G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Levosulpiride
CAS:23672-07-3
Levosulpiride (S-(-)-Sulpiride) is the (S)-enantiomer of sulpiride, which is a D2 receptor antagonist, an atypical …
Formula:
C15H23N3O4S
Purity:
99.88% - 99.93%
Color and Shape:
White Crystalline Powder
Molecular weight:
341.43
Ref: TM-T1211
| 100mg | 55.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
Haloperidol
CAS:52-86-8
Haloperidol (Serenace) is a highly potent neuroleptic by relieving nervous through the depression of nerve …
Formula:
C21H23ClFNO2
Purity:
99.69% - 99.76%
Color and Shape:
Crystals Solid
Molecular weight:
375.86
Ref: TM-T0025
| 25mg | 35.00 € | ||
| 50mg | 48.00 € | ||
| 100mg | 55.00 € | ||
| 200mg | 71.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
ZT 52656A hydrochloride
CAS:115730-24-0
ZT 52656A is a selective agonist of kappa opioid, and used for the prevention or …
Formula:
C19H26ClF3N2O
Purity:
98.78%
Color and Shape:
Solid
Molecular weight:
390.87
Ref: TM-T13414
| 1mg | 540.00 € | ||
| 5mg | 1,198.00 € | ||
| 10mg | 1,786.00 € | ||
| 25mg | 3,030.00 € | ||
| 50mg | 3,924.00 € | ||
| 100mg | 5,120.00 € | ||
| 1mL*10mM (DMSO) | 1,283.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
FTBMT
CAS:1358575-02-6
FTBMT is a selective GPR52 agonist (EC50: 75 nM) and it also has antipsychotic and …
Formula:
C19H16F4N4O
Purity:
99.12%
Color and Shape:
Solid
Molecular weight:
392.35
Ref: TM-T15352
| 5mg | 52.00 € | ||
| 10mg | 85.00 € | ||
| 25mg | 170.00 € | ||
| 50mg | 301.00 € | ||
| 100mg | 469.00 € | ||
| 200mg | 620.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
KGA-2727
CAS:666842-36-0
KGA-2727: potent, selective SGLT1 inhibitor (human Ki 97.4 nM, rat 43.5 nM), with high selectivity …
Formula:
C26H40N4O8
Purity:
98.95%
Color and Shape:
Solid
Molecular weight:
536.62
Ref: TM-T15656
| 1mg | 133.00 € | ||
| 2mg | 183.00 € | ||
| 5mg | 274.00 € | ||
| 10mg | 454.00 € | ||
| 25mg | 750.00 € | ||
| 50mg | 1,026.00 € | ||
| 100mg | 1,406.00 € | ||
| 1mL*10mM (DMSO) | 323.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
Phenothiazine
CAS:92-84-2
Phenothiazine (ENT 38) is a class of agents exhibiting antiemetic, antipsychotic, antihistaminic, and anticholinergic activities.
Formula:
C12H9NS
Purity:
99.94%
Color and Shape:
Yellow Solid Pellets
Molecular weight:
199.27
Ref: TM-T0776
| 1g | 42.00 € | ||
| 5g | 88.00 € | ||
| 10g | 115.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
LIT-001
CAS:2245072-21-1
LIT-001 improves social interaction in a mouse model of autism.It is the first nonpeptide oxytocin …
Formula:
C30H34F3N7O4S
Purity:
96.88% - 98.25%
Color and Shape:
Solid
Molecular weight:
645.7
Ref: TM-T11857
| 1mg | 70.00 € | ||
| 5mg | 153.00 € | ||
| 10mg | 273.00 € | ||
| 25mg | 432.00 € | ||
| 50mg | 638.00 € | ||
| 100mg | 908.00 € | ||
| 500mg | 1,825.00 € | ||
| 1mL*10mM (DMSO) | 212.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
Ceruletide
CAS:17650-98-5
Ceruletide is a decapeptide that is a safe and effective cholecystokinin and cholecystokinin receptor agonist.Cost-effective …
Formula:
C58H73N13O21S2
Purity:
97.54% - 98.47%
Color and Shape:
Solid
Molecular weight:
1352.4
Ref: TM-T14932
| 1mg | 159.00 € | ||
| 5mg | 430.00 € | ||
| 10mg | 605.00 € | ||
| 25mg | 938.00 € | ||
| 50mg | 1,283.00 € | ||
| 100mg | 1,738.00 € | ||
| 200mg | 2,337.00 € | ||
| 500µg | 107.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
AB928
CAS:2239273-34-6
AB928 is an orally bioavailable, selective dual adenosine receptor (A2aR/A2bR) antagonist. It has immunomodulatory activity[1].
Formula:
C23H22N8O
Purity:
100% - 98.55%
Color and Shape:
Solid
Molecular weight:
426.47
Ref: TM-T14078
| 1mg | 50.00 € | ||
| 5mg | 124.00 € | ||
| 10mg | 197.00 € | ||
| 25mg | 389.00 € | ||
| 50mg | 462.00 € | ||
| 100mg | 663.00 € | ||
| 1mL*10mM (DMSO) | 134.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
Frovatriptan succinate hydrate
CAS:158930-17-7
Frovatriptan treats all migraine types, nausea, vomiting, light/sound sensitivity, and prevents menstrual migraines; it targets …
Formula:
C18H25N3O6
Purity:
99.95%
Color and Shape:
Solid
Molecular weight:
379.41
Ref: TM-T11326
| 2mg | 35.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 144.00 € | ||
| 50mg | 207.00 € | ||
| 100mg | 306.00 € | ||
| 1mL*10mM (DMSO) | 59.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
Bambuterol hydrochloride
CAS:81732-46-9
Bambuterol hydrochloride (KWD-2183 hydrochloride) , a long-acting beta-adrenoceptor agonist, is utilized for the treating of …
Formula:
C18H30ClN3O5
Purity:
100% - 99.74%
Color and Shape:
White Solid
Molecular weight:
403.91
Ref: TM-T1446
| 10mg | 48.00 € | ||
| 25mg | 69.00 € | ||
| 50mg | 88.00 € | ||
| 100mg | 97.00 € | ||
| 200mg | 133.00 € | ||
| 500mg | 212.00 € | ||
| 1mL*10mM (DMSO) | 44.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
N6-Ethyladenosine
CAS:14357-08-5
N6-Ethyladenosine is an adenosine derivative, acts as an agonist of Adenosine receptor(hA1AR and hA3AR with …
Formula:
C12H17N5O4
Purity:
99.96%
Color and Shape:
Solid
Molecular weight:
295.29
Ref: TM-T12161
| 2mg | 34.00 € | ||
| 5mg | 50.00 € | ||
| 10mg | 80.00 € | ||
| 25mg | 131.00 € | ||
| 50mg | 212.00 € | ||
| 100mg | 313.00 € | ||
| 200mg | 452.00 € | ||
| 1mL*10mM (DMSO) | 86.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
Asenapine Maleate
CAS:85650-56-2
Asenapine Maleate (Org 5222 maleate) is a second generation (atypical) antipsychotic agent that is taken …
Formula:
C21H20ClNO5
Purity:
99.73%
Color and Shape:
Solid
Molecular weight:
401.84
Ref: TM-T1951
| 5mg | 35.00 € | ||
| 10mg | 51.00 € | ||
| 25mg | 80.00 € | ||
| 50mg | 96.00 € | ||
| 100mg | 135.00 € | ||
| 200mg | 225.00 € | ||
| 500mg | 373.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
AH 6809
CAS:33458-93-4
AH 6809 blocks EP1, EP2, EP3, DP receptors (Ki: 1217-1597 nM human, 350 nM mouse …
Formula:
C17H14O5
Purity:
97.59%
Color and Shape:
Solid
Molecular weight:
298.29
Ref: TM-T14148
| 1mg | 35.00 € | ||
| 5mg | 66.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 168.00 € | ||
| 50mg | 264.00 € | ||
| 100mg | 424.00 € | ||
| 200mg | 612.00 € | ||
| 1mL*10mM (DMSO) | 71.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
Adenosine A1 receptor activator T62
CAS:40312-34-3
Adenosine A1 receptor activator T62 is an allosteric enhancer of adenosine A1 receptor, and it …
Formula:
C15H14ClNOS
Purity:
95.00%
Color and Shape:
Solid
Molecular weight:
291.8
Ref: TM-T14127
| 1mg | 87.00 € | ||
| 5mg | 183.00 € | ||
| 10mg | 273.00 € | ||
| 25mg | 439.00 € | ||
| 50mg | 598.00 € | ||
| 100mg | 810.00 € | ||
| 200mg | 1,074.00 € | ||
| 1mL*10mM (DMSO) | 280.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
Doxylamine succinate
CAS:562-10-7
Doxylamine Succinate is a pyridine derivate histamine H1 antagonist with pronounced sedative properties.
Formula:
C21H28N2O5
Purity:
100%
Color and Shape:
5 1 (Ntp 1992)
Molecular weight:
388.46
Ref: TM-T1115
| 25mg | 44.00 € | ||
| 50mg | 55.00 € | ||
| 100mg | 66.00 € | ||
| 200mg | 100.00 € | ||
| 500mg | 164.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
Flopropione
CAS:2295-58-1
Flopropione (Phloropropiophenone), a spasmolytic or antispasmodic agent, is used as a 5-HT1A receptor antagonist.
Formula:
C9H10O4
Purity:
100%
Color and Shape:
Solid
Molecular weight:
182.17
Ref: TM-T0525
| 50mg | 35.00 € | ||
| 100mg | 48.00 € | ||
| 200mg | 62.00 € | ||
| 500mg | 90.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
JP1302 dihydrochloride
CAS:1259314-65-2
JP1302 dihydrochloride: selective α2C-adrenoceptor antagonist; Ki=28 nM, Kb=16 nM.
Formula:
C24H26Cl2N4
Purity:
99.61%
Color and Shape:
Solid
Molecular weight:
441.4
Ref: TM-T11726
| 1mg | 46.00 € | ||
| 2mg | 59.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 127.00 € | ||
| 25mg | 235.00 € | ||
| 50mg | 379.00 € | ||
| 100mg | 562.00 € | ||
| 500mg | 1,216.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
BI-671800
CAS:1093108-50-9
BI-671800 (AP-761) is a DP2/CRTH2 antagonist with IC50 values of 4.5 nM and 3.7 nM, …
Formula:
C25H26F3N5O3
Purity:
99.19%
Color and Shape:
Solid
Molecular weight:
501.5
Ref: TM-T14565
| 1mg | 58.00 € | ||
| 5mg | 131.00 € | ||
| 10mg | 207.00 € | ||
| 25mg | 373.00 € | ||
| 50mg | 530.00 € | ||
| 100mg | 718.00 € | ||
| 200mg | 938.00 € | ||
| 1mL*10mM (DMSO) | 144.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
Metoclopramide hydrochloride
CAS:7232-21-5
Metoclopramide hydrochloride (Metoclopramide HCl) is a selective dopamine D2 receptor antagonist, used as an antiemetic.
Formula:
C14H22ClN3O2·HCl
Purity:
99.94%
Color and Shape:
White To Off-White Powder
Molecular weight:
336.26
Ref: TM-T1069
| 10mg | 39.00 € | ||
| 25mg | 55.00 € | ||
| 50mg | 78.00 € | ||
| 100mg | 90.00 € | ||
| 200mg | 144.00 € | ||
| 500mg | 230.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Monday 3 Mar 2025
