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Transportador de membrana / canal de iones

Transportador de membrana / canal de iones

Los inhibidores de transportadores de membrana y canales iónicos son compuestos que bloquean la función de proteínas responsables del transporte de iones, nutrientes y otras moléculas a través de las membranas celulares. Estos inhibidores son cruciales para estudiar la regulación de la homeostasis celular, la transducción de señales y la neurotransmisión. Los inhibidores de transportadores de membrana y canales iónicos también son importantes para desarrollar tratamientos para trastornos como la epilepsia, las enfermedades cardiovasculares y los síndromes metabólicos. En CymitQuimica, ofrecemos una amplia selección de inhibidores de alta calidad de transportadores de membrana y canales iónicos para apoyar su investigación en fisiología, neurociencia y farmacología.

Subcategorías de "Transportador de membrana / canal de iones"

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Se han encontrado 2275 productos de "Transportador de membrana / canal de iones"

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  • SG-209

    CAS:
    <p>SG 209 is an analog of nicorandil and acts as a K+ channel opener and nitrate-free coronary vasodilator.</p>
    Fórmula:C10H12N2O3
    Pureza:99.84%
    Forma y color:Solid
    Peso molecular:208.21
  • Prilocaine

    CAS:
    <p>Prilocaine (NSC-40027) is a local anesthetic of the amino amide type, which acts on the sodium channel on the neuronal membrane and limits the spread of</p>
    Fórmula:C13H20N2O
    Pureza:98.49%
    Forma y color:Needles Solid
    Peso molecular:220.31
  • Transdermal Peptide Disulfide Acetate


    <p>Transdermal Peptide acetate(888486-23-5 free base) (TD 1 (peptide) acetate) is a 11-amino acid peptide, binds toNa+/K+-ATPase beta-subunit (ATP1B1), and mainly</p>
    Fórmula:C42H68N14O18S2
    Pureza:99.97%
    Forma y color:Solid
    Peso molecular:1121.2
  • 4-Chlorophenylguanidine hydrochloride

    CAS:
    <p>4-Chlorophenylguanidine hydrochloride is a potent inhibitor of urokinase selectivity.  </p>
    Fórmula:C7H9Cl2N3
    Pureza:99.75%
    Forma y color:Solid
    Peso molecular:206.07
  • Piperazine

    CAS:
    <p>Piperazine (1,4-Diazacyclohexane), a gamma-aminobutyric acid (GABA) agonist, serves as a crucial building block and core component in a wide range of marketed drugs known for their varied pharmacological activities.</p>
    Fórmula:C4H10N2
    Forma y color:Solid
    Peso molecular:86.14
  • BAY-8002

    CAS:
    <p>BAY-8002 is a potent dual MCT1/2 inhibitor (IC50 values are 3, 8, and 12 nM at rat (C6), human (DLD-1) and mouse (4T1) MCT1 respectively).</p>
    Fórmula:C20H14ClNO5S
    Pureza:98.7% - 99.13%
    Forma y color:Solid
    Peso molecular:415.85
  • AZ194

    CAS:
    <p>CRMP2-Ubc9-NaV1.7 inhibitor 194, is a CRMP2-Ubc9-NaV1.7 inhibitor.</p>
    Fórmula:C34H31F2N3O3
    Pureza:99.61%
    Forma y color:Solid
    Peso molecular:567.62
  • Tiludronate

    CAS:
    <p>Tiludronate, an oral bisphosphonate, treats metabolic bone disorders and inhibits osteoclasts.</p>
    Fórmula:C7H9ClO6P2S
    Forma y color:Solid
    Peso molecular:318.61
  • Esomeprazole

    CAS:
    <p>Esomeprazole is the S-isomer of omeprazole, inhibits the lysosomal cysteine protease legumain to prevent cancer metastasis.</p>
    Fórmula:C17H19N3O3S
    Pureza:97.3%
    Forma y color:Solid
    Peso molecular:345.42
  • Trofinetide

    CAS:
    <p>Trofinetide (NNZ-2566) is a synthetic analog of the endogenous N-terminus tripeptide. It has been shown to be neuroprotective in animal models of brain injury.</p>
    Fórmula:C13H21N3O6
    Pureza:98.70% - 99.50%
    Forma y color:Solid
    Peso molecular:315.32
  • Epaminurad

    CAS:
    <p>Epaminurad (UR-1102) is an oral URAT1 inhibitor for gout research with a Ki of 0.057 μM, modestly affects OAT1/3.</p>
    Fórmula:C14H10Br2N2O3
    Forma y color:Solid
    Peso molecular:414.05
  • HC-030031

    CAS:
    <p>HC-030031 (TOSLAB 829227) is a potent TRPA1 inhibitor, which antagonizes AITC- and formalin-evoked calcium influx with IC50s of 6.2 and 5.3 μM, respectively.</p>
    Fórmula:C18H21N5O3
    Pureza:99.69% - ≥95%
    Forma y color:Solid
    Peso molecular:355.39
  • ML335

    CAS:
    <p>ML335 is a selective activator of TREK-1 and TREK-2.</p>
    Fórmula:C15H14Cl2N2O3S
    Pureza:99.73% - 99.79%
    Forma y color:Solid
    Peso molecular:373.25
  • JNJ-26990990

    CAS:
    <p>"JNJ-26990990: broad-spectrum anticonvulsant, less side effects than topiramate, potential for pain and depression treatment; Phase II in 2007."</p>
    Fórmula:C9H10N2O2S2
    Pureza:97.37%
    Forma y color:Solid
    Peso molecular:242.32
  • Ipidacrine

    CAS:
    <p>Ipidacrine (NIK‐247) (NIK‐247) is an Antidementia Agent</p>
    Fórmula:C12H16N2
    Pureza:97.73%
    Forma y color:Solid
    Peso molecular:188.27
  • Licarbazepine

    CAS:
    <p>Licarbazepine (10,11-hydroxy-10,11 Dihydrocarbamezer) is the pharmacologically active metabolite of oxcarbazepine, a drug indicated for the treatment of partial</p>
    Fórmula:C15H14N2O2
    Pureza:99.11%
    Forma y color:Solid
    Peso molecular:254.28
  • YHO-13177

    CAS:
    <p>YHO-13177 is a potent and specific inhibitor of BCRP; potentiated the cytotoxicity of SN-38 in cancer cells.</p>
    Fórmula:C20H22N2O3S
    Pureza:98.78%
    Forma y color:Solid
    Peso molecular:370.47
  • CFTR corrector 2

    CAS:
    <p>CFTR corrector 2 (FDL169) is a novel and potent CFTR corrector for treating cystic fibrosis (CF) patients who carry the F508del mutation.</p>
    Fórmula:C27H23FN4O4
    Pureza:99.66%
    Forma y color:Solid
    Peso molecular:486.49
  • N4-benzyl-N2-methylquinazoline-2,4-diamine hydrochloride

    CAS:
    <p>N4-benzyl-N2-methylquinazoline-2,4-diamine hydrochloride is an inhibitor of TRPC4.</p>
    Fórmula:C16H17ClN4
    Pureza:99.25%
    Forma y color:Solid
    Peso molecular:300.79
  • Enflurane

    CAS:
    <p>Enflurane (Efrane), a volatile anaesthetic, inhibits Ca2+-activated K+ channels and is used to gauge anesthesia levels in gas chromatography.</p>
    Fórmula:C3H2ClF5O
    Pureza:99.64%
    Forma y color:Clear Colorless Liquid Ordinary Temperature And Pressure Bp 56 8°C Density 1 50 G Cm-3 At Room Temperature Used As An
    Peso molecular:184.49