Benzimidazole and Imidazole Derivatives
Benzimidazole is a compound consisting of a benzene ring fused to an imidazole ring, a five-membered structure containing two nitrogen atoms. Benzimidazole derivatives, such as albendazole, are known for their antiparasitic and antifungal activity, used in the treatment of parasitic infections and certain parasitic diseases in animals and humans. Imidazole, on the other hand, is a five-membered structure with two nitrogen atoms found in various biologically active compounds. Imidazole derivatives, such as metronidazole, have antimicrobial and antiparasitic properties. These compounds are also used in the pharmaceutical industry for treating bacterial infections, parasitic diseases, and some fungal infections, as well as in organic chemistry as catalysts.
At CymitQuimica, we offer high-purity benzimidazoles and imidazoles for research in medicinal chemistry, pharmacology, and biotechnology.
Found 10354 products of "Benzimidazole and Imidazole Derivatives"
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Imidapril
CAS:<p>Imidapril: oral ACE & MMP-9 inhibitor, lowers blood pressure, useful in hypertension, diabetic nephropathy, heart failure.</p>Formula:C20H27N3O6Color and Shape:SolidMolecular weight:405.44Ilaprazole
CAS:<p>Ilaprazole (IY-81149) is a proton pump inhibitor used in the treatment of dyspepsia gastroesophageal reflux disease (GORD/GERD) and duodenal ulcer.</p>Formula:C19H18N4O2SPurity:99.91%Color and Shape:SolidMolecular weight:366.44Galantamine EP Impurity E-13C,d3 (N-Desmethyl Galanthamine-13C,d3)
Formula:C1513CH16D3NO3Molecular weight:277.34(R,R)-Galantamine EP Impurity A L-DPTTA Salt ((+)-Narwedine L-DPTTA Salt, (+)-Galanthaminone L-DPTTA Salt)
CAS:Formula:C17H21NO3·C20H18O8Molecular weight:287.36 386.36Efinaconazole
CAS:<p>Efinaconazole (KP-103)(KP-103) is an Azole Antifungal currently under development as a topical treatment for onychomycosis.</p>Formula:C18H22F2N4OPurity:97.34% - 98%Color and Shape:SolidMolecular weight:348.39Varenicline dihydrochloride
CAS:<p>Varenicline dihydrochloride is a Selective α4β2 nicotinic acetylcholine receptor partial agonist.</p>Formula:C13H15Cl2N3Purity:99.88% - 99.97%Color and Shape:SolidMolecular weight:284.18Donepezil
CAS:<p>Donepezil (Aricept) is a piperidine-based, potent, specific, and reversible inhibitor of acetylcholinesterase (AChE).</p>Formula:C24H29NO3Purity:99.69%Color and Shape:White Or Almost White Crystal PowderMolecular weight:379.49Sertaconazole nitrate
CAS:<p>Sertaconazole nitrate, a broad-spectrum topical antifungal, treats skin and mucosal infections.</p>Formula:C20H15Cl3N2OS·HNO3Purity:98.66% - 99.65%Color and Shape:SolidMolecular weight:500.78Acotiamide
CAS:<p>Acotiamide, an oral AChE inhibitor (IC50: 1.79μM), improves gastric motility, targeting functional dyspepsia.</p>Formula:C21H30N4O5SColor and Shape:SolidMolecular weight:450.55Propiverine
CAS:<p>Propiverine reduces muscle spasms by limiting calcium influx, targeting bladder smooth muscles, aiding OAB research.</p>Formula:C23H29NO3Color and Shape:SolidMolecular weight:367.48Oxiconazole
CAS:<p>Oxiconazole is a broad-spectrum imidazole antifungal, inhibiting ergosterol biosynthesi by disrupting cytochrome P450 enzymes (lanosterol 14- α demethylase).</p>Formula:C18H13Cl4N3OPurity:99.99%Color and Shape:SolidMolecular weight:429.13Cyclopentolate Hydrochloride
CAS:<p>Cyclopentolate Hydrochloride is a muscarinic acetylcholine receptors antagonist with Kis of 1.62, 27.5, and 2.63 nM for M1, M2, and M3 receptors, respectively.</p>Formula:C17H26ClNO3Purity:99.91%Color and Shape:SolidMolecular weight:327.85Varenicline Tartrate
CAS:<p>Varenicline Tartrate (CP 526555-18) is a benzazepine derivative that functions as an ALPHA4/BETA2 NICOTINIC RECEPTOR partial agonist.</p>Formula:C13H13N3·C4H6O6Purity:98.23% - 98.32%Color and Shape:Tan SolidMolecular weight:361.35Benznidazol
CAS:<p>Benznidazol (Benznidazole)e has an antiprotozoal activity by interfering with parasite protein biosynthesis, influencing cytokines production and stimulating</p>Formula:C12H12N4O3Purity:99.53% - >99.99%Color and Shape:SolidMolecular weight:260.25(R)-Lansoprazole
CAS:<p>(R)-Lansoprazole (T 168390) is the R-isomer of lansoprazole and a substituted benzimidazole prodrug with selective and irreversible proton pump inhibitor</p>Formula:C16H14F3N3O2SPurity:98.09% - 98.99%Color and Shape:Brown SolidMolecular weight:369.36Fesoterodine
CAS:<p>Fesoterodine is an oral mAChR blocker (pKi: 7.3-8.0) for M1-M5, used to treat OAB.</p>Formula:C26H37NO3Purity:97.1%Color and Shape:SolidMolecular weight:411.58Fosravuconazole L-lysine ethanolate
CAS:<p>Fosravuconazole L-lysine ethanolate, a prodrug for ravuconazole, treats onychomycosis in Japan.</p>Formula:C31H40F2N7O8PSPurity:99.43%Color and Shape:SolidMolecular weight:739.7Eberconazole Nitrate
CAS:<p>Eberconazole Nitrate (Ebernet) is an azole antifungal agent and broad-spectrum imidazole derivative.</p>Formula:C18H15Cl2N3O3Purity:99.53%Color and Shape:SolidMolecular weight:392.23Propiverine hydrochloride
CAS:<p>Propiverine is a widely used antimuscarinic drug with a mixed mode of action in the treatment of symptoms associated with overactive bladder (OAB).</p>Formula:C23H30ClNO3Purity:99.93%Color and Shape:White Crystalling PowerMolecular weight:403.94Sulfamoxole
CAS:<p>Sulfamoxole (Sulfamoxol) is an antibacterial belonging to sulfonamide.</p>Formula:C11H13N3O3SPurity:97.8% - 99.41%Color and Shape:SolidMolecular weight:267.3L-Hyoscyamine sulfate
CAS:<p>L-Hyoscyamine sulfate (Levsin Sulfate) is a belladonna alkaloid derivative and the levorotatory form of racemic atropine which exhibits anticholinergic effect.</p>Formula:C34H48N2O10SPurity:96.7% - 99.61%Color and Shape:Long Orthorhombic Prisms From Acetone SolidMolecular weight:676.8Isoconazole nitrate
CAS:<p>Isoconazole nitrate (Fazol) (Travogen) is an azole antifungal reagent.</p>Formula:C18H14Cl4N2O·HNO3Purity:99.47%Color and Shape:White Crystals Or Crystalline PowderMolecular weight:479.14Aclidinium bromide
CAS:<p>Aclidinium bromide (LAS-W 330) is a synthetic anticholinergic agent that is used as an inhalant for treatment of acute bronchospasm due to chronic bronchitis.</p>Formula:C26H30NO4S2·BrPurity:99.53% - 99.69%Color and Shape:SolidMolecular weight:564.55Ipratropium Bromide
CAS:<p>Ipratropium Bromide (Sch 1000) is an antagonist of muscarinic receptors and is used in COPD and asthma studies.</p>Formula:C20H30BrNO3Purity:99.92%Color and Shape:SolidMolecular weight:412.37Vonoprazan
CAS:<p>Vonoprazan (TAK-438 (free base)) is an orally active potassium-competitive acid blocker.Vonoprazan can be used for the treatment of gastroduodenal ulcer and</p>Formula:C17H16FN3O2SPurity:99.87% - 99.92%Color and Shape:SolidMolecular weight:345.39Tetrazole
CAS:<p>Tetrazole (1H-TETRAZOLE) is the bioisoster of carboxylic acid, possess considerable antibacterial property.</p>Formula:CH2N4Purity:99.66%Color and Shape:White Crystalline SolidMolecular weight:70.053-Amino-1H-indazole-5-carboxylic acid
CAS:Formula:C8H7N3O2Purity:95.0%Color and Shape:SolidMolecular weight:177.163Thiabendazole-d4 (Major)
CAS:Controlled ProductFormula:C10D4H3N3SColor and Shape:Off WhiteMolecular weight:205.274-{[(1-methyl-1H-benzimidazol-2-yl)methyl]amino}benzoic acid
CAS:Purity:95.0%Molecular weight:281.31500244140625Midazolam
CAS:Controlled Product<p>Applications Anesthetic; anticonvulsant; sedative; hypnotic. Positive allosteric modulator of the GABAA receptor. Neuroprotective & Neuroresearch products.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Dundee, J. W., et al.: Drugs, 28, 519 (1984), Lahat, E., et al.: Br. Med. J., 321, 83 (2000)<br></p>Formula:C18H13ClFN3Color and Shape:White To Off-WhiteMolecular weight:325.77a-(Chloromethyl)-2,4-dichlorobenzyl Alcohol
CAS:Controlled Product<p>Impurity Isoconazole Impurity 6<br>Applications α-(Chloromethyl)-2,4-dichlorobenzyl alcohol is used in the synthesis of monocyclic nitroimidazole analogs of econazole. Isoconazole Impurity 6.<br>References Lee, S., et al.: Bioorg. Med. Chem. Lett., 21, 1515 (2011);<br></p>Formula:C8H7Cl3OColor and Shape:NeatMolecular weight:225.5((R)-1-phenyl-3,4-dihydroisoquinolin-2(1H)-yl)((S)-1-phenyl-3,4-dihydroisoquinolin-2(1H)-yl)methanone
CAS:Controlled Product<p>Impurity Solifenacin EP Impurity D<br>Applications ((R)-1-phenyl-3,4-dihydroisoquinolin-2(1H)-yl)((S)-1-phenyl-3,4-dihydroisoquinolin-2(1H)-yl)methanone is a possible impurity of solifenacin (S676700) which is a muscarinic M3 receptor antagoinst. Solifenacin is used in treatment of urinary incontinence.<br>References Ikeda K., et al.: Arch. Pharmacol., 366, 97, (2002); Chapple, C.R., et al.: Br. J. Urol., 93, 303 (2004); Ohtake, A., et al.: Eur. J. Pharmacol., 492, 243 (2004); Brunton, S., et al.: Curr. Med. Res. Opin., 21, 71 (2005); Habb, F., et al.: Eur. Urol. 47, 376 (2005); Payne, C.K., et al.: Drugs, 66, 175 (2006)<br></p>Formula:C31H28N2OColor and Shape:NeatMolecular weight:444.57(R)-4-Isopropyl-5,5-diphenyloxazolidin-2-one
CAS:Purity:95.0%Color and Shape:SolidMolecular weight:281.3550109863281Metronidazole-d4
CAS:Controlled Product<p>Applications Metronidazole-d4 is a labelled analog of Metronidazole (M338880). Used as an antibacterial in the treatment of rosacea. Antiprotozoal (trichomonas). A potential human carcinogen.<br>References Carballo, M., et al.: J. App. Toxicol., 29, 248 (2009), Leitsch, D., et al.: Mol. Microbiol., 72, 518 (2009), Sanderson, H., et al.: Toxicol. Lett., 187, 84 (2009),<br></p>Formula:C62H4H5N3O3Color and Shape:Light YellowMolecular weight:175.18N-(2-CHLORO-5-METHOXYPYRIMIDIN-4-YL)-1H-INDAZOL-6-AMINE
CAS:Purity:95.0%Molecular weight:275.70001220703125Mebendazole-d8
CAS:Controlled Product<p>Applications Labelled Mebendazole (M200500). Anthelmintic (Nematodes).<br>References Al-Badr, A.A., et al.: Anal. Profiles Drug Subs., 16, 291 (1987)<br></p>Formula:C162H3H10N3O3Color and Shape:NeatMolecular weight:298.31Omeprazole
CAS:Controlled Product<p>Applications Omeprazole covalently binds to proton pump. It inhibits gastric secretion. Used as an anttiulcerative.<br>References Muller, P., et al.: Arzneimittel-Forsch., 33, 1685 (1983), Wallmark, B., et al.: Biochim. Biophys. Acta., 778, 549 (1984), Morii, M., et al.: J. Biol. chem., 268, 21553 (1993), Ritter, M., et al.: Br. J. Pharmacol., 124, 627 (1998)<br></p>Formula:C17H19N3O3SColor and Shape:White To Light BrownMolecular weight:345.42Benzhydrol-d5
CAS:Controlled Product<p>Applications Intermediate in the preparation of labelled Modafinil (M482500).<br>References Kumar, C., et al.: Eur. J. Med. Chem., 44, 1223 (2009),<br></p>Formula:C13D5H7OColor and Shape:NeatMolecular weight:189.26Methyl 2-(1H-imidazol-1-yl)acetate
CAS:Formula:C6H8N2O2Purity:95.0%Color and Shape:SolidMolecular weight:140.142cis-[2-(2,4-Dichlorophenyl)-2-(1H-1,2,4-triazol-4-yl-methyl)-1,3-dioxolan-4-yl]methyl Methanesulfonate
CAS:<p>Impurity Itraconazole Impurity 16<br>Applications cis-[2-(2,4-Dichlorophenyl)-2-(1H-1,2,4-triazol-4-yl-methyl)-1,3-dioxolan-4-yl]methyl Methanesulfonate (Itraconazole Impurity 16) is an impurity in the synthesis of Itraconazole (I937500), an orally active antimycotic structurally related to Ketoconazole. Antifungal.<br>References Espinel-Ingroff, A., et al.: Antimicrob. Agents Chemother., 26, 5 (1984), Heykants, J., et al.: Mycoses, 32, Suppl 1, 67 (1989);<br></p>Formula:C14H15Cl2N3O5SColor and Shape:NeatMolecular weight:408.257Tebuconazole-d9
CAS:Controlled Product<p>Applications Isotope labelled Tebuconazole (T013000), which is an ergosterol biosynthesis inhibitor present in most pesticide formulations (1,2). Various uptake is observed in plants (3). Drinking water Contaminant Candidate List 3 - CCL 3 as per United States Environmental Protection Agency (EPA). Environmental contaminants; Food contaminants.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References 1. Grimalt S. et al.: Anal Bioanal Chem. 2015 Apr;407(11):3083-91 2. Gent, D. et al.: Plant Dis. 2003 May:87(5) p591-5973. Wang, C. et al.: Pest. Biochem. Physiol. 2007 Jan:87(1) p1-8<br></p>Formula:C16H13D9ClN3OColor and Shape:White To Light YellowMolecular weight:316.87N-(2-Hydroxyethyl)-5-methyl-1,2,4-oxadiazole-3-carboxamide
CAS:<p>Applications N-(2-Hydroxyethyl)-5-methyl-1,2,4-oxadiazole-3-carboxamide is a photolysis product of Metronidazole (M338880), an antibiotic.<br>References Moore, Douglas E., et al.: Radiation Phy. and Chem., 36(4), 547-50 (1990)<br></p>Formula:C6H9N3O3Color and Shape:NeatMolecular weight:171.154(S)-4-Isopropyl-5,5-diphenyloxazolidin-2-one
CAS:Purity:95.0%Color and Shape:SolidMolecular weight:281.35501098632811-[(furan-2-yl)methyl]-5-phenyl-2,3-dihydro-1H-imidazole-2-thione
Molecular weight:256.32000732421875Carbamazepine-d2,15N
CAS:Controlled ProductFormula:C15H10D2N15NOColor and Shape:Off White SolidMolecular weight:239.27Itraconazole Mono N-Oxide
Controlled ProductFormula:C35H38Cl2N8O5Color and Shape:NeatMolecular weight:721.63N-Ethyl-N-(4-picolyl)atropamide (>85%)
CAS:<p>Stability Light Sensitive<br>Applications N-Ethyl-N-(4-picolyl)atropamide is a major impurity of Tropicamide (T892650), a medication used to dilate the pupil.<br>References Stefanowicz, Zdzislawa, et al.: J. of Pharma. and Biomed. Analy., 49(2), 214-220 (2009)<br></p>Formula:C17H18N2OPurity:>85%Color and Shape:NeatMolecular weight:266.34O-Hydroxyethyl Metronidazole
CAS:Controlled Product<p>Applications O-Hydroxyethyl Metronidazole is the hydroxy ethyl analogue and impurity of the antiprotozoal agent Metronidazole (M338880). O-Hydroxyethyl Metronidazole as well as other 1-substituted-2-methyl-5-nitroimidazoles showed potential antitrichomonal activity.<br>References Kajfez, F. et al.: J. Med. Chem., 11, 167 (1968);<br></p>Formula:C8H13N3O4Color and Shape:Yellowish SolidMolecular weight:215.213a,4,5,6-Tetrahydro Midazolam
CAS:Controlled Product<p>Applications 3a,4,5,6-Tetrahydro Midazolam is an impurity of Midazolam (M343000), a drug used for the treatment of acute seizures and is also known to exhibit activities as an anticonvulsant, sedative, and hypnotic.<br>References Dundee, J. W., et al.: Drugs, 28, 519 (1984); Lahat, E., et al.: Br. Med. J., 321, 83 (2000); Sati, B., et al.: Acta Pharm., 63, 385 (2013);<br></p>Formula:C18H17ClFN3Color and Shape:NeatMolecular weight:329.801-(4-(3-Amino-1H-indazol-4-yl)phenyl)-3-(2-fluoro-5-methylphenyl)urea
CAS:Purity:95.0%Color and Shape:SolidMolecular weight:375.40701293945314-Cyanobenzyl Bromide
CAS:Controlled Product<p>Applications A benzyl halide as postemergence herbicides.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Singer, G.M., et al.: J. Med. Chem., 26, 309 (1983),<br></p>Formula:C8H6BrNColor and Shape:NeatMolecular weight:196.04
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