
Endocrinología / Hormonas
Los inhibidores de endocrinología/hormonas son compuestos que bloquean la acción de las hormonas o interfieren con las vías de señalización hormonal. Estos inhibidores son esenciales para estudiar la regulación de los sistemas endocrinos y para desarrollar tratamientos para enfermedades relacionadas con las hormonas, como la diabetes, los trastornos tiroideos y los cánceres dependientes de hormonas. Al modular la actividad hormonal, estos inhibidores pueden ayudar a dilucidar las complejas interacciones dentro del sistema endocrino. En CymitQuimica, ofrecemos una amplia gama de inhibidores de endocrinología/hormonas de alta calidad para apoyar su investigación en endocrinología, farmacología y ciencias médicas.
Subcategorías de "Endocrinología / Hormonas"
- Receptor de andrógenos(229 productos)
- Anexina A(16 productos)
- Aromatasa(22 productos)
- Receptor de estrógeno / progestágeno(59 productos)
- GPR(1 productos)
- Receptor de glucocorticoides(166 productos)
- LHRH(2 productos)
- Receptor de opioides(326 productos)
- Receptor de prostaglandinas(122 productos)
- RAAS(90 productos)
- Reductasa(50 productos)
- Somatostatina(57 productos)
- Receptor de la hormona tiroidea (THR)(32 productos)
- Receptor de vasopresina(48 productos)
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Se han encontrado 3373 productos de "Endocrinología / Hormonas"
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Akuammicine
CAS:Akuammicine, as an indole alkaloid from Catharanthus roseus, can be used in cancer cell eradication.Fórmula:C20H22N2O2Forma y color:SolidPeso molecular:322.408Glucocorticoids receptor agonist 1
CAS:<p>GRA-1, an arylpyrazole, is a potent glucocorticoid receptor agonist with robust anti-inflammatory effects and preserves insulin secretion.</p>Fórmula:C20H23FN2OForma y color:SolidPeso molecular:326.41ALR2-IN-1
CAS:ALR2-IN-1: potent, selective inhibitor of ALR2 (IC50=1.42 μM), antiglycemic, antioxidant; for diabetes research.Fórmula:C16H17N3O2SPureza:99.41%Forma y color:SoildPeso molecular:315.39MK-0773 FA
MK-0773 FA (MK-0773 FA (606101-58-0 Free base)) is an androgen receptor modulator used for the prevention and treatment of cancer-related muscle wasting.Fórmula:C28H36FN5O4Pureza:98.46%Forma y color:SoildPeso molecular:525.61Linuron
CAS:Linuron herbicide disrupts photosynthesis and acts as an androgen receptor antagonist.Fórmula:C9H10Cl2N2O2Pureza:99.08%Forma y color:White Crystalline Solid Linuron Is A Colorless Crystals Non Corrosive Used As An HerbicidePeso molecular:249.09(Rac)-Finerenone
CAS:Rac-Finerenone, or (Rac)-BAY 94-8862, is an oral nonsteroidal MR antagonist with high selectivity and an IC50 of 18 nM.Fórmula:C21H22N4O3Forma y color:SolidPeso molecular:378.432Montirelin
CAS:Montirelin is an analog of thyrotropin-releasing hormone.Fórmula:C17H24N6O4SForma y color:SolidPeso molecular:408.4821-hydroxy Eplerenone
CAS:21-hydroxy Eplerenone, a key eplerenone metabolite, is produced via CYP3A4.Fórmula:C24H30O7Forma y color:SolidPeso molecular:430.497GPCR agonist-2
CAS:GPCR agonist-2 (4-(Cyclopropylamino)-3-nitrobenzoic acid) is an agonist of the orphan human GPCR GPR109B.Fórmula:C10H10N2O4Pureza:99.96%Forma y color:SolidPeso molecular:222.2ER ligand-9
CAS:ER ligand-9 is a conjugate of an estrogen receptor (Estrogen Receptor/ERR) ligand and a linker, utilized in the synthesis of PROTACs ERD-1233.Fórmula:C31H33NO3Forma y color:SolidPeso molecular:467.599[(pF)Phe4]Nociceptin(1-13)NH2
CAS:<p>Potent, selective OP4 agonist; pKi=10.68, pEC50=9.80. >8000x selectivity vs other opioid receptors; long-lasting in vivo effects.</p>Fórmula:C61H99FN22O15Pureza:98%Forma y color:SolidPeso molecular:1399.6Dermorphin Analog
Dermorphin Analog, a heptapeptide from amphibian skin, binds μ-opioid receptors selectively and strongly.Fórmula:C44H59N11O10Pureza:98%Forma y color:SolidPeso molecular:901.43Tetrahydro Aldosterone
CAS:<p>Tetrahydro Aldosterone is a steroidal compound that inhibits the adrenal angiotensin II receptor, with an IC50 of 10 μM.</p>Fórmula:C21H32O5Forma y color:SolidPeso molecular:364.48OT-R antagonist 1
CAS:OT-R antagonist 1: Nonpeptide, selective, low-weight blocker of oxytocin; IC50 = 8 nM for Ca2+ disruption.Fórmula:C28H29N3O4Pureza:98%Forma y color:SolidPeso molecular:471.55[Orn5]-URP
CAS:Urotensin-II receptor antagonist, no agonist effect, pEC50 7.24, blocks U-II in rat aorta assay.Fórmula:C48H62N10O10S2Pureza:98%Forma y color:SolidPeso molecular:1003.2Olmesartan impurity
CAS:Olmesartan impurity, related to parent RNH-6270, is an AT1R antagonist used for hypertension research.Fórmula:C33H26N4OForma y color:SolidPeso molecular:494.598Piperidylthiambutene hydrochloride
CAS:Piperidylthiambutene hydrochloride is an opioid compound that exhibits analgesic effects in animal models.Fórmula:C17H22ClNS2Forma y color:SolidPeso molecular:339.95PRL 2915
CAS:<p>PRL 2915 is a potent antagonist of the human somatostatin subtype 2 receptor (hsst 2), exhibiting a binding affinity (K_i) of 12 nM [1].</p>Fórmula:C59H71ClN12O8S2Forma y color:SolidPeso molecular:1175.85Cgp 44099
CAS:Cgp 44099 is a potent plasma renin inhibitor from all subprimate species.Fórmula:C69H104N14O13Pureza:98%Forma y color:SolidPeso molecular:1337.676D3R/MOR antagonist 2
<p>Compound 121, a D3R/MOR antagonist with K i values of 361 nM and 85.2 nM for D3R and MOR respectively, has the potential for analgesic effects through MOR</p>Fórmula:C25H31ClN2OPureza:98%Forma y color:SolidPeso molecular:410.98

