
Endocrinología / Hormonas
Los inhibidores de endocrinología/hormonas son compuestos que bloquean la acción de las hormonas o interfieren con las vías de señalización hormonal. Estos inhibidores son esenciales para estudiar la regulación de los sistemas endocrinos y para desarrollar tratamientos para enfermedades relacionadas con las hormonas, como la diabetes, los trastornos tiroideos y los cánceres dependientes de hormonas. Al modular la actividad hormonal, estos inhibidores pueden ayudar a dilucidar las complejas interacciones dentro del sistema endocrino. En CymitQuimica, ofrecemos una amplia gama de inhibidores de endocrinología/hormonas de alta calidad para apoyar su investigación en endocrinología, farmacología y ciencias médicas.
Subcategorías de "Endocrinología / Hormonas"
- Receptor de andrógenos(229 productos)
- Anexina A(16 productos)
- Aromatasa(23 productos)
- Receptor de estrógeno / progestágeno(66 productos)
- GPR(1 productos)
- Receptor de glucocorticoides(165 productos)
- LHRH(2 productos)
- Receptor de opioides(327 productos)
- Receptor de prostaglandinas(122 productos)
- RAAS(89 productos)
- Reductasa(51 productos)
- Somatostatina(57 productos)
- Receptor de la hormona tiroidea (THR)(33 productos)
- Receptor de vasopresina(48 productos)
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Se han encontrado 3420 productos de "Endocrinología / Hormonas"
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Inocoterone acetate
CAS:Inocoterone acetate is a nonsteroidal antiandrogen that binds to the androgen receptor and possesses antiandrogenic activity in animal models.Fórmula:C18H26O3Forma y color:SolidPeso molecular:290.40AM-5262
CAS:AM-5262 is a potent GPR40 Full Agonist with improved rat PK profile and general selectivity profile.Fórmula:C33H35FO4Forma y color:SolidPeso molecular:514.63ER degrader 4
CAS:ER degrader 4, a selective and orally active compound, effectively degrades estrogen receptors and exhibits anti-tumor activity [1].Fórmula:C26H19FO4SForma y color:SolidPeso molecular:446.49Antidiabetic agent 15
Antidiabetic agent 15 (compound 1B15) acts as a dual inhibitor of AT1R and NEP, reducing oxidative stress and restoring mitochondrial membrane potential.Fórmula:C26H23NO5Forma y color:SolidPeso molecular:429.15762Nurr1 agonist 12
Nurr1 agonist 12 (Compound 37) acts as an agonist of the nuclear receptor-related protein 1 (Nurr1), enhancing its transcriptional activity with an EC50 of 0.06 μM. It stimulates human response elements NBRE, NurRE, and DR5 with EC50 values of 0.07 μM, 0.027 μM, and 0.014 μM, respectively. Additionally, Nurr1 agonist 12 induces the expression of neurotrophic genes regulated by Nurr1, such as tyrosine hydroxylase (TH), SOD1/2, BDNF, Sestrin 3, and BIRC5 (Survivin). The compound also demonstrates neuroprotective effects against neurotoxicity caused by Paraquat.Fórmula:C18H12ClN3OForma y color:SolidPeso molecular:321.76Myrciacetin
CAS:Myrciacetin from Rhododendron inhibits rat aldose reductase with IC50 of 13 μM.Fórmula:C17H16O6Forma y color:SolidPeso molecular:316.309Epi-Cryptoacetalide
Epi-Cryptoacetalide is a useful organic compound for research related to life sciences and the catalog number is T126054.Fórmula:C18H22O3Forma y color:SolidPeso molecular:286.371ODM-204
CAS:ODM-204 is novel nonsteroidal dual inhibitor of both androgen receptor and CYP17A1 enzyme(IC50s of 80 nM and 22 nM, respectively).Fórmula:C20H21F3N4Pureza:98%Forma y color:SolidPeso molecular:374.40MT-7716 hydrochloride
CAS:MT-7716 hydrochloride is a selective agonist of non-peptide nociceptin receptor (NOP)Fórmula:C27H29ClN4O2Pureza:98%Forma y color:SolidPeso molecular:477(S,S)-J-113397
CAS:(S,S)-J-113397 is an isomer of J-113397 . J-113397 is an Opioid Receptor antagonist [1] .Fórmula:C24H37N3O2Forma y color:SolidPeso molecular:399.57GPR88 agonist 2
GPR88 agonist 2 (compound 53) serves as a potent, brain-penetrant agonist of GPR88, exhibiting an EC50 of 14 µM in the GPR88 cAMP functional assay [1].Forma y color:Odour SolidGalloylalbiflorin
CAS:Galloylalbiflorin, an AR antagonist with IC50 53.3μM, is sourced from Paeonia lactiflora roots, exhibiting anti-androgenic properties.Fórmula:C30H32O15Forma y color:SolidPeso molecular:632.57TD-802
CAS:TD-802, an AR-targeting PROTAC with microsomal stability, shows promise for castration-resistant prostate cancer.Fórmula:C52H61ClN10O6Forma y color:SolidPeso molecular:957.56GNE-502
CAS:GNE-502 is an orally active and potent estrogen receptor (ER) degrader, specifically designed for research on breast cancer.Fórmula:C25H30FN3O3SForma y color:SolidPeso molecular:471.59Clocinnamox mesylate
CAS:Clocinnamox mesylate: irreversible μ-opioid blocker; Ki: 0.7 nM (mouse μ), 1.9 nM (δ), 5.7 nM (κ).Fórmula:C30H33ClN2O7SForma y color:SolidPeso molecular:601.11CP 85339
CAS:CP 85339 is an aspartic acid protease inhibitor for X-ray analysis of peptide-renin complexes.Fórmula:C31H49ClN4O6SForma y color:SolidPeso molecular:641.26PSDalpha
PSDalpha, a conjugate of PS, TB, and 17β-estradiol, degrades ERα with peak absorption at 465 nm, effectively inhibiting MCF-7 cell growth.Fórmula:C44H39N3O2SForma y color:SolidPeso molecular:673.86Bufrolin
CAS:Bufrolin is a potent GPR35 agonist, mast cell stabilizer, and anti-inflammatory research agent.Fórmula:C18H16N2O6Forma y color:SolidPeso molecular:356.33[Met5]-Enkephalin, amide
CAS:[Met5]-Enkephalin, amide activates δ and ζ opioid receptors; has multiple forms and varying plasma levels.Fórmula:C27H36N6O6SPureza:98%Forma y color:SolidPeso molecular:572.68Angiotensin II (1-4), human
CAS:Angiotensin II constricts blood vessels and boosts blood pressure by escalating norepinephrine release.Fórmula:C24H37N7O8Pureza:98%Forma y color:SolidPeso molecular:551.59

