Quinazoline and Quinoline Derivatives
Quinazolines and quinolines are nitrogen-containing heterocyclic compounds with aromatic structures that play a key role in the synthesis of drugs with anticancer, antimicrobial, and anti-inflammatory activity. Their derivatives feature structural modifications that optimise bioavailability and selectivity, enabling the development of new active ingredients for various therapeutic applications. These compounds are used in the manufacture of APIs for the treatment of cancer, infections, neurodegenerative diseases, and cardiovascular conditions. Additionally, quinazoline and quinoline derivatives are essential in the research of enzyme inhibitors and the design of innovative bioactive molecules.
At CymitQuimica, we offer high-purity quinazoline and quinoline derivatives for applications in chemical synthesis, pharmaceutical development, and biotechnology.
Found 65624 products of "Quinazoline and Quinoline Derivatives"
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3-Methoxy-6-(trifluoromethyl)picolinic acid
CAS:Formula:C8H6F3NO3Purity:98%Color and Shape:SolidMolecular weight:221.135(4-BROMO-1,3-DIMETHYL-1H-PYRAZOL-5-YL)METHANOL
CAS:Formula:C6H9BrN2OPurity:95.0%Molecular weight:205.0556-ethyl-3-(morpholin-4-ylcarbonyl)-4,5,6,7-tetrahydro-1-benzothiophen-2-amine
CAS:Formula:C15H22N2O2SPurity:95.0%Molecular weight:294.415-m-Tolyl-2H-pyrazol-3-ylamine
CAS:Formula:C10H11N3Purity:95+%Color and Shape:SolidMolecular weight:173.219Abiraterone acetate
CAS:Formula:C26H33NO2Purity:95.0%Color and Shape:White to off-white powderMolecular weight:391.5552-(4-Methoxyphenyl)pyridine
CAS:Formula:C12H11NOPurity:99%(GC-MS);RGColor and Shape:No data available.Molecular weight:185.2262-[4-(4-Benzyl-piperazin-1-yl)-butyl]-4-methyl-2H-[1,2,4]triazine-3,5-dione
Formula:C19H27N5O2Purity:95.0%Molecular weight:357.4585-Bromopyridine-2,3-dicarboxylic acid
CAS:Formula:C7H4BrNO4Purity:97%Color and Shape:SolidMolecular weight:246.0164-Bromo-1-ethyl-3-methyl-1H-pyrazole
CAS:Formula:C6H9BrN2Purity:95%Color and Shape:LiquidMolecular weight:189.0563,5-Dimethyl-1-phenyl-1H-pyrazole-4-sulfonylchloride
CAS:Formula:C11H11ClN2O2SPurity:95%Color and Shape:SolidMolecular weight:270.73(2-AMINOTHIOPHEN-3-YL)(4-BROMOPHENYL)METHANONE
CAS:Formula:C11H8BrNOSPurity:95.0%Molecular weight:282.165-Chloro-4-methoxy-thiophene-3-carbonyl chloride
CAS:Formula:C6H4Cl2O2SPurity:95.0%Molecular weight:211.063-(4-Bromo-phenylsulfanyl)-5-trifluoromethyl-pyridine-2-carboxylic acid
Formula:C13H7BrF3NO2SPurity:95.0%Molecular weight:378.165-(3-Methoxy-phenyl)-2H-pyrazol-3-ylamine
CAS:Formula:C10H11N3OPurity:≥98%Color and Shape:SolidMolecular weight:189.218{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}amine dihydrochloride
CAS:Formula:C11H15Cl2N3OPurity:95.0%Molecular weight:276.161-(2-(Trifluoromethyl)pyridin-4-yl)ethanamine dihydrochloride
CAS:Formula:C8H11Cl2F3N2Purity:95.0%Molecular weight:263.093-(2-thienyl)-1H-1,2,4-triazol-5-amine
CAS:Formula:C6H6N4SPurity:95.0%Color and Shape:White powderMolecular weight:166.2N-Methyl(3-(pyridin-4-yl)phenyl)methanamine
CAS:Formula:C13H14N2Purity:97%Color and Shape:LiquidMolecular weight:198.269Methyl 6-oxo-1-phenyl-1,6-dihydropyridine-3-carboxylate
CAS:Formula:C13H11NO3Purity:95.0%Molecular weight:229.2353-Fluoro-5-nitropyridin-2-ol
CAS:Formula:C5H3FN2O3Purity:98%Color and Shape:SolidMolecular weight:158.0886-Bromoquinoline-3-carbaldehyde
CAS:Formula:C10H6BrNOPurity:97%Color and Shape:SolidMolecular weight:236.068Ethyl 4-hydroxy-6-(trifluoromethyl)nicotinate
CAS:Formula:C9H8F3NO3Purity:95%Molecular weight:235.1621-(Pyridin-3-yl)cyclopropanamine dihydrochloride
CAS:Formula:C8H12Cl2N2Purity:95%Color and Shape:SolidMolecular weight:207.15-(5-Chloro-thiophen-2-yl)-[1,3,4]thiadiazol-2-ylamine
CAS:Formula:C6H4ClN3S2Purity:97.0%Molecular weight:217.69Methyl 3-amino-6-bromopicolinate
CAS:Formula:C7H7BrN2O2Purity:95%Color and Shape:SolidMolecular weight:231.0495-BROMOQUINOLINE-8-CARBALDEHYDE
CAS:Formula:C10H6BrNOPurity:97%Color and Shape:SolidMolecular weight:236.0683-Carbamoyl-1-((2R,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)tetrahydrofuran-2-yl)pyridin-1-ium
CAS:Purity:95%Color and Shape:Low Melting SolidMolecular weight:255.24899293-tert-butyl-1-(2-nitrophenyl)-1H-pyrazol-5-amine
CAS:Formula:C13H16N4O2Purity:95.0%Molecular weight:260.2974-(2-Methoxyethyl)-1-methyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazole
CAS:Purity:97%Molecular weight:266.1499939tert-Butyl 2-(pyridin-2-ylmethylene)hydrazinecarboxylate
CAS:Formula:C11H15N3O2Purity:95.0%Molecular weight:221.261-(2-Chloro-4-fluoro-benzyl)-3-isothiocyanato-1H-pyrazole
CAS:Formula:C11H7ClFN3SMolecular weight:267.71Ethyl 6-iodo-8-methyl-4-oxo-1,4-dihydroquinoline-3-carboxylate
CAS:Purity:95%Molecular weight:357.14700323-Chloro-2-hydroxypyridine-5-carboxylic acid
CAS:Formula:C6H4ClNO3Purity:95%Color and Shape:Solid, White to slightly pale yellow powderMolecular weight:173.55(S)-2-((2-oxo-3-(4-(3-oxomorpholino)phenyl)oxazolidin-5-yl)methyl)isoindoline-1,3-dione
CAS:Purity:97%Molecular weight:421.40899668-CHLOROISOQUINOLIN-3-AMINE
CAS:Formula:C9H7ClN2Purity:98%Color and Shape:SolidMolecular weight:178.624-Bromo-2-(pyridin-2-ylmethyl)pyridazin-3(2H)-one
Formula:C10H8BrN3OPurity:>95%Molecular weight:266.098Betrixaban
CAS:<p>Betrixaban is a non-VKORC1 anticoagulant targeting factor Xa, with low hERG affinity, used to prevent VTE in adults with mobility issues.</p>Formula:C23H22ClN5O3Purity:99.33%Color and Shape:SolidMolecular weight:451.91Ticlopidine
CAS:<p>Ticlopidine (PCR 5332) is an antiplatelet drug in the thienopyridine family which is an adenosine diphosphate (ADP) receptor inhibitor.</p>Formula:C14H14ClNSPurity:99.67%Color and Shape:SolidMolecular weight:263.79Meclofenamic acid
CAS:<p>Meclofenamic acid: non-selective gap-junction blocker, FTO inhibitor, anti-inflammatory.</p>Formula:C14H11Cl2NO2Purity:98%Color and Shape:SolidMolecular weight:296.15Prothioconazole
CAS:<p>Prothioconazole (Proline 480 SC Fungicide) is a chiral triazole fungicide in plant pathogen control.</p>Formula:C14H15Cl2N3OSPurity:99.77%Color and Shape:Un3077 9/Pg 3Molecular weight:344.26Pardoprunox
CAS:<p>Pardoprunox (SLV-308) is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties.</p>Formula:C12H15N3O2Purity:98%Color and Shape:SolidMolecular weight:233.27(3S,4S)-Tofacitinib
CAS:<p>(3S,4S)-Tofacitinib, a less active enantiomer of tofacitinib, is a Janus kinases inhibitor.</p>Formula:C16H20N6OPurity:98%Color and Shape:SolidMolecular weight:312.37Itopride free base
CAS:<p>Itopride HCl combats dyspepsia and GERD, inhibiting AChE and blocking D2 receptors.</p>Formula:C20H26N2O4Color and Shape:WhiteMolecular weight:358.43Mephenoxalone
CAS:<p>Mephenoxalone is a muscle relaxant and mild anxiolytic. It inhibits neuron transmission and relaxing skeletal muscles by inhibiting the reflex arc.</p>Formula:C11H13NO4Purity:98%Color and Shape:SolidMolecular weight:223.23Procymidone
CAS:<p>Procymidone is a broad-spectrum fungicide that inhibits fungal glycerol triester synthesis, thereby disrupting hyphal growth. androgen receptor (AR) antagonist</p>Formula:C13H11Cl2NO2Purity:99.86%Color and Shape:Colorless SolidMolecular weight:284.14Esmolol hydrochloride
CAS:Esmolol is a cardioselective beta-blocker used in parenteral forms in the treatment of arrhythmias and severe hypertension.Formula:C16H25NO4·HClPurity:98.72% - 99.48%Color and Shape:White SolidMolecular weight:331.15Icotinib
CAS:<p>Icotinib (Conmana) is an orally available quinazoline-based inhibitor of epidermal growth factor receptor (EGFR), with potential antineoplastic activity.</p>Formula:C22H21N3O4Purity:99.76% - 99.94%Color and Shape:SolidMolecular weight:391.42Penbutolol sulfate
CAS:<p>Penbutolol sulfate ((-)-Terbuclomine) is able to bind to both β2-adrenergic receptor and β1-adrenergic receptor, thus making it a non-selective β blocker.</p>Formula:C18H29NO2H2O4SPurity:98.55%Color and Shape:SolidMolecular weight:340.47Diphenidol
CAS:<p>Diphenidol, a muscarinic antagonist, is employed as an antivertigo and antiemetic agent.</p>Formula:C21H27NOColor and Shape:Needles From Petroleum Ether SolidMolecular weight:309.45Amfenac
CAS:<p>Amfenac promotes apoptosis in ARPE-19 cell culture.</p>Formula:C15H13NO3Color and Shape:SolidMolecular weight:255.271H-1-Ethyl-d5 Candesartan
CAS:Controlled Product<p>Applications Labelled Candesartan (C175575) impurity.<br></p>Formula:C26H19D5N6O3Color and Shape:Off-White To Light YellowMolecular weight:473.54N’-[2-[2,4-(Dimethylphenyl)thio]phenyl] Vortioxetine
Controlled Product<p>Applications N’-[2-[2,4-Dimethylphenyl)thio]phenyl] Vortioxetine is an impurity of Vortioxetine (V766000, HBr salt) which is a multimodal serotonergic agent, inhibits 5-HT1A, 5-HT1B, 5-HT3A, 5-HT7 receptor and SERT.<br>References Bang-Andersen, B., et al.: J. Med. Chem., 54, 3206 (2011); Mørk, A., et al.: J. Pharmacol. Exp. Ther., 340, 666 (2012); Mørk, A., et al.: Pharmacol. Biochem. Behav. 105C, 41 (2013)<br></p>Formula:C32H34N2S2Color and Shape:NeatMolecular weight:510.762-Amino-5-methyl-3-thiophenecarbonitrile
CAS:Controlled Product<p>Applications An impurity generated in the preparation of Olanzapine (O253750).<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Rao, R. et al.: J. Sep. Sci., 31, 107 (2008); Cui, D. et al.: Analyst, 136, 3149 (2011);<br></p>Formula:C6H6N2SColor and Shape:NeatMolecular weight:138.19δ-Valerolactam
CAS:Controlled Product<p>Applications δ-Valerolactam is a useful synthetic intermediate. It is an intermediate used to synthesize Cenicriviroc (C256550), an experimental drug candidate for the treatment of HIV infection. It is also a starting material for a new route to hexahydrojulolidines, using intramolecular 1,4-cycloaddition.<br>References Potts, K., et al. J. Org. Chem., 58, 5040 (1993); Klibanov, O., et al.: Curr. Opinion Invest. Drugs, 11, 940 (2010);<br></p>Formula:C5H9NOColor and Shape:NeatMolecular weight:99.131rac Toltrazuril Sulfoxide
CAS:<p>Applications Toltrazuril metabolite.<br>References Benoit, E., et al.: Biochem. Pharmacol., 46, 2337 (1993), Martinez-Villalba, A., et al.: Anal. Bioanal. Chem., 397, 2893 (2010),<br></p>Formula:C18H14F3N3O5SColor and Shape:Off-WhiteMolecular weight:441.381-(6-Methylpyridin-3-yl)-2-((4-(2-(6-methylpyridin-3-yl)-2-oxoethyl)phenyl)sulfonyl)ethanone
CAS:Controlled ProductFormula:C22H20N2O4SColor and Shape:NeatMolecular weight:408.47N-(4-Methoxybenzyl)-4-chloro-2-(trifluoroacetyl)aniline
CAS:Controlled ProductFormula:C16H13ClF3NO2Color and Shape:NeatMolecular weight:343.732S,3S,5S-5-Amino-2-[N-[[(5-thiozolyl)methoxy]carbonyl]amino]-1,6-diphenyl-3-hydroxyhexane
CAS:Controlled ProductFormula:C23H27N3O3SColor and Shape:NeatMolecular weight:425.54XL518
CAS:Controlled Product<p>Applications A potent, selective, orally bioavailable inhibitor of MEK1, a component of the RAS/RAF/MEK/ERK pathway. It inhibits proliferation and stimulates apoptosis in a variety of human tumor cell lines. In preclinical xenograft models, oral administration of XL518 results in sustained inhibition of pERK in tumor tissue, but not brain tissue, leading to tumor growth inhibition and regression at well tolerated doses.<br>References Rosen, L.S. et al.: J. Clin. Oncol., 26, 14585 (2008);<br></p>Formula:C21H21F3IN3O2Color and Shape:White To Off-WhiteMolecular weight:531.31rac Dropropizine
CAS:Controlled Product<p>Applications Dropropizine is a cough suppressant and central sedative therapeutic agent.<br>References Bakken, G., et al.: J. Med. Chem., 43, 4534 (2000), Salunkhe, M., et al.: Enz. Microb. Technol., 28, 333 (2001), Atul, B., et al.: J. Pharm. Sci., 91, 2067 (2002),<br></p>Formula:C13H20N2O2Color and Shape:WhiteMolecular weight:236.31(7-(4-{4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butoxy}butoxy)-3,4-dihydroquinolin-2(1H)-one)
CAS:Controlled Product<p>Impurity Aripiprazole USP Related Compound H<br>Applications (7-(4-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}butoxy)-3,4-dihydroquinolin-2(1H)-one) is an impurity of Aripiprazole (A771000), a selective dopamine D2-receptor antagonist with dopamine autoreceptor agonist activity. Aripiprazole USP Related Compound H.<br>References Zeidan, T.A., et al.: Crystal. Growth. Design., 13, 2036 (2013); Nagasaka, Y., et al.: Biopharma. Drug. Dispo., 33, 304 (2012); Chen, X., et al.: J. Med. Chem., 55, 7141 (2012);<br></p>Formula:C27H35Cl2N3O3Color and Shape:WhiteMolecular weight:520.494-Desisopropyl-4-ethyl Nateglinide
CAS:Controlled Product<p>Applications D-phenylanaline derivative and an analog Nateglinide (N379375) with similar hypoglycemic activity.<br>References Shinkai, H. et al.: J. Med. Chem., 32, 1436 (1989);<br></p>Formula:C18H25NO3Color and Shape:NeatMolecular weight:303.40
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