Quinazoline and Quinoline Derivatives
Quinazolines and quinolines are nitrogen-containing heterocyclic compounds with aromatic structures that play a key role in the synthesis of drugs with anticancer, antimicrobial, and anti-inflammatory activity. Their derivatives feature structural modifications that optimise bioavailability and selectivity, enabling the development of new active ingredients for various therapeutic applications. These compounds are used in the manufacture of APIs for the treatment of cancer, infections, neurodegenerative diseases, and cardiovascular conditions. Additionally, quinazoline and quinoline derivatives are essential in the research of enzyme inhibitors and the design of innovative bioactive molecules.
At CymitQuimica, we offer high-purity quinazoline and quinoline derivatives for applications in chemical synthesis, pharmaceutical development, and biotechnology.
Found 65497 products of "Quinazoline and Quinoline Derivatives"
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8-methyl-4-(pyridine-4-carbonyl)-1-oxa-4-azaspiro[4.5]decane-3-carboxylic acid
CAS:Purity:95.0%Molecular weight:304.346008300781252-(Thiophene-2-sulfonyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid
CAS:Purity:97%Molecular weight:323.38000488281254,6-Dimethyl-2-hydroxypyrimidine
CAS:Controlled Product<p>Applications 4,6-Dimethyl-2-hydroxypyrimidine is a component of Nicarbazine (N394530), a coccidiostat, which is an antiprotozoal agent that acts upon Coccidia parasites.<br>References Ksenija Sinigoj, G., et al.: Slovenski Kemijski Dnevi, (2012); Kyung-Woo, L., et al.: Han'guk Kagum Hakhoechi, 39, 17 (2012);<br></p>Formula:C6H8N2OColor and Shape:NeatMolecular weight:124.14(4S)-Brivaracetam
CAS:Controlled ProductFormula:C11H20N2O2Color and Shape:NeatMolecular weight:212.2895-(4-Nitrophenyl)-2-furaldehyde Azine
CAS:Controlled ProductFormula:C22H14N4O6Color and Shape:NeatMolecular weight:430.373-(4-CHLOROPHENYL)-1-PHENYL-1H-PYRAZOLE-4-CARBALDEHYDE
CAS:Purity:95.0%Molecular weight:282.7300109863281[1-(2-Thienyl)-3,4-dihydroisoquinolin-2(1H)-yl]acetic acid
CAS:Purity:95.0%Molecular weight:273.3500061035156Reserpic Acid Methyl Ester
CAS:Controlled Product<p>Applications Reserpine (R144600) derivative, an alkaloid found in Rauwolfia.<br>References Itoh, A. et al.: J. Nat. Prod. 68, 848 (2005)<br></p>Formula:C23H30N2O5Color and Shape:NeatMolecular weight:414.49Carboxymefloquine-d3
CAS:Controlled Product<p>Applications Labelled Carboxymefloquine (C178700). Carboxymefloquine is a metabolite of Mefloquine (M207050).<br>References Crevoisier, C., et al.: Eur. J. Clin. Pharmacol., 53, 135 (1997), Ridtitid, W., et al.: J. Pharm. Pharmacol., 52, 1265 (2000),<br></p>Formula:C12H2D3F6NO2Color and Shape:NeatMolecular weight:312.181,3-Diphenyl-1 H -pyrazole-4-carboxylic acid
CAS:Purity:95.0%Color and Shape:SolidMolecular weight:264.28399658203125Kynurenic Acid-d5
CAS:Controlled Product<p>Applications A labelled product of L-Tryptophan metabolism, possessing neruoactive activity having antiexcitotoxic and anticonvulsant properties.<br>References Wejksza, K., et al.: Pharmacol. Rep., 61, 751 (2009), Gohil, V., et al.: Nat. Biotechnol., 28, 249 (2010), Di Natale, B., et al.: Toxicol. Sci., 115, 89 (2010),<br></p>Formula:C102H5H2NO3Color and Shape:BeigeMolecular weight:194.20Darunavir
CAS:<p>Applications Second generation HIV-1-protease inhibitor; structurally similar to amprenavir. Antiviral. It is a COVID19-related research product.<br>References Koh, Y., et al.: Antimicrob. Agents Chemother., 47, 3123 (2003), Arasteh, K., et al.: AIDS, 19, 943 (2005), Surleraux, D.L.N.G., et al.: J. Med. Chem., 48, 1813 (2005),<br></p>Formula:C27H37N3O7SColor and Shape:BeigeMolecular weight:547.66PTC-124
CAS:Controlled Product<p>Applications PTC-124 is a nonaminoglycoside that has been reported to induce ribosomes to read through premature nonsense stop signals on mRNA, allowing the production of full-length functional proteins,<br>References Yu, H. et al.: Int. J. Mol. Med., 33, 729 (2014); Aditya, S. et al.: J. Biomed. Pharm. Res., 2, 21 (2013);<br></p>Formula:C15H9FN2O3Color and Shape:White To Off-WhiteMolecular weight:284.24Primidone-d5
CAS:Controlled Product<p>Applications Anticonvulsant.<br>References Bogue, C., et al.: Br. J. Pharmacol., 8, 230 (1953), Daley, R.D., Anal. Profiles Drug Subs., 2, 409 (1973),<br></p>Formula:C122H5H9N2O2Color and Shape:Off-WhiteMolecular weight:223.28N-Nitroso Desmethyl Olopatadine
Controlled ProductFormula:C20H20N2O4Color and Shape:NeatMolecular weight:352.384rac Naproxen-d3
CAS:Controlled Product<p>Applications Labelled Naproxen. An anti-inflammatory, analgesic, antipyretic. A non-steroidal anti-inflammatory.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Harrison, I.T., et al.: J. Med. Chem., 13, 203 (1970)<br></p>Formula:C142H3H11O3Color and Shape:Off-WhiteMolecular weight:233.28(R)-6-(4-Aminophenyl)-4,5-dihydro-5-methyl-3(2H)-pyridazinone
CAS:Controlled Product<p>Applications A metabolite of Levosimendan.<br>References Rubinstein, A., et al.: J. Pharmacol. Met., 19, 213 , (1988), Pollesello, P., et al.: J. Biol. Chem., 269, 28584 (1994), Yokoshiki, H., et al.: Eur. J. Pharmacol., 333, 249 (1997)<br></p>Formula:C11H13N3OColor and Shape:NeatMolecular weight:203.24Tamsulosin
CAS:<p>Tamsulosin: an alpha1A blocker for easing urination in BPH by relaxing prostate and bladder muscles.</p>Formula:C20H28N2O5SPurity:99.93%Color and Shape:White CrystalsMolecular weight:408.51Ref: 10-F014390
1g247.00€5g624.00€10gTo inquire2.5g375.00€50mg67.00€100mg97.00€250mg128.00€500mg194.00€2-(PYRIDIN-2-YLMETHYL)-1H-BENZO[D]IMIDAZOLE-6-CARBOXYLIC ACID
Purity:90.0%Molecular weight:253.261001586914068-Bromo-3-methyl-7-(2-butynyl)-xanthine
CAS:Controlled ProductFormula:C10H9BrN4O2Color and Shape:NeatMolecular weight:297.108Norfloxacin Nicotinate
CAS:Controlled Product<p>Applications Norfloxacin nicotinate is a fluoroquinolone antibacterial agent that is a norfloxacin derivative with improved solubility in water.<br></p>Formula:C16H18FN3O3·C6H5NO2Color and Shape:NeatMolecular weight:319.33 + (123.11)Afatinib Dimaleate
CAS:Controlled Product<p>Applications Afatinib Dimaleate is a salt of Afatinib {BIBW 2992) (B377000), an aminocrotonylamino-substituted quinazoline derivative used for treating cancer and diseases of the respiratory tract, lungs, gastrointestinal tract, bile duct, and gallbladder. An anilino-quinazoline that irreversibly inhibits EGFR and HER2 kinase activity.<br>References D, Li. et al.: Oncogene., 27, 4702 (2008); Wang, X. et al.: Cancer Res., 74, 4431 (2014);<br></p>Formula:C24H25ClFN5O3·2C4H4O4Color and Shape:NeatMolecular weight:718.08N,N'-Methylene Ambroxol Hydrochloride
CAS:Controlled Product<p>Impurity Ambroxol EP Impurity B Hydrochloride<br>Stability Hygroscopic<br>Applications Ambroxol Cyclic Impurity is a metabolite as well as an impurity of the bronchosecretolytic drug, Ambroxol (A575900).<br>References Hammer, R. et al.: Arzneim.-Forsch., 28, 899 (1978); Nieder, M. et al.: HRC & CC, 9, 561 (1986); Huq, F. et al.: J. Pharmacol. Toxicol., 3, 147 (2008);<br></p>Formula:C14H18Br2N2O·ClHColor and Shape:White To Off-WhiteMolecular weight:426.571-[3-(4-tert-Butylbenzoyl)propyl]-4-hydroxypiperidine
CAS:Controlled ProductFormula:C19H29NO2Color and Shape:WhiteMolecular weight:303.44Raltitrexed
CAS:Controlled Product<p>Applications Folate-based inhibitor of thymidylate synthase; rapidly and extensively metabolized to its more potent polyglutamate derivatives. Antineoplastic.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Jodrell, D.I., et al.: Cancer Chemother. Pharmacol., 28, 331 (1991), Jackman, A.L., et al.: Eur. J. Cancer, 31A, 1277 (1995)<br></p>Formula:C21H22N4O6SColor and Shape:NeatMolecular weight:458.49(5,6-Difluoropyridin-3-yl)boronic acid
CAS:Formula:C5H4BF2NO2Purity:96%Color and Shape:No data available.Molecular weight:158.95-Methyl-2-(2,4,6-trichlorophenyl)-2H-pyrazol-3-ylamine
CAS:Formula:C10H8Cl3N3Purity:97.0%Molecular weight:276.55(S)-N-((2-oxo-3-(4-(3-oxomorpholino)phenyl)oxazolidin-5-yl)methyl)thiophene-2-carboxamide
CAS:Purity:98%Molecular weight:401.440002441406251-(4-Fluorophenyl)-3-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-1H-pyrazole-4-carbaldehyde
CAS:Molecular weight:324.3110046386719N-Benzyl Hydroxymedetomidine
CAS:Controlled Product<p>Applications N-Benzyl Hydroxymedetomidine is an impurity of Medetomidine (M203250, HCl); an α2-adrenergic agonist, sedative, and analgesic.<br>References Scheinin, M., et al.: Br. J. Clin. Pharmacol., 24, 443 (1987); Stenberg, D., et al.: J. Vet. Pharmacol. Ther., 10, 319 (1987); Virtanen, R., et al.: Eur. J. Pharmacol., 150, 9 (1988); Cullen, L.K., et al.: Br. Vet. J., 152, 519 (1996)<br></p>Formula:C20H22N2OColor and Shape:NeatMolecular weight:306.4N-Nitroso-Vildagliptin
CAS:Controlled ProductFormula:C17H24N4O3Color and Shape:NeatMolecular weight:332.4(4-(Diisopropylcarbamoyl)-2-ethoxypyridin-3-yl)boronic acid
CAS:Purity:95+%Molecular weight:294.1600036621094Arotinolol
CAS:Controlled Product<p>Applications Arotinolol is both and alpha- and beta-adrenoceptor antagonist and is used to treat essential tremors and hypertension.<br>References Kuroda, Y., et al.: Neurology, 38, 650 (1988); Miyagishi, A., et al.: Arch. Pharmacodyn. Ther., 271, 249 (1984); Wu, H., et al.: Hypertens. Res.: Off. J. Jpn. Soc. Hypertens., 24, 605 (2001)<br></p>Formula:C15H21N3O2S3Color and Shape:NeatMolecular weight:371.541-(4-morpholinyl)cyclohexanecarboxylic acid hydrochloride hydrate
Purity:95.0%Molecular weight:267.753’-Anhydro Ezetimibe
CAS:Controlled ProductFormula:C24H19F2NO2Color and Shape:NeatMolecular weight:391.41[1-(2-thienyl)butyl]amine hydrochloride
CAS:Formula:C8H14ClNSPurity:95.0%Color and Shape:SolidMolecular weight:191.72
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