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Apoptosis

Apoptosis

Los inhibidores de la apoptosis son compuestos que previenen o retrasan el proceso de muerte celular programada, conocido como apoptosis. Estos inhibidores son vitales para estudiar los mecanismos de supervivencia celular y se utilizan para investigar enfermedades donde la apoptosis está desregulada, como el cáncer, los trastornos neurodegenerativos y las enfermedades autoinmunes. Al modular la apoptosis, estos inhibidores pueden ayudar en el desarrollo de terapias dirigidas a controlar la muerte celular. En CymitQuimica, ofrecemos una amplia selección de inhibidores de la apoptosis de alta calidad para apoyar su investigación en biología celular, oncología y campos relacionados.

Subcategorías de "Apoptosis"

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Se han encontrado 5622 productos de "Apoptosis"

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  • Sophocarpine

    CAS:
    <p>Sophocarpine, a major ingredient of Sophora alopecuroides, has a wide range of pharmacological effects.</p>
    Fórmula:C15H22N2O
    Pureza:99.89%
    Forma y color:Solid
    Peso molecular:246.35
  • CDPPB

    CAS:
    <p>CDPPB is a modulator of mGluR5 positive allosteric(with an EC50 of 27 nM in Chinese hamster ovary cells expressing human mGluR5).</p>
    Fórmula:C23H16N4O
    Pureza:99.16%
    Forma y color:Solid
    Peso molecular:364.4
  • Iproniazid

    CAS:
    <p>Iproniazid is an irreversible monoamine oxidase inhibitor. It is used as an antidepressive agent.</p>
    Fórmula:C9H13N3O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:179.22
  • CCPA

    CAS:
    <p>CCPA (2-chloro-N(6)cyclopentyladenosine) is a potent and selective agonist of adenosine A1 receptor</p>
    Fórmula:C15H20ClN5O4
    Pureza:99.1%
    Forma y color:Off-White To Light Yellow Solid
    Peso molecular:369.8
  • Candesartan Cilexetil

    CAS:
    <p>Candesartan Cilexetil, an angiotensin II blocker (IC50: 0.26 nM), turns to candesartan in the body, which dilates blood vessels by hindering AT1.</p>
    Fórmula:C33H34N6O6
    Pureza:98.22% - >99.99%
    Forma y color:White Crystalline Powder
    Peso molecular:610.66
  • Oprozomib

    CAS:
    <p>Oprozomib inhibits 20S proteasome β5/LMP7, is orally available, and may have cancer-fighting properties. IC50: β5 - 36 nM; LMP7 - 82 nM.</p>
    Fórmula:C25H32N4O7S
    Pureza:98% - 99.87%
    Forma y color:Solid
    Peso molecular:532.61
  • NVP-ADW742

    CAS:
    <p>NVP-ADW742 (ADW) is an IGF-1R inhibitor with IC50 of 0.17 μM, &gt;16-fold more potent against IGF-1R than InsR; little activity to HER2, PDGFR, VEGFR-2, Bcr-Abl</p>
    Fórmula:C28H31N5O
    Pureza:96.14% - 98.70%
    Forma y color:Solid
    Peso molecular:453.58
  • Glafenine Hydrochloride

    CAS:
    <p>Glafenine Hydrochloride is an anti-inflammatory agent.</p>
    Fórmula:C19H17ClN2O4·HCl
    Pureza:98.89%
    Forma y color:Solid
    Peso molecular:409.26
  • TASIN-1 Hydrochloride

    CAS:
    <p>TASIN-1 Hydrochloride (TASIN-1 HCl) is a selective inhibitor of truncated APC that acts by selectively killing colorectal cancer cells that express truncated</p>
    Fórmula:C18H29ClN2O3S
    Pureza:99.94%
    Forma y color:Solid
    Peso molecular:388.95
  • 1R,3S-RSL 3

    CAS:
    1R,3S-RSL 3 is a harmala alkaloid.
    Fórmula:C23H21ClN2O5
    Pureza:99.51%
    Forma y color:Solid
    Peso molecular:440.88
  • Amcasertib

    CAS:
    <p>Amcasertib (BBI503) is an orally administered investigational agent designed to inhibit cancer stem cell pathways via targeting stemness kinases.</p>
    Fórmula:C31H33N5O2S
    Pureza:97.56% - >99.99%
    Forma y color:Solid
    Peso molecular:539.69
  • Paroxetine

    CAS:
    <p>Paroxetine is a inhibitor of serotonin uptake that is effective in the treatment of depression.</p>
    Fórmula:C19H20FNO3
    Pureza:98.89% - 99.45%
    Forma y color:White To Off-White Powder
    Peso molecular:329.37
  • Parcetasal

    CAS:
    <p>Parcetasal (MR-897) is a non-steroidal anti-inflammatory agent that can be used in pain relief studies.</p>
    Fórmula:C17H15NO5
    Pureza:99.07%
    Forma y color:Solid
    Peso molecular:313.3
  • Romidepsin

    CAS:
    Romidepsin (NSC-630176), an IV histone deacetylase inhibitor, treats refractory cutaneous/peripheral T-cell lymphomas.
    Fórmula:C24H36N4O6S2
    Pureza:99.4% - 99.94%
    Forma y color:Solid
    Peso molecular:540.7
  • PX-12

    CAS:
    <p>PX-12, a Trx-1 inhibitor, promotes apoptosis, reduces HIF-1α/VEGF, and inhibits tumor growth, suggesting use in advanced cancer therapy.</p>
    Fórmula:C7H12N2S2
    Pureza:98% - 99.21%
    Forma y color:Solid
    Peso molecular:188.31
  • L524-0366

    CAS:
    <p>L524-0366 ([1-(3-chlorophenyl)triazol-4-yl]-thiomorpholino-methanone) is a TWEAK-Fn14 signaling cascade inhibitor.</p>
    Fórmula:C13H13ClN4OS
    Pureza:98.6% - 99.13%
    Forma y color:Solid
    Peso molecular:308.79
  • Saquinavir

    CAS:
    <p>Saquinavir (Ro 31-8959) is a potent HIV protease inhibitor, is an antiretroviral drug used together with other medications to treat or prevent HIV/AIDS.</p>
    Fórmula:C38H50N6O5
    Pureza:99.50% - >99.99%
    Forma y color:Solid
    Peso molecular:670.84
  • PCNA-I1

    CAS:
    <p>PCNA-I1 is an inhibitor targeting PCNA chromatin association in prostate cancer.</p>
    Fórmula:C17H14N2O2S
    Pureza:97.64%
    Forma y color:Solid
    Peso molecular:310.37
  • 4-IBP

    CAS:
    4-IBP is a selective σ1 agonist with a high level of affinity for the σ1 receptor (Ki = 1.7 nM) and a moderate affinity for the σ2 receptor (Ki = 25.2 nM) .
    Fórmula:C19H21IN2O
    Pureza:98.99%
    Forma y color:Solid
    Peso molecular:420.29
  • Lubiprostone

    CAS:
    <p>Lubiprostone (RU-0211), an activator of ClC-2 chloride channels, is used in the therapy of idiopathic chronic constipation.</p>
    Fórmula:C20H32F2O5
    Pureza:97.31% - 98.54%
    Forma y color:White Odorless Crystals Or Crystalline Powder
    Peso molecular:390.46
  • RH01687

    CAS:
    <p>RH01687 is a potent β-cell protector , exhibits β-cell-protective activities against endoplasmic reticulum (ER) stress.</p>
    Fórmula:C12H9ClN6O2S
    Pureza:97.93%
    Forma y color:Solid
    Peso molecular:336.76
  • Clodronic acid disodium salt

    CAS:
    <p>Clodronic acid disodium salt (Lodronate), a bisphosphonate, is a potent antiosteolytic agent which inhibits bone resorption.</p>
    Fórmula:CH4Cl2O6P0·2Na
    Pureza:>99.99% - ≥98%
    Forma y color:White Solid
    Peso molecular:288.86
  • Sodium benzoate

    CAS:
    <p>Sodium benzoate (Benzoic acid sodium salt) is a D-Amino Acid Oxidase Inhibitor.Sodium Benzoate is a Food Preservative.</p>
    Fórmula:C7H5NaO2
    Pureza:99.72%
    Forma y color:White Solid Crystalline
    Peso molecular:144.10
  • HX 531

    CAS:
    <p>HX 531 is a RXR antagonist (IC50 of 18 nM).Cost-effective and quality-assured.</p>
    Fórmula:C29H29N3O4
    Pureza:98.59% - 99.86%
    Forma y color:Solid
    Peso molecular:483.56
  • Benzarone

    CAS:
    <p>Benzarone (Benzarona) is a potent inhibitor of human uric acid transporter 1 (URAT1, IC50 = 2.8 μM in oocyte). Benzarone lowers the level of uric acid serum.</p>
    Fórmula:C17H14O3
    Pureza:99.77%
    Forma y color:Solid
    Peso molecular:266.29
  • 3-hydroxy-3-phenylpentanamide

    CAS:
    <p>Chiral 3-hydroxy-3-phenylpentanamide: neuroprotective, may treat anxiety/depression/addiction, anticancer.</p>
    Fórmula:C11H15NO2
    Pureza:98.42%
    Forma y color:Solid
    Peso molecular:193.24
  • Ceftiofur

    CAS:
    <p>Ceftiofur is a semisynthetic antibiotic, with activity against various gram-positive/negative, anaerobic and aerobic bacteria encountered by domestic animals.</p>
    Fórmula:C19H17N5O7S3
    Pureza:98.26%
    Forma y color:Solid
    Peso molecular:523.56
  • Dantrolene sodium hemiheptahydrate

    CAS:
    <p>Dantrolene depresses excitation-contraction coupling in skeletal muscle by binding to the ryanodine receptor 1 and decreasing intracellular calcium</p>
    Fórmula:C14H9N4NaO5·5H2O
    Pureza:99.72%
    Forma y color:Orange Powder
    Peso molecular:399.29
  • GYY4137

    CAS:
    <p>GYY4137 (GYY 4137 morpholine salt) is a novel water-soluble and slow releasing H2S donor with antihypertensive, anti-inflammatory and anticancer activity.</p>
    Fórmula:C11H16NO2PS2·C4H9NO
    Pureza:95.54% - 99.97%
    Forma y color:Solid
    Peso molecular:376.47
  • DIM-C-pPhCO2Me

    CAS:
    <p>DIM-C-pPhCO2Me is a nuclear receptor 4A1 (NR4A1) antagonist.</p>
    Fórmula:C25H20N2O2
    Pureza:99.55% - 99.86%
    Forma y color:Solid
    Peso molecular:380.44
  • Desciclovir

    CAS:
    <p>Desciclovir (DCV), a prodrug of the antiherpetic agent acyclovir (ACV), is converted in humans to ACV, presumably by xanthine oxidase.</p>
    Fórmula:C8H11N5O2
    Pureza:99.54%
    Forma y color:Solid
    Peso molecular:209.21
  • 2-HBA

    CAS:
    <p>2-HBA, a synthetic analog of curcumin, is an indirect inducer of enzymes that catalyze detoxification reactions through the Keap1-Nrf2-ARE pathway.</p>
    Fórmula:C17H14O3
    Pureza:99.76%
    Forma y color:Solid
    Peso molecular:266.29
  • NSC 3852

    CAS:
    <p>NSC 3852 is a potent inhibitor of histone deacetylase.</p>
    Fórmula:C9H6N2O2
    Pureza:99.64%
    Forma y color:Slightly Yellow To Yellow-Green Powder
    Peso molecular:174.16
  • 3,4 Dichloroisocoumarin

    CAS:
    <p>3,4 Dichloroisocoumarin is a granzyme, cathepsin G, and neutrolphil elastase inhibitor</p>
    Fórmula:C9H4Cl2O2
    Pureza:97.94%
    Forma y color:Solid
    Peso molecular:215.03
  • Thalidomide-NH-CH2-COOH TFA

    CAS:
    <p>2-{[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]amino}acetic acid (trifluoroacetic acid) is mainly used in compounds Synthesis.</p>
    Fórmula:C17H14F3N3O8
    Pureza:95.00%
    Forma y color:Solid
    Peso molecular:445.3036
  • Hexamethylene bisacetamide

    CAS:
    <p>Hexamethylene bisacetamide inhibits BET Bromodomain Proteins.</p>
    Fórmula:C10H20N2O2
    Pureza:99.94%
    Forma y color:White Flakes
    Peso molecular:200.28
  • PDL-1 cpd 10

    CAS:
    <p>PDL-1 cpd 10 is a novel small molecule PD-L1 inhititor.</p>
    Fórmula:C21H23N5O2
    Pureza:97.08%
    Forma y color:Solid
    Peso molecular:377.44
  • Acenocoumarol

    CAS:
    <p>Acenocoumarol is a Vitamin K antagonist and used as an anticoagulant.</p>
    Fórmula:C19H15NO6
    Pureza:99.95%
    Forma y color:Crystals Solid
    Peso molecular:353.33
  • OTS964 hydrochloride

    CAS:
    <p>OTS964 hydrochloride (OTS964) is a potent and selective TOPK inhibitor with potential anticancer activity.</p>
    Fórmula:C23H24N2O2S·HCl
    Pureza:96.5% - 98.03%
    Forma y color:Solid
    Peso molecular:428.97
  • Z-VAD-FMK

    CAS:
    <p>Z-VAD-FMK (Caspase Inhibitor VI) is a broad-spectrum inhibitor of caspases.Z-VAD-FMK binds to activated caspases and inhibits apoptosis.Z-VAD-FMK does not</p>
    Fórmula:C21H28FN3O7
    Pureza:98.24% - 99.79%
    Forma y color:Solid
    Peso molecular:453.46
  • Sinapinic Acid

    CAS:
    <p>Sinapinic Acid (Synapoic acid) is a phenolic isolated from the roots of Hydnophytum formicarumJack. It is an HDAC inhibitor and also inhibits ACE-I activity.</p>
    Fórmula:C11H12O5
    Pureza:99.88% - >99.99%
    Forma y color:Solid
    Peso molecular:224.21
  • Nocodazole

    CAS:
    Nocodazole: synthetic microtubule polymerization blocker, also impedes Abl with low IC50; binds to beta-tubulin.
    Fórmula:C14H11N3O3S
    Pureza:98% - 99.91%
    Forma y color:Physical Description White Powder (Ntp 1992)
    Peso molecular:301.32
  • Tyrphostin AG1296

    CAS:
    Tyrphostin AG1296 (Tyrphostin AG 1296) is an inhibitor of PDGFR with IC50 of 0.3-0.5 μM, no activity to EGFR.
    Fórmula:C16H14N2O2
    Pureza:99.94% - >99.99%
    Forma y color:Solid
    Peso molecular:266.29
  • Euscaphic acid

    CAS:
    <p>Euscaphic acid has anti-diabetic and anti-inflammatory effects, blocking IKK/MAPKs and NF-κB activation by disrupting TRAF6/IRAK1/TAK1 clustering.</p>
    Fórmula:C30H48O5
    Pureza:98.93%
    Forma y color:Solid
    Peso molecular:488.7
  • Licochalcone B

    CAS:
    <p>Licochalcone B inhibits human bladder cancer cells, reduces inflammation by NO, TNFalpha, and MCP-1, and a derivative protects against endotoxin shock.</p>
    Fórmula:C16H14O5
    Pureza:99.33% - 99.93%
    Forma y color:Solid
    Peso molecular:286.28
  • Z-DEVD-FMK

    CAS:
    <p>Z-DEVD-FMK (Caspase-3 Inhibitor) is a selective, irreversible Caspase-3 inhibitor, and also exhibits effective inhibition activity on caspase-6, caspase-7,</p>
    Fórmula:C30H41FN4O12
    Pureza:96.19% - 99.69%
    Forma y color:Solid
    Peso molecular:668.66
  • Rebastinib

    CAS:
    <p>DCC-2036 (Rebastinib (DCC-2036)) is a conformational control Bcr-Abl inhibitor for Abl1(WT, IC50: 0.8 nM) and Abl1(T315I, IC50: 4 nM), also inhibits LYN, SRC,</p>
    Fórmula:C30H28FN7O3
    Pureza:99.53% - 99.79%
    Forma y color:Solid
    Peso molecular:553.59
  • Pitstop 2

    CAS:
    <p>Pitstop2 is an amphipathic protein-bound inhibitor of the clathrin terminal domain. Pitstop2 has antitumor activity. Cost-effective, quality assurance.</p>
    Fórmula:C20H13BrN2O3S2
    Pureza:99.54%
    Forma y color:Solid
    Peso molecular:473.36
  • ZM 336372

    CAS:
    <p>ZM 336372 is a potent and selective c-Raf inhibitor.</p>
    Fórmula:C23H23N3O3
    Pureza:97.24% - 97.51%
    Forma y color:Solid
    Peso molecular:389.45
  • Avelumab

    CAS:
    <p>Avelumab is a fully human IgG1 anti-PD-L1 monoclonal antibody. Avelumab shows potential antibody-dependent cell-mediated cytotoxicity.</p>
    Pureza:95% - 97.17% (SDS-PAGE)
    Forma y color:Liquid
    Peso molecular:143.8 kDa