G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
Read more
Tegaserod maleate
CAS:189188-57-6
Tegaserod (SDZ-HTF-919), a 5-HT4 agonist for irritable bowel syndrome, was withdrawn by FDA on March …
Formula:
C20H27N5O5
Purity:
98% - 99.06%
Color and Shape:
White Powder
Molecular weight:
417.46
Ref: TM-T1551
| 10mg | 46.00 € | ||
| 25mg | 78.00 € | ||
| 50mg | 118.00 € | ||
| 100mg | 194.00 € | ||
| 200mg | 295.00 € | ||
| 500mg | 497.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Paroxetine hydrochloride
CAS:78246-49-8
Paroxetine hydrochloride (Paroxetine HCl) is a serotonin uptake inhibitor that is effective in the treatment …
Formula:
C19H21ClFNO3
Purity:
98% - 99.91%
Color and Shape:
White Crystalline Powder
Molecular weight:
365.826
Ref: TM-T1636
| 25mg | 54.00 € | ||
| 50mg | 63.00 € | ||
| 100mg | 89.00 € | ||
| 200mg | 113.00 € | ||
| 500mg | 153.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Betahistine mesylate
CAS:54856-23-4
Betahistine mesylate (Extovyl), an H1 agonist and vasodilator, treats Meniere's disease and vascular headaches; risks …
Formula:
C8H12N2·2(CH4O3S)
Purity:
98%
Color and Shape:
Coa
Molecular weight:
328.4
Ref: TM-T0246L
| 10mg | 35.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Ethamsylate
CAS:2624-44-4
Ethamsylate (Dicynene) enhances capillary stability, platelet adhesion, and blocks prostaglandins to act as a hemostatic …
Formula:
C10H17NO5S
Purity:
99.98%
Color and Shape:
White Crystals Or Crystalline Powder
Molecular weight:
263.31
Ref: TM-T0002
| 5g | 88.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Dapoxetine hydrochloride
CAS:129938-20-1
Dapoxetine hydrochloride (LY-210448 hydrochloride) is a selectivity short-acting serotonin reuptake inhibitor, used for the therapy …
Formula:
C21H23NO·HCl
Purity:
100% - 99%
Color and Shape:
White To Off-White Crystalline Solid
Molecular weight:
341.87
Ref: TM-T6461
| 10mg | 35.00 € | ||
| 25mg | 57.00 € | ||
| 50mg | 74.00 € | ||
| 100mg | 99.00 € | ||
| 200mg | 154.00 € | ||
| 500mg | 241.00 € | ||
| 1mL*10mM (DMSO) | 65.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Prasugrel
CAS:150322-43-3
Prasugrel (CS-747) is a piperazine derivative and PLATELET AGGREGATION INHIBITOR that is used to prevent …
Formula:
C20H20FNO3S
Purity:
98.62% - 99.76%
Color and Shape:
White Solid
Molecular weight:
373.44
Ref: TM-T0230
| 25mg | 46.00 € | ||
| 50mg | 60.00 € | ||
| 100mg | 76.00 € | ||
| 200mg | 117.00 € | ||
| 500mg | 190.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Sulfisoxazole
CAS:127-69-5
Sulfisoxazole: a short-acting antibacterial targeting gram-positive/negative bacteria and inhibits breast cancer exosome by affecting endothelin …
Formula:
C11H13N3O3S
Purity:
99.98%
Color and Shape:
White To Cream Powder
Molecular weight:
267.3
Ref: TM-T0750
| 1g | 73.00 € | ||
| 200mg | 37.00 € | ||
| 500mg | 52.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Pranlukast
CAS:103177-37-3
Pranlukast (ONO-1078) is a cysteinyl leukotriene receptor-1 antagonist.
Formula:
C27H23N5O4
Purity:
99.85%
Color and Shape:
Off-White Solid
Molecular weight:
481.5
Ref: TM-T0694
| 25mg | 54.00 € | ||
| 50mg | 78.00 € | ||
| 100mg | 87.00 € | ||
| 200mg | 124.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
ONC206
CAS:1638178-87-6
ONC206, an analogue of the TRAIL inducer ONC201, acts as a selective antagonist of the …
Formula:
C23H22F2N4O
Purity:
99.93%
Color and Shape:
Solid
Molecular weight:
408.44
Ref: TM-T16392
| 2mg | 34.00 € | ||
| 5mg | 49.00 € | ||
| 10mg | 81.00 € | ||
| 25mg | 117.00 € | ||
| 50mg | 203.00 € | ||
| 100mg | 302.00 € | ||
| 1mL*10mM (DMSO) | 50.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Amisulpride
CAS:71675-85-9
Amisulpride (Solian/Deniban), a dopamine antagonist antipsychotic, treats psychosis and schizophrenia in Europe/Australia, not in the …
Formula:
C17H27N3O4S
Purity:
100%
Color and Shape:
White Or Almost White Crystalline Powder
Molecular weight:
369.48
Ref: TM-T0811
| 1g | 346.00 € | ||
| 25mg | 49.00 € | ||
| 50mg | 68.00 € | ||
| 100mg | 90.00 € | ||
| 200mg | 138.00 € | ||
| 500mg | 238.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Oxolinic acid
CAS:14698-29-4
Oxolinic acid (Nidantin) is a synthetic antimicrobial related to NALIDIXIC ACID and used in URINARY …
Formula:
C13H11NO5
Purity:
98.15% - 98.39%
Color and Shape:
Crystals From Dimethylformamide White Crystalline Powder
Molecular weight:
261.23
Ref: TM-T1233
| 1g | 53.00 € | ||
| 250mg | 40.00 € | ||
| 500mg | 50.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
BP 897 hydrochloride
CAS:314776-92-6
BP 897: potent D3 agonist (Ki: 0.92 nM), weak D2 antagonist (Ki: 61 nM), low …
Formula:
C26H32ClN3O2
Purity:
99.42%
Color and Shape:
Solid
Molecular weight:
454
Ref: TM-T14767
| 1mg | 36.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 109.00 € | ||
| 25mg | 212.00 € | ||
| 50mg | 346.00 € | ||
| 100mg | 553.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Chlorpheniramine maleate
CAS:113-92-8
Chlorpheniramine maleate (NCI-C55265) is a histamine H1 antagonist used in allergic reactions, hay fever, rhinitis, …
Formula:
C20H23ClN2O4
Purity:
99.67%
Color and Shape:
Odorless White Crystalline Solid Or White Powder With A Bitter Taste
Molecular weight:
390.87
Ref: TM-T1553
| 200mg | 34.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Pimethixene
CAS:314-03-4
Pimethixene (Calmixen) blocks 5-HT1A, 2A/B/C, H1, D2/D4.4 & muscarinic M1/M2 receptors; potent with pKis 7.54-10.44.
Formula:
C19H19NS
Purity:
99.1%
Color and Shape:
Solid
Molecular weight:
293.43
Ref: TM-T12489
| 2mg | 34.00 € | ||
| 5mg | 50.00 € | ||
| 10mg | 63.00 € | ||
| 25mg | 103.00 € | ||
| 50mg | 152.00 € | ||
| 100mg | 218.00 € | ||
| 200mg | 326.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Nylidrin hydrochloride
CAS:849-55-8
Nylidrin HCl inhibits IgG1-induced histamine release in guinea pigs and IgE-induced release in rat mast …
Formula:
C19H26ClNO2
Purity:
100%
Color and Shape:
Solid
Molecular weight:
335.87
Ref: TM-T0173
| 1g | 277.00 € | ||
| 25mg | 37.00 € | ||
| 50mg | 52.00 € | ||
| 100mg | 68.00 € | ||
| 200mg | 95.00 € | ||
| 500mg | 185.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Itopride hydrochloride
CAS:122892-31-3
Itopride hydrochloride (Ganaton) is an AChE and D2DR inhibitor.
Formula:
C20H27ClN2O4
Purity:
99.76%
Color and Shape:
White Or Pale Brownish Crystal
Molecular weight:
394.9
Ref: TM-T1552
| 50mg | 41.00 € | ||
| 100mg | 54.00 € | ||
| 500mg | 85.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Bromperidol
CAS:10457-90-6
Bromperidol (R-11333) is a butyrophenone derivative and it is a potent and long-acting neuroleptic.
Formula:
C21H23BrFNO2
Purity:
99.89%
Color and Shape:
Tan Solid
Molecular weight:
420.32
Ref: TM-T14830
| 10mg | 43.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Roxatidine Acetate hydrochloride
CAS:93793-83-0
Roxatidine Acetate hydrochloride (HOE 760) is a specific and competitive histamin H2-receptor antagonist. Roxatidine inhibits …
Formula:
C19H29ClN2O4
Purity:
99.61%
Color and Shape:
Solid
Molecular weight:
384.9
Ref: TM-T0157
| 200mg | 34.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
MRGPRX1 agonist 1
CAS:2377379-39-8
MRGPRX1 agonist 1 is a highly potent MRGPRX1 (Mas-related G-protein-coupled receptor X1)agonist(EC50 of 50 nM).
Formula:
C23H21N3O4S
Purity:
99.59%
Color and Shape:
Solid
Molecular weight:
435.5
Ref: TM-T12104
| 1mg | 87.00 € | ||
| 5mg | 206.00 € | ||
| 10mg | 330.00 € | ||
| 25mg | 599.00 € | ||
| 50mg | 820.00 € | ||
| 100mg | 1,169.00 € | ||
| 1mL*10mM (DMSO) | 228.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Terbutaline
CAS:23031-25-6
Terbutaline is a short-acting agonist of β2-adrenergic receptor (β2-AR) . It is an active metabolite …
Formula:
C12H19NO3
Purity:
99.46%
Color and Shape:
Solid
Molecular weight:
225.3
Ref: TM-T8810
| 5mg | 42.00 € | ||
| 10mg | 55.00 € | ||
| 25mg | 90.00 € | ||
| 50mg | 115.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
