G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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PF-06882961
CAS:2230198-02-2
PF-06882961 is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.
Formula:
C31H30FN5O4
Purity:
95.1% - 99.54%
Color and Shape:
Solid
Molecular weight:
555.6
Ref: TM-T12431
| 1mg | 50.00 € | ||
| 5mg | 88.00 € | ||
| 10mg | 153.00 € | ||
| 25mg | 195.00 € | ||
| 50mg | 249.00 € | ||
| 100mg | 427.00 € | ||
| 1mL*10mM (DMSO) | 109.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Brompheniramine maleate
CAS:980-71-2
Brompheniramine maleate (Dimotane) is an antagonist against histamine H1 receptors.
Formula:
C16H19BrN2·C4H4O4
Purity:
99.3%
Color and Shape:
Crystal Powder
Molecular weight:
435.31
Ref: TM-T0205
| 25mg | 34.00 € | ||
| 50mg | 43.00 € | ||
| 100mg | 51.00 € | ||
| 200mg | 94.00 € | ||
| 500mg | 144.00 € | ||
| 1mL*10mM (DMSO) | 37.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
ONC206
CAS:1638178-87-6
ONC206, an analogue of the TRAIL inducer ONC201, acts as a selective antagonist of the …
Formula:
C23H22F2N4O
Purity:
99.93%
Color and Shape:
Solid
Molecular weight:
408.44
Ref: TM-T16392
| 2mg | 34.00 € | ||
| 5mg | 49.00 € | ||
| 10mg | 81.00 € | ||
| 25mg | 117.00 € | ||
| 50mg | 203.00 € | ||
| 100mg | 302.00 € | ||
| 1mL*10mM (DMSO) | 50.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Mirabegron
CAS:223673-61-8
Mirabegron (YM178) is a beta-3 adrenergic agonist that is used for treatment of overactive bladder …
Formula:
C21H24N4O2S
Purity:
99.14%
Color and Shape:
Light Yellow To Yellow Solid
Molecular weight:
396.51
Ref: TM-T1671
| 1mg | 35.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 74.00 € | ||
| 10mg | 113.00 € | ||
| 25mg | 189.00 € | ||
| 50mg | 343.00 € | ||
| 100mg | 493.00 € | ||
| 500mg | 1,095.00 € | ||
| 1mL*10mM (DMSO) | 82.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Bithionol
CAS:97-18-7
Bithionol (Actamer), formerly marketed as an active ingredient in various topical drug products, was shown …
Formula:
C12H6Cl4O2S
Purity:
99.27%
Color and Shape:
White Or Grayish-White Crystalline Powder Phenolic Odor (Ntp 1992)
Molecular weight:
356.05
Ref: TM-T0830
| 500mg | 54.00 € | ||
| 1mL*10mM (DMSO) | 60.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Naltrexone hydrochloride
CAS:16676-29-2
Naltrexone hydrochloride (Naltrexone HCl) is a synthetic opioid antagonist used in the prevention of relapse …
Formula:
C20H24ClNO4
Purity:
100% - 99%
Color and Shape:
White Crystalline Powder
Molecular weight:
377.862
Ref: TM-T0963
| 100mg | 54.00 € | ||
| 200mg | 68.00 € | ||
| 500mg | 110.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Silodosin
CAS:160970-54-7
Silodosin (KAD 3213) is an alpha-Adrenergic Blocker. The mechanism of action of silodosin is as …
Formula:
C25H32F3N3O4
Purity:
99.63% - 99.76%
Color and Shape:
Colorless To Pink Solid
Molecular weight:
495.53
Ref: TM-T1504
| 5mg | 38.00 € | ||
| 10mg | 56.00 € | ||
| 25mg | 81.00 € | ||
| 50mg | 88.00 € | ||
| 100mg | 104.00 € | ||
| 200mg | 130.00 € | ||
| 1mL*10mM (DMSO) | 43.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Desvenlafaxine
CAS:93413-62-8
Desvenlafaxine, a venlafaxine metabolite, is an SNRI used as an antidepressant.
Formula:
C16H25NO2
Purity:
99.46% - 99.86%
Color and Shape:
White Crystalline Powder
Molecular weight:
263.38
Ref: TM-T1580
| 50mg | 36.00 € | ||
| 100mg | 47.00 € | ||
| 500mg | 87.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Ro 10-5824 dihydrochloride
CAS:189744-94-3
Ro 10-5824 dihydrochloride is a selective agonist of dopamine D4 receptor partial, (Ki of 5.2 …
Formula:
C17H22Cl2N4
Purity:
99.95%
Color and Shape:
Solid
Molecular weight:
353.29
Ref: TM-T12761
| 5mg | 34.00 € | ||
| 10mg | 49.00 € | ||
| 25mg | 83.00 € | ||
| 50mg | 121.00 € | ||
| 1mL*10mM (DMSO) | 41.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
PF-5190457
CAS:1334782-79-4
PF-5190457 is an effective and selective ghrelin receptor inverse agonist (pKi: 8.36).
Formula:
C29H32N6OS
Purity:
99.34%
Color and Shape:
Solid
Molecular weight:
512.67
Ref: TM-T16508
| 1mg | 36.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 123.00 € | ||
| 25mg | 269.00 € | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 90.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Hyodeoxycholic acid
CAS:83-49-8
Hyodeoxycholic acid (NSC 60672) has been used in trials studying the treatment of Hypercholesterolemia.
Formula:
C24H40O4
Purity:
97.26%
Color and Shape:
Solid
Molecular weight:
392.57
Ref: TM-T2968
| 50mg | 45.00 € | ||
| 100mg | 57.00 € | ||
| 1mL*10mM (DMSO) | 63.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Clozapine
CAS:5786-21-0
Clozapine (HF 1854) is a tricylic dibenzodiazepine, classified as an atypical antipsychotic agent.
Formula:
C18H19ClN4
Purity:
99.91% - 99.93%
Color and Shape:
Yellow Crystals From Acetone-Petroleum Ether Solid
Molecular weight:
326.82
Ref: TM-T0455
| 1g | 440.00 € | ||
| 10mg | 35.00 € | ||
| 25mg | 52.00 € | ||
| 50mg | 69.00 € | ||
| 100mg | 99.00 € | ||
| 200mg | 167.00 € | ||
| 500mg | 296.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Ursodeoxycholic acid
CAS:128-13-2
Ursodeoxycholic acid (UDCA) can be used to dissolve gallstones and reduce cholesterol absorption.
Formula:
C24H40O4
Purity:
99.74% - ≥95%
Color and Shape:
White - Almost White Solid Powder
Molecular weight:
392.57
Ref: TM-T0700
| 1g | 54.00 € | ||
| 5g | 111.00 € | ||
| 1mL*10mM (DMSO) | 65.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Luzindole
CAS:117946-91-5
Luzindole (N-0774) is a selective melatonin receptor antagonist.
Formula:
C19H20N2O
Purity:
98.53%
Color and Shape:
Off-White Amorphous Solid
Molecular weight:
292.37
Ref: TM-T15795
| 1mg | 51.00 € | ||
| 5mg | 143.00 € | ||
| 10mg | 233.00 € | ||
| 25mg | 389.00 € | ||
| 50mg | 577.00 € | ||
| 100mg | 812.00 € | ||
| 500mg | 1,625.00 € | ||
| 1mL*10mM (DMSO) | 155.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Ziprasidone hydrochloride monohydrate
CAS:138982-67-9
Ziprasidone hydrochloride monohydrate (CP 88059) is a united 5-HT (serotonin) and dopamine receptor antagonist which …
Formula:
C21H21ClN4OS·HCl·H2O
Purity:
98% - 99.95%
Color and Shape:
Off-White Powder
Molecular weight:
467.12
Ref: TM-T0031
| 10mg | 55.00 € | ||
| 25mg | 88.00 € | ||
| 50mg | 111.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Bisoprolol hemifumarate
CAS:104344-23-2
Bisoprolol, a selective beta-1 adrenergic receptor antagonist, selectively and competitively binds to and blocks beta-1 …
Formula:
C20H33NO6
Purity:
99% - 99.95%
Color and Shape:
White To Offf-White Powder
Molecular weight:
383.49
Ref: TM-T0143
| 50mg | 51.00 € | ||
| 1mL*10mM (DMSO) | 56.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Ramelteon
CAS:196597-26-9
Ramelteon (TAK-375) is a Melatonin Receptor Agonist. The mechanism of action of ramelteon is as …
Formula:
C16H21NO2
Purity:
97.21% - 99.92%
Color and Shape:
Crystalline Solid
Molecular weight:
259.34
Ref: TM-T1463
| 2mg | 44.00 € | ||
| 5mg | 64.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 133.00 € | ||
| 50mg | 198.00 € | ||
| 100mg | 319.00 € | ||
| 500mg | 503.00 € | ||
| 1mL*10mM (DMSO) | 71.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Tamsulosin hydrochloride
CAS:106463-17-6
Tamsulosin hydrochloride (Flomax hydrochloride) is the hydrochloride salt of tamsulosin, a sulfonamide derivative with α1 …
Formula:
C20H29ClN2O5S
Purity:
100% - 99.95%
Color and Shape:
White To Off-White Solid
Molecular weight:
444.97
Ref: TM-T0210
| 10mg | 35.00 € | ||
| 25mg | 52.00 € | ||
| 50mg | 73.00 € | ||
| 100mg | 95.00 € | ||
| 1mL*10mM (DMSO) | 46.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Talipexole dihydrochloride
CAS:36085-73-1
Talipexole dihydrochloride (Domnin) is a dopamine D2 receptor agonist, α2-adrenoceptor agonist, and 5-HT3 receptor antagonist …
Formula:
C10H17Cl2N3S
Purity:
98.64%
Color and Shape:
Light Yellow Solid
Molecular weight:
282.23
Ref: TM-T14490
| 2mg | 38.00 € | ||
| 5mg | 55.00 € | ||
| 10mg | 89.00 € | ||
| 25mg | 151.00 € | ||
| 50mg | 259.00 € | ||
| 100mg | 417.00 € | ||
| 200mg | 602.00 € | ||
| 500mg | 930.00 € | ||
| 1mL*10mM (DMSO) | 63.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Benserazide hydrochloride
CAS:14919-77-8
Benserazide hydrochloride (Ro 4-4602) is a peripherally-acting L-amino acid decarboxylase (AAAD) or DOPA decarboxylase inhibitor.
Formula:
C10H15N3O5·HCl
Purity:
98.63% - 99.74%
Color and Shape:
White Crystalline Solid
Molecular weight:
293.7
Ref: TM-T1517
| 1g | 66.00 € | ||
| 500mg | 50.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
