Apoptosis
Los inhibidores de la apoptosis son compuestos que previenen o retrasan el proceso de muerte celular programada, conocido como apoptosis. Estos inhibidores son vitales para estudiar los mecanismos de supervivencia celular y se utilizan para investigar enfermedades donde la apoptosis está desregulada, como el cáncer, los trastornos neurodegenerativos y las enfermedades autoinmunes. Al modular la apoptosis, estos inhibidores pueden ayudar en el desarrollo de terapias dirigidas a controlar la muerte celular. En CymitQuimica, ofrecemos una amplia selección de inhibidores de la apoptosis de alta calidad para apoyar su investigación en biología celular, oncología y campos relacionados.
Subcategorías de "Apoptosis"
- ASK(6 productos)
- BCL(11 productos)
- Caspasa(125 productos)
- FOXO1(3 productos)
- IAP(66 productos)
- Mdm2(12 productos)
- PD-1 / PD-L1(125 productos)
- PDK(9 productos)
- PERK(25 productos)
- Serina / treonina quinasa(15 productos)
- Survivin(13 productos)
- TNF(92 productos)
- c-RET(51 productos)
- p53(62 productos)
Mostrar 6 subcategorías más
Se han encontrado 5600 productos de "Apoptosis"
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Tetrahydropalmatine
CAS:<p>Tetrahydropalmatine (DL-Tetrahydropalmatine) is an active component isolated from corydalis, suppressing amygdaloid release of dopamine to inhibit an epileptic</p>Fórmula:C21H25NO4Pureza:99.59% - 99.95%Forma y color:SolidPeso molecular:355.43Geniposidic Acid
CAS:<p>Geniposidic acid, an iridoid glucoside, used in therapy of jaundice, inflammation and hepatic disorders.</p>Fórmula:C16H22O10Pureza:99.77% - >99.99%Forma y color:SolidPeso molecular:374.34Pemetrexed disodium
CAS:<p>Pemetrexed disodium treats lung cancer/mesothelioma; may cause moderate serum enzyme elevation, rarely acute liver injury.</p>Fórmula:C20H19N5Na2O6Pureza:99.29% - 99.49%Forma y color:Crystalline SolidPeso molecular:471.37NVP-2
CAS:<p>NVP-2 selectively inhibits CDK9 (IC50: 0.514 nM), prompts apoptosis, and affects other CDKs (IC50: 0.584-0.706 μM).</p>Fórmula:C27H37ClN6O2Pureza:99.13%Forma y color:SolidPeso molecular:513.07Salicylic acid
CAS:<p>Salicylic acid (2-Hydroxybenzoic acid), a natural compound extracted from Willow bark, is an anti-inflammatory inhibitor of activity cyclooxygenase.</p>Fórmula:C7H6O3Pureza:98.04% - 98.83%Forma y color:White Solid PowderPeso molecular:138.12(20S)-Protopanaxadiol
CAS:(20S)-Protopanaxadiol (20-Epiprotopanaxadiol) (20-Epiprotopanaxadiol), an apoptosis inducer, is an aglycon metabolic derivative of the protopanaxadiol-typeFórmula:C30H52O3Pureza:97.07% - 98.91%Forma y color:SolidPeso molecular:460.73Cetrimonium bromide
CAS:<p>Cetrimonium bromide (Lauroseptol) is is a mixture of different quaternary ammonium salts, which is a known component of the broad-spectrum antiseptic cetrimide.</p>Fórmula:C19H42BrNPureza:≥95%Forma y color:SolidPeso molecular:364.46Thioridazine hydrochloride
CAS:<p>Thioridazine hydrochloride (Mellaril) , an antipsychotic drug, is used in the therapy of psychosis and schizophrenia and shows serotonin antagonism or D4</p>Fórmula:C21H27ClN2S2Pureza:99.55% - 99.957%Forma y color:White To Off-White SolidPeso molecular:407.04Onvatilimab
CAS:<p>Onvatilimab (JNJ-61610588) is a human IgG1 κ monoclonal antibody with antitumor effects for advanced head and neck cancers.</p>Pureza:98.11% (SEC-HPLC) - > 95%Forma y color:LiquidPeso molecular:144.52 kDaLinagliptin
CAS:<p>Linagliptin (BI 1356) is a potent, orally bioavailable dihydropurinedione-based inhibitor of dipeptidyl peptidase 4 (DPP-4), with hypoglycemic activity.</p>Fórmula:C25H28N8O2Pureza:99.15% - >99.99%Forma y color:SolidPeso molecular:472.54Cytarabine
CAS:<p>Cytarabine (Ara-C) is a nucleoside analog, an inhibitor of DNA synthesis (IC50=16 nM).</p>Fórmula:C9H13N3O5Pureza:99.83% - 99.93%Forma y color:Fine Off-White Crystalline PowderPeso molecular:243.22Vorinostat
CAS:<p>Vorinostat (SAHA) is a pan-histone deacetylase (HDAC) inhibitor (IC50=10 nM) with inhibitory activity against HDAC1/2/3/6/7/11.</p>Fórmula:C14H20N2O3Pureza:99.47% - 99.65%Forma y color:White Crystalline SolidPeso molecular:264.32Abacavir
CAS:<p>Abacavir (Ziagen) is a nucleoside reverse transcriptase inhibitor analog of guanosine.</p>Fórmula:C14H18N6OPureza:99.36% - 99.81%Forma y color:White PowderPeso molecular:286.33Topotecan hydrochloride
CAS:<p>Topotecan hydrochloride (NSC609699) is an antineoplastic agent used to treat ovarian cancer.</p>Fórmula:C23H24ClN3O5Pureza:97.88% - 99.41%Forma y color:White Crystalline SolidPeso molecular:457.92IBR2
CAS:<p>IBR2 is a potent RAD51 inhibitor that disrupts DNA repair, inhibits cancer cell growth, and induces apoptosis.</p>Fórmula:C24H20N2O2SPureza:99.5%Forma y color:SolidPeso molecular:400.49DCZ0415
CAS:<p>DCZ0415: Potent TRIP13 inhibitor; combats myeloma in vitro, in vivo, and in drug-resistant patients; hinders DNA repair and NF-κB activity.</p>Fórmula:C23H20N2O2Pureza:99.34% - 99.95%Forma y color:SolidPeso molecular:356.42Crolibulin
CAS:<p>Crolibulin (EPC2407) is an inhibitor of small molecule tubulin polymerization.</p>Fórmula:C18H17BrN4O3Pureza:98.04%Forma y color:SolidPeso molecular:417.26Oxcarbazepine
CAS:<p>Oxcarbazepine (GP 47680), an anti-epileptic, reduces CNS disorganized electrical activity.</p>Fórmula:C15H12N2O2Pureza:98.46%Forma y color:Crystals From Ethanol SolidPeso molecular:252.27Piceatannol
CAS:<p>Piceatannol (Astringenin) is a synthetic anti-inflammatory that blocks p56lck, syk kinases, and NF-κB, made from resveratrol.</p>Fórmula:C14H12O4Pureza:98.66% - 99.73%Forma y color:Light Tan To Yellow PowderPeso molecular:244.24BAM 15
CAS:<p>BAM 15 is an uncoupler of mitochondrial protonophore.</p>Fórmula:C16H10F2N6OPureza:99.75% - 99.92%Forma y color:SolidPeso molecular:340.29JTE-013
CAS:<p>JTE-013 is an effective and specific antagonist of S1P2.</p>Fórmula:C17H19Cl2N7OPureza:97.69%Forma y color:SolidPeso molecular:408.29Bithionol
CAS:<p>Bithionol (Actamer), formerly marketed as an active ingredient in various topical drug products, was shown to be a potent photosensitizer with the potential to</p>Fórmula:C12H6Cl4O2SPureza:99.04%Forma y color:White Or Grayish-White Crystalline Powder Phenolic Odor (Ntp 1992)Peso molecular:356.05Benzethonium chloride
CAS:<p>Benzethonium chloride (Quatrachlor) is a synthetic quaternary ammonium salt with surfactant, antiseptic, and broad spectrum antimicrobial properties.</p>Fórmula:C27H42ClNO2Pureza:99.91%Forma y color:White To Off-White Solid Solid Particulate/PowderPeso molecular:448.09Olanzapine
CAS:<p>Olanzapine (LY170053) is an atypical antipsychotic that is used currently in the treatment of schizophrenia and bipolar illness.</p>Fórmula:C17H20N4SPureza:99.86% - ≥95%Forma y color:Yellowish Crystalline PowderPeso molecular:312.43BH3I-1
CAS:<p>BH3I-1 (BHI1) is a Bcl-2 antagonist.</p>Fórmula:C15H14BrNO3S2Pureza:97.6% - 98.2%Forma y color:SolidPeso molecular:400.319-ING-41
CAS:<p>9-ING-41 is a glycogen synthase kinase-3 inhibitor.</p>Fórmula:C22H13FN2O5Pureza:99.32%Forma y color:SolidPeso molecular:404.35(E/Z)-BCI
CAS:<p>(E/Z)-BCI (NSC-150117), a dual-specificity phosphatase 6 (DUSP6) inhibitor with anti-inflammatory properties, reduces LPS-induced inflammatory mediators and ROS</p>Fórmula:C22H23NOPureza:99.94%Forma y color:SolidPeso molecular:317.42Nimbolide
CAS:<p>Nimbolide, from neem, inhibits CDK4/6, NF-κB, Wnt, PI3K-Akt, MAPK, JAK-STAT pathways and induces apoptosis.</p>Fórmula:C27H30O7Pureza:95.84% - 99.4%Forma y color:SolidPeso molecular:466.52Estradiol benzoate
CAS:<p>Estradiol benzoate (Benzhormovarine) is the synthetic benzoate ester of estradiol, a steroid sex hormone vital to the maintenance of fertility in females.</p>Fórmula:C25H28O3Pureza:99.7% - 99.93%Forma y color:SolidPeso molecular:376.49Docetaxel
CAS:<p>Docetaxel (RP-56976) is a semi-synthetic analog of paclitaxel, a microtubule depolymerization inhibitor (IC50=0.2 μM).</p>Fórmula:C43H53NO14Pureza:98.6% - 99.29%Forma y color:Off-White CrystPeso molecular:807.88Tiratricol
CAS:<p>Tiratricol, a thyroid hormone metabolite for hyperlipidemia and obesity, studied in Allan-Herndon-Dudley Syndrome treatment.</p>Fórmula:C14H9I3O4Pureza:98.77% - 99.16%Forma y color:SolidPeso molecular:621.93(11β)-17-(Acetyloxy)-11-[4-(dimethylamino)phenyl]-19-norpregna-4,9-diene-3,20-dione
CAS:Fórmula:C30H37NO4Pureza:98%Forma y color:SolidPeso molecular:475.6191Norcantharidin, mixture of endo/exo
CAS:Fórmula:C8H8O4Pureza:97%Forma y color:SolidPeso molecular:168.1467Phenformin
CAS:<p>Phenformin: a biguanide with anti-cancer, anti-glycemic effects, inhibits skin tumors, enhances keratinocyte differentiation/apoptosis.</p>Fórmula:C10H15N5Pureza:99.72%Forma y color:SolidPeso molecular:205.26Cl-amidine hydrochloride
CAS:<p>Cl-amidine hydrochloride is an orally available PAD inhibitor that blocks histone 3 deimination.Cost-effective and quality-assured.</p>Fórmula:C14H20Cl2N4O2Pureza:92.34% - 98.14%Forma y color:SolidPeso molecular:347.24Oxireno[9,10]cyclodeca[1,2-b]furan-9(1aH)-one, 2,3,6,7,7a,8,10a,10b-octahydro-1a,5-dimethyl-8-methylene-, (1aR,4E,7aS,10aS,10bR)-
CAS:Fórmula:C15H20O3Pureza:97%Forma y color:SolidPeso molecular:248.3175Roxadustat
CAS:<p>Roxadustat (FG-4592) is an orally bioavailable, hypoxia-inducible factor prolyl hydroxylase inhibitor (HIF-PHI), with potential anti-anemic activity.</p>Fórmula:C19H16N2O5Pureza:99% - 99.88%Forma y color:SolidPeso molecular:352.34Ruplizumab
CAS:<p>PF-03732010 is a humanized antibody targeting P-calmodulin with antitumor and antimetastatic activity.</p>Pureza:98.5% (SDS-PAGE); 98.7% (SEC-HPLC) - 98.5% (SDS-PAGE); 98.7% (SEC-HPLC)Forma y color:LiquidRef: IN-DA00365L
1g285,00€5gA consultar10gA consultar1mg44,00€25gA consultar50gA consultar25mg68,00€50mg102,00€100mg120,00€250mg157,00€500mg184,00€[1,4'-Bipiperidine]-1'-carboxylic acid,(4S)-4,11-diethyl-3,4,12,14-tetrahydro-4-hydroxy-3,14-dioxo-1H-pyrano[3',4':6,7]indolizino[1,2-b]quinolin-9-yl ester, monohydrochloride
CAS:Fórmula:C33H39ClN4O6Pureza:98%Forma y color:SolidPeso molecular:623.1390β-Elemene
CAS:<p>β-Elemene (Levo-β-elemene) is a natural product isolated from Curcuma wenyujin, with an antitumor activity and induce cell apoptosis.</p>Fórmula:C15H24Pureza:99.165% - 99.35%Forma y color:SolidPeso molecular:204.35(E)-Methyl 4-coumarate
CAS:<p>(E)-Methyl 4-coumarate (OMpCA) is a predicted metabolite generated by BioTransformer1 that is produced by the metabolism of methyl 3-phenylprop-2-enoate.</p>Fórmula:C10H10O3Pureza:99.68% - 99.97%Forma y color:White Crystal PowderPeso molecular:178.18Cinchonine
CAS:<p>Cinchonine (LA40221), a potent amide local anesthetic for surface use, is toxic and limited to spinal anesthesia.</p>Fórmula:C19H22N2OPureza:99.45%Forma y color:White Or Almost White Solid PowderPeso molecular:294.39Tigatuzumab
CAS:<p>Tigatuzumab (CS-1008) is a humanized monoclonal antibody targeting DR5 and is a TRAIL-R2 agonist with antitumor activity that induces apoptosis in cancer cells.</p>Pureza:98.9% (SDS-PAGE); 96.6% (SEC-HPLC) - 98.9% (SDS-PAGE); 96.6% (SEC-HPLC)Forma y color:LiquidPeso molecular:144.6 (kDa)1,8,9-Trihydroxy-3-methoxy-6H-benzofuro[3,2-c][1]benzopyran-6-one
CAS:Fórmula:C16H10O7Pureza:98%Forma y color:SolidPeso molecular:314.2464Dostarlimab
CAS:<p>Dostarlimab (TSR-042) is an immune checkpoint inhibitor targeting PD-1, blocking its interaction with its ligands PD-L1 and PD-L2.</p>Pureza:>95%Forma y color:Liquid(2E)-3-[(4-Methylbenzene)sulfonyl]prop-2-enenitrile
CAS:Fórmula:C10H9NO2SPureza:98%Forma y color:SolidPeso molecular:207.2490Eragidomide
CAS:<p>Eragidomide (Cereblon modulator 1) is a CRBN E3 ligase modulator, specifically binds to CRBN, thereby affecting the activity of the ubiquitin E3 ligase complex.</p>Fórmula:C22H18ClF2N3O4Pureza:97.51% - 99.63%Forma y color:SolidPeso molecular:461.85Lomefloxacin hydrochloride
CAS:<p>Lomefloxacin hydrochloride (Okacyn) is a fluoroquinolone that inhibits DNA replication in bacteria, causing cell death.</p>Fórmula:C17H20ClF2N3O3Pureza:99.43% - 99.75%Forma y color:White PowderPeso molecular:387.81Bax inhibitor peptide V5 acetate
<p>Bax inhibitor peptide V5 acetate (Bax inhibitor peptide V5 acetate（579492-81-2 free base)) is a Bax-mediated apoptosis inhibitor, used for cancer treatment.</p>Fórmula:C29H54N6O8SPureza:99.2%Forma y color:SolidPeso molecular:646.85Azilsartan
CAS:<p>Azilsartan (TAK-536) is an Angiotensin II Type 1 receptor antagonist that lowers blood pressure.</p>Fórmula:C25H20N4O5Pureza:99.35% - 99.62%Forma y color:SolidPeso molecular:456.45Phenol, 2-methoxy-5-[(1Z)-2-(3,4,5-trimethoxyphenyl)ethenyl]-
CAS:Fórmula:C18H20O5Pureza:98%Forma y color:SolidPeso molecular:316.3484GLYCINE, N-[(3Α,5Β,12Α)-3,12-DIHYDROXY-24-OXOCHOLAN-24-YL]-, SODIUM SALT (1:1)
CAS:Fórmula:C26H42NNaO5Pureza:98%Forma y color:SolidPeso molecular:471.6051Amiloride hydrochloride
CAS:<p>Amiloride hydrochloride (Amiloride HCl) 是上皮钠通道和尿激酶型纤溶酶原激活物受体的抑制剂，也是 polycystin-2通道阻断剂。</p>Fórmula:C6H9Cl2N7OPureza:99.72% - 99.95%Forma y color:Physical Description Crystalline Solid Or Very Light Yellow Powder (Ntp 1992)Peso molecular:266.09Tioxolone
CAS:<p>Tioxolone is a metalloenzyme carbonic anhydrase I inhibitor.</p>Fórmula:C7H4O3SPureza:97.79%Forma y color:Light Yellow To Beige PowderPeso molecular:168.17Chlorhexidine diacetate
CAS:<p>Chlorhexidine diacetate (Bactigras) is a disinfectant and topical anti-infective agent used also as mouthwash to prevent oral plaque.</p>Fórmula:C26H38Cl2N10O4Pureza:99.61% - 99.69%Forma y color:White To Pale Yellow PowderPeso molecular:625.55IMB-XH1
CAS:<p>IMB-XH1 (Mcl1-IN-2) is a myeloid cell factor 1 (Mcl-1) inhibitor.</p>Fórmula:C19H15N3OSPureza:98%Forma y color:SolidPeso molecular:333.41Lucatumumab
CAS:<p>Lucatumumab (HCD122) is a fully human anti-CD40 monoclonal antibody with anti-tumor activity for the study of multiple myeloma.</p>Pureza:95.5% (SDS-PAGE); 98.4% (SEC-HPLC) - 95.5% (SDS-PAGE); 98.4% (SEC-HPLC)Forma y color:LiquidIrbesartan
CAS:<p>Irbesartan (SR-47436) is an Angiotensin 2 Receptor Blocker. The mechanism of action of irbesartan is as an Angiotensin 2 Receptor Antagonist.</p>Fórmula:C25H28N6OPureza:99.79% - 99.81%Forma y color:White Crystalline PowderPeso molecular:428.53Nortriptyline hydrochloride
CAS:<p>Nortriptyline HCl, a metabolite of amitriptyline, treats major and atypical depression, dysthymia.</p>Fórmula:C19H22ClNPureza:99.85% - ≥95%Forma y color:SolidPeso molecular:299.844-[1-(5,6,7,8-Tetrahydro-3,5,5,8,8-pentamethyl-2-naphthalenyl)ethenyl]benzoic acid
CAS:Fórmula:C24H28O2Pureza:95%Forma y color:SolidPeso molecular:348.4779Ref: IN-DA00389U
1g253,00€10gA consultar1mg39,00€25gA consultar50gA consultar10mg49,00€50mg52,00€250mg111,00€Zonisamide
CAS:<p>Zonisamide (AD 810), a sulfonamide anticonvulsant, is approved for use as an adjunctive treatment in adults with partial-onset seizures.</p>Fórmula:C8H8N2O3SPureza:99.05% - 99.9%Forma y color:Off-White PowderPeso molecular:212.23Acetylcysteine
CAS:<p>Acetylcysteine (NAC) is an N-acetyl derivative of cysteine, a ROS inhibitor and mucolytic agent.</p>Fórmula:C5H9NO3SPureza:98.01% - >99.99%Forma y color:Crystals From Water SolidPeso molecular:163.19Lidocaine hydrochloride
CAS:<p>Lidocaine HCl: local anesthetic, antiarrhythmic, stronger & longer-lasting than procaine but shorter than bupivacaine/prilocaine.</p>Fórmula:C14H23ClN2OPureza:99.81% - 99.92%Forma y color:White Crystal PowderPeso molecular:270.798Adenosine
CAS:<p>Adenosine (D-Adenosine) is a ribonucleoside. Adenosine has vasodilatory, antiarrhythmic and analgesic effects. Cost-effective and quality-assured.</p>Fórmula:C10H13N5O4Pureza:98.76% - 99.86%Forma y color:Needles (From Water +3/2) Physical Description White To Off-White Crystalline Powder (Ntp 1992)Peso molecular:267.24Hydralazine hydrochloride
CAS:<p>Hydralazine hydrochloride, an antihypertensive phthalazine, induces vasodilation and may inhibit tumor DNA methylation.</p>Fórmula:C8H9ClN4Pureza:99.85% - 99.86%Forma y color:Yellow Crystals White Crystalline SolidPeso molecular:196.64Diclofenac sodium
CAS:<p>Diclofenac sodium (GP 45840) is a non-steroidal anti-inflammatory agent (NSAID) with antipyretic and analgesic actions.</p>Fórmula:C14H10Cl2NNaO2Pureza:98.21% - 99.73%Forma y color:White Or Off-White PowderPeso molecular:318.13Amcinonide
CAS:<p>Amcinonide (CL-34699) is a Corticosteroid. The mechanism of action of amcinonide is as a Corticosteroid Hormone Receptor Agonist.</p>Fórmula:C28H35FO7Pureza:98.33% - 99.62%Forma y color:SolidPeso molecular:502.5717-ODYA
CAS:<p>17-ODYA (Alkynyl Stearic Acid) is an alkyl chain-based PROTAC linker that can be used in the synthesis of PROTACs.</p>Fórmula:C18H32O2Pureza:98.21%Forma y color:SolidPeso molecular:280.452-Butenamide, 2-cyano-N-(2,5-dibromophenyl)-3-hydroxy-
CAS:Fórmula:C11H8Br2N2O2Pureza:98%Forma y color:SolidPeso molecular:360.0014Metronidazole
CAS:<p>Metronidazole (Metronidazol) is a synthetic nitroimidazole derivative with antiprotozoal and antibacterial activities.</p>Fórmula:C6H9N3O3Pureza:99.46% - 99.96%Forma y color:Cream-Colored CrystalsPeso molecular:171.15Amrinone
CAS:<p>Amrinone (Inocor) is a positive inotropic cardiotonic (cardiotonic agent) with vasodilator properties, phosphodiesterase 3 inhibitory activity.</p>Fórmula:C10H9N3OPureza:98.88% - 99.45%Forma y color:SolidPeso molecular:187.2Gefitinib
CAS:<p>Gefitinib (ZD1839) is an EGFR first-generation inhibitor with oral activity that inhibits the EGFR 19 Del and L858R mutations.</p>Fórmula:C22H24ClFN4O3Pureza:99.92% - >99.99%Forma y color:Light-Yellow Crystalline PowderPeso molecular:446.9Ecabet Sodium
CAS:<p>Ecabet Sodium (TA-2711) is a potential new agent in the management of distal colitis.</p>Fórmula:C20H27NaO5SPureza:99.90%Forma y color:SolidPeso molecular:402.48Hexylresorcinol
CAS:<p>Hexylresorcinol (4-Hexylresorcinol) is a substituted dihydroxybenzene used topically as an antiseptic for the treatment of minor skin infections.</p>Fórmula:C12H18O2Pureza:99.26% - 99.51%Forma y color:Solid Solid Particulate/PowderPeso molecular:194.27Gemcitabine
CAS:<p>Gemcitabine (LY188011) is a synthetic cytosine nucleoside derivative and an inhibitor of DNA synthesis.</p>Fórmula:C9H11F2N3O4Pureza:98.66% - 99.67%Forma y color:SolidPeso molecular:263.2Fenobam
CAS:Fenobam shows inverse agonist activity which blocks the mGlu5 receptor basal activity(IC50: 84 nM).Fórmula:C11H11ClN4O2Pureza:99.93%Forma y color:SolidPeso molecular:266.68Bergenin
CAS:<p>Bergenin (Bengenin) is a polyphenol, which is an effective antinarcotic agent with antioxidant action.</p>Fórmula:C14H16O9Pureza:99.55% - 99.60%Forma y color:The Loose White Needle Crystal Powder Or CrystallinePeso molecular:328.27Dipyridamole
CAS:<p>Dipyridamole (Persantin) is a Platelet Aggregation Inhibitor. The physiologic effect of dipyridamole is by means of Decreased Platelet Aggregation.</p>Fórmula:C24H40N8O4Pureza:99.47% - 99.84%Forma y color:SolidPeso molecular:504.63Trifluridine
CAS:<p>Trifluridine is a fluorinated thymidine analog with antineoplastic and antiviral properties, disrupting DNA and protein synthesis, leading to apoptosis.</p>Fórmula:C10H11F3N2O5Pureza:99.39% - 99.82%Forma y color:White Crystalline PowderPeso molecular:296.2Tegaserod maleate
CAS:<p>Tegaserod (SDZ-HTF-919), a 5-HT4 agonist for irritable bowel syndrome, was withdrawn by FDA on March 30, 2007, due to heart risk concerns.</p>Fórmula:C20H27N5O5Pureza:98% - 99.06%Forma y color:White PowderPeso molecular:417.46N-Oleoyl-L-Serine
CAS:<p>N-Oleoyl-L-Serine (N-Oleoylserine) is a lipid modulator of bone remodeling and stimulates osteoclast apoptosis for the study of osteoporosis.</p>Fórmula:C21H39NO4Pureza:99.76%Forma y color:SolidPeso molecular:369.54Pranoprofen
CAS:<p>Pranoprofen (Pyranoprofen) (INN) is a non-steroidal anti-inflammatory drug used in ophthalmology.</p>Fórmula:C15H13NO3Pureza:97.98% - 99.85%Forma y color:SolidPeso molecular:255.27Mevastatin
CAS:<p>Mevastatin (ML236B) is an HMG-CoA reductase inhibitor that was initially isolated from the mold Pythium ultimum.</p>Fórmula:C23H34O5Pureza:99.12%Forma y color:White-Yellowish To Yellow Powder Solid PowderPeso molecular:390.51Lenalidomide
CAS:<p>Lenalidomide (CC-5013) is an orally immunomodulator. Lenalidomide is a ligand for the ubiquitin E3 ligase cereblon (CRBN). Cost-effective and quality-assured.</p>Fórmula:C13H13N3O3Pureza:98% - 99.97%Forma y color:Yellow SolidPeso molecular:259.26Benufutamab
CAS:<p>Benufutamab (GEN1029) is an agonistic antibody targeting death receptor 5 (DR5) with anti-tumor activity, used in the study of solid tumors.</p>Pureza:98.6% (SEC-HPLC) - 98.62% (SEC-HPLC)Forma y color:LiquidMyricetin
CAS:<p>Myricetin (Cannabiscetin) is a natural flavonoid and MEK1 inhibitor. Myricetin has hypoglycemic and antioxidant activities. Cost-effective and quality-assured.</p>Fórmula:C15H10O8Pureza:97.92% - 99.85%Forma y color:Yellow Needles From Dilute Alcohol SolidPeso molecular:318.24Temozolomide
CAS:<p>Temozolomide (TMZ) is a DNA alkylating agent with blood-brain barrier permeability and oral activity.</p>Fórmula:C6H6N6O2Pureza:98% - 99.87%Forma y color:Off-White To Light-Pink Crystalline SolidPeso molecular:194.15Oxaliplatin
CAS:<p>Oxaliplatin (L-OHP) is a DNA alkylating agent, an inhibitor of DNA synthesis.</p>Fórmula:C8H14N2O4PtPureza:97% - 99.93%Forma y color:SolidPeso molecular:397.29YS-67
CAS:<p>YS-67 is an orally available, selective and potent EGFR inhibitor with antitumor activity, inhibits p-EGFR and p-AKT, and inhibits the proliferation of A549, PC-9, and A431 cells.YS-67 blocks cell cycle progression and induces apoptosis in the G0/G1 phase, and can be used in the study of non-small-cell lung cancer.</p>Fórmula:C32H34N4O3Pureza:98.88%Forma y color:SoildPeso molecular:522.64Propafenone
CAS:<p>Propafenone: a drug for ventricular arrhythmias with mild beta-blocker activity, prolongs refractory period, and reduces heart automaticity.</p>Fórmula:C21H27NO3Pureza:99.02%Forma y color:SolidPeso molecular:341.44Levetiracetam
CAS:<p>Levetiracetam (SIB-S1) is a relatively unique anticonvulsant that is typically used in combination with other antiepileptic medications for partial onset</p>Fórmula:C8H14N2O2Pureza:99.67% - 99.86%Forma y color:White Crystalline PowderPeso molecular:170.21Risedronic Acid
CAS:<p>Risedronic Acid (Risedronate), a pyridinyl biphosphonate, can inhibit osteoclast-mediated bone resorption.</p>Fórmula:C7H11NO7P2Pureza:99.85% - 99.87%Forma y color:White Crystalline PowderPeso molecular:283.119H-Xanthene-4-aceticacid, 5,6-dimethyl-9-oxo-
CAS:Fórmula:C17H14O4Pureza:98%Forma y color:SolidPeso molecular:282.2907Ref: IN-DA0035WP
1g205,00€5gA consultar10gA consultar25gA consultar50gA consultar5mg37,00€25mg54,00€100mg72,00€250mg108,00€Formononetin
CAS:<p>Formononetin (Flavosil) is an O-methylated isoflavone and a phytoestrogen from the root of Astragalus membranaceus.</p>Fórmula:C16H12O4Pureza:97.39% - 99.94%Forma y color:SolidPeso molecular:268.26GPNA hydrochloride
CAS:<p>GPNA hydrochloride inhibits Gln transporter ASCT2, induces apoptosis in A549 cells, blocks SNAT1/2/4/5 & LAT1/2 transporters, and is a GGT substrate.</p>Fórmula:C11H14ClN3O5Pureza:99.13%Forma y color:SolidPeso molecular:303.7AUNP-12 acetate
<p>AUNP-12 acetate is a polypeptide inhibitor of PD-1 that is equivalent to PD-1 and PD-2 in inhibiting lymphocyte proliferation and effector fuction, in addition</p>Fórmula:C144H230N40O50Pureza:95.07%Forma y color:SolidPeso molecular:3321.61α-Lipoic Acid
CAS:<p>α-Lipoic Acid, a sulfur-containing octanoic acid derivative, is biosynthesized from linoleic acid and used in dietary supplements.</p>Fórmula:C8H14O2S2Pureza:98.39% - 99.73%Forma y color:Forms Yellowish Flakes Light Yellow To Yellow PowderPeso molecular:206.33Tamoxifen
CAS:<p>Tamoxifen is an orally active selective estrogen receptor modulator (SERM) that acts as an estrogen antagonist in breast cells and an agonist in bone, liver, and uterine cells. It can be used to induce gene knockout and liver injury models in mice, and also exhibits multiple biological activities, including activation of Hsp90, induction of autophagy and apoptosis, and inhibition of EBOV and MARV viral infections.</p>Fórmula:C26H29NOPureza:98.46% - 99.92%Forma y color:Fine Off-White Crystalline PowderPeso molecular:371.51Moroxydine hydrochloride
CAS:<p>Moroxydine hydrochloride (ABOB hydrochloride) is a synthetic antiviral drug chemically belonging to the series of the heterocyclic biguanidines.</p>Fórmula:C6H13N5O·HClPureza:99.15%Forma y color:White Crystalline PowderPeso molecular:207.66Dantrolene sodium
CAS:<p>Dantrolene sodium treats spasticity by disrupting muscle contraction; not central in action, grouped with central relaxants.</p>Fórmula:C14H9N4NaO5Pureza:98% - 99.87%Forma y color:CoaPeso molecular:336.23Spartalizumab
CAS:<p>"Spartalizumab (PDR001), a humanized IgG4 monoclonal antibody, targets PD-1 to inhibit PD-L1/L2 interactions, useful in ATC research."</p>Pureza:SDS-PAGE:95.2%;SEC-HPLC:96.3%Forma y color:LiquidPeso molecular:145.74 kDaInavolisib
CAS:<p>Inavolisib (GDC-0077) is an orally available selective PI3Kα inhibitor with an IC50 value of 0.038 nM.Cost-effective and quality-assured.</p>Fórmula:C18H19F2N5O4Pureza:97.36% - 99.87%Forma y color:SolidPeso molecular:407.37ZX-29
CAS:<p>ZX-29: Strong ALK inhibitor; IC50 - ALK 2.1 nM, L1196M 1.3 nM, G1202R 3.9 nM; triggers autophagy; anti-cancer.</p>Fórmula:C23H28ClN7O3SPureza:98.32%Forma y color:SolidPeso molecular:518.03CITCO
CAS:<p>CITCO, an imidazothiazole, selectively inhibits BTSCs growth with 49 nM EC50 on PXR and is a CAR agonist.</p>Fórmula:C19H12Cl3N3OSPureza:99.24%Forma y color:SolidPeso molecular:436.74Pranlukast
CAS:<p>Pranlukast (ONO-1078) is a cysteinyl leukotriene receptor-1 antagonist.</p>Fórmula:C27H23N5O4Pureza:99.41%Forma y color:Off-White SolidPeso molecular:481.5Deracoxib
CAS:<p>Deracoxib (SC 46) is a selective COX-2 inhibitor, non-steroidal, non-narcotic anti-inflammatory drug with an IC50 of 70-150 μM for osteosarcoma cells.</p>Fórmula:C17H14F3N3O3SPureza:98.94% - 99.81%Forma y color:SolidPeso molecular:397.37AZD4320
CAS:<p>AZD4320 inhibits BCL2/BCLxL; IC50: KPUM-MS3=26nM, KPUM-UH1=17nM, STR-428=170nM.</p>Fórmula:C45H48ClF3N4O7S3Pureza:98.13% - 99.71%Forma y color:SolidPeso molecular:945.534-(4-Fluorophenyl)-2-(4-methylsulfinylphenyl)-5-(4-pyridyl)-1H-imidazole
CAS:Fórmula:C21H16FN3OSPureza:98%Forma y color:SolidPeso molecular:377.4346Ref: IN-DA003K1L
1gA consultar5mg50,00€25mg105,00€50mg139,00€100mg157,00€250mg488,00€500mgA consultarClofilium tosylate
CAS:<p>Clofilium tosylate is a potassium channel blocker, induces apoptosis on human promyelocytic leukemia (HL-60) cells.</p>Fórmula:C28H44ClNO3SPureza:99.68%Forma y color:SolidPeso molecular:510.17NBDHEX
CAS:<p>NBDHEX is a potent inhibitor of glutathione S-transferase P1-1 (GSTP1-1).</p>Fórmula:C12H15N3O4SPureza:97.38%Forma y color:SolidPeso molecular:297.33Sodium diatrizoate
CAS:<p>Sodium diatrizoate is an X-ray contrast medium for angiography, urography; may cause oxidative stress and apoptosis.</p>Fórmula:C11H8I3N2NaO4Pureza:99.29% - 99.96%Forma y color:SolidPeso molecular:635.9Clofarabine
CAS:<p>Clofarabine (Clofarex)m, a second generation purine nucleoside analog with antineoplastic activity, inhibits the enzymatic activities of ribonucleotide</p>Fórmula:C10H11ClFN5O3Pureza:99.94% - >99.99%Forma y color:White SolidPeso molecular:303.68Cusatuzumab
CAS:<p>Cusatuzumab (ARGX-110) is a human CD70 monoclonal antibody with enhanced antibody-dependent cytotoxic activity.</p>Pureza:95% - 95%Forma y color:LiquidLevonorgestrel
CAS:<p>Levonorgestrel (D-Norgestrel) is a Progestin and Progestin-containing Intrauterine Device.</p>Fórmula:C21H28O2Pureza:99.42% - 99.44%Forma y color:Crystals From Methanol SolidPeso molecular:312.45Iproniazid Phosphate
CAS:<p>Iproniazid Phosphate is a non-selective, irreversible monoamine oxidase inhibitor (MAOI).</p>Fórmula:C9H13N3O·H3PO4Pureza:99.6% - 99.87%Forma y color:SolidPeso molecular:277.211(3H)-Isobenzofuranone, 6,7-dimethoxy-3-[(5R)-5,6,7,8-tetrahydro-4-methoxy-6-methyl-1,3-dioxolo[4,5-g]isoquinolin-5-yl]-, hydrochloride (1:1), (3S)-
CAS:Fórmula:C22H24ClNO7Pureza:98%Forma y color:SolidPeso molecular:449.8815L-Leucinamide, N-[(phenylmethoxy)carbonyl]-L-leucyl-N-[(1S)-1-formyl-3-methylbutyl]-
CAS:Fórmula:C26H41N3O5Pureza:98%Forma y color:SolidPeso molecular:475.6208Ref: IN-DA0072SK
1gA consultar5mg68,00€10mg90,00€25mg124,00€50mg168,00€100mg229,00€250mg500,00€500mgA consultarMIM1
CAS:<p>MIM1 (Inhibitor of Mcl-1) is an myeloid cell factor 1 (Mcl-1) inhibitor.</p>Fórmula:C17H21N3O3SPureza:99.84%Forma y color:SolidPeso molecular:347.43Sterigmatocystine
CAS:<p>Sterigmatocystine, a G1 phase and DNA synthesis inhibitor, curbs p21 and is a mycotoxin precursor from Aspergillus versicolor.</p>Fórmula:C18H12O6Pureza:98%Forma y color:Pale-Yellow Crystals Pale Yellow SolidPeso molecular:324.28F1324 acetate
<p>F1324 acetate is an efficient, high-affinity b-cell lymphoma inhibitor with IC50 of 1 nM.</p>Fórmula:C85H125N21O22SPureza:98%Forma y color:SolidPeso molecular:1825.09Episilvestrol
CAS:<p>Episilvestrol is a derivative of silvestrol with eIF4A-targeted antitumor properties, found in Aglaia silvestris fruits and twigs.</p>Fórmula:C34H38O13Pureza:98%Forma y color:SolidPeso molecular:654.66mTOR inhibitor-27
<p>mTORinhibitor-27 (Compound 7e) is an inhibitor of mammalian target of rapamycin (mTOR) with an IC50 value of 5.47 μM. It can induce apoptosis in tumor cells and arrest the cell cycle in the S phase, thereby inhibiting cancer cell growth. mTORinhibitor-27 presents potential for research in cancer, including skin cancer.</p>Forma y color:Odour SolidDeoxynyboquinone
CAS:<p>Deoxynyboquinone is a potent inducer of cancer cell death with IC(50) values between 16 and 210 nM.</p>Fórmula:C15H12N2O4Pureza:98%Forma y color:SolidPeso molecular:284.27rac-CCT-250863 HCl
<p>rac-CCT-250863 HCl: NEK 2 inhibitor, halts cell cycle, anti-cancer growth, boosts Pomalidomide-induced apoptosis.</p>Fórmula:C24H26ClF3N4O2SPureza:98.21%Forma y color:SoildPeso molecular:527KWCN-41
CAS:<p>KWCN-41, a RIPK1 inhibitor with 88 nM IC50, blocks necrosis, spares apoptosis, and is anti-inflammatory.</p>Fórmula:C18H17N3O2Forma y color:SolidPeso molecular:307.35Psalmotoxin 1
CAS:<p>Psalmotoxin 1 is a potent and selective acid-sensing ion channel 1a (ASIC1a) blocker.</p>Fórmula:C200H312N62O57S6Pureza:98%Forma y color:SolidPeso molecular:4689.41SP3N hydrochloride
<p>SP3N hydrochloride is a specific degrader of the prolyl isomerase (FKBP12). Its alkylamine moiety is metabolized into an active aldehyde (SP3CHO), which recruits the SCFFBXO22 ligase for the degradation of FKBP12. SP3N hydrochloride is applicable in cancer research.</p>Forma y color:Odour SolidSuramin
CAS:<p>Suramin is an RdRp and PTPase inhibitor with anti-parasitic, anti-tumor, and anti-angiogenic activities, inhibiting sirtuins and DNA topoisomerase II.</p>Fórmula:C51H40N6O23S6Pureza:99.80%Forma y color:SolidPeso molecular:1297.28SDH-IN-26
<p>SDH-IN-26 (Compound C3) is a succinate dehydrogenase (SDH) inhibitor with significant inhibitory activity against various plant pathogenic fungi, including solanrhizoctonia and Botrytis cinerea. It exhibits an EC50 value of 0.270 μg/mL against solanrhizoctonia. SDH-IN-26 compromises fungal cell membrane integrity, increases membrane permeability, disrupts cell structure, reduces mitochondrial count, and affects normal hyphal growth. It also decreases mitochondrial membrane potential, inducing apoptosis. SDH-IN-26 holds potential for studying plant diseases caused by fungi.</p>Forma y color:Odour SolidMG-277
<p>MG-277 is a molecular glue compound transformed from PROTAC degradation agent, MG-277 potently inhibits tumor cell growth in a p53-independent manner.</p>Fórmula:C41H42Cl2FN5O5Pureza:98%Forma y color:SolidPeso molecular:774.71PL120131
<p>PL120131 is a PD-1/PD-L1 inhibitory peptide that disrupts the interaction between PD-1 and PD-L1 by binding to PD-1. This compound can inhibit the apoptosis signaling pathway mediated by PD-1, thereby preventing apoptosis (apoptosis) in Jurkat cells and primary lymphocytes. Additionally, PL120131 supports cytotoxic T lymphocytes (CTL) in exhibiting antitumor activity.</p>Fórmula:C62H105N19O18Forma y color:SolidPeso molecular:1404.61RIPK3-IN-3
<p>RIPK3-IN-3 (compound 20) is a selective RIPK3 inhibitor that demonstrates potent activity with an IC50 value of 10 nM.</p>Fórmula:C16H11N5SForma y color:SolidPeso molecular:305.36(±)-Enterodiol
CAS:<p>"(±)-Enterodiol, the racemate of Enterodiol, is metabolized from lignans found in whole-grain cereals, nuts, legumes, flaxseed, and vegetables by human intestinal bacteria. This compound exhibits apoptotic effects in colorectal cancer (CRC) cells and has been identified to possess anti-cancer activities [1] [2]."</p>Fórmula:C18H22O4Forma y color:SolidPeso molecular:302.36Pantoprazole Sodium Hydrate
CAS:<p>Pantoprazole Sodium Hydrate (BY1023 (sodium hydrate)) is a proton pump inhibitor drug, used for short-term treatment of erosion and ulceration of the esophagus</p>Fórmula:C16H14F2N3NaO4SH2OPureza:98.32%Forma y color:SolidPeso molecular:432.37MAO-B-IN-30
CAS:<p>MAO-B-IN-30 is a selective and potent MAO-B inhibitor that crosses the blood-brain barrier with antiproliferative activity and inhibits both MAO-A and MAO-B.MAO-B-IN-30 reduces the levels of TNF-alpha, IL-6, and NF-kB in organisms, and can be used to study Parkinson's-type neurological disorders.</p>Fórmula:C15H10BrN3O2Pureza:98.31%Forma y color:SoildPeso molecular:344.16CYP51/PD-L1-IN-4
<p>CYP51/PD-L1-IN-4 (compound 14a-2) is a potent dual-target inhibitor of CYP51/PD-L1, displaying IC50 values of 0.17 and 0.021 μM, respectively.</p>Fórmula:C27H28N4O3Forma y color:SolidPeso molecular:456.54PG-11047 2HCl
<p>PG-11047 2HCl treats genitourinary, immune, genetic, ocular, blood/lymphatic disorders, and aids lymphoma/prostate cancer research.</p>Fórmula:C14H34Cl2N4Pureza:97.47%Forma y color:SolidPeso molecular:329.35Kdo2-Lipid A ammonium
CAS:<p>Kdo2-Lipid A ammonium (KLA) is a selective and potent TLR4 agonist, a lipopolysaccharide.Kdo2-Lipid A ammonium induces the release of TNF and PGE2.</p>Fórmula:C110H214N6O39P2Pureza:98%Forma y color:SolidPeso molecular:2306.84APG-1387
CAS:<p>APG-1387 inhibits IAPs, degrades cIAP1/2, XIAP, boosts chemosensitivity, and induces apoptosis in NPC.</p>Fórmula:C60H72N10O10S2Forma y color:SolidPeso molecular:1157.41Dynorphin A
CAS:<p>Dynorphin A is a endogenous opioid peptide and a κ-opioid receptor (KOR) agonist,a neurotransmitter and regulator in the central and peripheral nervous systems</p>Fórmula:C99H155N31O23Pureza:95.93%Forma y color:SolidPeso molecular:2147.48PROTAC Bcl2 degrader-1
CAS:<p>PROTAC Bcl2 degrader-1 is a PROTAC, which potently and selectively induces the degradation of Mcl-1 (IC50: 11.81 μM) and Bcl-2 (IC50: 4.94 μM; DC50: 3.0 μM).</p>Fórmula:C45H45BrN6O10SPureza:98%Forma y color:SolidPeso molecular:941.84Dapirolizumab
<p>Dapirolizumab is an anti-CD40 monoclonal antibody used in research on systemic lupus erythematosus (SLE) and other autoimmune diseases.</p>Pureza:>95%Forma y color:LiquidPeso molecular:145.5 kDaAS-99 free base
CAS:<p>AS-99 is a first-in-class, potent and selective ASH1L histone methyltransferase inhibitor (IC50= 0.79 μM, Kd= 0.89 μM) with anti-leukemic activity.</p>Fórmula:C27H30F3N5O3S2Forma y color:SolidPeso molecular:593.68(-)-Mcl-1 inhibitor 21
CAS:<p>(-)-Mcl-1 inhibitor 21 (Example 1-38) is an Mcl-1 inhibitor with an IC50 of 7.51 μM. It exhibits pro-apoptotic and anti-proliferative activity against SUDHL5 and SUDHL10 cell lines, making it useful for cancer research.</p>Fórmula:C32H33N3O4Forma y color:SolidPeso molecular:523.622KH16
<p>KH16 is an HDAC inhibitor.KH16 stimulates apoptosis and is able to inhibit gene expression patterns in a variety of tumor cells.</p>Fórmula:C18H20N6O2Pureza:98.15%Forma y color:SolidPeso molecular:352.39TD1092
<p>TD1092, a pan-IAP degrader, activates caspase 3/7, induces apoptosis in cancer cells, inhibits NF-κB, and is used in cancer research.</p>Fórmula:C55H70N8O9Forma y color:SolidPeso molecular:987.19CAY10678
CAS:<p>CAY10678 is an mPGES-1 inhibitor that inhibits PD-1.CAY10678 reduces collagen deposition and T-cell depletion, and may be used to study melanoma.CASHIPS</p>Fórmula:C23H34N4OPureza:99.66%Forma y color:SolidPeso molecular:382.54HEMTAC CDK4/6 degrader 1
CAS:<p>HEMTAC CDK4/6 degrader 1, a PROTAC targeting HSP90/CDK4/6, Kd of 35.7 μM, disrupts B16F10 melanoma cell cycle, and induces apoptosis.</p>Fórmula:C48H53ClN16O4Forma y color:SolidPeso molecular:953.49Delmitide
CAS:<p>Delmitide, a TNF-alpha production inhibitor, is used potentially for the treatment of Crohn's disease and ulcerative colitis.</p>Fórmula:C59H105N17O11Pureza:98%Forma y color:SolidPeso molecular:1228.57Thalidomide-O-amido-C3-COOH
CAS:<p>Thalidomide-O-amido-C3-COOH is a cereblon ligand-linker for PROTACs, melding Thalidomide with a standard linker.</p>Fórmula:C19H19N3O8Pureza:98%Forma y color:SolidPeso molecular:417.37BODIPY FL thalidomide
CAS:<p>BODIPY FL thalidomide is a fluorescent probe that binds human cereblon protein with high affinity, exhibiting a dissociation constant (Kd) of 3.6 nM [1].</p>Fórmula:C37H43BF2N6O7Forma y color:SolidPeso molecular:732.58Thalidomide-Piperazine 5-fluoride hydrochloride
CAS:<p>Thalidomide-Piperazine 5-fluoride hydrochloride, a derivative of the cereblon (CRBN) inhibitor Thalidomide, serves as a ligand for E3 ubiquitin ligase (Ligands for E3 Ligase), facilitating the synthesis of PROTACs [1].</p>Fórmula:C17H18ClFN4O4Forma y color:SolidPeso molecular:396.8Chlopynostat
<p>Chlopynostat (Compound 6c) is an HDAC1 inhibitor with an IC50 value of 67 nM. It induces apoptosis by inhibiting HDAC1, thereby reversing STAT4/p66Shc defects.</p>Fórmula:C22H17ClN4O2Peso molecular:404.104Beclin1-Bcl-2 interaction inhibitor 1
<p>Beclin1-Bcl-2 Interaction Inhibitor 1 effectively disrupts the binding of Beclin 1 to Bcl-2, and is utilized in cancer and neurodegeneration research [1].</p>Forma y color:Odour SolidEGFR-PK/JNK-2-IN-1
<p>EGFR-PK/JNK-2-IN-1 (Compound 6c) is a dual inhibitor of EGFR-PK and JNK-2, with IC50 values of 2.7 and 3.0 μM, respectively. It can induce apoptosis and cause cell cycle arrest at various stages. This compound is applicable in cancer research.</p>Fórmula:C22H17ClN4O3SPeso molecular:452.07099DA5-HTL
<p>DA5-HTL is a compound that combines dasatinib with the HaloTag system, effectively inhibiting the growth of tumor cells, with a GI50 of 1.923 nM.</p>Fórmula:C39H58Cl2N8O8SPeso molecular:868.34754WD6305
WD6305 is an effective and selective METTL3-METTL14 PROTAC degrader, with DC50 values of 140 nM and 194 nM for METTL3 and METTL14, respectively. It inhibits m6A modification and the proliferation of acute myeloid leukemia cells while inducing apoptosis. WD6305 also exhibits antitumor activity.Fórmula:C61H75F2N11O5SPeso molecular:1111.56414WEE1-IN-7
<p>WEE1-IN-7 (compound 12h) is a potent, orally active WEE1 inhibitor with an IC50 value of 2.1 nM. This compound induces apoptosis and causes cell cycle arrest in the S phase, demonstrating antitumor activity.</p>Topoisomerase II inhibitor 17
<p>TopoisomeraseII inhibitor 17 (compound 4c) is a thiazolopyrimidine-based inhibitor of Topoisomerase II with an IC50 of 0.23 μM. This compound significantly disrupts the cell cycle and induces apoptosis.</p>Fórmula:C25H22Cl3N3O5SPeso molecular:581.03458WK369
WK369 is an innovative small molecule inhibitor of BCL6, demonstrating remarkable bioactivity against ovarian cancer by inducing cell cycle arrest and triggering apoptosis. It binds directly to the BCL6-BTB domain, obstructing the interaction between BCL6 and SMRT, which results in the reactivation of p53, ATR, and CDKN1A.Fórmula:C19H20FN5O2Peso molecular:369.1601YX-02-030
CAS:<p>YX-02-030M is a PROTACMDM2 degrader. It inhibits the binding of MDM2 to p53 and VHL to HIF1α, with IC50 values of 63 nM and 1.35 μM, respectively. YX-02-030M binds to MDM2 and recruits the VHL E3 ubiquitin ligase to initiate MDM2 degradation, effectively killing p53 mutant or deficient triple-negative breast cancer (TNBC) cells.</p>Fórmula:C66H85Cl2N9O10SPeso molecular:1267.41PD-1/PD-L1-IN-48
<p>PD-1/PD-L1-IN-48 (compound HD10) is an effective inhibitor of the PD-1/PD-L1 interaction, exhibiting an IC50 of 3.1 nM. It plays a vital role in cancer research.</p>Forma y color:Odour SolidFR900359
CAS:<p>FR900359 is a macrocyclic Gq protein inhibitor that inhibits melanoma cell proliferation and can be used to study asthma, inflammation and cancer.</p>Fórmula:C49H75N7O15Pureza:98%Forma y color:SolidPeso molecular:1002.16BMSpep-57
CAS:<p>BMSpep-57: Macrocyclic peptide, inhibits PD-1/PD-L1, IC50=7.68 nM, binds PD-L1 (Kd=19 nM/MST, 19.88 nM/SPR), boosts T cell IL-2 in PBMCs.</p>Fórmula:C89H126N24O19SForma y color:SolidPeso molecular:1868.2CDC20-IN-2
<p>CDC20-IN-2 (14c) is an inhibitor of Cdc20 with a KD of 7.65 μM, inducing G2/M phase arrest, promoting DNA damage accumulation, and stabilizing key substrates such as Cyclin B1 and Bim. This leads to enhanced apoptosis, as well as inhibition of tumor cell proliferation and migration.</p>Forma y color:Odour SolidMKC-1
CAS:<p>MKC-1 (Ro-31-7453) is an oral bisindolylmaleimide inhibitor that disrupts tubulin polymerization, potentially halting cancer cell division.</p>Fórmula:C22H16N4O4Pureza:99.63% - 99.85%Forma y color:SolidPeso molecular:400.39FOXO4-DRI
CAS:<p>FOXO4-DRI: a peptide blocking FOXO4/p53 interaction; induces senescent cells' apoptosis.</p>Fórmula:C228H388N86O64Forma y color:SolidPeso molecular:5358.06d-(KLAKLAK)2, Proapoptotic Peptide
CAS:<p>d-(KLAKLAK)2 is an antimicrobial and antitumor peptide, notable within the group of antimicrobial peptides, and exhibits strong anticancer properties. It kills bacteria by disrupting their cell membranes, causing leakage of cell contents. Additionally, d-(KLAKLAK)2 inhibits tumor cell proliferation by inducing apoptosis through mitochondrial swelling and membrane damage.</p>Fórmula:C72H139N21O14Forma y color:SolidPeso molecular:1523.01Tubulin polymerization-IN-67
<p>Tubulin polymerization-IN-67 (Compound 5h) serves as an inhibitor of microtubule protein polymerization at the colchicine binding site, exhibiting an IC50 value of 2.92 μM. It effectively inhibits the proliferation of various cancer cell lines including HT29, A549, U2OS, MG-63, and HeLa, with IC50 values ranging from 0.12 to 4.13 μM. Additionally, Tubulin polymerization-IN-67 induces cell cycle arrest at the G2/M phase and triggers apoptosis in U2OS cells. It also inhibits cell migration in A549 and reduces mitochondrial membrane potential (MMP) while increasing intracellular ROS levels, thereby suppressing angiogenesis in HUVEC cells. Furthermore, this compound demonstrates antitumor activity in mice.</p>Forma y color:Odour SolidTrilexium
CAS:<p>Trilexium (TRX-E-009-1), a third-generation benzopyran structurally related to TRX-E-002-1, increases p21 protein expression, induces apoptosis, depolymerizes microtubules, and demonstrates broad anti-cancer activity [1] [2].</p>Fórmula:C24H23FO6Forma y color:SolidPeso molecular:426.43PBE-AMF
<p>PBE-AMF is a prodrug that activates H2O2 and exhibits anticancer activity. It impedes tumor proliferation by inhibiting DNA synthesis, reducing ATP levels, inducing cell death (apoptosis), and blocking the cell cycle. PBE-AMF effectively and selectively inhibits the proliferation of MDA-MB-231 cells (IC50=6.4 μM) while sparing non-cancerous MCF-10A cells.</p>Forma y color:Odour SolidNarasin (sodium salt)
CAS:<p>Narasin (sodium salt) (HainanMycin) induces tumor necrosis factor-related apoptosis-induced ligand (TRAIL)-mediated apoptosis by ER stress in glioma cells and</p>Fórmula:C43H71NaO11Pureza:98%Forma y color:SolidPeso molecular:787.01RLX HCl
CAS:<p>RLX HCl is anticancer, inhibits tumour proliferation by suppressing the PI3K/Akt/FoxO3a in experimental colon cancer, antiproliferative.</p>Fórmula:C13H15ClN2OPureza:99.43%Forma y color:SoildPeso molecular:250.72Ac-Trp-Glu-His-Asp-Aldehyde
CAS:<p>Ac-Trp-Glu-His-Asp-Aldehyde is a powerful and selective inhibitor of caspase-1, demonstrating a K_i value of 56 pM [1] [2].</p>Fórmula:C28H33N7O9Forma y color:SolidPeso molecular:611.6Mepacrine
CAS:<p>Mepacrine (Erion) is an acridine derivative formerly widely used as an antimalarial.</p>Fórmula:C23H30ClN3OPureza:98.78%Forma y color:Bright Yellow CrystalsPeso molecular:399.96FL118
CAS:<p>FL118 is a novel survivin inhibitor that inhibits cancer stem cell-like properties.FL118 is a novel camptothecin analog with anticancer activity that inhibits</p>Fórmula:C21H16N2O6Pureza:98.99%Forma y color:SoildPeso molecular:392.36TRAP1-IN-1
CAS:<p>TRAP1-IN-1 is a selective TRAP1 inhibitor, induces degradation of TRAP1 downstream proteins, inhibits OXPHOS, and disrupts mitochondrial membrane potential.</p>Fórmula:C45H39F7N2O4P2Pureza:98%Forma y color:SolidPeso molecular:866.74CDK2-IN-45
<p>CDK2-IN-45 is a CDK2 inhibitor with an IC50 value of 0.64 μM. It effectively inhibits the proliferation of DU-145 and PC-3 cell lines, with IC50 values of 2.20 μM and 4.17 μM, respectively. Additionally, CDK2-IN-45 induces G0/G1 phase cell cycle arrest and apoptosis. It is utilized in prostate cancer research.</p>Fórmula:C25H16ClN5SForma y color:SolidPeso molecular:453.95Thalidomide-O-amido-PEG1-(C1-PEG)2-C2-NH2
<p>Thalidomide-PEG conjugate for E3 ligase in PROTACs; has cereblon ligand and 3-unit PEG linker.</p>Fórmula:C27H35F3N4O11Pureza:98%Forma y color:SolidPeso molecular:648.58PAK4-IN-3
<p>PAK4-IN-3 (compound 27e) is a PAK4 inhibitor exhibiting an IC50 of 10 nM and demonstrates antiproliferative effects on A549 cells with an IC50 of 0.61μM.</p>Pureza:98%Forma y color:Odour SolidCot inhibitor-1 hydrochloride
<p>Cot inhibitor-1 hydrochloride blocks TPL-2 kinase (IC50=28nM) and TNF-α synthesis (IC50=5.7nM) in human blood.</p>Fórmula:C27H28Cl3FN8Pureza:98.26%Forma y color:SoildPeso molecular:589.92cpm-1285
CAS:<p>CPM-1285 induces apoptosis by effectively inhibiting the function of intracellular Bcl-2 and associated death antagonists.</p>Fórmula:C153H240N44O42SPureza:98%Forma y color:SolidPeso molecular:3399.88Ferroptosis-IN-17
<p>Ferroptosis-IN-17 (Compound 18) is an inhibitor of ferroptosis with an EC50 value of 0.57 μM. It effectively reduces the accumulation of intracellular ferrous ions and lipid peroxidation while restoring levels of glutathione (GSH) and glutathione peroxidase 4 (GPX4). In rat plasma, Ferroptosis-IN-17 demonstrates good solubility and notable metabolic stability. This compound holds potential for research in tumor suppression, neurodegenerative diseases, and cardiovascular disorders.</p>Fórmula:C21H26N4O5SForma y color:SolidPeso molecular:446.52FD2157
<p>FD2157, a photosensitive PI3K inhibitor, exhibits inhibitory IC50 values of 43 nM for PI3Kα, 83 nM for PI3Kβ, 84 nM for PI3Kγ, and 14 nM for PI3Kδ.</p>Fórmula:C27H21ClN6O8SPureza:98%Forma y color:SolidPeso molecular:625.01UZH1a
CAS:<p>UZH1a: METTL3 inhibitor, IC50 280 nM, used for epitranscriptomic modulation and has antitumor properties.</p>Fórmula:C32H42N6O3Forma y color:SoildPeso molecular:558.71Anticancer agent 106
<p>Compound 106 (compound 10ic) induces apoptosis in B16-F10 melanoma cells and potently inhibits metastatic nodules in mouse models of lung metastatic melanoma,</p>Fórmula:C26H25N3O4SPureza:98%Forma y color:SolidPeso molecular:475.56CPT2
CAS:<p>Carnitine palmitoyltransferase 2 (CPT2), an enzyme involved in fatty acid oxidation, serves as a prognostic biomarker for colorectal cancer (CRC).</p>Pureza:98%Forma y color:SolidThalidomide-O-PEG4-amine
CAS:<p>Thalidomide-O-PEG4-amine is a PEG-based PROTAC linker that can be used in the synthesis of PROTACs[1].</p>Fórmula:C23H31N3O9Pureza:98%Forma y color:SolidPeso molecular:493.51SACLAC
CAS:<p>SACLAC is a cysteine asparaginase activation inhibitor with antitumor activity used in the study of acute myeloid leukemia and cancer.</p>Fórmula:C20H40ClNO3Pureza:97.03%Forma y color:SoildPeso molecular:377.99TAT-NEP1-40
<p>TAT-NEP1-40, a blood-brain barrier (BBB) permeable peptide, confers protection to PC12 cells against oxygen and glucose deprivation (OGD) while promoting</p>Fórmula:C268H438N88O77Pureza:98%Forma y color:SolidPeso molecular:6124.89Flaccidoside II
CAS:<p>Flaccidoside II, an active triterpenoid saponin from Anemone flaccida rhizome, both inhibits proliferation and induces apoptosis in Malignant Peripheral Nerve</p>Fórmula:C59H96O25Pureza:98%Forma y color:SolidPeso molecular:1205.38Antitumor agent-96
<p>"Antitumor agent-96 (Compound D34) is a potent MRE11 inhibitor that down-regulates the homologous recombination (HR) pathway by binding to and suppressing the</p>Fórmula:C27H32N2O2Pureza:98%Forma y color:SolidPeso molecular:416.56Asparanin A
CAS:<p>Asparanin A, an apoptosis inducer with anticancer properties, arrests the cell cycle in the G0/G1 phase via the mitochondria and PI3K/AKT signaling pathways.</p>Fórmula:C39H64O13Pureza:98%Forma y color:SolidPeso molecular:740.92
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