G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Agomelatine
CAS:138112-76-2
Agomelatine (Valdoxan), like melatonin, boosts mood by targeting melatonin and 5-HT2C receptors.
Formula:
C15H17NO2
Purity:
99.92%
Color and Shape:
White Solid
Molecular weight:
243.3
Ref: TM-T1445
| 5mg | 67.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 138.00 € | ||
| 50mg | 237.00 € | ||
| 100mg | 306.00 € | ||
| 500mg | 732.00 € | ||
| 1mL*10mM (DMSO) | 69.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Fluoxetine hydrochloride
CAS:56296-78-7
Fluoxetine HCl (Lilly110140), a selective serotonin reuptake inhibitor (SSRI), is an antidepressant with fewer side …
Formula:
C17H19ClF3NO
Purity:
99.6% - 99.98%
Color and Shape:
White To Off-White Crystalline Solid White To Off-White Powder
Molecular weight:
345.787
Ref: TM-T0450L
| 25mg | 57.00 € | ||
| 50mg | 74.00 € | ||
| 100mg | 93.00 € | ||
| 200mg | 148.00 € | ||
| 500mg | 239.00 € | ||
| 1mL*10mM (DMSO) | 69.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Loxapine succinate
CAS:27833-64-3
Loxapine succinate (Loxapac), a D2DR and D4DR inhibitor, is utilized in schizophrenia.
Formula:
C22H24ClN3O5
Purity:
99.92%
Color and Shape:
White To Of-White Solid
Molecular weight:
445.9
Ref: TM-T1412
| 50mg | 39.00 € | ||
| 100mg | 51.00 € | ||
| 200mg | 82.00 € | ||
| 500mg | 161.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Roxatidine Acetate hydrochloride
CAS:93793-83-0
Roxatidine Acetate hydrochloride (HOE 760) is a specific and competitive histamin H2-receptor antagonist. Roxatidine inhibits …
Formula:
C19H29ClN2O4
Purity:
99.61%
Color and Shape:
Solid
Molecular weight:
384.9
Ref: TM-T0157
| 200mg | 34.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Fenoterol
CAS:13392-18-2
Fenoterol is an agonist of β2-adrenergic receptor It is classed as sympathomimetic beta agonist and …
Formula:
C17H21NO4
Purity:
99.56%
Color and Shape:
Solid
Molecular weight:
303.35
Ref: TM-T8358
| 2mg | 38.00 € | ||
| 5mg | 54.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 158.00 € | ||
| 50mg | 227.00 € | ||
| 1mL*10mM (DMSO) | 71.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Pimethixene
CAS:314-03-4
Pimethixene (Calmixen) blocks 5-HT1A, 2A/B/C, H1, D2/D4.4 & muscarinic M1/M2 receptors; potent with pKis 7.54-10.44.
Formula:
C19H19NS
Purity:
99.1%
Color and Shape:
Solid
Molecular weight:
293.43
Ref: TM-T12489
| 2mg | 34.00 € | ||
| 5mg | 50.00 € | ||
| 10mg | 63.00 € | ||
| 25mg | 103.00 € | ||
| 50mg | 152.00 € | ||
| 100mg | 218.00 € | ||
| 200mg | 326.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
(+)-Dropropizine
CAS:99291-24-4
(+)-Dropropizine can inhibit histamine receptor, anti-allergic, and reduce a cough by modulation of neuropeptides involved …
Formula:
C13H20N2O2
Purity:
99.92%
Color and Shape:
White Or Off White Crystalline Powder
Molecular weight:
236.31
Ref: TM-T0217L
| 1g | 49.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Brompheniramine maleate
CAS:980-71-2
Brompheniramine maleate (Dimotane) is an antagonist against histamine H1 receptors.
Formula:
C16H19BrN2·C4H4O4
Purity:
99.3%
Color and Shape:
Crystal Powder
Molecular weight:
435.31
Ref: TM-T0205
| 25mg | 34.00 € | ||
| 50mg | 43.00 € | ||
| 100mg | 51.00 € | ||
| 200mg | 94.00 € | ||
| 500mg | 144.00 € | ||
| 1mL*10mM (DMSO) | 37.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
2-(1-Piperazinyl)pyrimidine
CAS:20980-22-7
2-(1-Piperazinyl)pyrimidine is used as an anti-anxiety drug.
Formula:
C8H12N4
Purity:
98.86%
Color and Shape:
Liquid - Crystal - Lump
Molecular weight:
164.21
Ref: TM-T1696
| 1g | 38.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Adenosine A1 receptor activator T62
CAS:40312-34-3
Adenosine A1 receptor activator T62 is an allosteric enhancer of adenosine A1 receptor, and it …
Formula:
C15H14ClNOS
Purity:
95.00%
Color and Shape:
Solid
Molecular weight:
291.8
Ref: TM-T14127
| 1mg | 95.00 € | ||
| 5mg | 177.00 € | ||
| 10mg | 263.00 € | ||
| 25mg | 424.00 € | ||
| 50mg | 577.00 € | ||
| 100mg | 781.00 € | ||
| 200mg | 1,035.00 € | ||
| 1mL*10mM (DMSO) | 271.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Zolmitriptan
CAS:139264-17-8
Zolmitriptan targets 5-HT 1B/1D receptors, constricts cranial vessels, inhibits pain signals, and stops pro-inflammatory neuropeptides, …
Formula:
C16H21N3O2
Purity:
98.8% - 99.91%
Color and Shape:
White Or Kind Of White Powder
Molecular weight:
287.36
Ref: TM-T1092
| 10mg | 62.00 € | ||
| 25mg | 102.00 € | ||
| 50mg | 144.00 € | ||
| 100mg | 217.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Naltrexone hydrochloride
CAS:16676-29-2
Naltrexone hydrochloride (Naltrexone HCl) is a synthetic opioid antagonist used in the prevention of relapse …
Formula:
C20H24ClNO4
Purity:
100% - 99%
Color and Shape:
White Crystalline Powder
Molecular weight:
377.862
Ref: TM-T0963
| 100mg | 54.00 € | ||
| 200mg | 68.00 € | ||
| 500mg | 110.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
ZT 52656A hydrochloride
CAS:115730-24-0
ZT 52656A is a selective agonist of kappa opioid, and used for the prevention or …
Formula:
C19H26ClF3N2O
Purity:
98.78%
Color and Shape:
Solid
Molecular weight:
390.87
Ref: TM-T13414
| 1mg | 528.00 € | ||
| 5mg | 1,169.00 € | ||
| 10mg | 1,744.00 € | ||
| 25mg | 2,959.00 € | ||
| 50mg | 3,831.00 € | ||
| 100mg | 5,000.00 € | ||
| 1mL*10mM (DMSO) | 1,253.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
EMPA
CAS:680590-49-2
EMPA is a selective, high-affinity and reversible antagonist of orexin OX2 receptor(human and rat OX2-HEK293 …
Formula:
C23H26N4O4S
Purity:
99.91%
Color and Shape:
Solid
Molecular weight:
454.54
Ref: TM-T11186
| 1mg | 51.00 € | ||
| 5mg | 110.00 € | ||
| 10mg | 172.00 € | ||
| 25mg | 327.00 € | ||
| 50mg | 482.00 € | ||
| 100mg | 688.00 € | ||
| 1mL*10mM (DMSO) | 130.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Ro 10-5824 dihydrochloride
CAS:189744-94-3
Ro 10-5824 dihydrochloride is a selective agonist of dopamine D4 receptor partial, (Ki of 5.2 …
Formula:
C17H22Cl2N4
Purity:
99.95%
Color and Shape:
Solid
Molecular weight:
353.29
Ref: TM-T12761
| 5mg | 34.00 € | ||
| 10mg | 49.00 € | ||
| 25mg | 83.00 € | ||
| 50mg | 121.00 € | ||
| 1mL*10mM (DMSO) | 41.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
PF-5190457
CAS:1334782-79-4
PF-5190457 is an effective and selective ghrelin receptor inverse agonist (pKi: 8.36).
Formula:
C29H32N6OS
Purity:
99.34%
Color and Shape:
Solid
Molecular weight:
512.67
Ref: TM-T16508
| 1mg | 36.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 123.00 € | ||
| 25mg | 269.00 € | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 90.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Hydroxyzine Pamoate
CAS:10246-75-0
Hydroxyzine Pamoate (Bobsule) is a histamine H1 receptor antagonist that is effective in the treatment …
Formula:
C44H43ClN2O8
Purity:
99.71%
Color and Shape:
Solid
Molecular weight:
763.27
Ref: TM-T0053
| 10mg | 35.00 € | ||
| 25mg | 52.00 € | ||
| 50mg | 88.00 € | ||
| 100mg | 131.00 € | ||
| 200mg | 171.00 € | ||
| 500mg | 282.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Clozapine
CAS:5786-21-0
Clozapine (HF 1854) is a tricylic dibenzodiazepine, classified as an atypical antipsychotic agent.
Formula:
C18H19ClN4
Purity:
99.91% - 99.93%
Color and Shape:
Yellow Crystals From Acetone-Petroleum Ether Solid
Molecular weight:
326.82
Ref: TM-T0455
| 1g | 440.00 € | ||
| 10mg | 35.00 € | ||
| 25mg | 52.00 € | ||
| 50mg | 69.00 € | ||
| 100mg | 99.00 € | ||
| 200mg | 167.00 € | ||
| 500mg | 296.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Pheniramine maleate
CAS:132-20-7
Pheniramine maleate (Trimetose), an alkylamine derivative with antihistaminic and vasodilatory properties, binds to histamine H1 …
Formula:
C16H20N2·C4H4O4
Purity:
99.79%
Color and Shape:
Physical Description White Powder With A Faint Amine-Like Odor Melting Point 107°C
Molecular weight:
356.42
Ref: TM-T0370
| 25mg | 36.00 € | ||
| 50mg | 45.00 € | ||
| 100mg | 55.00 € | ||
| 200mg | 65.00 € | ||
| 500mg | 91.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Fluphenazine dihydrochloride
CAS:146-56-5
Fluphenazine dihydrochloride (Prolixin) is an inhibitor of phenothiazine-class D1DR and D2DR. Fluphenazine can be used …
Formula:
C22H28Cl2F3N3OS
Purity:
100%
Color and Shape:
Off-White Solid
Molecular weight:
510.44
Ref: TM-T0068
| 50mg | 55.00 € | ||
| 100mg | 61.00 € | ||
| 200mg | 86.00 € | ||
| 500mg | 115.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
