G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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FTBMT
CAS:1358575-02-6
FTBMT is a selective GPR52 agonist (EC50: 75 nM) and it also has antipsychotic and …
Formula:
C19H16F4N4O
Purity:
99.12%
Color and Shape:
Solid
Molecular weight:
392.35
Ref: TM-T15352
| 5mg | 52.00 € | ||
| 10mg | 85.00 € | ||
| 25mg | 170.00 € | ||
| 50mg | 301.00 € | ||
| 100mg | 469.00 € | ||
| 200mg | 620.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Levocarnitine propionate hydrochloride
CAS:119793-66-7
Levocarnitine propionate hydrochloride (ST-261) is used for the treatment of the deterioration of renal function, …
Formula:
C10H20ClNO4
Purity:
90% - 98%
Color and Shape:
Solid
Molecular weight:
253.72
Ref: TM-T1182
| 25mg | 35.00 € | ||
| 50mg | 50.00 € | ||
| 100mg | 65.00 € | ||
| 500mg | 153.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Duloxetine hydrochloride
CAS:136434-34-9
Duloxetine hydrochloride is an SNRI used for depression, anxiety, and pain in diabetes and fibromyalgia.
Formula:
C18H20ClNOS
Purity:
100% - 99.97%
Color and Shape:
White Or White Crystalline Powder
Molecular weight:
333.88
Ref: TM-T1471
| 10mg | 52.00 € | ||
| 50mg | 86.00 € | ||
| 100mg | 106.00 € | ||
| 200mg | 133.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Dexchlorpheniramine Maleate
CAS:2438-32-6
Dexchlorpheniramine Maleate, an antihistamine with anticholinergic effects, treats allergies like hay fever. It's the active …
Formula:
C20H23ClN2O4
Purity:
99.58%
Color and Shape:
White Or Almost White Crystalline Powder
Molecular weight:
390.86
Ref: TM-T0785
| 100mg | 34.00 € | ||
| 1mL*10mM (DMSO) | 42.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Rimonabant hydrochloride
CAS:158681-13-1
Rimonabant hydrochloride (SR 141716A) 是中心大麻素受体 1 的高效选择性反向激动剂, Ki 值为1.8 nM。它也能够抑制分枝杆菌膜蛋白3。
Formula:
C22H22Cl4N4O
Purity:
100% - 99.5%
Color and Shape:
Off-White To White Crystalline Powder
Molecular weight:
500.25
Ref: TM-T1519
| 5mg | 46.00 € | ||
| 10mg | 66.00 € | ||
| 25mg | 116.00 € | ||
| 50mg | 207.00 € | ||
| 100mg | 310.00 € | ||
| 500mg | 743.00 € | ||
| 1mL*10mM (DMSO) | 74.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
(+)-Dropropizine
CAS:99291-24-4
(+)-Dropropizine can inhibit histamine receptor, anti-allergic, and reduce a cough by modulation of neuropeptides involved …
Formula:
C13H20N2O2
Purity:
99.92%
Color and Shape:
White Or Off White Crystalline Powder
Molecular weight:
236.31
Ref: TM-T0217L
| 1g | 49.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Olodaterol
CAS:868049-49-4
Olodaterol is a novel, long-acting beta2-adrenergic agonist (LABA) that exerts its pharmacological effect by binding …
Formula:
C21H26N2O5
Purity:
98.9%
Color and Shape:
Solid
Molecular weight:
386.45
Ref: TM-T3457
| 1mg | 49.00 € | ||
| 5mg | 87.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
PF-04995274
CAS:1331782-27-4
PF-04995274: potent, selective partial 5-HT4R agonist; EC50 0.26-0.47 nM; brain penetrant; may treat Alzheimer's cognitive …
Formula:
C23H32N2O6
Purity:
99.52%
Color and Shape:
Solid
Molecular weight:
432.51
Ref: TM-T16481
| 1mg | 35.00 € | ||
| 5mg | 74.00 € | ||
| 10mg | 124.00 € | ||
| 25mg | 197.00 € | ||
| 50mg | 350.00 € | ||
| 100mg | 505.00 € | ||
| 1mL*10mM (DMSO) | 73.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
SR59230A
CAS:174689-39-5
SR59230A is a potent, selective antagonist of β3-adrenergic receptor(β3, β1, and β2 receptors with IC50s …
Formula:
C23H29NO6
Purity:
98.84%
Color and Shape:
Solid
Molecular weight:
415.48
Ref: TM-T13016
| 1mg | 52.00 € | ||
| 2mg | 77.00 € | ||
| 5mg | 107.00 € | ||
| 10mg | 172.00 € | ||
| 25mg | 343.00 € | ||
| 50mg | 510.00 € | ||
| 100mg | 737.00 € | ||
| 1mL*10mM (DMSO) | 125.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Citalopram hydrobromide
CAS:59729-32-7
Citalopram hydrobromide (XU-62-320) , a selective serotonin reuptake inhibitor (SSRI), selectively inhibits the CNS neuronal …
Formula:
C20H22BrFN2O
Purity:
99.81%
Color and Shape:
White Crystalline Powder
Molecular weight:
405.304
Ref: TM-T1483
| 10mg | 48.00 € | ||
| 25mg | 71.00 € | ||
| 50mg | 89.00 € | ||
| 100mg | 110.00 € | ||
| 200mg | 155.00 € | ||
| 500mg | 246.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Amitraz
CAS:33089-61-1
Amitraz (NSC 324552): white monoclinic crystals, mp 86-87°C, water-insoluble, used as acaricide and in canine …
Formula:
C19H23N3
Purity:
99.62%
Color and Shape:
White/Pale Yellow Crystalline Solid
Molecular weight:
293.41
Ref: TM-T1632
| 1g | 52.00 € | ||
| 500mg | 39.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Anamorelin
CAS:249921-19-5
Anamorelin (ONO-7643) is a novel ghrelin receptor agonist (EC50: 0.74 nM in the FLIPR assay).
Formula:
C31H42N6O3
Purity:
99.35% - 99.88%
Color and Shape:
Solid
Molecular weight:
546.7
Ref: TM-T10319
| 5mg | 60.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 127.00 € | ||
| 50mg | 177.00 € | ||
| 1mL*10mM (DMSO) | 73.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Atomoxetine hydrochloride
CAS:82248-59-7
Atomoxetine HCl (LY 139603) is a selective non-stimulant ADHD drug that blocks norepinephrine reuptake, enhancing …
Formula:
C17H22ClNO
Purity:
99.86%
Color and Shape:
White Solid
Molecular weight:
291.82
Ref: TM-T0869
| 25mg | 48.00 € | ||
| 50mg | 59.00 € | ||
| 100mg | 85.00 € | ||
| 200mg | 115.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Tripelennamine hydrochloride
CAS:154-69-8
Tripelennamine hydrochloride (Pyribenzamine hydrochloride) is a histamine H1 antagonist with low sedative action but frequent …
Formula:
C16H21N3·HCl
Purity:
100% - 99.54%
Color and Shape:
White Solid
Molecular weight:
291.82
Ref: TM-T1269
| 1g | 139.00 € | ||
| 100mg | 37.00 € | ||
| 500mg | 97.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Talipexole dihydrochloride
CAS:36085-73-1
Talipexole dihydrochloride (Domnin) is a dopamine D2 receptor agonist, α2-adrenoceptor agonist, and 5-HT3 receptor antagonist …
Formula:
C10H17Cl2N3S
Purity:
98.64%
Color and Shape:
Light Yellow Solid
Molecular weight:
282.23
Ref: TM-T14490
| 2mg | 38.00 € | ||
| 5mg | 56.00 € | ||
| 10mg | 89.00 € | ||
| 25mg | 154.00 € | ||
| 50mg | 264.00 € | ||
| 100mg | 424.00 € | ||
| 200mg | 613.00 € | ||
| 500mg | 949.00 € | ||
| 1mL*10mM (DMSO) | 63.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
AMG 487
CAS:473719-41-4
AMG 487: potent CXCR3 antagonist, blocks CXCL10/CXCL11 binding, IC50s: 8.0/8.2 nM.
Formula:
C32H28F3N5O4
Purity:
99.89%
Color and Shape:
Solid
Molecular weight:
603.59
Ref: TM-T10297L
| 1mg | 52.00 € | ||
| 2mg | 77.00 € | ||
| 5mg | 115.00 € | ||
| 10mg | 164.00 € | ||
| 25mg | 268.00 € | ||
| 50mg | 398.00 € | ||
| 100mg | 587.00 € | ||
| 1mL*10mM (DMSO) | 154.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Centanafadine hydrochloride
CAS:923981-14-0
Centanafadine HCl is a NE/DA reuptake inhibitor, also affects serotonin (IC50: NE 6 nM, DA …
Formula:
C15H16ClN
Purity:
99.65%
Color and Shape:
Solid
Molecular weight:
245.75
Ref: TM-T10758L
| 1mg | 59.00 € | ||
| 5mg | 126.00 € | ||
| 10mg | 202.00 € | ||
| 25mg | 406.00 € | ||
| 50mg | 653.00 € | ||
| 100mg | 1,026.00 € | ||
| 200mg | 1,378.00 € | ||
| 500mg | 2,052.00 € | ||
| 1mL*10mM (DMSO) | 140.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Naphazoline hydrochloride
CAS:550-99-2
Naphazoline hydrochloride (Naphazoline HCl) is an adrenergic vasoconstrictor agent used as a decongestant.
Formula:
C14H15ClN2
Purity:
97.6%
Color and Shape:
White Crystalline Powder White Crystalline Powder
Molecular weight:
246.74
Ref: TM-T0446
| 1g | 34.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
PF-06882961
CAS:2230198-02-2
PF-06882961 is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.
Formula:
C31H30FN5O4
Purity:
95.1% - 99.54%
Color and Shape:
Solid
Molecular weight:
555.6
Ref: TM-T12431
| 1mg | 49.00 € | ||
| 5mg | 89.00 € | ||
| 10mg | 156.00 € | ||
| 25mg | 197.00 € | ||
| 50mg | 253.00 € | ||
| 100mg | 434.00 € | ||
| 1mL*10mM (DMSO) | 109.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Terlipressin Acetate
CAS:1884420-36-3
Terlipressin Acetate, a highly selective vasopressin V1 receptor agonist, on OGD/R-induced damage in intestinal epithelial …
Formula:
C56H82N16O19S2
Purity:
98.50% - 99.69%
Color and Shape:
Solid
Molecular weight:
1347.5
Ref: TM-T13920L
| 5mg | 48.00 € | ||
| 10mg | 62.00 € | ||
| 25mg | 103.00 € | ||
| 50mg | 136.00 € | ||
| 100mg | 207.00 € | ||
| 200mg | 310.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
