
Transportador de membrana / canal de iones
Los inhibidores de transportadores de membrana y canales iónicos son compuestos que bloquean la función de proteínas responsables del transporte de iones, nutrientes y otras moléculas a través de las membranas celulares. Estos inhibidores son cruciales para estudiar la regulación de la homeostasis celular, la transducción de señales y la neurotransmisión. Los inhibidores de transportadores de membrana y canales iónicos también son importantes para desarrollar tratamientos para trastornos como la epilepsia, las enfermedades cardiovasculares y los síndromes metabólicos. En CymitQuimica, ofrecemos una amplia selección de inhibidores de alta calidad de transportadores de membrana y canales iónicos para apoyar su investigación en fisiología, neurociencia y farmacología.
Subcategorías de "Transportador de membrana / canal de iones"
- ABC(3 productos)
- ATPasa(93 productos)
- Receptor de adiponectina(5 productos)
- CFTR(64 productos)
- Receptor CGRP(52 productos)
- Canal de calcio(496 productos)
- Canal de cloruro(49 productos)
- Receptor GABA(336 productos)
- Transportador de monoamina(23 productos)
- Transportador de monocarboxilato(17 productos)
- NKCC(2 productos)
- NPC1L1(3 productos)
- Cotransportador de Na-K-Cl(8 productos)
- OAT(27 productos)
- OCT(7 productos)
- P-gp(53 productos)
- Canal de potasio(277 productos)
- Bomba de protones(39 productos)
- SGLT(30 productos)
- Canal de sodio(202 productos)
- Canal TRP / TRPV(93 productos)
Mostrar 13 subcategorías más
Se han encontrado 2290 productos de "Transportador de membrana / canal de iones"
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Ethacizine hydrochloride
CAS:<p>Ethacizine hydrochloride (NIK-244) has antiarrhythmic activity and can be used to study arrhythmias and myocardial infarction.</p>Fórmula:C22H28ClN3O3SPureza:98.08% - 98.08%Forma y color:SolidPeso molecular:449.99PF-05198007
CAS:PF-05198007 is a compound with a similar pharmacodynamic profile to PF-05089771. PF-05198007 is an effective and selective arylsulfonamide Nav1.7 inhibitor.Fórmula:C19H12ClF4N5O3S2Pureza:98%Forma y color:SolidPeso molecular:533.91Dipropofol
CAS:<p>Dipropofol (4,4-Bis(2,6-di-isopropylphenol)) is a small molecule GABAA receptor agonist that can be used to study epilepsy.</p>Fórmula:C24H34O2Pureza:99.51%Forma y color:SolidPeso molecular:354.53NS 383
CAS:<p>ASIC blocker with varying IC50: 0.12 μM in hASIC1a, and ineffective on hASIC2a/3; <5 μM on rASIC1a/2a/3; alleviates pain in inflamed/CCI rats.</p>Fórmula:C19H19N3O2Forma y color:SolidPeso molecular:321.37Lesinurad sodium
CAS:<p>Lesinurad sodium (RDEA594 sodium) is a selective inhibitor of uric acid reabsorption and is used in the study of cardiovascular diseases.</p>Fórmula:C17H13BrN3NaO2SPureza:99.97%Forma y color:SolidPeso molecular:426.26Lubiprostone hemiketal
CAS:Lubiprostone (hemiketal) (RU-0211 (hemiketal)), a selective activator of the chloride channel 2 (CLCN2), facilitates the treatment of chronic idiopathic constipation and opioid-induced constipation. It functions by enhancing CLCN2 channel activity, which boosts chloride ion secretion in the intestines, subsequently increasing fluid secretion and improving intestinal peristalsis. Additionally, Lubiprostone (hemiketal) may be utilized in research related to chronic constipation and cancer.Fórmula:C20H32F2O5Forma y color:SolidPeso molecular:390.46AM-2099
CAS:<p>AM-2099 is a selective voltage-gated sodium channel Nav1.7 inhibitor used in pain research.</p>Fórmula:C19H13F3N4O3S2Forma y color:SolidPeso molecular:466.46BTD
CAS:<p>BTD is a TRPC5 activator that activates heteromeric channel complexes composed of TRPC5 and its closest relatives TRPC1 or TRPC4.</p>Fórmula:C24H33N3O4SForma y color:SolidPeso molecular:459.6Vigabatrin Hydrochloride
CAS:<p>Vigabatrin Hydrochloride (γ-Vinyl-GABA hydrochloride) is a structural analog of the GABA, irreversibly inhibiting the catabolism of GABA by GABA transaminase.</p>Fórmula:C6H11NO2·HClPureza:98%Forma y color:SolidPeso molecular:165.62CGP 36742
CAS:<p>CGP 36742 blocks GABAB receptor, crosses blood-brain barrier, aids depression treatment (IC50: 32 μM).</p>Fórmula:C7H18NO2PForma y color:SolidPeso molecular:179.2Bamaquimast
CAS:Bamaquimast (L 0042) is a proton pump inhibitor for the study of asthma-like immune system disorders and respiratory diseases.Fórmula:C16H21N3O3Pureza:98.47%Forma y color:SolidPeso molecular:303.36Neosolaniol
CAS:Neosolaniol, a type A trichothecene mycotoxin produced by Fusarium species, strongly induces an anorectic (loss of appetite) response.Fórmula:C19H26O8Pureza:98%Forma y color:SolidPeso molecular:382.4Valnoctamide
CAS:Valnoctamide (Valmethamide) has antiepileptic and anticonvulsant activity and may be used in the study of neurological disorders.Fórmula:C8H17NOPureza:98%Forma y color:SolidPeso molecular:143.23Crinecerfont hydrochloride
CAS:<p>SSR-125543, a potent CRF1 receptor non-peptide antagonist, effective in CAH research, taken orally.</p>Fórmula:C27H29Cl2FN2OSForma y color:SolidPeso molecular:519.5Mepivacaine
CAS:<p>Mepivacaine (Carbocaine) is an amide local anesthetic, blocking sodium channels for nerve blocks and epidurals.</p>Fórmula:C15H22N2OPureza:99.35%Forma y color:SolidPeso molecular:246.35GYKI 52466 dihydrochloride
CAS:GYKI 52466 dihydrochloride is an AMPA/Kainate receptor antagonist with anticonvulsant activity and can be used to study neurological diseases.Fórmula:C17H17Cl2N3O2Pureza:99.38%Forma y color:SolidPeso molecular:366.24(+)-SJ733
CAS:<p>(+)-SJ733 (SJ000557733) is a potent Na+-ATPase PfATP4 inhibitor with antimalarial activity for the study of malaria.</p>Fórmula:C24H16F4N4O2Pureza:99.21%Forma y color:SolidPeso molecular:468.4(R)-3-Amino-4-hydroxybutanoic acid
CAS:<p>(R)-3-Amino-4-hydroxybutanoic acid,L-beta-Homoserine, is a full agonist at the human recombinant rho1 GABAC receptor, a modulator of GABAA and GABAB receptors.</p>Fórmula:C4H9NO3Pureza:99.92%Forma y color:SolidPeso molecular:119.12(R)-BPO-27
CAS:(R)-BPO-27 is an orally active and potent ATP-competitive CFTR inhibitor (IC50: 4 nM) for the study of diarrhoea and polycystic kidney.Fórmula:C26H18BrN3O6Pureza:99.1%Forma y color:SolidPeso molecular:548.34Fanapanel hydrate
CAS:<p>Fanapanel hydrate selectively blocks AMPA/kainate over NMDA; Ki: 3.2 nM (quisqualate), 100 nM (kainate), 8.5 μM (NMDA).</p>Fórmula:C14H17F3N3O7PForma y color:SolidPeso molecular:427.27
