Quinazoline and Quinoline Derivatives
Quinazolines and quinolines are nitrogen-containing heterocyclic compounds with aromatic structures that play a key role in the synthesis of drugs with anticancer, antimicrobial, and anti-inflammatory activity. Their derivatives feature structural modifications that optimise bioavailability and selectivity, enabling the development of new active ingredients for various therapeutic applications. These compounds are used in the manufacture of APIs for the treatment of cancer, infections, neurodegenerative diseases, and cardiovascular conditions. Additionally, quinazoline and quinoline derivatives are essential in the research of enzyme inhibitors and the design of innovative bioactive molecules.
At CymitQuimica, we offer high-purity quinazoline and quinoline derivatives for applications in chemical synthesis, pharmaceutical development, and biotechnology.
Found 65615 products of "Quinazoline and Quinoline Derivatives"
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2-Quinolin-2-yl-1-[3-(trifluoromethyl)phenyl]ethanone
CAS:Formula:C18H12F3NOPurity:95.0%Color and Shape:SolidMolecular weight:315.2955-(1,3-Dioxolan-2-yl)-2-(3-nitrobenzoyl)thiophene
CAS:Purity:97.0%Molecular weight:305.29998779296875ETHYL 1-CYCLOPROPYL-6,7-DIFLUORO-8-METHOXY-4-OXO-1,4-DIHYDRO-QUINOLINE-3-CARBOXYLATE
CAS:Purity:97.0%Color and Shape:SolidMolecular weight:323.2959899902344Destriazolyl Bromo Propiconazole (Mixture of Diastereomers)
CAS:<p>Applications Destriazolyl Bromo Propiconazole is an impurity of Propiconazole (P770100).<br>References Godefroi, E.F., et al.: J. Med. Chem., 12, 784 (1969), Buchel, K.H., et al.: Arzneim.-Forsch., 22, 1260 (1972),<br></p>Formula:C13H15BrCl2O2Color and Shape:NeatMolecular weight:354.071’-Hydroxy Bufuralol (Mixture of Diastereomers)
CAS:Controlled Product<p>Stability Hygroscopic<br>Applications A metabolite of Bufuralol, a β-Adrenergic blocker with peripheral vasodilating activity.<br>References Boobis, A.R., et al.: Biochem. Pharmacol., 34, 65 (1985), Yamazaki, H., et al.: Mol. Pharmacol., 46, 568 (1994), Mast, N., et al.: Biochem., 42, 14284 (2003),<br></p>Formula:C16H23NO3Color and Shape:BeigeMolecular weight:277.36R-(-)-N-Demethyl Deprenyl-d5
CAS:Controlled Product<p>Applications A labelled metabolite of Deprenyl (D288641) (Selegiline).<br>References Dyck, L., et al.: Drug Metab. Dispos., 29, 1156 (2001), Damaj, M., et al.: J. Pharmacol. Exp. Ther., 320, 250 (2007),<br></p>Formula:C12H10D5NColor and Shape:NeatMolecular weight:178.291,3-Bis(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)thiourea
CAS:Purity:98%Molecular weight:448.549987792968752-[4-[2-(1-Piperidinyl)ethoxy]benzoyl]benzoic Acid
CAS:<p>Applications 2-[4-[2-(1-Piperidinyl)ethoxy]benzoyl]benzoic Acid is a research reagent with antispasmodic<br>References Bal-Tembe, S., et al.: Bioorg. Med. Chem., 5, 1381(1997);Punekar, N., et al.: Biotech. App. Biochem, 14, 378 (1991);<br></p>Formula:C21H23NO4Color and Shape:NeatMolecular weight:353.41ent-Rivaroxaban
CAS:<p>Applications ent-Rivaroxaban is the R-isomer of Rivaroxaban (R538000), which is a novel antithrombotic agent. A highly potent and selective, direct FXa inhibitor.<br>References Ansell, J., et al.: Drugs, 64, 1 (2004), Eriksson, B., et al.: J. Thromb. Haemost., 3, 103 (2005), Kubitza, D., et al.: Clin. Pharmacol. Ther., 78, 412 (2005),<br></p>Formula:C19H18ClN3O5SColor and Shape:White To Off-WhiteMolecular weight:435.88(E)-3-(2-Cyclopropyl-4-(4-fluorophenyl)quinolin-3-yl)acrylaldehyde
CAS:Purity:95%Molecular weight:317.36300659179692-n-Propyl-4-methyl-6-(1-methylbenzimidazol-2-yl)-benzimidazole
CAS:Formula:C19H20N4Color and Shape:WhiteMolecular weight:304.391-(2,4,5-Trimethoxybenzyl)piperazine Dihydrochloride
CAS:Controlled Product<p>Stability Hygroscopic<br>Applications 1-(2,4,5-Trimethoxybenzyl)piperazine Dihydrochloride is an impurity of Trimetazidine (T795610). Trimetazidine impurity E.<br></p>Formula:C14H22N2O3·2ClHColor and Shape:NeatMolecular weight:339.26Nateglinide Ethyl Ester
CAS:Controlled Product<p>Applications The ethyl ester of the oral hypoglycemic agent Nateglinide (N379375). It showed no effects on gross behavior in mice.<br>References Maeda, K. et al.: Yak. Chir., 25, S157 (1997);<br></p>Formula:C21H31NO3Color and Shape:NeatMolecular weight:345.48N-(2-Succinyl) Phenylephrine(Mixture of Diastereomers) ( >85%)
CAS:<p>Impurity N-(2-Succinyl) Phenylephrine Impurity<br>Applications The major degradation product identified in Acetaminophen, Phenylephrine hydrochloride, and Chlorpheniramine maleate.<br>References Wong, J., et al.: Anal. Chem., 78, 7891 (2006),<br></p>Formula:C13H17NO6Purity:>85%Color and Shape:NeatMolecular weight:283.283-[5-(1,5-Dioxo-5-(p-fluophenylpentyl]-4(S)-phenyl-2-oxazolidinone
CAS:Controlled ProductFormula:C20H18FNO4Color and Shape:NeatMolecular weight:355.3596Topiramate-d12
CAS:Controlled Product<p>Applications Labelled Topiramate, which is used as an anticonvulsant.<br></p>Formula:C122H12H9NO8SColor and Shape:Off WhiteMolecular weight:351.447-Hydroxy Risperidone
CAS:Controlled ProductFormula:C23H27FN4O3Color and Shape:NeatMolecular weight:426.48Alogliptin Benzoate
CAS:<p>Applications Alogliptin Benzoate is an oral antihyperglycemic agent that is a selective inhibitor of the enzyme dipeptidyl peptidase-4 (DPP-4). Alogliptin Benzoate is used in the treatment of type 2 diabetes.<br>References Wang, Y., et. al.: Drugs Future, 33, 7 (2008); Lynn, F., et al.: Diabetes, 50, 1004 (2001); Trumper, A., et al.: J. Endocrinol., 174, 233 (2002); Vollmer, K., et al.: J. Clin. Endocrinol. Metab., 94, 1379 (2009)<br></p>Formula:C18H21N5O2·C7H6O2Color and Shape:NeatMolecular weight:461.512,3-Dichlorothiophene-5-sulfonyl chloride
CAS:Formula:C4HCl3O2S2Purity:≥97%Color and Shape:SolidMolecular weight:251.52Mitotane-13C6
CAS:Controlled Product<p>Applications Mitotane-13C6 is the isotope labelled analogue of Mitotane (M372500), an antineoplastic and adrenolytic agent.<br>References Das, S., and Thomas, P.: Endocrinology, 140, 1953 (1999), Andersen, A., et al.: Ther. Drug. Monit., 21, 355 (1999), Leblond, V.S., and Hontela, T.: Toxicol. Appl. Pharmacol., 157, 16 (1999)<br></p>Formula:C6C8H10Cl4Color and Shape:Light YellowMolecular weight:326.03-Chloromethyl-5-methylpyridine Hydrochloride
CAS:Controlled Product<p>Applications 3-Chloromethyl-5-methylpyridine is an intermediate in the synthesis of Rupatadine (R701650).<br>References Merlos, M., et al.: Pharmacol. Exp. Therap., 280, 114 (1997), Bell, I., et al.: J. Med. Chem., 41, 2146 (1998),<br></p>Formula:C7H8ClN·ClHColor and Shape:White To BeigeMolecular weight:178.06(R)-9-Hydroxy Risperidone-d4
CAS:Controlled ProductFormula:C23H23D4FN4O3Color and Shape:NeatMolecular weight:430.512-Hydroxy-5-methylpyridine
CAS:Controlled Product<p>Applications 2-Hydroxy-5-methylpyridine (cas# 1003-68-5) is a useful compound for organic synthesis. In particular it has been used for the diastereoselective preparation of cyclobutane-fused pyridinyl sulfonyl fluorides.<br>References Liu, J., et al.: Org. Biomol. Chem., 18, 4019 (2020)<br></p>Formula:C6H7NOColor and Shape:Light YellowMolecular weight:109.13Dehydro Nifedipine-d6
CAS:Controlled Product<p>Applications The main labelled Nifedipine metabolite in human plasma.<br>References Guengerich, F., et al.: J. Biol. Chem., 261, 5051 (1986), Bork, R., et al.: J. Biol. Chem., 264, 910 (1989), Kerla, V., et al.: Biochem. Pharmacol., 44, 1745 (1992),<br></p>Formula:C17H10D6N2O6Color and Shape:NeatMolecular weight:350.362-{[3-(4-Chlorophenyl)-1-phenyl-1H-pyrazol-4-yl]methylidene}-5,5-dimethylcyclohexane-1,3-dione
CAS:Molecular weight:404.8900146484375Lornoxicam
CAS:Controlled Product<p>Applications Cyclooxygenase inhibitor; structurally similar to Tenoxicam. Anti-inflammatory; analgesic.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Ankier, S.I., et al.: Postgrad. Med. J., 64, 752 (1988), Tricerri, M., et al.: Chem. Phys. Lipids, 71, 61 (1994), Santos, N., et al.: Biochemistry, 37, 8674 (1998), Pellicano, A., et al.: Infect. Immun., 75, 1738 (2007),<br></p>Formula:C13H10ClN3O4S2Color and Shape:Yellow Crystalline PowderMolecular weight:371.823-((3-(N-Cyclopropylsulfamoyl)-7-(2,4-dimethoxypyrimidin-5-yl)quinolin-4-yl)amino)-5-(3,5-difluorophenoxy)benzoic acid
CAS:Purity:98%Molecular weight:649.630004882813Ref: 10-F867169
5mgTo inquire10mgTo inquire25mgTo inquire50mgTo inquire100mgTo inquire250mgTo inquire3-(Pyridin-3-yl)-[1,2,4]triazolo[4,3-a]pyridine-6-carboxylic acid
CAS:Molecular weight:240.2220001220703Metomidate Hydrochloride
CAS:Controlled Product<p>Applications Metomidate Hydrochloride is used as an anesthetic for veterinary use.<br>References Harvey, B., et al.: Vet. Rec. 122(8), 174-7 (1988); Green, C. J., et al.: Lab. Anim., 15(2), 171-5 (1981); Cadle, D. R., et al.: Vet. Rec., 98(5), 91-2 1976); Massee, K. C., et al.: Aquaculture, 134(3-4), 351-359 (1995)<br></p>Formula:C13H14N2O2·ClHColor and Shape:White To Off-WhiteMolecular weight:266.72Loxapine N-Oxide
CAS:<p>Stability Hygroscopic, Light Sensitive<br>Applications Loxapine N-Oxide is a metabolite of Loxapine (L472750), a D2/D4-Dopamine receptor antagonist. It is a serotonergic receptor antagonist that acts as a dibenzoxazepine antipsychotic agent.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Shen, Y., et al.: J. Biol. Chem., 268, 18200 (1993), Fiorella, D., et al.: Psychopharmacology, 121, 347 (1995), Glusa, E., et al.: Br. J. Pharmacol., 130, 692 (2000)<br></p>Formula:C18H18ClN3O2Color and Shape:NeatMolecular weight:343.815,5',5''-(1,3,5-Triazine-2,4,6-triyl)tris(pyridin-2-amine)
CAS:Purity:95%Color and Shape:SolidMolecular weight:357.38101196289066-Fluoro-3-(4-piperidinyl)-1,2-benzisoxazole Hydrochloride
CAS:Controlled Product<p>Impurity Risperidone EP Impurity M; Paliperidone USP Related Compound B<br>Applications 6-Fluoro-3-(4-piperidinyl)-1,2-benzisoxazole Hydrochloride (Risperidone EP Impurity M; Paliperidone USP Related Compound B) is a novel antiproliferative agent.<br>References Benaka P. et al.: Invest. New Drugs., 27, 534 (2009);<br></p>Formula:C12H13FN2O·ClHColor and Shape:NeatMolecular weight:256.70Zaltoprofen
CAS:Controlled Product<p>Applications Zaltoprofen is a non-steroidal anti-inflammatory drug. It inhibits bradykinin-induced pain responses without blocking bradykinin receptors.<br>References Hirate, K., et al.: Nerosci. Res., 54, 288 (2006); Yamamoto, M., et al.: Chirality, 2, 280 (1990); Inoue, M., et al.: J Pharmacol. Exp. Ther., 293, 662 (2000); Graven-Nielsen, T., et al.: Clin. J. Pain, 17, 2 (2001)<br></p>Formula:C17H14O3SColor and Shape:NeatMolecular weight:298.366-methoxy-N-(pyridin-2-ylmethyl)-1,3-benzothiazol-2-amine
CAS:Purity:95.0%Molecular weight:271.3399963378906Nizatidine
CAS:Controlled Product<p>Applications Histamine H2-receptor antagonist related to Ranitidine (R120000). Antiulcerative.<br>References Callaghan, J.T., et al.: Clin. Pharmacol. Ther., 37, 162 (1985), Secor, J.W., et al.: Br. J. Clin. Pharmacol., 20, 710 (1985), Knadler, M.P., et al.: Drug Metab. Dispos., 14, 175 (1986), Wozniak, T.J., et al.: Anal. Profiles Drug Subs., 19, 397(1990)<br></p>Formula:C12H21N5O2S2Color and Shape:Off-White To Light YellowMolecular weight:331.46N”Nitrosoprotriptyline
CAS:Controlled ProductFormula:C19H20N2OColor and Shape:NeatMolecular weight:292.3752-[3,5-Dichloro-4-[(4-chlorophenyl)methyl]phenyl]-1,2,4-triazine-3,5(2H,4H)-dione
CAS:Controlled Product<p>Applications An anticoccidal triazine used for the treatment of coccidiosis in chickens. An impurity of Diclazuril (D436200).<br>References McFarland, J. et al.: J. Med. Chem., 35, 2543 (1992);<br></p>Formula:C16H10Cl3N3O2Color and Shape:NeatMolecular weight:382.63
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