Transportador de membrana / canal de iones
Los inhibidores de transportadores de membrana y canales iónicos son compuestos que bloquean la función de proteínas responsables del transporte de iones, nutrientes y otras moléculas a través de las membranas celulares. Estos inhibidores son cruciales para estudiar la regulación de la homeostasis celular, la transducción de señales y la neurotransmisión. Los inhibidores de transportadores de membrana y canales iónicos también son importantes para desarrollar tratamientos para trastornos como la epilepsia, las enfermedades cardiovasculares y los síndromes metabólicos. En CymitQuimica, ofrecemos una amplia selección de inhibidores de alta calidad de transportadores de membrana y canales iónicos para apoyar su investigación en fisiología, neurociencia y farmacología.
Subcategorías de "Transportador de membrana / canal de iones"
- ABC(3 productos)
- ATPasa(97 productos)
- Receptor de adiponectina(5 productos)
- CFTR(66 productos)
- Receptor CGRP(51 productos)
- Canal de calcio(573 productos)
- Canal de cloruro(54 productos)
- Receptor GABA(371 productos)
- Transportador de monoamina(30 productos)
- Transportador de monocarboxilato(18 productos)
- NKCC(2 productos)
- NPC1L1(3 productos)
- Cotransportador de Na-K-Cl(10 productos)
- OAT(32 productos)
- OCT(7 productos)
- P-gp(55 productos)
- Canal de potasio(302 productos)
- Bomba de protones(42 productos)
- SGLT(31 productos)
- Canal de sodio(257 productos)
- Canal TRP / TRPV(96 productos)
Mostrar 13 subcategorías más
Se han encontrado 2703 productos de "Transportador de membrana / canal de iones"
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Z433927330
CAS:Z433927330 is a potent and selective Aquaporin-7 (AQP7) inhibitor(IC50s of 0.2).
Fórmula:C20H20N4O3Pureza:99.78%Forma y color:SolidPeso molecular:364.4Caloxin 2A1 TFA
Caloxin 2A1 TFA is a PM Ca2+ pump inhibitor that inhibits human red blood cell Ca2+-Mg2+-ATPase leakage.Fórmula:C66H92F3N19O24Pureza:99.89%Forma y color:SolidPeso molecular:1592.55AZD 7009
CAS:AZD 7009 is a novel antiarrhythmic compound that inhibits the sodium current of hNav1.5 in CHO K1 cells with an IC50 of 11 uM.Fórmula:C23H34N4O5Pureza:98.42% - 98.51%Forma y color:SoildPeso molecular:446.54Vocacapsaicin hydrochloride
CAS:Vocacapsaicin hydrochloride (CA-008 hydrochloride) is a non-opioid TRPV1 agonist, a raw material for capsaicin, and is used for pain relief.Fórmula:C26H42ClN3O4Pureza:99.66% - 99.80%Forma y color:SolidPeso molecular:496.08Cycloleucine
CAS:Cycloleucine is an antagonist of NMDA receptor associated glycine receptor with a Ki of 600 μM.Fórmula:C6H11NO2Pureza:99.90%Forma y color:SolidPeso molecular:129.16CIQ
CAS:CIQ is a subunit-selective potentiator of NMDA receptors containing the NR2C or NR2D subunit. EC50 value: 2.7 μM for NR2C and 2.8 μM for NR2D.Fórmula:C26H26ClNO5Pureza:99.5%Forma y color:SolidPeso molecular:467.94Flumazenil
CAS:Flumazenil (Ro 15-1788) antagonizes the benzodiazepine binding site of the gamma-aminobutyric acid (GABA)/benzodiazepine receptor complex in the central nervousFórmula:C15H14FN3O3Pureza:99.72% - 99.98%Forma y color:Less Crystals Colourless CrystalsPeso molecular:303.29Trichlormethiazide
CAS:Trichlormethiazide (Naqua) is a short-acting, 3-dichloromethyl derivative of hydrochlorothiazide, belonging to the class of thiazide diuretics.Fórmula:C8H8Cl3N3O4S2Pureza:98.8% - 99.54%Forma y color:SolidPeso molecular:380.66DCPIB
CAS:DCPIB, a known specific and potent inhibitor of volume-regulated anion channels (VRAC),DCPIB displayed superior selectivity toward TRESK with an IC50 of 0.14 μMFórmula:C22H28Cl2O4Pureza:99.79% - 99.87%Forma y color:SolidPeso molecular:427.36Ref: TM-T10979
2mg39,00€5mg57,00€10mg87,00€25mg177,00€50mg301,00€100mg485,00€200mg690,00€1mL*10mM (DMSO)63,00€Indapamide
CAS:Indapamide (Noranat) is a non-thiazide sulphonamide diuretic compound, generally used in the treatment of hypertension, as well as decompensated cardiac failure.Fórmula:C16H16ClN3O3SPureza:98.97% - 99.83%Forma y color:SolidPeso molecular:365.835,5-Dimethyloxazolidine-2,4-dione
CAS:5,5-Dimethyloxazolidine-2,4-dione (Dimethadione) is an anticonvulsant that is the active metabolite of TRIMETHADIONE.Fórmula:C5H7NO3Pureza:99.12%Forma y color:Drypowder PelletslargecrystalsPeso molecular:129.11Disopyramide
CAS:Disopyramide, or Triombrin, a class I anti-arrhythmic with membrane-stabilizing effects, has heart depressant, anticholinergic, and anesthetic properties.Fórmula:C21H29N3OPureza:99.62%Forma y color:SolidPeso molecular:339.47Ethaverine hydrochloride
CAS:Ethaverine hydrochloride is a homologue of papaverine and is used as a vasodilator and antispasmodic.Cost-effective and quality-assured.Fórmula:C24H30ClNO4Pureza:99.66% - 99.90%Forma y color:SolidPeso molecular:431.96Ref: TM-T0369
2mg44,00€5mg63,00€10mg102,00€25mg167,00€50mg250,00€100mg358,00€200mg530,00€1mL*10mM (DMSO)85,00€NMDA-IN-1
CAS:NMDA-IN-1 is a potent and NR2B-selective antagonist of NMDA(NMDA Ki of 0.85 nM; NR2B Ca2+ influx IC50 is 9.7 nM).Fórmula:C20H23ClFN3OPureza:99.57%Forma y color:SolidPeso molecular:375.87VU6036720
VU6036720 is a potent and selective inhibitor of the isomeric Kir4.1/5.1.VU6036720 inhibits Kir4.1/5.1 activity by decreasing the channel open-circuit
Fórmula:C20H22ClFN4O2SPureza:98.1%Forma y color:SoildPeso molecular:436.93Eleclazine hydrochloride
CAS:Eleclazine hydrochloride (GS 6615 hydrochloride) is a novel inhibitor of late Na+ current (IC50: 0.7 uM).Fórmula:C21H17ClF3N3O3Pureza:99.86%Forma y color:SolidPeso molecular:451.83Ref: TM-T15207
1mg58,00€5mg110,00€10mg166,00€25mg268,00€50mg403,00€100mg532,00€200mg705,00€1mL*10mM (DMSO)122,00€Dooku1
CAS:Dooku1, Yoda1 analog, blocks Piezo1 channels, halting Ca2+ entry. IC50: 1.3μM in HEK 293, 1.5μM in HUVEC, stops Yoda1's aortic relaxation.Fórmula:C13H9Cl2N3OSPureza:98.87% - 99.74%Forma y color:SolidPeso molecular:326.2Ref: TM-T11076
1mg43,00€2mg56,00€5mg93,00€10mg133,00€25mg259,00€50mg482,00€100mg695,00€1mL*10mM (DMSO)90,00€Penicillin G sodium salt
CAS:Penicillin G sodium(Benzylpenicillin sodium) salt is a penicillin derivative commonly used in the form of its sodium or potassium salts in the treatment of a
Fórmula:C16H17N2NaO4SPureza:98.11%Forma y color:White To Off-White Crystalline PowderPeso molecular:356.37Diphenidol hydrochloride
CAS:Diphenidol hydrochloride (Difenidol hydrochloride), a muscarinic antagonist, is employed as an anti-vertigo and as an antiemetic drug.Fórmula:C21H28ClNOPureza:99.15% - 99.33%Forma y color:Crystals Soluble In Methanol WaterPeso molecular:345.91Tocainide hydrochloride
CAS:Tocainide hydrochloride (2-amino-n-(2,6-dimethylphenyl)propanamide hydrochloride) is a sodium channel blocker.Fórmula:C11H17ClN2OPureza:97%Forma y color:SolidPeso molecular:228.723,4,5-Trimethoxycinnamic acid
CAS:3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) (TMCA) is one of the constituents of Polygalae Radix and may exert anti-seizure activity by acting at theFórmula:C12H14O5Pureza:98.91%Forma y color:SolidPeso molecular:238.24MRZ 2-514
CAS:MRZ 2-514 (8-bromo-4,5-dihydroxypyridazino[4,5-b]quinolin-1-one) is a strychnine-insensitive modulatory site of the NMDA receptor (glycineB)antagonist with KiFórmula:C11H6BrN3O3Pureza:98.459%Forma y color:SolidPeso molecular:308.09Ref: TM-T12110
1mg92,00€5mg192,00€10mg313,00€25mg620,00€50mg1.044,00€100mg1.404,00€1mL*10mM (DMSO)212,00€Moxidectin
CAS:Moxidectin (CL301423) is an anthelmintic for heartworm/intestinal worms in dogs, cats, horses, cattle, and sheep; oral/topical/injectable.Fórmula:C37H53NO8Pureza:97.38%Forma y color:Appearance White Or Pale Yellow Amorphous PowderPeso molecular:639.82Bemegride
CAS:Bemegride (3-Ethyl-3-methylglutarimide), a central nervous system stimulant, serves as an antidote for barbiturate poisoning.Fórmula:C8H13NO2Pureza:99.89%Forma y color:Physical Description White Crystalline Solid Sublimes At 212°F And 200 Mm Pressure (Ntp 1992)Peso molecular:155.19NS13001
CAS:NS13001, an oral SK channel modulator, shows promise for SCA2 therapy; EC50: 1.8 µM (SK2), 0.14 µM (SK3).Fórmula:C17H16ClN7Pureza:99.55%Forma y color:SolidPeso molecular:353.81Riparin III
CAS:Riparin III is an alcamide isolated from Aniba riparia that has exhibited effects of antidepressant and anxiolytic activities in acute stress behavioral models.Fórmula:C16H17NO4Pureza:95.13%Forma y color:SolidPeso molecular:287.31Flindokalner
CAS:Flindokalner (BMS-204352) modulates potassium channels, enhances Kv7 subtypes and BKca, inhibits Kv7.1 (Ki=3.7μM), GABAA; has anxiolytic effects in vivo.Fórmula:C16H10ClF4NO2Pureza:99.96%Forma y color:SolidPeso molecular:359.7TPC2-A1-P
CAS:TPC2-A1-P is a TPC2 agonist that can differentially activate two-pore channel 2 (TPC2) and mimic the activation of TPC2 with NAADP and PIP (2).Fórmula:C20H21BrF3NO3Pureza:98.49%Forma y color:SolidPeso molecular:460.29Ref: TM-T36806
1mg92,00€5mg225,00€10mg374,00€25mg710,00€50mg1.153,00€100mg1.755,00€1mL*10mM (DMSO)226,00€Manidipine dihydrochloride
CAS:Manidipine dihydrochloride (Manidipine 2HCl) is a potent calcium channel blocker for Ca2+ current(IC50=2.6 nM).Fórmula:C35H40Cl2N4O6Pureza:99.76% - 99.86%Forma y color:SolidPeso molecular:683.62Torsemide
CAS:Torsemide (AC-4464), a sulfonylurea loop diuretic, has a long action duration, high plasma protein binding, and a long half-life.Fórmula:C16H20N4O3SPureza:99.81%Forma y color:Crystalline SolidPeso molecular:348.42Lotilaner
CAS:Lotilaner is a parasiticide.Fórmula:C20H14Cl3F6N3O3SPureza:99.56%Forma y color:SolidPeso molecular:596.76Ref: TM-T15775
1mg44,00€2mg58,00€5mg94,00€10mg144,00€25mg335,00€50mg550,00€100mg882,00€200mg1.188,00€1mL*10mM (DMSO)111,00€Baclofen
CAS:Baclofen (Lioresal), a chlorophenyl-butanoic acid derivative, treats spasms from spinal cord injury and MS by mimicking GABA at GABA-B receptors.Fórmula:C10H12ClNO2Pureza:98% - >99.99%Forma y color:1992)Peso molecular:213.66Phenibut
CAS:Phenibut (Aminophenylbutyric acid) is a central depressant and derivative of the naturally occurring inhibitory neurotransmitter γ-aminobutyric acid (GABA).Fórmula:C10H13NO2Pureza:99.55%Forma y color:SolidPeso molecular:179.224-Aminopyridine
CAS:4-Aminopyridine (Dalfampridine) is a nonselective potassium (K+) channel blocker that binds to the cytoplasmic side of the cell membrane.Fórmula:C5H6N2Pureza:91.61%Forma y color:SolidPeso molecular:94.11Pramocaine hydrochloride
CAS:Pramocaine hydrochloride (Pramoxine HCl), a topical anesthetic, is served as an antipruritic.Fórmula:C17H27NO3·HClPureza:99.15% - 99.61%Forma y color:Crystals White Or Off White Crystalline PowderPeso molecular:329.86γ-Aminobutyric acid
CAS:γ-Aminobutyric acid (4-Aminobutyric acid) is the most common inhibitory neurotransmitter in the central nervous system.Fórmula:C4H9NO2Pureza:99.95%Forma y color:White Or Almost White(According To Quality Test Specification It Can Be White Or Almost White ) Solid PowderPeso molecular:103.12Bupivacaine hydrochloride
CAS:Bupivacaine hydrochloride (Vivacaine) is a long-lasting, amide local anesthetic that blocks sodium channels, inhibiting nerve impulses and sensation.Fórmula:C18H28N2O·HClPureza:99.89% - 99.9%Forma y color:SolidPeso molecular:324.89VU0134992 hydrochloride
CAS:VU0134992 hydrochloride is the first subtype-preferring, orally active and selective blocker of Kir4.1 potassium channel pore(IC50 : 0.97 μM).Fórmula:C20H32BrClN2O2Pureza:>99.99%Forma y color:SolidPeso molecular:447.84Fluxametamide
CAS:Fluxametamide, an isoxazoline insecticide, targets insect chloride channels with IC50s of 1.95 nM (GABA) and 225 nM (glutamate).Fórmula:C20H16Cl2F3N3O3Pureza:99.49%Forma y color:SolidPeso molecular:474.26DSP-2230
CAS:DSP-2230 is a selective blocker of Nav1.7/Nav1.8.
Fórmula:C20H20F3N5O2Pureza:97.14%Forma y color:SolidPeso molecular:419.4Suloctidil
CAS:Suloctidil is a peripheral vasodilator that was formerly used in the management of peripheral and cerebral vascular disorders.Fórmula:C20H35NOSPureza:99.75% - >99.99%Forma y color:SolidPeso molecular:337.56Omeprazole sulfide
CAS:Omeprazole sulfide (Ufiprazole), a metabolite of Omeprazole, functions as a proton pump inhibitor.Fórmula:C17H19N3O2SPureza:98.83%Forma y color:White To Slightly Collored Solid Solid CrystallinePeso molecular:329.42NaV1.7 inhibitor-1
CAS:NaV1.7 inhibitor-1, an efficacious inhibitor of voltage-gated sodium channel (NaV) 1.7 (IC50 of 0.6 nM for hNaV1.7).Fórmula:C23H30FNO4SPureza:99.89%Forma y color:SolidPeso molecular:435.55Ref: TM-T12181
1mg99,00€5mg241,00€10mg385,00€25mg663,00€50mg888,00€100mg1.305,00€1mL*10mM (DMSO)265,00€Nefiracetam
CAS:Nefiracetam (DM9384), in Phase 2 trials, enhances GABA, choline, monoamine systems, and treats Ro 5-4864 convulsions.Fórmula:C14H18N2O2Pureza:97.37%Forma y color:White To Off-White Crystalline PowderPeso molecular:246.3ML418
CAS:ML418 is a potent, selective and CNS penetrating Kir7.1 potassium channel blocker (IC50 = 310 nM), and also potently inhibits Kir6.2/SUR1.Fórmula:C19H24ClN3O3Pureza:99.3%Forma y color:SolidPeso molecular:377.87Ref: TM-T16110
1mg37,00€5mg79,00€10mg111,00€25mg178,00€50mg288,00€100mg414,00€200mg583,00€1mL*10mM (DMSO)88,00€1-EBIO
CAS:1-EBIO (1-EBIO) is a calium channel agonist.Fórmula:C9H10N2OPureza:98.75%Forma y color:SolidPeso molecular:162.19IK1 inhibitor PA-6
CAS:IK1 inhibitor PA-6 (PA-6) is a selective and potent inhibitor of IK1 (KIR2.x ion-channel-carried inward rectifier current)(IC50 of 12-15 nM for human and mouseFórmula:C31H32N4O2Pureza:98.9%Forma y color:SolidPeso molecular:492.61Methocarbamol
CAS:Methocarbamol (AHR 85) is a centrally acting muscle relaxant whose mode of action has not been established.Fórmula:C11H15NO5Pureza:99.96%Forma y color:Crystals From Benzene SolidPeso molecular:241.24Prilocaine hydrochloride
CAS:Prilocaine HCl: local amino amide anesthetic, blocks voltage-gated sodium channels in neurons, inhibits Na+ permeability.Fórmula:C13H21ClN2OPureza:99.97%Forma y color:Needles White Or Off White Crystalline PowderPeso molecular:256.77BMS-195270
CAS:BMS-195270 is a bio-active chemical.Fórmula:C15H9ClF3N3O2Pureza:98.7%Forma y color:SolidPeso molecular:355.7
