Endocrinología / Hormonas
Los inhibidores de endocrinología/hormonas son compuestos que bloquean la acción de las hormonas o interfieren con las vías de señalización hormonal. Estos inhibidores son esenciales para estudiar la regulación de los sistemas endocrinos y para desarrollar tratamientos para enfermedades relacionadas con las hormonas, como la diabetes, los trastornos tiroideos y los cánceres dependientes de hormonas. Al modular la actividad hormonal, estos inhibidores pueden ayudar a dilucidar las complejas interacciones dentro del sistema endocrino. En CymitQuimica, ofrecemos una amplia gama de inhibidores de endocrinología/hormonas de alta calidad para apoyar su investigación en endocrinología, farmacología y ciencias médicas.
Subcategorías de "Endocrinología / Hormonas"
- Receptor de andrógenos(229 productos)
- Anexina A(16 productos)
- Aromatasa(22 productos)
- Receptor de estrógeno / progestágeno(64 productos)
- GPR(1 productos)
- Receptor de glucocorticoides(165 productos)
- LHRH(2 productos)
- Receptor de opioides(325 productos)
- Receptor de prostaglandinas(122 productos)
- RAAS(86 productos)
- Reductasa(51 productos)
- Somatostatina(57 productos)
- Receptor de la hormona tiroidea (THR)(32 productos)
- Receptor de vasopresina(48 productos)
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Se han encontrado 3369 productos de "Endocrinología / Hormonas"
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NH-3
CAS:NH-3, an orally active THR antagonist with a 55 nM IC50, blocks thyroid hormone binding and cofactor recruitment.Fórmula:C28H27NO6Pureza:97.79% - 99.40%Forma y color:SolidPeso molecular:473.52Ref: TM-T40548
1mg217,00€5mg550,00€10mg792,00€25mg1.206,00€50mg1.605,00€100mg2.175,00€500mg4.389,00€1mL*10mM (DMSO)492,00€AM-5262
CAS:AM-5262 is a potent GPR40 Full Agonist with improved rat PK profile and general selectivity profile.Fórmula:C33H35FO4Forma y color:SolidPeso molecular:514.63ER degrader 4
CAS:ER degrader 4, a selective and orally active compound, effectively degrades estrogen receptors and exhibits anti-tumor activity [1].Fórmula:C26H19FO4SForma y color:SolidPeso molecular:446.49ER ligand-6
CAS:ER ligand-6 serves as the target protein ligand for the PROTAC ER Degrader-14.
Fórmula:C29H32FNO4Forma y color:SolidPeso molecular:477.567ER ligand-7
ER ligand-7 is a ligand for the estrogen receptor (ER) that can be used as a target protein ligand for synthesizing PROTAC ER Degrader-15.
Fórmula:C27H23F4NO3Forma y color:SolidPeso molecular:485.47Tamoxifen-PEG-Clozapine
Tamoxifen-PEG-Clozapine is an estrogen receptor α (ERα) PROTAC degrader. It targets ERα for degradation through the ubiquitin-proteasome system by utilizing the E3 ubiquitin ligase component N-recognin 5. This compound is applicable in cancer research. (Pink: ERα inhibitor; Black: linker; Blue: CRBN Ligand)Fórmula:C54H63ClN6O7Forma y color:SolidPeso molecular:943.567Antidiabetic agent 15
Antidiabetic agent 15 (compound 1B15) acts as a dual inhibitor of AT1R and NEP, reducing oxidative stress and restoring mitochondrial membrane potential.Fórmula:C26H23NO5Forma y color:SolidPeso molecular:429.15762AR ligand-33
AR ligand-33 is a ligand for the androgen receptor (AR), and it can be used as a target protein ligand for the synthesis of PROTAC AR Degrader-8.Fórmula:C25H28N2O3Forma y color:SolidPeso molecular:404.501Nurr1 agonist 12
Nurr1 agonist 12 (Compound 37) acts as an agonist of the nuclear receptor-related protein 1 (Nurr1), enhancing its transcriptional activity with an EC50 of 0.06 μM. It stimulates human response elements NBRE, NurRE, and DR5 with EC50 values of 0.07 μM, 0.027 μM, and 0.014 μM, respectively. Additionally, Nurr1 agonist 12 induces the expression of neurotrophic genes regulated by Nurr1, such as tyrosine hydroxylase (TH), SOD1/2, BDNF, Sestrin 3, and BIRC5 (Survivin). The compound also demonstrates neuroprotective effects against neurotoxicity caused by Paraquat.Fórmula:C18H12ClN3OForma y color:SolidPeso molecular:321.76Paramethasone
CAS:Parametasone is a glucocorticoid with the general properties of corticosteroids.Fórmula:C22H29FO5Forma y color:SolidPeso molecular:392.46Myrciacetin
CAS:Myrciacetin from Rhododendron inhibits rat aldose reductase with IC50 of 13 μM.Fórmula:C17H16O6Forma y color:SolidPeso molecular:316.309Epi-Cryptoacetalide
Epi-Cryptoacetalide is a useful organic compound for research related to life sciences and the catalog number is T126054.Fórmula:C18H22O3Forma y color:SolidPeso molecular:286.371ODM-204
CAS:ODM-204 is novel nonsteroidal dual inhibitor of both androgen receptor and CYP17A1 enzyme(IC50s of 80 nM and 22 nM, respectively).Fórmula:C20H21F3N4Pureza:98%Forma y color:SolidPeso molecular:374.40MT-7716 hydrochloride
CAS:MT-7716 hydrochloride is a selective agonist of non-peptide nociceptin receptor (NOP)Fórmula:C27H29ClN4O2Pureza:98%Forma y color:SolidPeso molecular:477(S,S)-J-113397
CAS:(S,S)-J-113397 is an isomer of J-113397 . J-113397 is an Opioid Receptor antagonist [1] .Fórmula:C24H37N3O2Forma y color:SolidPeso molecular:399.57Human PTHrP-(1-36)
CAS:Human PTHrP-(1-36) is a secreted form of parathyroid hormone-related protein that exhibits anticalciuric effects and promotes beta cell function andFórmula:C191H305N59O52Forma y color:SolidPeso molecular:4259.83Demoxytocin
CAS:Demoxytocin, oxytocin analog, enhances smooth muscle contraction by increasing calcium ion permeability. Used in labor research.Fórmula:C43H65N11O12S2Forma y color:SolidPeso molecular:992.17PROTAC ER Degrader-12
PROTACER Degrader-12 (Compound 70) is an estrogen receptor PROTAC degrader with a degradation concentration (DC50) of less than 10 nM. It inhibits the proliferation of MCF-7 cells at a DC50 of under 10 nM and exhibits anticancer properties.Fórmula:C47H48F3N5O5Peso molecular:819.36075Angiotensin II (3-8), human TFA
Angiotensin II (3-8), human (TFA) is an angiotensin AT1 receptor agonist with less activity.Fórmula:C42H55F3N8O10Pureza:98%Forma y color:SolidPeso molecular:888.93
