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Transportador de membrana / canal de iones

Transportador de membrana / canal de iones

Los inhibidores de transportadores de membrana y canales iónicos son compuestos que bloquean la función de proteínas responsables del transporte de iones, nutrientes y otras moléculas a través de las membranas celulares. Estos inhibidores son cruciales para estudiar la regulación de la homeostasis celular, la transducción de señales y la neurotransmisión. Los inhibidores de transportadores de membrana y canales iónicos también son importantes para desarrollar tratamientos para trastornos como la epilepsia, las enfermedades cardiovasculares y los síndromes metabólicos. En CymitQuimica, ofrecemos una amplia selección de inhibidores de alta calidad de transportadores de membrana y canales iónicos para apoyar su investigación en fisiología, neurociencia y farmacología.

Subcategorías de "Transportador de membrana / canal de iones"

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Se han encontrado 2272 productos de "Transportador de membrana / canal de iones"

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  • Procyclidine hydrochloride

    CAS:
    <p>Procyclidine hydrochloride ((±)-Procyclidine hydrochlorid) is a potent anticholinergic agent and also have NMDA antagonist properties.</p>
    Fórmula:C19H30ClNO
    Pureza:99.24% - 99.88%
    Forma y color:Crystals From Petroleum Ether White Powder
    Peso molecular:323.9
  • CTP disodium dihydrate

    CAS:
    <p>CTP disodium dihydrate is an agonist of P2X4 purinergic receptor</p>
    Fórmula:C9H18N3Na2O16P3
    Pureza:98.51%
    Forma y color:White Crystalline Powder
    Peso molecular:563.15
  • AZ194

    CAS:
    <p>CRMP2-Ubc9-NaV1.7 inhibitor 194, is a CRMP2-Ubc9-NaV1.7 inhibitor.</p>
    Fórmula:C34H31F2N3O3
    Pureza:99.61%
    Forma y color:Solid
    Peso molecular:567.62
  • KPT185

    CAS:
    <p>KPT185 (KPT 185) is a selective CRM1 inhibitor, inducing apoptosis, cell-cycle arrest.</p>
    Fórmula:C16H16F3N3O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:355.31
  • JNJ 303

    CAS:
    <p>JNJ 303 is a potent blocker of IKs (IC50 : 64 nM).</p>
    Fórmula:C21H29ClN2O4S
    Pureza:99.28%
    Forma y color:Solid
    Peso molecular:440.98
  • PF-06869206

    CAS:
    <p>PF-06869206 is an oral selective inhibitor of the sodium-phosphate cotransporter NaPi2a (SLC34A1, IC50: 380 nM).</p>
    Fórmula:C15H14ClF3N4O2
    Pureza:99.79% - 99.88%
    Forma y color:Solid
    Peso molecular:374.75
  • Anthracene-9-carboxylic acid

    CAS:
    <p>Anthracene-9-carboxylic acid is an inhibitor of chloride transport with a moderate to strong inhibitory action on PKA activated cardiac IcI.</p>
    Fórmula:C15H10O2
    Pureza:99.05%
    Forma y color:Yellow Cystalline Powder
    Peso molecular:222.24
  • FGH10019

    CAS:
    <p>FGH10019 is a novel inhibitor of sterol regulatory element-binding protein (SREBP) ( IC50 :1 μM).</p>
    Fórmula:C18H19N3O2S2
    Pureza:98.93%
    Forma y color:Solid
    Peso molecular:373.49
  • Evenamide

    CAS:
    <p>Evenamide (NW-3509) is a sodium channel blocker. Which shows efficacy in a broad spectrum of rodent models of psychosis, mania, depression, and aggressiveness.</p>
    Fórmula:C16H26N2O2
    Pureza:96.74% - 99.15%
    Forma y color:Solid
    Peso molecular:278.39
  • Trofinetide

    CAS:
    <p>Trofinetide (NNZ-2566) is a synthetic analog of the endogenous N-terminus tripeptide. It has been shown to be neuroprotective in animal models of brain injury.</p>
    Fórmula:C13H21N3O6
    Pureza:98.70% - 99.50%
    Forma y color:Solid
    Peso molecular:315.32
  • Prilocaine

    CAS:
    <p>Prilocaine (NSC-40027) is a local anesthetic of the amino amide type, which acts on the sodium channel on the neuronal membrane and limits the spread of</p>
    Fórmula:C13H20N2O
    Pureza:98.49%
    Forma y color:Needles Solid
    Peso molecular:220.31
  • Transdermal Peptide Disulfide Acetate


    <p>Transdermal Peptide acetate(888486-23-5 free base) (TD 1 (peptide) acetate) is a 11-amino acid peptide, binds toNa+/K+-ATPase beta-subunit (ATP1B1), and mainly</p>
    Fórmula:C42H68N14O18S2
    Pureza:99.97%
    Forma y color:Solid
    Peso molecular:1121.2
  • Omecamtiv mecarbil

    CAS:
    <p>Omecamtiv mecarbil (CK-1827452) has been used in trials studying the treatment and basic science of Heart Failure, Echocardiogram, Pharmacokinetics, Chronic</p>
    Fórmula:C20H24FN5O3
    Pureza:98% - 99.23%
    Forma y color:Solid
    Peso molecular:401.43
  • 4-Chlorophenylguanidine hydrochloride

    CAS:
    <p>4-Chlorophenylguanidine hydrochloride is a potent inhibitor of urokinase selectivity.  </p>
    Fórmula:C7H9Cl2N3
    Pureza:99.75%
    Forma y color:Solid
    Peso molecular:206.07
  • HC067047 Hydrochloride(883031-03-6 free base)

    CAS:
    <p>HC-067047 hydrochloride, a TRPV4 antagonist, selectively inhibits human, rat, and mouse currents with IC50s: 486 nM, 133 nM, and 17 nM.</p>
    Fórmula:C26H29ClF3N3O2
    Pureza:99.95%
    Forma y color:Solid
    Peso molecular:507.98
  • Esomeprazole

    CAS:
    <p>Esomeprazole is the S-isomer of omeprazole, inhibits the lysosomal cysteine protease legumain to prevent cancer metastasis.</p>
    Fórmula:C17H19N3O3S
    Pureza:97.3%
    Forma y color:Solid
    Peso molecular:345.42
  • Epaminurad

    CAS:
    <p>Epaminurad (UR-1102) is an oral URAT1 inhibitor for gout research with a Ki of 0.057 μM, modestly affects OAT1/3.</p>
    Fórmula:C14H10Br2N2O3
    Forma y color:Solid
    Peso molecular:414.05
  • ML335

    CAS:
    <p>ML335 is a selective activator of TREK-1 and TREK-2.</p>
    Fórmula:C15H14Cl2N2O3S
    Pureza:99.73% - 99.79%
    Forma y color:Solid
    Peso molecular:373.25
  • Glibenclamide potassium

    CAS:
    <p>Glibenclamide potassium, a more soluble form of Glibenclamide, exists as anhydrous and hydrate salts.</p>
    Fórmula:C23H27ClKN3O5S
    Forma y color:Solid
    Peso molecular:532.09
  • JNJ-26990990

    CAS:
    <p>"JNJ-26990990: broad-spectrum anticonvulsant, less side effects than topiramate, potential for pain and depression treatment; Phase II in 2007."</p>
    Fórmula:C9H10N2O2S2
    Pureza:97.37%
    Forma y color:Solid
    Peso molecular:242.32