
Transportador de membrana / canal de iones
Los inhibidores de transportadores de membrana y canales iónicos son compuestos que bloquean la función de proteínas responsables del transporte de iones, nutrientes y otras moléculas a través de las membranas celulares. Estos inhibidores son cruciales para estudiar la regulación de la homeostasis celular, la transducción de señales y la neurotransmisión. Los inhibidores de transportadores de membrana y canales iónicos también son importantes para desarrollar tratamientos para trastornos como la epilepsia, las enfermedades cardiovasculares y los síndromes metabólicos. En CymitQuimica, ofrecemos una amplia selección de inhibidores de alta calidad de transportadores de membrana y canales iónicos para apoyar su investigación en fisiología, neurociencia y farmacología.
Subcategorías de "Transportador de membrana / canal de iones"
- ABC(3 productos)
- ATPasa(93 productos)
- Receptor de adiponectina(5 productos)
- CFTR(64 productos)
- Receptor CGRP(51 productos)
- Canal de calcio(493 productos)
- Canal de cloruro(49 productos)
- Receptor GABA(336 productos)
- Transportador de monoamina(23 productos)
- Transportador de monocarboxilato(17 productos)
- NKCC(2 productos)
- NPC1L1(3 productos)
- Cotransportador de Na-K-Cl(8 productos)
- OAT(27 productos)
- OCT(7 productos)
- P-gp(53 productos)
- Canal de potasio(276 productos)
- Bomba de protones(39 productos)
- SGLT(30 productos)
- Canal de sodio(202 productos)
- Canal TRP / TRPV(93 productos)
Mostrar 13 subcategorías más
Se han encontrado 2275 productos de "Transportador de membrana / canal de iones"
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SG-209
CAS:<p>SG 209 is an analog of nicorandil and acts as a K+ channel opener and nitrate-free coronary vasodilator.</p>Fórmula:C10H12N2O3Pureza:99.84%Forma y color:SolidPeso molecular:208.21Prilocaine
CAS:<p>Prilocaine (NSC-40027) is a local anesthetic of the amino amide type, which acts on the sodium channel on the neuronal membrane and limits the spread of</p>Fórmula:C13H20N2OPureza:98.49%Forma y color:Needles SolidPeso molecular:220.31Transdermal Peptide Disulfide Acetate
<p>Transdermal Peptide acetate(888486-23-5 free base) (TD 1 (peptide) acetate) is a 11-amino acid peptide, binds toNa+/K+-ATPase beta-subunit (ATP1B1), and mainly</p>Fórmula:C42H68N14O18S2Pureza:99.97%Forma y color:SolidPeso molecular:1121.24-Chlorophenylguanidine hydrochloride
CAS:<p>4-Chlorophenylguanidine hydrochloride is a potent inhibitor of urokinase selectivity. </p>Fórmula:C7H9Cl2N3Pureza:99.75%Forma y color:SolidPeso molecular:206.07Piperazine
CAS:<p>Piperazine (1,4-Diazacyclohexane), a gamma-aminobutyric acid (GABA) agonist, serves as a crucial building block and core component in a wide range of marketed drugs known for their varied pharmacological activities.</p>Fórmula:C4H10N2Forma y color:SolidPeso molecular:86.14BAY-8002
CAS:<p>BAY-8002 is a potent dual MCT1/2 inhibitor (IC50 values are 3, 8, and 12 nM at rat (C6), human (DLD-1) and mouse (4T1) MCT1 respectively).</p>Fórmula:C20H14ClNO5SPureza:98.7% - 99.13%Forma y color:SolidPeso molecular:415.85AZ194
CAS:<p>CRMP2-Ubc9-NaV1.7 inhibitor 194, is a CRMP2-Ubc9-NaV1.7 inhibitor.</p>Fórmula:C34H31F2N3O3Pureza:99.61%Forma y color:SolidPeso molecular:567.62Tiludronate
CAS:<p>Tiludronate, an oral bisphosphonate, treats metabolic bone disorders and inhibits osteoclasts.</p>Fórmula:C7H9ClO6P2SForma y color:SolidPeso molecular:318.61Esomeprazole
CAS:<p>Esomeprazole is the S-isomer of omeprazole, inhibits the lysosomal cysteine protease legumain to prevent cancer metastasis.</p>Fórmula:C17H19N3O3SPureza:97.3%Forma y color:SolidPeso molecular:345.42Trofinetide
CAS:<p>Trofinetide (NNZ-2566) is a synthetic analog of the endogenous N-terminus tripeptide. It has been shown to be neuroprotective in animal models of brain injury.</p>Fórmula:C13H21N3O6Pureza:98.70% - 99.50%Forma y color:SolidPeso molecular:315.32Epaminurad
CAS:<p>Epaminurad (UR-1102) is an oral URAT1 inhibitor for gout research with a Ki of 0.057 μM, modestly affects OAT1/3.</p>Fórmula:C14H10Br2N2O3Forma y color:SolidPeso molecular:414.05HC-030031
CAS:<p>HC-030031 (TOSLAB 829227) is a potent TRPA1 inhibitor, which antagonizes AITC- and formalin-evoked calcium influx with IC50s of 6.2 and 5.3 μM, respectively.</p>Fórmula:C18H21N5O3Pureza:99.69% - ≥95%Forma y color:SolidPeso molecular:355.39ML335
CAS:<p>ML335 is a selective activator of TREK-1 and TREK-2.</p>Fórmula:C15H14Cl2N2O3SPureza:99.73% - 99.79%Forma y color:SolidPeso molecular:373.25JNJ-26990990
CAS:<p>"JNJ-26990990: broad-spectrum anticonvulsant, less side effects than topiramate, potential for pain and depression treatment; Phase II in 2007."</p>Fórmula:C9H10N2O2S2Pureza:97.37%Forma y color:SolidPeso molecular:242.32Ipidacrine
CAS:<p>Ipidacrine (NIK‐247) (NIK‐247) is an Antidementia Agent</p>Fórmula:C12H16N2Pureza:97.73%Forma y color:SolidPeso molecular:188.27Licarbazepine
CAS:<p>Licarbazepine (10,11-hydroxy-10,11 Dihydrocarbamezer) is the pharmacologically active metabolite of oxcarbazepine, a drug indicated for the treatment of partial</p>Fórmula:C15H14N2O2Pureza:99.11%Forma y color:SolidPeso molecular:254.28YHO-13177
CAS:<p>YHO-13177 is a potent and specific inhibitor of BCRP; potentiated the cytotoxicity of SN-38 in cancer cells.</p>Fórmula:C20H22N2O3SPureza:98.78%Forma y color:SolidPeso molecular:370.47CFTR corrector 2
CAS:<p>CFTR corrector 2 (FDL169) is a novel and potent CFTR corrector for treating cystic fibrosis (CF) patients who carry the F508del mutation.</p>Fórmula:C27H23FN4O4Pureza:99.66%Forma y color:SolidPeso molecular:486.49N4-benzyl-N2-methylquinazoline-2,4-diamine hydrochloride
CAS:<p>N4-benzyl-N2-methylquinazoline-2,4-diamine hydrochloride is an inhibitor of TRPC4.</p>Fórmula:C16H17ClN4Pureza:99.25%Forma y color:SolidPeso molecular:300.79Enflurane
CAS:<p>Enflurane (Efrane), a volatile anaesthetic, inhibits Ca2+-activated K+ channels and is used to gauge anesthesia levels in gas chromatography.</p>Fórmula:C3H2ClF5OPureza:99.64%Forma y color:Clear Colorless Liquid Ordinary Temperature And Pressure Bp 56 8°C Density 1 50 G Cm-3 At Room Temperature Used As AnPeso molecular:184.49
