Enzyme Modulators
Enzyme modulators are compounds that can enhance or inhibit the activity of enzymes, thereby regulating the rate of biochemical reactions. These modulators play a critical role in controlling metabolic pathways, cell signaling, and various physiological processes. Enzyme modulators are widely used in research and drug development to study enzyme functions and to develop therapeutic agents. At CymitQuimica, we offer a comprehensive range of high-quality enzyme modulators to support your research in enzyme regulation and drug discovery.
Subcategories of "Enzyme Modulators"
Found 691 products for "Enzyme Modulators".
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Zileuton- Bio-X ™
CAS:Zileuton is an inhibitor of the 5-lipoxygenase enzyme, thus preventing the leukotrienes LTE4, LDT4, LTB4 and LTC4 from being formed. This in turn reduces inflammation, bronchoconstriction and mucus secretion in the airways. As a result, Zileuton can be used in the treatment and management of asthma and allergic rhinitis. Studies have shown that Zileuton has the potential to reverse dementia-related brain damage.Formula:C11H12N2O2SPurity:(%) Min. 95%Color and Shape:PowderMolecular weight:236.29 g/mol4-Deoxyuridine
CAS:A cytidine analogue and inhibitor of DNA methyl transferases (DNMTs) with anti-cancer activity. This stable, hydrophilic compound forms covalent complexes between DNMT and zebularine-substrate DNA. It causes DNA lesions that block replication and cause replication fork collapse, leading to the formation of DNA double-strand breaks. It was also shown that zebularine-induced DNA methylation decrease in the IL-1β promoter region and disrupts molecular mechanisms of neuroinflammation. Moreover, this molecule down-regulates the DNA-methylation profile in the pluripotency genes’ promoters, which leads to improved development of somatic cell nuclear transfer (SCNT) embryos.Formula:C9H12N2O5Purity:Min. 95%Color and Shape:PowderMolecular weight:228.21 g/molPelitinib
CAS:EGFR tyrosine kinase inhibitor; pro-apoptotic; antiproliferative in cancer cellsFormula:C24H23ClFN5O2Purity:Min. 95%Color and Shape:PowderMolecular weight:467.92 g/molApremilast - Bio-X ™
CAS:Apremilast is the commercial name of a phosphodiesterase-4 (PDE4) inhibitor developed to treat chronic inflammatory disorders. Similarly to thalidomide, the apremilast molecule carries a phthalimide ring, but it lacks however the glutarimide ring needed to bind to cereblon, specifically targeted by thalidomide. As a drug, apremilast is indicated for the treatment of psoriasis and psoriatic arthritis.Formula:C22H24N2O7SPurity:Min. 99 Area-%Color and Shape:White/Off-White SolidMolecular weight:460.5 g/molVatalanib HCl
CAS:VEGFR tyrosine kinase inhibitor
Formula:C20H15ClN4•HClPurity:Min. 95%Molecular weight:383.27 g/molU 0126 monoethanolate
CAS:Inhibitor of MEK1 and MEK2 kinasesFormula:C18H16N6S2•C2H6OPurity:Min. 95%Color and Shape:White To Beige SolidMolecular weight:426.56 g/molNolatrexed dihydrochloride
CAS:Thymidylate synthase inhibitorFormula:C14H14Cl2N4OSPurity:Min. 95%Color and Shape:White To Light (Or Pale) Yellow SolidMolecular weight:357.26 g/molMeloxicam - Bio-X ™
CAS:Meloxicam is a non-steroidal anti-inflammatory drug (NSAID) which is used to treat various types of pain and inflammation caused by arthritis. It is also a COX-2 inhibitor which reduces gastrointestinal effects of this drug. Inhibiting these enzymes, allow for a decrease in inflammatory symptoms.Formula:C14H13N3O4S2Purity:Min. 95%Color and Shape:PowderMolecular weight:351.4 g/molPimecrolimus
CAS:Immune suppressant; prevents pro-inflammatory cytokine releaseFormula:C43H68ClNO11Purity:Min. 95%Color and Shape:PowderMolecular weight:810.45 g/molMK 886 sodium salt
CAS:Inhibitor of 5-lipoxygenase activating protein_x000D_
Formula:C27H33ClNNaO2SPurity:Min. 95%Color and Shape:PowderMolecular weight:494.06 g/molCA3
CAS:Inhibits YAP/Tead transcriptional activity. Has anti-tumour effects on oesophageal adenocarcinoma with therapeutic potential in combination with 5-FU. Involved in ferroptosis, mediated by iron-dependent ROS.
Formula:C23H27N3O5S2Purity:Min. 95%Color and Shape:White Off-White PowderMolecular weight:489.61 g/molRipasudil HCl hydrate
CAS:Inhibitor of Rho-kinases
Formula:C15H18FN3O2S•HCl•(H2O)2Purity:Min. 95%Color and Shape:White Off-White PowderMolecular weight:395.88 g/molBIX 02188
CAS:A selective inhibitor of MEK5 protein kinase with an IC50 value of 4.3 nM. Blocks transcriptional activation of myocyte-specific enhancer factor 2C (MEF2C). Inhibits phosphorylation of ERK5 protein kinase and thereby reverses inhibition of TNF signaling induced by fluid shear stress in endothelial cells. Induces apoptosis in FLT3-ITD cells.
Formula:C25H24N4O2Purity:Min. 95%Molecular weight:412.18993A 939572 - Bio-X ™
CAS:A 939572 is an inhibitor of stearoyl-CoA desaturase 1 (SCD1). It exhibits anticancer activity as it inhibits cell growth and promotes cell death in human non-small cell lung carcinoma cells.Formula:C20H22ClN3O3Purity:Min. 95%Color and Shape:PowderMolecular weight:387.86 g/molAtorvastatin sodium salt - Bio-X ™
CAS:Atorvastatin is an HMG-CoA reductase inhibitor which is used to lower lipid levels and to reduce the risk of cardiovascular disease. This drug belongs to the class of medicines called statins. It lowers abnormal levels of cholesterol and lipids to reduce the risk of cardiovascular disease by inhibiting the enzyme HMG-CoA.Formula:C33H35FN2O5•NaPurity:(%) Min. 95%Color and Shape:PowderMolecular weight:581.63 g/molDrotaverine HCl - Bio-X ™
CAS:Drotaverine is an antispasmodic drug that is used to alleviate gastrointestinal and genitourinary smooth muscle spasms. This drug works by inhibiting phosphodiesterase-4 and increasing levels of cAMP leading to smooth muscle relaxation.Formula:C24H31NO4•HClPurity:Min. 95%Color and Shape:PowderMolecular weight:433.97 g/molDeracoxib
CAS:Inhibitor of COX-2 and PDE4 enzymes; NSAID of coxib classFormula:C17H14F3N3O3SPurity:Min. 95%Color and Shape:White To Off-White To Brown SolidMolecular weight:397.37 g/molIWP-2
CAS:Antagonist of Wnt signalling pathway by inhibiting the activity of Porcn, a member of the membrane-bound O-acyltransferase (MBOAT) family. Porcn is required for the palmitoylation of Wnt, mediating its secretion and signalling. Inhibits self-renewal in embryonic stem cells, whilst promoting differentiation to epiblast stem cells.Formula:C22H18N4O2S3Purity:Min. 95%Color and Shape:White To Off-White SolidMolecular weight:466.05919Rofecoxib - Bio-X ™
CAS:Controlled ProductRofecoxib is a non-steroidal anti-inflammatory drug that is used to treat osteoarthritis, acute pain and migraine attacks. This drug is also a COX-2 inhibitor. As a result, it reduces inflammation and pain.Formula:C17H14O4SPurity:Min. 95%Color and Shape:PowderMolecular weight:314.36 g/mol
