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Endocrinología / Hormonas

Endocrinología / Hormonas

Los inhibidores de endocrinología/hormonas son compuestos que bloquean la acción de las hormonas o interfieren con las vías de señalización hormonal. Estos inhibidores son esenciales para estudiar la regulación de los sistemas endocrinos y para desarrollar tratamientos para enfermedades relacionadas con las hormonas, como la diabetes, los trastornos tiroideos y los cánceres dependientes de hormonas. Al modular la actividad hormonal, estos inhibidores pueden ayudar a dilucidar las complejas interacciones dentro del sistema endocrino. En CymitQuimica, ofrecemos una amplia gama de inhibidores de endocrinología/hormonas de alta calidad para apoyar su investigación en endocrinología, farmacología y ciencias médicas.

Subcategorías de "Endocrinología / Hormonas"

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Se han encontrado 3415 productos de "Endocrinología / Hormonas"

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  • (Glu2)-TRH

    CAS:
    (Glu2)-TRH: Stable TRH analog; reduces TRH's cholinergic action; no thyroliberinase metabolism; neuroprotective with antidepressant, anticonvulsant effects.
    Fórmula:C15H22N4O6
    Forma y color:Solid
    Peso molecular:354.36

    Ref: TM-T76493

    5mg
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    50mg
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  • Osteostatin

    CAS:
    Osteostatin, derived from parathyroid hormone-related protein (PTHrP) 107-111, has demonstrated properties conducive to bone repair in animal models presenting
    Fórmula:C27H41N9O8
    Forma y color:Solid
    Peso molecular:619.67

    Ref: TM-T81592

    5mg
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    50mg
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  • 7α-(Thiomethyl)spironolactone

    CAS:
    7α-(Thiomethyl)spironolactone is a steroid receptor antagonist and major spironolactone metabolite, steroid metabolism, nuclear receptor, and coronavirus.
    Fórmula:C23H32O3S
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:388.56

    Ref: TM-T37362

    1mg
    237,00€
    5mg
    707,00€
    10mg
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    25mg
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  • NPFF1-R antagonist 1


    NPFF1-R antagonist 1 (compound 8b) is a piperidine analog and an effective neuropeptide FF (NPFF) receptor antagonist. It exhibits 15-fold selectivity for the NPFF1-R subtype, with Ki values of 211 nM and 3270 nM for NPFF1-R and NPFF2-R, respectively.
    Fórmula:C37H44N4O
    Peso molecular:560.35151

    Ref: TM-T209569

    10mg
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    50mg
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  • VinclozolinM2-2204


    VinclozolinM2-2204 is an androgen receptor AUTOTAC degrader with a DC50 of 200 nM in LNCaP prostate cancer cells. It induces the formation of AR+LC3+ autophagic membranes and is applicable for cancer research.
    Fórmula:C43H51Cl2N3O9
    Peso molecular:823.30024

    Ref: TM-T210394

    10mg
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    50mg
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  • DP50


    DP50 is a bifunctional compound containing both an opioid receptor agonist (MOP) and a neuropeptide FF receptor (NPFFR) antagonist. It can be utilized in studies related to analgesia.
    Fórmula:C58H72N8O7
    Peso molecular:992.5524

    Ref: TM-TP3590

    10mg
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    50mg
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  • PIPE-3297


    PIPE-3297 (compound 25) is a selective kappa opioid receptor (KOR) agonist that activates the G protein signaling pathway with an EC50 of 1.1 nM and exhibits low β-arrestin-2 recruitment activity (10%). Additionally, PIPE-3297 promotes myelination and has anti-inflammatory properties.
    Fórmula:C23H30N2O
    Peso molecular:350.23581

    Ref: TM-T209195

    10mg
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    50mg
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  • Nurr1 agonist 9


    Nurr1 agonist 9 (Compound 36) acts as an agonist for Nurr1, with an EC50 of 0.090 µM and a Kd of 0.17 µM. It activates Nurr1 homodimers (NurRE, EC50 = 0.094 µM) and Nurr1-RXR heterodimers (DR5, EC50 = 0.165 µM). This compound induces the expression of Nurr1-regulated tyrosine hydroxylase (TH) in Parkinson's disease organoid models and can penetrate the human brain endothelial cell barrier.

    Fórmula:C21H19ClN4O2
    Peso molecular:394.11965

    Ref: TM-T210048

    10mg
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    50mg
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  • Awl 60

    CAS:
    Awl 60 is a substance P (6-11) non-competitive antagonist.
    Fórmula:C57H65N9O8S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:1036.25

    Ref: TM-T25122

    25mg
    1.369,00€
  • SB 205607 dihydrobromide

    CAS:
    non-peptide δ1 opioid receptor agonist
    Fórmula:C23H24N2O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:344.45

    Ref: TM-T23313

    10mg
    672,00€
  • Ethamoxytriphetol

    CAS:
    Ethamoxytriphetol is a non-steroidal estrogen antagonist.
    Fórmula:C27H33NO3
    Forma y color:Solid
    Peso molecular:419.56

    Ref: TM-T25395

    25mg
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    50mg
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    100mg
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  • Bradykinin potentiator-5

    CAS:
    Bradykinin potentiator-5 is a peptide inflammatory mediator, causes blood vessels to dilate (enlarge), and therefore causes blood pressure to fall.
    Fórmula:C30H41N7O7
    Pureza:98%
    Forma y color:Solid
    Peso molecular:611.69

    Ref: TM-T25173

    25mg
    2.718,00€
    50mg
    3.582,00€
    100mg
    4.950,00€
  • Enalapril

    CAS:
    Enalapril is a dicarbocyl-containing peptide and angiotensin-converting enzyme (ACE) inhibitor with antihypertensive activity.
    Fórmula:C20H28N2O5
    Pureza:99.47% - 99.51%
    Forma y color:Solid
    Peso molecular:376.45

    Ref: TM-T1605

    100mg
    34,00€
    1mL*10mM (DMSO)
    33,00€
  • 5-O-β-D-Glucopyranosylmyricanol


    5-O-beta-D-Glucopyranosylmyricanol is a useful organic compound for research related to life sciences and the catalog number is T123967.
    Fórmula:C27H36O10
    Forma y color:Solid
    Peso molecular:520.575

    Ref: TM-T123967

    1mg
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    5mg
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  • RU-39411

    CAS:
    RU-39411 is a steroidal anti-estrogen.
    Fórmula:C28H37NO3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:435.60

    Ref: TM-T26158

    25mg
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    50mg
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    100mg
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  • Acetiromate

    CAS:
    Acetiromate is a drug of antilipidemic. It is used to treat hyperlipidemia.
    Fórmula:C15H9I3O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:649.94

    Ref: TM-T23611

    25mg
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    50mg
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    100mg
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  • LY301875

    CAS:
    LY301875 is an antagonist of nonpeptide angiotensin receptor.
    Fórmula:C31H36N4O10S
    Forma y color:Solid
    Peso molecular:656.70

    Ref: TM-T27940

    25mg
    3.078,00€
    50mg
    3.853,00€
    100mg
    5.040,00€
  • AT2R antagonist 2


    Compound I-16 (AT2R antagonist 2) is an orally active AT2R antagonist.
    Fórmula:C20H23F3N8S
    Forma y color:Solid
    Peso molecular:464.51

    Ref: TM-T201045

    10mg
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    50mg
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  • TRIP13-IN-1


    TRIP13-IN-1 (compound 20) is a potent ligand and inhibitor of TRIP13, demonstrating anticancer effects both in vivo and in vitro.
    Fórmula:C24H25NO9S
    Forma y color:Solid
    Peso molecular:503.52

    Ref: TM-T201292

    10mg
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    50mg
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  • Trioxifene mesylate

    CAS:
    Trioxifene mesylate is an antiestrogen that suppresses growth hormone secretion.
    Fórmula:C31H35NO6S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:549.68

    Ref: TM-T26295

    25mg
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    50mg
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    100mg
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