Endocrinología / Hormonas
Los inhibidores de endocrinología/hormonas son compuestos que bloquean la acción de las hormonas o interfieren con las vías de señalización hormonal. Estos inhibidores son esenciales para estudiar la regulación de los sistemas endocrinos y para desarrollar tratamientos para enfermedades relacionadas con las hormonas, como la diabetes, los trastornos tiroideos y los cánceres dependientes de hormonas. Al modular la actividad hormonal, estos inhibidores pueden ayudar a dilucidar las complejas interacciones dentro del sistema endocrino. En CymitQuimica, ofrecemos una amplia gama de inhibidores de endocrinología/hormonas de alta calidad para apoyar su investigación en endocrinología, farmacología y ciencias médicas.
Subcategorías de "Endocrinología / Hormonas"
- Receptor de andrógenos(229 productos)
- Anexina A(16 productos)
- Aromatasa(23 productos)
- Receptor de estrógeno / progestágeno(66 productos)
- GPR(1 productos)
- Receptor de glucocorticoides(165 productos)
- LHRH(2 productos)
- Receptor de opioides(327 productos)
- Receptor de prostaglandinas(122 productos)
- RAAS(89 productos)
- Reductasa(51 productos)
- Somatostatina(57 productos)
- Receptor de la hormona tiroidea (THR)(33 productos)
- Receptor de vasopresina(48 productos)
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Se han encontrado 3420 productos de "Endocrinología / Hormonas"
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Olmesartan medoxomil impurity C
CAS:Impurity C of Olmesartan medoxomil is a selective AT1 inhibitor with an IC50 of 66.2 μM.Fórmula:C29H28N6O5Forma y color:SolidPeso molecular:540.57Azilsartan Medoxomil Potassium
CAS:Azilsartan Medoxomil Potassium (TAK-491 Potassium) is an orally administered angiotensin II receptor type 1 antagonist with IC50 of 0.62 nM, which used in the treatment of adults with essential hypertension.Fórmula:C30H23N4O8·KPureza:99.99%Forma y color:SolidPeso molecular:606.62Hydrocortisone sodium succinate
CAS:Hydrocortisone sodium succinate is a glucocorticoid which is used to alleviate allergic reactions, particularly those of the skin and gums.Fórmula:C25H34NaO8Forma y color:SolidPeso molecular:485.529L 363564
CAS:L 363564 is a kidney renin inhibitor.Fórmula:C54H76N12O10Forma y color:SolidPeso molecular:1053.276ST-CY14
ST-CY14 is an inhibitor of the Nur77-PPARγ interaction with an EC50 of 3.15 μM. It binds to Nur77 (Kd=32 nM) to prevent its ubiquitination and degradation by PPARγ, reducing fatty acid uptake and mitochondrial respiration, and inhibiting the transcription of CD36 and FABP4. ST-CY14 suppresses proliferation and migration of MCF7 and MDA-MB-231 cancer cells and impedes tumor growth and bone metastasis in mouse models.Fórmula:C139H237N57O31S2Forma y color:SolidPeso molecular:3266.86PTP1B/AKR1B1-IN-2
PTP1B/AKR1B1-IN-2 (Compound 7f) is a potent inhibitor targeting both PTP1B and AKR1B1 with IC50 values of 3.2 and 2.1 μM, respectively, and K i values of 4.0Fórmula:C23H23NO4S2Pureza:98%Forma y color:SolidPeso molecular:441.56AZ 1729
CAS:FFA2 modulator; inhibits cAMP, enhances 35SGTPγS binding (pEC50: 6.9, 7.23); alters Gi/Gq signaling; affects lipolysis, neutrophil migration.Fórmula:C18H16FN5OSForma y color:SolidPeso molecular:369.42Estrogen receptor modulator 6
CAS:ER modulator 6 (3a) is a potent ERβ agonist with a K i of 0.44 nM; 19x more selective for ERβ than ERα.
Fórmula:C18H16F2O3Forma y color:SolidPeso molecular:318.32Ro 64-6198
CAS:Ro 64-6198: Nonpeptide, selective NOP agonist, high brain uptake, EC50=25.6 nM, 100x NOP>opioid affinity.Fórmula:C26H31N3OPureza:98%Forma y color:SolidPeso molecular:401.54AKR1B10-IN-1
CAS:AKR1B10-IN-1: potent AKR1B10 inhibitor, IC50 3.5 nM; hinders lung cancer cell growth, spread, and Cisplatin resistance.Fórmula:C19H16FNO4Forma y color:SolidPeso molecular:341.338UFP-101
CAS:Strong, selective NOP receptor antagonist with pKi=10.24; >3000x selectivity over δ, μ, κ receptors; blocks nociceptin effects.
Fórmula:C82H138N32O21Pureza:98%Forma y color:SolidPeso molecular:1908.19T4-ATA (S-isomer)
T4-ATA S-isomer, the active form of the thyroid hormone, represents the S-isomer of T4-ATA.Fórmula:C19H15I4NO6SPureza:98%Forma y color:SolidPeso molecular:893.01U-54494A hydrochloride
CAS:U-54494A hydrochloride is a benzamide derivative related to kappa opioid receptor agonists. U-54494A hydrochloride has anticonvulsant activity.Fórmula:C18H25Cl3N2OForma y color:SolidPeso molecular:391.76[Sar1, Ile8]-Angiotensin II TFA
[Sar1,Ile8]-Angiotensin II (TFA) contracts arteries and affects cell growth in vascular muscle.Fórmula:C48H74F3N13O12Pureza:98%Forma y color:SolidPeso molecular:1082.18Herkinorin
CAS:Herkinorin: μ-opioid agonist with 100x μ-affinity, 50x less κ-affinity than Salvinorin A, from Salvia divinorum. Semi-synthetic from Salvinorin B.Fórmula:C28H30O8Forma y color:SolidPeso molecular:494.53PROTAC ER Degrader-3
CAS:PROTAC ER Degrader-3 from patent WO2017201449A1 is a PAC synthesis intermediate for ADC/PROTAC antibody conjugates, boosting ERα degradation.Fórmula:C71H77N7O12Pureza:98%Forma y color:SolidPeso molecular:1220.434Alclometasone
CAS:Alclometasone is a glucocorticoid that reduces inflammation and treats various skin conditions like eczema and psoriasis.Fórmula:C22H29ClO5Pureza:98%Forma y color:SolidPeso molecular:408.92Dynorphin B (1-13)
CAS:Dynorphin B (1-13) acts as an agonist on opioid κ-receptor.Fórmula:C74H115N21O17Pureza:98%Forma y color:SolidPeso molecular:1570.84Antihypertensive agent 3
Antihypertensive agent 3 (compound 4a), an angiotensin II receptor 1 antagonist, demonstrates antihypertensive activity in spontaneously hypertensive rats (SHRsFórmula:C16H13NO4SForma y color:SolidPeso molecular:315.34Neuropeptide AF (human)
CAS:Neuropeptide AF (93-110), Human is an endogenous antiopioid peptide.Fórmula:C90H132N26O25Pureza:98%Forma y color:SolidPeso molecular:1978.17
