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Transportador de membrana / canal de iones

Transportador de membrana / canal de iones

Los inhibidores de transportadores de membrana y canales iónicos son compuestos que bloquean la función de proteínas responsables del transporte de iones, nutrientes y otras moléculas a través de las membranas celulares. Estos inhibidores son cruciales para estudiar la regulación de la homeostasis celular, la transducción de señales y la neurotransmisión. Los inhibidores de transportadores de membrana y canales iónicos también son importantes para desarrollar tratamientos para trastornos como la epilepsia, las enfermedades cardiovasculares y los síndromes metabólicos. En CymitQuimica, ofrecemos una amplia selección de inhibidores de alta calidad de transportadores de membrana y canales iónicos para apoyar su investigación en fisiología, neurociencia y farmacología.

Subcategorías de "Transportador de membrana / canal de iones"

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Se han encontrado 2272 productos de "Transportador de membrana / canal de iones"

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  • N-Acetylglycyl-D-glutamic acid

    CAS:
    <p>Excitatory peptide that induces seizures</p>
    Fórmula:C9H14N2O6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:246.22
  • Pradigastat

    CAS:
    <p>Pradigastat (LCQ-908) is a diacylglycerol acyltransferase 1 (DGAT1) inhibitor for the treatment of constipation and can be used in the study of obesity</p>
    Fórmula:C25H24F3N3O2
    Pureza:95.21% - 95.21%
    Forma y color:Solid
    Peso molecular:455.47
  • A-317491 sodium salt hydrate


    <p>A-317491 sodium salt hydrate is a non-nucleotide P2X3 and P2X2/3 receptor antagonist, which inhibits calcium flux mediated by the receptors.</p>
    Fórmula:C33H29NNaO9
    Pureza:98%
    Forma y color:Solid
    Peso molecular:606.57
  • MNI-caged-NMDA

    CAS:
    <p>NMDA caged with the photosensitive 4-methoxy-7-nitroindolinyl group</p>
    Fórmula:C14H17N3O6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:323.30
  • R-(-)-Niguldipine hydrochloride

    CAS:
    <p>R-(-)-Niguldipine HCl: L-type Ca2+ blocker, K+ agonist, α1A antagonist; lowers blood pressure; weaker enantiomer.</p>
    Fórmula:C36H40ClN3O6
    Forma y color:Solid
    Peso molecular:646.17
  • Clopamide

    CAS:
    <p>Clopamide (Brinaldix) is a piperidine and sulfamoylbenzamide-based diuretic with thiazide-like diuretic activity.</p>
    Fórmula:C14H20ClN3O3S
    Pureza:99.71%
    Forma y color:White To Yellowish Crystalline Powder
    Peso molecular:345.84
  • Verapamil

    CAS:
    <p>Verapamil (CP-16533-1), an oral calcium channel blocker, inhibits P-gp and CYP3A4, used for hypertension, arrhythmias, and angina research.</p>
    Fórmula:C27H38N2O4
    Pureza:99.61% - 99.93%
    Forma y color:Oil
    Peso molecular:454.6
  • IEM 1754 2HBr

    CAS:
    <p>IEM 1754 2HBr (IEM 1754 dihydrobromide) is a selective AMPA/kainate receptor blockers for GluR1 and GluR3 with IC50 of 6 μM.</p>
    Fórmula:C16H30N2·2HBr
    Pureza:99.71% - 99.72%
    Forma y color:Solid
    Peso molecular:412.25
  • Psora 4

    CAS:
    <p>Psora 4 (5-(4-Phenylbutoxy)psoralen) is a Kv1.3 blocker and a caloric restriction mimetic.</p>
    Fórmula:C21H18O4
    Forma y color:Solid
    Peso molecular:334.37
  • SCH 50911 hydrochloride

    CAS:
    <p>SCH 50911 hydrochloride is a selective, orally-active and competitive antagonist of γ-Aminobutyric acid B GABA(B) receptor(IC50 : 1.1 μM).</p>
    Fórmula:C8H16ClNO3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:209.67
  • PPNDS

    CAS:
    <p>P2X1 receptor antagonist</p>
    Fórmula:C18H15N4NaO14PS2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:629.42
  • NO 711

    CAS:
    <p>NO 711(NNC-711 free acid) is a selective inhibitor of GAT-1, which enhances non-rapid eye movement sleep, and prevents paclitaxel-induced neuropathic pain.</p>
    Fórmula:C21H22N2O3
    Pureza:99.70%
    Forma y color:Solid
    Peso molecular:350.41
  • (±)-Homoproline Hydrochloride

    CAS:
    <p>(±)-Homoproline Hydrochloride. Affordable Excellence: Reliable Quality You Can Trust</p>
    Fórmula:C6H12ClNO2
    Pureza:99.69%
    Forma y color:Solid
    Peso molecular:165.62
  • VU0405601

    CAS:
    <p>VU0405601 is a hERG channel activator that protects against drug-induced cardiac arrhythmias.</p>
    Fórmula:C17H13BrN2O2
    Pureza:99.16%
    Forma y color:Solid
    Peso molecular:357.2
  • JTV-519 hemifumarate

    CAS:
    <p>JTV-519 hemifumarate: Ca2+ blocker, SERCA inhibitor, ryanodine receptor partial agonist; antiarrhythmic, cardioprotective.</p>
    Fórmula:C54H68N4O8S2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:965.28
  • HN37

    CAS:
    <p>HN37, KCNQ2 activator (EC50=37 nM). Affordable Excellence: Reliable Quality You Can Trust</p>
    Fórmula:C20H21FN2O2
    Pureza:99.27%
    Forma y color:Solid
    Peso molecular:340.39
  • ICA

    CAS:
    <p>ICA (N-[4-(2-Pyridinyl)-2-thiazolyl]-2-pyridinamine) is a SK channel inhibitor and exhibits antileishmanial activity (IC50: 2.1 µM).</p>
    Fórmula:C13H10N4S
    Pureza:99.68%
    Forma y color:Solid
    Peso molecular:254.31
  • Benzamil hydrochloride

    CAS:
    <p>Benzamil hydrochloride is a specific and potent sodium channel (ENaC) blocker.</p>
    Fórmula:C13H15Cl2N7O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:356.21
  • V-9302

    CAS:
    <p>V-9302 (V9302) is a competitive antagonist of transmembrane glutamine flux that selectively and potently targets the amino acid transporter ASCT2 (IC50: 9.6 uM</p>
    Fórmula:C34H38N2O4
    Pureza:98% - 99.54%
    Forma y color:Solid
    Peso molecular:538.68
  • Nifekalant hydrochloride

    CAS:
    <p>Nifekalant hydrochloride is an IKr potassium channel blocker with an IC50 of 10 µM.</p>
    Fórmula:C19H28ClN5O5
    Pureza:99.91%
    Forma y color:Solid
    Peso molecular:441.91
  • CFTR corrector 9

    CAS:
    <p>CFTR corrector 9 is a CF modulator used to research cystic fibrosis and related disorders.</p>
    Fórmula:C16H14N2O4
    Pureza:98.24%
    Forma y color:Solid
    Peso molecular:298.29
  • L-4FPG

    CAS:
    <p>L-4FPG is a Glycine derivative, inhibits the neutral amino acid transporters ASCT1 and ASCT2.</p>
    Fórmula:C8H8FNO2
    Pureza:99.26%
    Forma y color:Solid
    Peso molecular:169.15
  • TRPC6-PAM-C20

    CAS:
    <p>TRPC6-PAM-C20, a selective enhancer for TRPC6, boosts calcium in HEK cells and OAG-related platelet clumping, EC50: 2.37μM.</p>
    Fórmula:C22H21NO4
    Pureza:98.16%
    Forma y color:Solid
    Peso molecular:363.41
  • CP-100356 hydrochloride

    CAS:
    <p>CP-100356 hydrochloride is an MDR1 (P-gp) and BCRP inhibitor, a nucleotide-derived substrate analog that induces stomatal opening in the dark.</p>
    Fórmula:C31H37ClN4O6
    Pureza:99.19%
    Forma y color:Solid
    Peso molecular:597.1
  • Nav1.7 inhibitor

    CAS:
    <p>Nav1.7 inhibitor is a Nav1.7 inhibitor for research in the field of pain and anesthesia.</p>
    Fórmula:C15H11Cl3FNO4S
    Pureza:97.52%
    Forma y color:Solid
    Peso molecular:426.68
  • CP-457920

    CAS:
    <p>CP-457920 is a selective α5 GABAA receptor inverse agonist that is suitable for investigating dementia in Alzheimer's disease.</p>
    Fórmula:C18H17N3O3
    Pureza:99.06% - 99.74%
    Forma y color:Solid
    Peso molecular:323.35
  • FSBA hydrochloride

    CAS:
    <p>FSBA hydrochloride(5'-p-Fluorosulfonylbenzoyladenosine) is an ATP analogue serving as an affinity probe for the ATP site of Na/K-ATPase.</p>
    Fórmula:C17H17ClFN5O7S
    Pureza:97.96%
    Forma y color:Solid
    Peso molecular:489.86
  • Sodium Channel inhibitor 2

    CAS:
    <p>Sodium Channel inhibitor 2 is a blocker of sodium channel.</p>
    Fórmula:C26H25Cl2N3O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:466.4
  • Cilobradine hydrochloride

    CAS:
    <p>Cilobradine hydrochloride (DK-AH 269) is an HCN Channel blocker and an open channel blocker of neuronal Ih and related cardiac If channels.</p>
    Fórmula:C28H39ClN2O5
    Pureza:98.40%
    Forma y color:Solid
    Peso molecular:519.07
  • TC-AQP1-1

    CAS:
    <p>TC-AQP1-1 blocks aquaporin 1; found via virtual screening; hinders water flux in Xenopus oocytes at low µM.</p>
    Fórmula:C12H10O4
    Pureza:97.59%
    Forma y color:Solid
    Peso molecular:218.21
  • Bamaluzole

    CAS:
    <p>Bamaluzole is an agonist of GABA receptor.</p>
    Fórmula:C14H12ClN3O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:273.72
  • BK 129

    CAS:
    <p>BK 129 is a local anesthetic with relaxant properties. BK 129 inhibits Ca2+ entry into the smooth muscle cell and Ca2+ release from sarcoplasmic reticulum.</p>
    Fórmula:C22H36N2O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:392.53
  • Almokalant

    CAS:
    <p>Almokalant: Class III antiarrhythmic, K+ channel blocker, inhibits Ikr current.</p>
    Fórmula:C18H28N2O3S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:352.49
  • V116517

    CAS:
    <p>V-116517, a TRPV1 antagonist, is used potentially for the treatment of severe pain due to osteoarthritis and chronic pain due postherpetic neuralgia (PHN).</p>
    Fórmula:C19H18ClF3N4O3
    Forma y color:Solid
    Peso molecular:442.82
  • AMG8788

    CAS:
    <p>AMG8788 is a selective, potent and orally active TRPM8 antagonist (IC50: 63.2 nM).</p>
    Fórmula:C23H18F4N2O
    Forma y color:Solid
    Peso molecular:414.4
  • JTV-519 fumarate

    CAS:
    <p>Ryanodine receptor (RyR) inhibitor; stabilizes RyR2 in a closed conformation. Exhibits antiarrhythmic and cardioprotective properties in vivo.</p>
    Fórmula:C29H36N2O6S
    Forma y color:Solid
    Peso molecular:540.67
  • PD 122860

    CAS:
    <p>PD 122860 is a dihydropyridine enhancing heart contractility, altering ECG, and relaxing aortic rings.</p>
    Fórmula:C23H20F3N3O4S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:491.48
  • DS1

    CAS:
    <p>DS1 is a GABAA receptor agonist which can stimulate gonadotropin subunit gene expression in mouse.</p>
    Fórmula:C18H10Br2ClN3OS
    Forma y color:Solid
    Peso molecular:511.62
  • Sodium Channel inhibitor 1

    CAS:
    <p>Sodium Channel inhibitor1 is a novel and selective voltage-gated sodium channel for pain treatment.</p>
    Fórmula:C24H19F4N3O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:473.42
  • VU625

    CAS:
    <p>VU625 (VU007625) is an AeKir1 inhibitor (IC50: 96.8nM) that acts as a mosquito killer and inhibits AeKir1-mediated currents.</p>
    Fórmula:C19H22N2O4S
    Pureza:99.08%
    Forma y color:Solid
    Peso molecular:374.45
  • Terodiline

    CAS:
    <p>Terodiline is an orally available selective muscarinic M1 receptor and calcium channel antagonist for the study of diseases caused by abnormal bladder function.</p>
    Fórmula:C20H27N
    Pureza:98.20% - 99.59%
    Forma y color:Solid
    Peso molecular:281.44
  • Asivatrep

    CAS:
    <p>Asivatrep (PAC14028) is a selective and potent antagonist of transient receptor potential vanilloid subtype 1 (TRPV1) for the study of atopic dermatitis.</p>
    Fórmula:C21H22F5N3O3S
    Pureza:95.13%
    Forma y color:Solid
    Peso molecular:491.48
  • AMG9678

    CAS:
    <p>AMG9678 is a selective, potent, orally active TRPM8 antagonist (IC50: 31.2 nM).</p>
    Fórmula:C20H18F6N2O
    Forma y color:Solid
    Peso molecular:416.36
  • Topiramate lithium

    CAS:
    <p>Topiramate lithium: antiepileptic, GluR5 antagonist, enhances GABA, inhibits kainate/AMPA, Na+/Ca2+ channels; ↑ K+ conductance; ↓ carbonic anhydrase.</p>
    Fórmula:C12H20LiNO8S
    Forma y color:Solid
    Peso molecular:345.29
  • MC-70

    CAS:
    <p>MC-70 is a potent P-glycoprotein (P-gp) inhibitor (EC50 = 0.69 μM).</p>
    Fórmula:C24H25NO3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:375.46
  • ORM-10962

    CAS:
    <p>ORM-10962 is a potent, highly selective inhibitor of sodium-calcium exchanger (NCX) (for the reverse and forward mode inhibition with IC50 values of 67 and 55</p>
    Fórmula:C27H29N3O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:459.54
  • Caldaret

    CAS:
    <p>Caldaret is an intracellular Ca2+ handling modulator that acts through reverse mode Na+/Ca2+ exchanger inhibition.</p>
    Fórmula:C11H16N2O3S
    Forma y color:Solid
    Peso molecular:256.32
  • UBP 296

    CAS:
    <p>GluR5-subunit containing kainate receptor antagonist</p>
    Fórmula:C15H15N3O6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:333.3
  • Y 23684

    CAS:
    <p>Y-23684 is an anxiolytic drug with a novel chemical structure. It has similar effects to benzodiazepine drugs and is classed as a nonbenzodiazepine anxiolytic.</p>
    Fórmula:C18H13ClN2O2S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:356.83
  • Nav1.7-IN-3

    CAS:
    <p>Nav1.7-IN-3 is a selective and orally bioavailable inhibitor of voltage-gated sodium channel Nav1.7(IC50 of 8 nM).</p>
    Fórmula:C17H20ClFN4O2S2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:430.95
  • CGP 46381

    CAS:
    <p>CGP 46381 is a GABAB receptor antagonist.</p>
    Fórmula:C10H22NO2P
    Pureza:98%
    Forma y color:White Solid
    Peso molecular:219.26
  • YS-201

    CAS:
    <p>YS-201 is an antagonist of dihydropyridine-type calcium channel.</p>
    Fórmula:C24H31N3O6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:457.52
  • IEM 1460

    CAS:
    <p>AMPA receptors blocker</p>
    Fórmula:C19H38Br2N2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:454.33
  • (S)-ML753286

    CAS:
    <p>(S)-ML753286 is a breast cancer resistance protein (BCRP) inhibitor (IC50: 0.6 μM on BCRP efflux transporter).</p>
    Fórmula:C20H25N3O3
    Forma y color:Solid
    Peso molecular:355.43
  • Indantadol HCl

    CAS:
    <p>Indantadol HCl (CHF-3381) is a NMDA antagonist and nonselective MAO inhibitor.</p>
    Fórmula:C11H15ClN2O
    Pureza:98.24%
    Forma y color:Solid
    Peso molecular:226.7
  • GABAA receptor agent 5

    CAS:
    <p>Compound 018 is a potent γ-GABAAR antagonist, Ki of 0.020 μM, with low membrane permeability.</p>
    Fórmula:C21H25N3O2S
    Forma y color:Solid
    Peso molecular:383.51
  • CP-409092 hydrochloride

    CAS:
    <p>CP-409092 hydrochloride is a partial agonist of the GABAA receptor with anti-anxiety activity.</p>
    Fórmula:C17H20ClN3O2
    Forma y color:Solid
    Peso molecular:333.81
  • BGT1-IN-9

    CAS:
    <p>BGT1-IN-9 is an M1 muscarinic agonist.</p>
    Fórmula:C5H10ClN3O2
    Forma y color:Solid
    Peso molecular:179.605
  • Atomoxetine

    CAS:
    <p>Atomoxetine (HSDB 7352) is a selective norepinephrine inhibitor that may cause an increase in blood pressure by increasing norepinephrine concentrations in</p>
    Fórmula:C17H21NO
    Pureza:98%
    Forma y color:Solid
    Peso molecular:255.35
  • Flordipine

    CAS:
    <p>Flordipine is used as a calcium channel blocker.</p>
    Fórmula:C26H33F3N2O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:510.55
  • Omeprazole magnesium

    CAS:
    <p>Omeprazole magnesium: oral PPI that reduces stomach acid, treats acid reflux and heartburn.</p>
    Fórmula:C34H36MgN6O6S2
    Forma y color:Solid
    Peso molecular:713.12
  • Ro 04-5595 hydrochloride

    CAS:
    <p>NR2B-containing NMDA receptors antagonist</p>
    Fórmula:C19H23Cl2NO2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:368.3
  • TTA-Q6(isomer)

    CAS:
    <p>TTA-Q6(isomer) is an isomer of TTA-Q6. TTA-Q6 is a selective antagonist of the T-type Ca2+ channel.</p>
    Fórmula:C20H15ClF3N3O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:405.8
  • Apimostinel

    CAS:
    <p>Apimostinel (NRX-1074; AGN-241660) is a partial agonist of NMDA receptor.</p>
    Fórmula:C25H37N5O6
    Forma y color:Solid
    Peso molecular:503.59
  • NMDA receptor antagonist 4

    CAS:
    <p>NMDA antagonist 4 (IIc) is an oral, voltage-dependent blocker with IC50 of 1.93 μM and may penetrate the BBB, useful in Alzheimer's research.</p>
    Fórmula:C15H18FN
    Forma y color:Solid
    Peso molecular:231.31
  • Istaroxime

    CAS:
    <p>Istaroxime is an effective inhibitor of Na+, K+-ATPase (IC50: 0.11 μM).</p>
    Fórmula:C21H32N2O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:360.49
  • JNJ-56022486

    CAS:
    <p>JNJ-56022486 is a selective TARP γ‑8 AMPA receptor modulator.</p>
    Fórmula:C15H10ClN3O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:283.71
  • KCa1.1 channel activator-2


    <p>KCa1.1 channel activator-2, a Quercetin hybrid, selectively stimulates vascular KCa1.1 channel, with strong myorelaxant effects.</p>
    Fórmula:C23H22O8S2
    Forma y color:Solid
    Peso molecular:490.55
  • PPDA

    CAS:
    <p>Subtype-selective NMDA receptor antagonist</p>
    Fórmula:C21H18N2O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:378.38
  • (R)-3C4HPG

    CAS:
    <p>NMDA and AMPA/kainate receptor antagonist</p>
    Fórmula:C9H9NO5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:211.17
  • GoSlo-SR-5-69

    CAS:
    <p>BK channel activator (EC50 = 251 nM). Shifts the voltage required for half maximal negatively (DV1/2 = -104 mV).</p>
    Fórmula:C24H20N2NaO5S
    Forma y color:Solid
    Peso molecular:471.48
  • Hyperforin dicyclohexylammonium salt

    CAS:
    <p>Hyperforin dicyclohexylammonium is a TRPC6 activator and antidepressant that modulates Ca2+ levels.</p>
    Fórmula:C47H75NO4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:718.1
  • TRPC6-IN-2

    CAS:
    <p>TRPC6-IN-2 is a TRPC protein inhibitor, specifically inhibiting TRPC6 protein.</p>
    Fórmula:C19H17Cl2FN6
    Forma y color:Solid
    Peso molecular:419.28
  • Metapramine

    CAS:
    <p>Metapramine, a tricyclic antidepressant, blocks norepinephrine reuptake and is a low-affinity NMDA antagonist.</p>
    Fórmula:C16H18N2
    Pureza:99.03% - 99.67%
    Forma y color:Solid
    Peso molecular:238.33
  • SB-237376 HCl

    CAS:
    <p>SB-237376 HCl (SB-237376 hydrochloride) is a calcium and potassium channel antagonist used in the treatment of cardiac arrhythmias.</p>
    Fórmula:C20H26ClN3O5
    Pureza:98.70%
    Forma y color:Solid
    Peso molecular:423.89
  • GNE-5729

    CAS:
    <p>GNE-5729 is a positive allosteric modulator of NMDAR blood-brain barrier orally available, GluN2A, GluN2C and GluN2D, neurological and psychiatric disorders.</p>
    Fórmula:C17H10Cl2F3N5O
    Pureza:99.40% - 99.85%
    Forma y color:Solid
    Peso molecular:428.2
  • JNc-440

    CAS:
    <p>JNc-440, a strong anti-hypertensive, boosts TRPV4-KCa2.3 interaction and vasodilation, lowering blood pressure in mice.</p>
    Fórmula:C26H24N4O3
    Forma y color:Solid
    Peso molecular:440.49
  • ML252

    CAS:
    <p>ML252 selectively inhibits KCNQ2 (IC50=69nM) and Cytochrome P450 isoforms CYP1A2, CYP2C9, CYP3A4, CYP2D6 with low nanomolar IC50s.</p>
    Fórmula:C20H24N2O
    Forma y color:Solid
    Peso molecular:308.42
  • XPC-6444

    CAS:
    <p>XPC-6444 is a isoform-selective, and CNS-penetrant inhibitor of NaV1.6 with IC50 of41 nM for hNaV1.6,with anticonvulsant activity.</p>
    Fórmula:C22H25F3N4O2S2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:498.58
  • (BrMT)2

    CAS:
    <p>(BrMT)2 is an activator of the Kv1.1 potassium ion channel.</p>
    Fórmula:C20H20Br2N4S2
    Forma y color:Solid
    Peso molecular:540.34
  • RPR-260243

    CAS:
    <p>RPR-260243 is a novel activator of HERG and modifies HERG currents inhibited by dofetilide (IC50 = 58 nM).</p>
    Fórmula:C28H25F3N2O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:510.5
  • β-CCB

    CAS:
    <p>benzodiazepine receptor ligand</p>
    Fórmula:C16H16N2O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:268.31
  • UCL-1848 trifluoroacetate salt

    CAS:
    <p>UCL-1848 trifluoroacetate salt is a selective Ca2+-activated, SK potassium channel blocker.</p>
    Fórmula:C32H34F6N4O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:652.638
  • UBP714

    CAS:
    <p>UBP714, derived from UBP608, boosts NMDAR in CA1 hippocampus, promising for schizophrenia and cognitive deficits treatment.</p>
    Fórmula:C11H7BrO4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:283.07
  • ZD-9379

    CAS:
    <p>ZD-9379 is a NMDA receptor antagonist.</p>
    Fórmula:C19H14ClN3O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:383.79
  • Ro 8-4304 hydrochloride

    CAS:
    <p>Ro 8-4304 hydrochloride is a NMDA receptor antagonist.</p>
    Fórmula:C21H24ClFN2O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:406.88
  • YM 244769 hydrochloride

    CAS:
    <p>inhibitor of the reverse mode of Na+/Ca2+ exchange (NCX)</p>
    Fórmula:C26H23ClFN3O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:479.93
  • WX-081

    CAS:
    <p>WX-081 is an anti-TB drug effective against DS-TB (MIC: 0.083 μg/ml) and MDR-TB strains (MIC: 0.11 μg/ml) with hERG inhibition (IC50: 1.89 μM).</p>
    Fórmula:C34H33ClN2O2
    Forma y color:Solid
    Peso molecular:537.09
  • RH 3421

    CAS:
    <p>RH 3421 is used as a neuroactive dihydropyrazole insecticide.</p>
    Fórmula:C20H17ClF3N3O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:439.82
  • Ro 25-6981 HCl

    CAS:
    <p>Ro 25-6981 HCl is an effective and selective NMDA glutamate receptors containing the NR2B subunit antagonist.</p>
    Fórmula:C22H30ClNO2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:375.93
  • Biricodar dicitrate

    CAS:
    <p>Biricodar dicitrate (VX-710) is a potent MDR inhibitor with no anticancer activity and can be used to study prostate cancer.</p>
    Fórmula:C46H57N3O21
    Pureza:97.78% - 99.78%
    Forma y color:Solid
    Peso molecular:987.95
  • Sabiporide

    CAS:
    <p>Sabiporide is a NHE-1 inhibitor and a cardioprotective agent.</p>
    Fórmula:C18H20ClF3N6O2
    Forma y color:Solid
    Peso molecular:444.84
  • LY339434

    CAS:
    <p>LY339434 is a potent and selective agonist of the kainate receptor GluK1, GluR5.</p>
    Fórmula:C18H19NO4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:313.35
  • Abeprazan

    CAS:
    <p>Abeprazan is a potassium-competitive acid blocker targeting acid-related diseases without acid activation.</p>
    Fórmula:C19H17F3N2O3S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:410.41
  • Homoquinolinic acid

    CAS:
    <p>NMDA receptor agonist</p>
    Fórmula:C8H7NO4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:181.15
  • CCD-3693

    CAS:
    <p>CCD-3693 is a gamma-aminobutyric acid (GABA) receptor agonist.</p>
    Fórmula:C21H31F3O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:372.46
  • GABA-AT-IN-1

    CAS:
    <p>GABA-AT-IN-1 (Compound 6) is an inhibitor of γ-aminobutyric acid transaminase (GABA-AT) that crosses the blood-brain barrier.</p>
    Fórmula:C23H18N2O6
    Forma y color:Solid
    Peso molecular:418.4
  • KRN4884

    CAS:
    <p>KRN 4884 activates KATP channels (EC50=0.55 μM) at 0.1-3 μM with 1 mM ATP.</p>
    Fórmula:C15H14ClN5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:299.76
  • Farnesyl pyrophosphate

    CAS:
    <p>Farnesyl pyrophosphate: 15-C isoprenoid, TRPM2 agonist, crucial for cholesterol, ubiquinones, protein farnesylation, and GGPP synthesis.</p>
    Fórmula:C15H28O7P2
    Forma y color:Solid
    Peso molecular:382.33
  • Picoprazole

    CAS:
    <p>Picoprazole is a specific H+/K+-ATPase inhibitor (IC50 of 3.1±0.4 μM).</p>
    Fórmula:C17H17N3O3S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:343.4
  • Nav1.8-IN-2

    CAS:
    <p>Nav1.8-IN-2 (compound 35A) strongly inhibits Nav1.8 (IC50: 0.4 nM), useful for researching pain, cough, and pruritus.</p>
    Fórmula:C18H13Cl2F3N2O3
    Forma y color:Solid
    Peso molecular:433.21
  • FR-168888 mesylate

    CAS:
    <p>FR-168888, a new Na+/H+ exchange inhibitor, can protect the heart from arrhythmia and myocardial cell death in ischemic and reperfused situations.</p>
    Fórmula:C14H18N4O5S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:354.38
  • Istaroxime oxalate

    CAS:
    <p>Istaroxime (PST-2744) is a positive inotrope that inhibits Na+/K+ ATPase, raising intracellular sodium and calcium levels.</p>
    Fórmula:C23H34N2O7
    Forma y color:Solid
    Peso molecular:450.53
  • Terodiline hydrochloride

    CAS:
    <p>Terodiline hydrochloride is an antagonist of M1-selective muscarinic receptor (mAChR)(Kbs of 15, 160, 280, and 198 nM in rabbit vas deferens (M1), atria (M2),</p>
    Fórmula:C20H28ClN
    Pureza:98%
    Forma y color:Solid
    Peso molecular:317.9
  • Nav1.7-IN-6

    CAS:
    <p>Nav1.7-IN-6, a selective inhibitor of Nav1.7.</p>
    Fórmula:C25H25ClF6N2O4S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:598.99
  • PKF050-638

    CAS:
    <p>PKF050-638 disrupts CRM1-NES, inhibits HIV-1 Rev export; selective with IC50=0.04 μM.</p>
    Fórmula:C13H13ClN4O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:292.72
  • Lemildipine

    CAS:
    <p>Lemildipine is a new blocker of dihydropyridine calcium entry.</p>
    Fórmula:C20H22Cl2N2O6
    Forma y color:Solid
    Peso molecular:457.3
  • CGP 36216 hydrochloride

    CAS:
    <p>CGP 36216 hydrochloride is a potent and selective antagonist of GABAB receptors (IC50: 43 μM).</p>
    Fórmula:C5H14NO2P
    Pureza:98%
    Forma y color:Solid
    Peso molecular:151.14
  • CP-465022 (maleate)

    CAS:
    <p>CP-465022 Maleate: A selective noncompetitive AMPA antagonist with IC50 of 25 nM, showing anticonvulsant effects and useful for AMPA-related studies.</p>
    Fórmula:C30H28ClFN4O5
    Forma y color:Solid
    Peso molecular:579.02
  • TC-T 6000

    CAS:
    <p>TC-T 6000 (hENT4-IN-1) is an ENT4 inhibitor with vasodilator activity that inhibits hENT1 and hENT2 for the study of cancer and cardiovascular damage.</p>
    Fórmula:C26H48N8O2
    Pureza:98.14%
    Forma y color:Solid
    Peso molecular:504.71
  • GNE-6901

    CAS:
    <p>GNE-6901 is a selective GluN2A PAM.</p>
    Fórmula:C18H17FN2O3S
    Forma y color:Solid
    Peso molecular:360.4
  • Diproteverine

    CAS:
    <p>Diproteverine is a calcium antagonist, it has antianginal property.</p>
    Fórmula:C26H35NO4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:425.56
  • Nav1.1 activator 1

    CAS:
    <p>Nav1.1 activator 1 is a highly potent activator of Nav1.1 with BBB penetration.</p>
    Fórmula:C24H23F3N4O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:440.46
  • NMDA receptor antagonist 5

    CAS:
    <p>Compound 10e: potent, non-toxic, brain-permeable NMDA receptor antagonist; key for neurological research.</p>
    Fórmula:C19H16BrNO2
    Forma y color:Solid
    Peso molecular:370.24
  • (S)-(-)-HA 966

    CAS:
    <p>(S)-(-)-HA 966 is a NMDA receptor antagonist.</p>
    Fórmula:C4H8N2O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:116.12
  • Nav1.7-IN-2

    CAS:
    <p>Nav1.7-IN-2 is avoltage-gated sodium channels (Nav) inhibitor in particular Nav 1.7(IC50 of 80 nM).</p>
    Fórmula:C22H22FN5O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:407.44
  • KRP-199

    CAS:
    <p>KRP-199, a highly potent and selective antagonist for the AMPA receptors, exhibits good neuroprotective effects in vivo.</p>
    Fórmula:C22H14F3N5O7
    Pureza:98%
    Forma y color:Solid
    Peso molecular:517.37
  • GABAA receptor agent 8

    CAS:
    <p>Compound 5e, a GABAA receptor modulator, shows potent anticonvulsant effects with low neurotoxicity for epilepsy research.</p>
    Fórmula:C19H16N4O
    Forma y color:Solid
    Peso molecular:316.36
  • Aprindine hydrochloride

    CAS:
    <p>Aprindine HCl, a Class 1b antiarrhythmic, treats heart arrhythmias, outperforming digoxin in delaying atrial fibrillation. It's effective orally.</p>
    Fórmula:C22H31ClN2
    Forma y color:Solid
    Peso molecular:358.95
  • UBP141

    CAS:
    <p>UBP141 is a antagonist of N-methyl-D-aspartate (NMDA) receptor.</p>
    Fórmula:C21H18N2O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:378.38
  • NHE3-IN-3

    CAS:
    <p>NHE3-IN-3 inhibits human/rat NHE3 with pIC50s 6.2/6.6; 98% oral bioavailability in rats.</p>
    Fórmula:C16H16Cl2N2O2S
    Forma y color:Solid
    Peso molecular:371.28
  • 3-Chlorodiphenylamine

    CAS:
    3-Cl-DPA, a cardiac troponin activator, acts by a mechanism distinct from bepridil or TFP.
    Fórmula:C12H10ClN
    Forma y color:Solid
    Peso molecular:203.67
  • Eltanexor Z-isomer

    CAS:
    <p>Eltanexor Z-isomer, less active than KPT-8602, inhibits Z138, MM1S, and 3T3 cells with IC50s: 100 nM-50 μM, &lt;100 nM, &gt;30 μM.</p>
    Fórmula:C17H10F6N6O
    Forma y color:Solid
    Peso molecular:428.29
  • KMUP-4

    CAS:
    <p>Kmup-4 is an enhancer of cGMP activity and an aortic smooth muscle relaxant.</p>
    Fórmula:C19H23N7O4
    Forma y color:Solid
    Peso molecular:413.43
  • H100

    CAS:
    <p>H100 inhibits Cl- transport, mildly affects NaK2Cl cotransporter and Band 3 anion exchanger, not KCl cotransporter.</p>
    Fórmula:C18H16N2O6S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:388.4
  • LY 233536

    CAS:
    <p>LY 233536 is a novel, competitive antagonist of NMDA receptor.</p>
    Fórmula:C12H19N5O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:265.31
  • L-701252

    CAS:
    <p>L-701252, a potent glycine site NMDA receptor antagonist, exhibits an inhibition concentration (IC50) of 420 nM.</p>
    Fórmula:C13H10ClNO3
    Pureza:97.7%
    Forma y color:White Crystalline Solid
    Peso molecular:263.68
  • D-AP4

    CAS:
    <p>broad spectrum excitatory amino acid receptor antagonist</p>
    Fórmula:C4H10NO5P
    Pureza:98%
    Forma y color:White Powder
    Peso molecular:183.1
  • GSK-5503A

    CAS:
    <p>GSK-5503A is a novel channel blocker of CRAC.</p>
    Fórmula:C23H17F2N3O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:405.4
  • UT-B-IN-1

    CAS:
    <p>UT-B-IN-1: reversible UT-B inhibitor, IC50: 10 nM (human), 25 nM (mouse), low toxicity, diuretic research tool.</p>
    Fórmula:C20H17N5O2S3
    Forma y color:Solid
    Peso molecular:455.58
  • Quinine hemisulfate

    CAS:
    <p>Quinidine: antiarrhythmic, orally active, inhibits cytochrome P450db, blocks K+ channels (IC50: 19.9μM), may aid in malaria research.</p>
    Fórmula:C40H50N4O8S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:746.92
  • (RS)-CPP

    CAS:
    <p>(RS)-CPP is a NMDA antagonist.</p>
    Fórmula:C8H17N2O5P
    Pureza:98%
    Forma y color:Solid
    Peso molecular:252.2
  • PF-05214030

    CAS:
    <p>PF-05214030 is a novel potent TRPV4 antagonist (hTRPV4 IC50 4nM; rTRPV4 IC50 27nM).</p>
    Fórmula:C17H13Cl2FN2O4S
    Forma y color:Solid
    Peso molecular:431.27
  • FG8119

    CAS:
    <p>FG8119 is a novel benzodiazepine agonist with potential anticonvulsant and antiepileptic activity for the study of neurological disorders.</p>
    Fórmula:C17H15N5O2
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:321.33
  • GABAA receptor agent 6

    CAS:
    <p>GABAA receptor agent 6 (compound 2027) is a potent γ-GABAAR antagonist with low cellular membrane permeability (Ki = 0.56 μM) [1].</p>
    Fórmula:C18H25N3O2
    Forma y color:Solid
    Peso molecular:315.41
  • GSK-5498A

    CAS:
    <p>GSK-5498A: Selective CARC blocker, inhibits release of mediators from mast cells and cytokines from T-cells (IC50, 1 μM).</p>
    Fórmula:C18H11F6N3O
    Forma y color:Solid
    Peso molecular:399.29
  • TB 21007

    CAS:
    <p>GABAA receptor inverse agonist</p>
    Fórmula:C15H17NO2S3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:339.5
  • D-3263

    CAS:
    <p>D-3263 is an agonist of transient receptor potential melatonin member 8 (TRPM8) with potential antitumor activity.</p>
    Fórmula:C21H31N3O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:373.49
  • Gea 857

    CAS:
    <p>Gea 857 is a potassium conductance putative blocker.</p>
    Fórmula:C15H22ClNO2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:283.79
  • N20C hydrochloride

    CAS:
    <p>N20C hydrochloride (2-((3,3-diphenylpropyl)amino)acetamide hydrochloride) is a non-competitive NMDA receptor open-channel blocker.</p>
    Fórmula:C17H21ClN2O
    Pureza:99.9%
    Forma y color:Solid
    Peso molecular:304.81
  • PNU 37883 hydrochloride

    CAS:
    <p>Kir6 (KATP) channel antagonist</p>
    Fórmula:C21H36ClN3O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:381.98
  • TRPC5-IN-1

    CAS:
    <p>TRPC5-IN-1 is a TRPC5 inhibitor active in various animal models of chronic kidney disease.</p>
    Fórmula:C20H16N4O
    Forma y color:Solid
    Peso molecular:328.37
  • 4-(Phenyldiazenyl)benzoic acid

    CAS:
    <p>4-(Phenyldiazenyl)benzoic acid is a photosensitive and photoswitchable TRPA1 agonist that can be used as pharmacological tool to study pain signaling.</p>
    Fórmula:C13H10N2O2
    Forma y color:Solid
    Peso molecular:226.23
  • MPO-IN-5

    CAS:
    <p>MPO-IN-5: strong, irreversible MPO blocker; IC50s: 0.22 μM for peroxidation, 2.8 μM for hERG.</p>
    Fórmula:C24H24N6O2
    Forma y color:Solid
    Peso molecular:428.49
  • KC 12291 hydrochloride

    CAS:
    <p>voltage-gated sodium channel blocker</p>
    Fórmula:C22H28ClN3O3S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:449.99
  • NMDA receptor potentiator-1

    CAS:
    <p>Compound 1368 is a selective NMDA receptor enhancer; IC50s: 4 μM for NR2C, 5 μM for NR2D.</p>
    Fórmula:C26H26ClNO5
    Forma y color:Solid
    Peso molecular:467.94
  • (RS)-3,4-DCPG

    CAS:
    <p>antagonist of AMPA receptors and agonist of mGluR8</p>
    Fórmula:C10H9NO6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:239.18
  • SOCE inhibitor 1

    CAS:
    <p>SOCE inhibitor 1 is a inhibitor of store-operated calcium entry (SOCE)(IC50 of 4.4 μM).</p>
    Fórmula:C25H22F3N5O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:513.47
  • ZAPA sulfate

    CAS:
    <p>GABAA receptors agonist</p>
    Fórmula:C4H8N2O6S2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:244.25
  • NMDA receptor modulator 5

    CAS:
    <p>NMDA receptor modulator 5 (Compound 195), a potent NMDA receptor modulator, exhibits potential for neurological disorder research [1].</p>
    Fórmula:C14H11F3N2O3S
    Forma y color:Solid
    Peso molecular:344.31
  • TPMPA

    CAS:
    <p>GABAA-ρ antagonist</p>
    Fórmula:C6H12NO2P
    Pureza:98%
    Forma y color:Solid
    Peso molecular:161.14
  • Glisoxepide

    CAS:
    <p>Glisoxepide: sulphonamide, oral K(ATP) blocker, antihyperglycemic, affects heart.</p>
    Fórmula:C20H27N5O5S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:449.52
  • JNJ-55511118

    CAS:
    <p>JNJ-55511118 is a TARP γ8 allosteric modulator with anticonvulsant activity, which can be used in research on chronic operant alcohol self-administration.</p>
    Fórmula:C14H8ClF3N2O2
    Forma y color:Solid
    Peso molecular:328.67
  • S3337

    CAS:
    <p>S3337 is an inhibitor of H+, K+-ATPase</p>
    Fórmula:C18H21N3O3S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:359.44
  • (2R,3S)-Chlorpheg

    CAS:
    <p>(2R,3S)-Chlorpheg is a NMDA receptor antagonist.</p>
    Fórmula:C11H12ClNO4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:257.67
  • PF-0713

    CAS:
    <p>PF 0713, a GABAA receptor agonist, is used as an intravenous sedative-hypnotic for general anaesthesia, ICU sedation, procedural sedation, chemotherapy.</p>
    Fórmula:C14H22O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:206.32
  • Lidoflazine

    CAS:
    <p>Lidoflazine: antianginal, blocks HERG K+ &amp; Ca channels, risks QT prolongation &amp; arrhythmia.</p>
    Fórmula:C30H35F2N3O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:491.62
  • NMDA receptor modulator 3

    CAS:
    <p>NMDA receptor modulator 3 (Compound 99) is a potent modulator of NMDA receptor that can be used in the research of neurological disorder [1].</p>
    Fórmula:C12H9F3N2O2S
    Forma y color:Solid
    Peso molecular:302.27
  • Corrector C4

    CAS:
    <p>Corrector C4, a corrector commonly used to study cystic fibrosis mutants, works by alleviating the interaction between CFTR transmembrane domain mutants and</p>
    Fórmula:C21H17ClN4O2S2
    Pureza:98.36%
    Forma y color:Solid
    Peso molecular:456.97
  • CAY10719

    CAS:
    <p>CAY10719 selectively inhibits ABCG2 (IC50 = 0.23 μM), reverses SN 38 resistance, and inhibits ATPase, with low ABCG1 activity.</p>
    Fórmula:C25H20Cl2N2O2
    Forma y color:Solid
    Peso molecular:451.34
  • TG41

    CAS:
    <p>TG41 is a GABAA receptors positive modulator.</p>
    Fórmula:C18H13BrCl2N2O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:440.12
  • MK-7145

    CAS:
    <p>MK-7145 is an inhibitor of ROMK(IC50 of 0.045 μM).</p>
    Fórmula:C26H30N2O6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:466.53
  • RN-9893 (hydrochloride)

    CAS:
    <p>RN-9893 is a TRPV4 antagonist with human/rat IC50s of 0.42/0.66 μM; selective over TRPV1, TRPV3, TRPM8. Reduces rat TRPV4 activity (IC50: 0.57-2.1 μM).</p>
    Fórmula:C21H24ClF3N4O5S
    Forma y color:Solid
    Peso molecular:536.95
  • (S)-Lercanidipine hydrochloride

    CAS:
    <p>(S)-Lercanidipine hydrochloride is the S-enantiomer of Lercanidipine hydrochloride. (S)-lercanidipine hydrochloride is a potent blocker of calcium channel.</p>
    Fórmula:C36H42ClN3O6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:648.19
  • Kadethrin

    CAS:
    <p>Kadethrin is a synthetic pyrethroid. It was used as a pesticide.</p>
    Fórmula:C23H24O4S
    Pureza:98%
    Forma y color:Yellow-Brown Viscous Oil Solid
    Peso molecular:396.5
  • HZ166

    CAS:
    <p>HZ-166 is a positive GABAA receptor modulator and a GABAA receptor subtype-selective benzodiazepine site ligand.</p>
    Fórmula:C21H16N4O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:356.38
  • NCS-382

    CAS:
    <p>γ-Hydroxybutyric acid antagonist</p>
    Fórmula:C13H14O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:218.25
  • L-trans-2,4-PDC

    CAS:
    <p>L-trans-2,4-PDC is an EAAT1-4 inhibitor/non-transportable EAAT5 inhibitor.</p>
    Fórmula:C6H9NO4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:159.14
  • Anipamil

    CAS:
    <p>Anipamil is a long-acting blocker of calcium channel,and for the treatment of cardiovascular disease.</p>
    Fórmula:C34H52N2O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:520.79
  • SL-651498

    CAS:
    <p>SL-651498, a GABAA receptor agonist, is used potentially for the treatment of anxiety.</p>
    Fórmula:C23H20FN3O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:389.42
  • Norbormide

    CAS:
    <p>Norbormide is a toxic compound used as a rodenticide. It has several mechanisms of action, acting as a vasoconstrictor and calcium channel blocker.</p>
    Fórmula:C33H25N3O3
    Pureza:98%
    Forma y color:Crystals From Methylene Chloride + Ether Norbormide Is A Colorless To Off-White Crystalline Powder Used As A Selective Rat Poison (Epa 1998)
    Peso molecular:511.57
  • Neramexane Mesylate

    CAS:
    <p>Neramexane: NMDA &amp; nicotinic receptor blocker with neuroprotective, antidepressant, and cognitive-enhancing effects.</p>
    Fórmula:C12H27NO3S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:265.41
  • Dofequidar

    CAS:
    <p>Dofequidar (MS-209 free base) is a quinoline derivative that inhibits the efflux of chemotherapeutic agents.</p>
    Fórmula:C30H31N3O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:481.59
  • MRS4719

    CAS:
    <p>MRS4719: potent P2X4 antagonist, IC50 0.503 μM. Reduces infarct, brain atrophy, Ca2+ influx. Used in ischemic stroke research.</p>
    Fórmula:C26H13N5O3S·C6H15N
    Forma y color:Solid
    Peso molecular:504.6
  • Clathrodin

    CAS:
    <p>Clathrodin is a voltage-gated sodium (NaV) channels modulator.</p>
    Fórmula:C11H13N5O
    Forma y color:Solid
    Peso molecular:231.25
  • GABAA receptor agent 4

    CAS:
    <p>Compound 1e is a potent γ-GABAAR antagonist with a Ki of 0.18 µM, offering immunomodulatory effects on T cell proliferation.</p>
    Fórmula:C17H24N2O
    Forma y color:Solid
    Peso molecular:272.39
  • UBP 302

    CAS:
    <p>UBP 302 is a selective GLUK5 kainate receptor antagonist with Kd 402 nM; low GluK2 affinity.</p>
    Fórmula:C15H15N3O6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:333.3
  • GNE-0439

    CAS:
    <p>GNE-0439 is a Nav1.7-selective inhibitor (IC50 0.34 μM), also targeting Nav1.5 and mutant N1742K channels, valuable for ion channel research.</p>
    Fórmula:C21H31NO3
    Pureza:99.60%
    Forma y color:Solid
    Peso molecular:345.48
  • Ro 41-3290

    CAS:
    <p>Ro 41-3290 is the desethylated derivative of Ro 41-3696, which is an agonist of nonbenzodiazepine partial at the benzodiazepine receptor.</p>
    Fórmula:C24H21ClN2O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:420.89
  • BIIB-513

    CAS:
    <p>BIIB-513 is an inhibitor of Na+/H+ exchange.</p>
    Fórmula:C19H25N5O8S2
    Forma y color:Solid
    Peso molecular:515.56
  • RuBi-4AP

    CAS:
    <p>voltage-dependent K+ channel blocker</p>
    Fórmula:C30H28Cl2N8Ru
    Pureza:98%
    Forma y color:Solid
    Peso molecular:672.57
  • (S)-(-)-5-Iodowillardiine

    CAS:
    <p>hGluR5 kainate receptor agonist</p>
    Fórmula:C7H8IN3O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:325.06
  • Laniquidar

    CAS:
    <p>Laniquidar (R101933) inhibits P-glycoprotein (IC50: 0.51 μM), poor oral bioavailability, modulates drug resistance transporters.</p>
    Fórmula:C37H36N4O3
    Forma y color:Solid
    Peso molecular:584.71
  • LUF7346

    CAS:
    <p>LUF7346 is an allosteric modulator of hERG.</p>
    Fórmula:C20H15BrN2O3
    Forma y color:Solid
    Peso molecular:411.25
  • Lu AE98134

    CAS:
    <p>Lu AE98134 enhances Nav1.1, Nav1.2, and Nav1.5 sodium channels, but not Nav1.4/1.6/1.7; studied in CNS diseases like schizophrenia.</p>
    Fórmula:C21H23N5O3S
    Forma y color:Solid
    Peso molecular:425.5
  • YS-035 hydrochloride

    CAS:
    <p>inhibitor of outward K+ currents</p>
    Fórmula:C21H30ClNO4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:395.92
  • VU0529331

    CAS:
    <p>VU0529331 activates non-GIRK1 potassium channels (EC50: ~5.1 μM GIRK2, 5.2 μM GIRK1/2) and GIRK4 channels.</p>
    Fórmula:C22H20N6O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:384.43
  • QAQ dichloride

    CAS:
    <p>QAQ dichloride is a photoswitchable blocker of Na v/K v channels, active in trans form, and a light-sensitive analgesic targeting pain neurons.</p>
    Fórmula:C28H44N6O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:496.69
  • CGP11952

    CAS:
    <p>CGP11952 is same the benzodiazepines in its pharmacological action and it also is an experimental benzodiazepine derivative.</p>
    Fórmula:C21H21Cl2N5O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:446.33
  • Cyphenothrin

    CAS:
    <p>Cyphenothrin, a synthetic pyrethroid, combats carbamate-resistant cockroaches.</p>
    Fórmula:C24H25NO3
    Forma y color:Faint Yellow Sticky Liquid
    Peso molecular:375.46
  • AMP-PNP tetralithium

    CAS:
    <p>AMP analog that blocks Kir6 channels, inhibits axonal transport, and stabilizes organelle-microtubule interactions.</p>
    Fórmula:C10H13Li4N6O12P3
    Forma y color:Solid
    Peso molecular:529.93
  • ML67-33

    CAS:
    <p>ML67-33 selectively activates K2P channels; EC50: 36.3 μM (cell-free), 9.7 μM (HEK293). Reversible TREK-1 modulation.</p>
    Fórmula:C18H17Cl2N5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:374.27
  • Pregabalin arenacarbil

    CAS:
    <p>Pregabalin arenacarbil is a gabamimetic.</p>
    Fórmula:C15H27NO6
    Forma y color:Solid
    Peso molecular:317.38
  • Alilusem

    CAS:
    <p>Alilusem is a new diuretic that is beneficial to the clinical treatment of hypertension.</p>
    Fórmula:C17H15ClKN2O5S
    Forma y color:Solid
    Peso molecular:433.92
  • TRPV antagonist 1

    CAS:
    <p>TRPV antagonist 1 is an antagonist of transient receptor potential vanilloid (TRPV; IC50 &lt; 250 nM).</p>
    Fórmula:C26H21F3N2O4S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:514.52
  • URAT1 inhibitor 4

    CAS:
    <p>URAT1 inhibitor 4 is a potent, orally active Lesinurad derivative with a 7.56 μM IC50, showing greater in vivo efficacy.</p>
    Fórmula:C27H20BrN3O4S3
    Forma y color:Solid
    Peso molecular:626.56
  • UK-52831

    CAS:
    <p>UK-52831, a calcium channel antagonist, is used potentially for the treatment of hypertension and myocardia ischemia.</p>
    Fórmula:C22H26Cl2N6O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:525.39
  • DS2

    CAS:
    <p>Positive allosteric modulator of δ-subunit containing GABAA receptors</p>
    Fórmula:C18H12ClN3OS
    Pureza:98%
    Forma y color:Solid
    Peso molecular:353.83
  • ATPA

    CAS:
    <p>ATPA activates GluR5 glutamate receptors; EC50s range 0.66-32 μM across GluR5 variants.</p>
    Fórmula:C10H16N2O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:228.24
  • Ro 19-4603

    CAS:
    <p>Benzodiazepine inverse agonist</p>
    Fórmula:C15H17N3O3S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:319.38