
Endocrinología / Hormonas
Los inhibidores de endocrinología/hormonas son compuestos que bloquean la acción de las hormonas o interfieren con las vías de señalización hormonal. Estos inhibidores son esenciales para estudiar la regulación de los sistemas endocrinos y para desarrollar tratamientos para enfermedades relacionadas con las hormonas, como la diabetes, los trastornos tiroideos y los cánceres dependientes de hormonas. Al modular la actividad hormonal, estos inhibidores pueden ayudar a dilucidar las complejas interacciones dentro del sistema endocrino. En CymitQuimica, ofrecemos una amplia gama de inhibidores de endocrinología/hormonas de alta calidad para apoyar su investigación en endocrinología, farmacología y ciencias médicas.
Subcategorías de "Endocrinología / Hormonas"
- Receptor de andrógenos(229 productos)
- Anexina A(16 productos)
- Aromatasa(22 productos)
- Receptor de estrógeno / progestágeno(64 productos)
- GPR(1 productos)
- Receptor de glucocorticoides(165 productos)
- LHRH(2 productos)
- Receptor de opioides(326 productos)
- Receptor de prostaglandinas(122 productos)
- RAAS(86 productos)
- Reductasa(51 productos)
- Somatostatina(57 productos)
- Receptor de la hormona tiroidea (THR)(33 productos)
- Receptor de vasopresina(48 productos)
Mostrar 6 subcategorías más
Se han encontrado 3415 productos de "Endocrinología / Hormonas"
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(Glu2)-TRH
CAS:(Glu2)-TRH: Stable TRH analog; reduces TRH's cholinergic action; no thyroliberinase metabolism; neuroprotective with antidepressant, anticonvulsant effects.Fórmula:C15H22N4O6Forma y color:SolidPeso molecular:354.36Osteostatin
CAS:Osteostatin, derived from parathyroid hormone-related protein (PTHrP) 107-111, has demonstrated properties conducive to bone repair in animal models presentingFórmula:C27H41N9O8Forma y color:SolidPeso molecular:619.677α-(Thiomethyl)spironolactone
CAS:7α-(Thiomethyl)spironolactone is a steroid receptor antagonist and major spironolactone metabolite, steroid metabolism, nuclear receptor, and coronavirus.Fórmula:C23H32O3SPureza:>99.99%Forma y color:SolidPeso molecular:388.56NPFF1-R antagonist 1
NPFF1-R antagonist 1 (compound 8b) is a piperidine analog and an effective neuropeptide FF (NPFF) receptor antagonist. It exhibits 15-fold selectivity for the NPFF1-R subtype, with Ki values of 211 nM and 3270 nM for NPFF1-R and NPFF2-R, respectively.Fórmula:C37H44N4OPeso molecular:560.35151VinclozolinM2-2204
VinclozolinM2-2204 is an androgen receptor AUTOTAC degrader with a DC50 of 200 nM in LNCaP prostate cancer cells. It induces the formation of AR+LC3+ autophagic membranes and is applicable for cancer research.Fórmula:C43H51Cl2N3O9Peso molecular:823.30024DP50
DP50 is a bifunctional compound containing both an opioid receptor agonist (MOP) and a neuropeptide FF receptor (NPFFR) antagonist. It can be utilized in studies related to analgesia.Fórmula:C58H72N8O7Peso molecular:992.5524PIPE-3297
PIPE-3297 (compound 25) is a selective kappa opioid receptor (KOR) agonist that activates the G protein signaling pathway with an EC50 of 1.1 nM and exhibits low β-arrestin-2 recruitment activity (10%). Additionally, PIPE-3297 promotes myelination and has anti-inflammatory properties.Fórmula:C23H30N2OPeso molecular:350.23581Nurr1 agonist 9
Nurr1 agonist 9 (Compound 36) acts as an agonist for Nurr1, with an EC50 of 0.090 µM and a Kd of 0.17 µM. It activates Nurr1 homodimers (NurRE, EC50 = 0.094 µM) and Nurr1-RXR heterodimers (DR5, EC50 = 0.165 µM). This compound induces the expression of Nurr1-regulated tyrosine hydroxylase (TH) in Parkinson's disease organoid models and can penetrate the human brain endothelial cell barrier.
Fórmula:C21H19ClN4O2Peso molecular:394.11965Awl 60
CAS:Awl 60 is a substance P (6-11) non-competitive antagonist.Fórmula:C57H65N9O8SPureza:98%Forma y color:SolidPeso molecular:1036.25SB 205607 dihydrobromide
CAS:non-peptide δ1 opioid receptor agonistFórmula:C23H24N2OPureza:98%Forma y color:SolidPeso molecular:344.45Ethamoxytriphetol
CAS:Ethamoxytriphetol is a non-steroidal estrogen antagonist.Fórmula:C27H33NO3Forma y color:SolidPeso molecular:419.56Bradykinin potentiator-5
CAS:Bradykinin potentiator-5 is a peptide inflammatory mediator, causes blood vessels to dilate (enlarge), and therefore causes blood pressure to fall.Fórmula:C30H41N7O7Pureza:98%Forma y color:SolidPeso molecular:611.69Enalapril
CAS:Enalapril is a dicarbocyl-containing peptide and angiotensin-converting enzyme (ACE) inhibitor with antihypertensive activity.Fórmula:C20H28N2O5Pureza:99.47% - 99.51%Forma y color:SolidPeso molecular:376.455-O-β-D-Glucopyranosylmyricanol
5-O-beta-D-Glucopyranosylmyricanol is a useful organic compound for research related to life sciences and the catalog number is T123967.Fórmula:C27H36O10Forma y color:SolidPeso molecular:520.575RU-39411
CAS:RU-39411 is a steroidal anti-estrogen.Fórmula:C28H37NO3Pureza:98%Forma y color:SolidPeso molecular:435.60Acetiromate
CAS:Acetiromate is a drug of antilipidemic. It is used to treat hyperlipidemia.Fórmula:C15H9I3O5Pureza:98%Forma y color:SolidPeso molecular:649.94LY301875
CAS:LY301875 is an antagonist of nonpeptide angiotensin receptor.Fórmula:C31H36N4O10SForma y color:SolidPeso molecular:656.70AT2R antagonist 2
Compound I-16 (AT2R antagonist 2) is an orally active AT2R antagonist.Fórmula:C20H23F3N8SForma y color:SolidPeso molecular:464.51TRIP13-IN-1
TRIP13-IN-1 (compound 20) is a potent ligand and inhibitor of TRIP13, demonstrating anticancer effects both in vivo and in vitro.Fórmula:C24H25NO9SForma y color:SolidPeso molecular:503.52Trioxifene mesylate
CAS:Trioxifene mesylate is an antiestrogen that suppresses growth hormone secretion.Fórmula:C31H35NO6SPureza:98%Forma y color:SolidPeso molecular:549.68

