.2
Ref: TM-T77340L
| 1mg | 182.00 € | ||
| 5mg | 401.00 € | ||
| 10mg | 593.00 € | ||
| 25mg | 917.00 € | ||
| 50mg | 1,268.00 € | ||
| 100mg | 1,706.00 € | ||
| 500mg | 3,418.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
AMI-193
CAS:510-74-7
AMI-193 (Spiramide) is a selective 5-HT2 & D2 receptor antagonist with antipsychotic properties.
Formula:
C22H26FN3O2
Purity:
99.04%
Color and Shape:
Solid
Molecular weight:
383.46
Ref: TM-T21855
| 5mg | 45.00 € | ||
| 10mg | 63.00 € | ||
| 25mg | 131.00 € | ||
| 50mg | 208.00 € | ||
| 100mg | 310.00 € | ||
| 1mL*10mM (DMSO) | 50.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Cortistatin-14
CAS:186901-48-4
Cortistatin-14, a neuropeptide structurally similar to growth inhibitor-14, is used to study sepsis-induced cognitive impairment.
Formula:
C81H114N20O18S2
Purity:
98.06%
Color and Shape:
Solid
Molecular weight:
1720.03
Ref: TM-TP1570
| 1mg | 97.00 € | ||
| 5mg | 374.00 € | ||
| 10mg | 671.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
WAY-298630
CAS:303134-93-2
Fluorophenoxy benzimidazole, a CRTH2 blocker, IC50 < 10 μM for rhinitis, COPD, arthritis, eczema, conjunctivitis.
Formula:
C17H15FN2O3S
Purity:
97.13%
Color and Shape:
Liquid
Molecular weight:
346.38
Ref: TM-T77601
| 1mg | 181.00 € | ||
| 5mg | 400.00 € | ||
| 10mg | 595.00 € | ||
| 25mg | 917.00 € | ||
| 50mg | 1,263.00 € | ||
| 100mg | 1,710.00 € | ||
| 500mg | 3,428.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
GLP-1 receptor agonist 9 citrate
GLP-1 receptor agonist 9 citrate is an agonist of GLP-1.
Formula:
C38H39ClFN3O12
Purity:
95%
Color and Shape:
Liquid
Molecular weight:
784.18
Ref: TM-T9579L
| 1mg | 181.00 € | ||
| 5mg | 406.00 € | ||
| 10mg | 600.00 € | ||
| 25mg | 920.00 € | ||
| 50mg | 1,287.00 € | ||
| 100mg | 1,738.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Litoxetine HCl
Litoxetine HCl, an SSRI and 5-HT antagonist, treats urinary incontinence and relaxes rat oesophageal muscles …
Formula:
C16H20ClNO
Purity:
98.98% - 99.19%
Color and Shape:
Soild
Molecular weight:
277.79
Ref: TM-T67956L
| 1mg | 95.00 € | ||
| 5mg | 213.00 € | ||
| 10mg | 319.00 € | ||
| 25mg | 545.00 € | ||
| 50mg | 782.00 € | ||
| 100mg | 1,078.00 € | ||
| 1mL*10mM (DMSO) | 207.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Brexpiprazole S-oxide
CAS:1191900-51-2
Brexpiprazole S-oxide is the main metabolite of Brexpiprazole, a human 5-HT1A and dopamine receptor partial …
Formula:
C25H27N3O3S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
449.57
Ref: TM-T10612
| 100mg | To inquire | ||
| 500mg | To inquire |
Estimated delivery in United States, on Thursday 12 Dec 2024
Ro60-0175
CAS:169675-08-5
Ro60-0175 is a selective 5-HT2B and 5-HT2C serotonin receptor agonist, often used as fumarate.
Formula:
C11H12ClFN2
Purity:
97.09%
Color and Shape:
Liquid
Molecular weight:
226.68
Ref: TM-T39161
| 1mg | 96.00 € | ||
| 5mg | 212.00 € | ||
| 10mg | 346.00 € | ||
| 25mg | 606.00 € | ||
| 50mg | 828.00 € | ||
| 100mg | 1,141.00 € | ||
| 1mL*10mM (DMSO) | 193.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
O-Desethyl Dapagliflozin
CAS:864070-37-1
O-Desethyl Dapagliflozin (Empagliflozin-4) is a SGLT2 inhibitor, IC50=33nM.
Formula:
C19H21ClO6
Purity:
97.09%
Color and Shape:
Liquid
Molecular weight:
380.82
Ref: TM-T67849
| 1mg | 56.00 € | ||
| 5mg | 119.00 € | ||
| 10mg | 182.00 € | ||
| 25mg | 314.00 € | ||
| 50mg | 460.00 € | ||
| 100mg | 667.00 € | ||
| 1mL*10mM (DMSO) | 132.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
LY 344864 racemate
CAS:186543-64-6
LY 344864 racemate is a 5-HT1F receptor agonist.
Formula:
C21H22FN3O
Purity:
99.47%
Color and Shape:
Soild
Molecular weight:
351.42
Ref: TM-T2344L
| 5mg | 45.00 € | ||
| 10mg | 69.00 € | ||
| 25mg | 103.00 € | ||
| 50mg | 172.00 € | ||
| 100mg | To inquire | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Upacicalcet HCl
Upacicalcet HCl, a calcium mimetic, reduces blood PTH by targeting parathyroid receptors; treats secondary hyperparathyroidism.
Formula:
C11H15Cl2N3O6S
Purity:
98.56%
Color and Shape:
Soild
Molecular weight:
388.22
Ref: TM-T29067L
| 1mg | 172.00 € | ||
| 5mg | 424.00 € | ||
| 10mg | 621.00 € | ||
| 25mg | 989.00 € | ||
| 50mg | 1,337.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
![(1R,5S,6r)-N-(2-methyl-1-((3-methylpyridin-2-yl)oxy)propan-2-yl)-3-azabicyclo[3.1.0]hexane-6-carbo…](https://static.cymitquimica.com/products/TM/thumb/T77670.jpg)
(1R,5S,6r)-N-(2-methyl-1-((3-methylpyridin-2-yl)oxy)propan-2-yl)-3-azabicyclo[3.1.0]hexane-6-carboxamide L(+)-Tartaric acid
CAS:2919211-45-1
(1R,5S,6r)-N-(2-methyl-1-((3-methylpyridin-2-yl)oxy)propan-2-yl)-3-azabicyclo[3.1.0]hexane-6-carboxamide L(+)-Tartaric acid is a potential SSTR4 agonist.
Formula:
C20H29N3O8
Purity:
99.23%
Color and Shape:
Soild
Molecular weight:
439.46
Ref: TM-T77670
| 1mg | 182.00 € | ||
| 5mg | 402.00 € | ||
| 10mg | 591.00 € | ||
| 25mg | 917.00 € | ||
| 50mg | 1,271.00 € | ||
| 100mg | 1,706.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
RS 15385-198
CAS:121961-55-5
RS 15385-198 is a less active isomer of Delequamine. Delequamine is a selective alpha2-adrenergic receptor …
Formula:
C18H26N2O3S
Purity:
98.81%
Color and Shape:
Soild
Molecular weight:
350.48
Ref: TM-T68051L
| 1mg | 183.00 € | ||
| 5mg | 453.00 € | ||
| 10mg | 648.00 € | ||
| 25mg | 1,011.00 € | ||
| 50mg | 1,395.00 € | ||
| 100mg | 1,844.00 € | ||
| 500mg | 3,679.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Pranazepide
CAS:150408-73-4
Pranazepide (FK 480) is a small molecule cholecystokinin receptor antagonist used to study digestive disorders …
Formula:
C26H19FN4O2
Purity:
98.20% - 99.68%
Color and Shape:
Solid
Molecular weight:
438.45
Ref: TM-T34123
| 1mg | 513.00 € | ||
| 5mg | 1,129.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Sufotidine
CAS:80343-63-1
Sufotidine (AH 25352X) is a highly selective competitive H2 receptor antagonist.
Formula:
C20H31N5O3S
Purity:
99% - 99.28%
Color and Shape:
Liquid
Molecular weight:
421.56
Ref: TM-T68146
| 1mg | 233.00 € | ||
| 5mg | 582.00 € | ||
| 10mg | 824.00 € | ||
| 25mg | 1,236.00 € | ||
| 50mg | 1,654.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Eledoisin Related Peptide
CAS:2990-43-4
Eledoisin Related Peptide (Eledoisin RP) is a tachykinin receptor ligand.
Formula:
C34H58N8O6S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
706.94
Ref: TM-T7631
| 1mg | 153.00 € | ||
| 5mg | 641.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Donitriptan hydrochloride
CAS:170911-68-9
Donitriptan hydrochloride (Donitriptan monohydrochloride) is a potent, high efficacy agonist of 5-HT1B/1D receptors with pKis …
Formula:
C23H26ClN5O2
Purity:
99.8% - 99.8%
Color and Shape:
Solid
Molecular weight:
439.94
Ref: TM-T21666
| 2mg | 40.00 € | ||
| 5mg | 49.00 € | ||
| 10mg | 63.00 € | ||
| 25mg | 132.00 € | ||
| 50mg | 234.00 € | ||
| 100mg | 332.00 € | ||
| 200mg | 430.00 € | ||
| 500mg | To inquire |
Estimated delivery in United States, on Thursday 12 Dec 2024
Tiaprost
CAS:71116-82-0
Tiaprost is a analog of prostaglandin F2α .
Formula:
C20H28O6S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
396.5
Ref: TM-T17092
| 1mg | 162.00 € | ||
| 5mg | 650.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Ebalzotan
CAS:149494-37-1
NAE-086 is a high-affinity and selective 5-HT(1A) receptor ligand with a K(i) value of 4.5 …
Formula:
C19H30N2O2
Purity:
99.08% - 99.41%
Color and Shape:
Liquid
Molecular weight:
318.45
Ref: TM-T68059
| 1mg | 271.00 € | ||
| 5mg | 737.00 € | ||
| 10mg | 1,101.00 € | ||
| 25mg | 2,001.00 € | ||
| 50mg | 2,624.00 € | ||
| 100mg | 3,492.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Meclinertant
CAS:146362-70-1
Meclinertant: selective NTS1 antagonist, blocks Ca2+ mobilization, with anxiolytic and anti-addictive properties.
Formula:
C32H31ClN4O5
Purity:
99.35%
Color and Shape:
Solid
Molecular weight:
587.07
Ref: TM-T16034
| 1mg | 86.00 € | ||
| 2mg | 131.00 € | ||
| 5mg | 282.00 € | ||
| 10mg | 546.00 € | ||
| 25mg | 857.00 € | ||
| 50mg | 1,170.00 € | ||
| 100mg | 1,569.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
