Transportador de membrana / canal de iones
Los inhibidores de transportadores de membrana y canales iónicos son compuestos que bloquean la función de proteínas responsables del transporte de iones, nutrientes y otras moléculas a través de las membranas celulares. Estos inhibidores son cruciales para estudiar la regulación de la homeostasis celular, la transducción de señales y la neurotransmisión. Los inhibidores de transportadores de membrana y canales iónicos también son importantes para desarrollar tratamientos para trastornos como la epilepsia, las enfermedades cardiovasculares y los síndromes metabólicos. En CymitQuimica, ofrecemos una amplia selección de inhibidores de alta calidad de transportadores de membrana y canales iónicos para apoyar su investigación en fisiología, neurociencia y farmacología.
Subcategorías de "Transportador de membrana / canal de iones"
- ABC(3 productos)
- ATPasa(93 productos)
- Receptor de adiponectina(5 productos)
- CFTR(64 productos)
- Receptor CGRP(51 productos)
- Canal de calcio(493 productos)
- Canal de cloruro(49 productos)
- Receptor GABA(336 productos)
- Transportador de monoamina(23 productos)
- Transportador de monocarboxilato(17 productos)
- NKCC(2 productos)
- NPC1L1(3 productos)
- Cotransportador de Na-K-Cl(8 productos)
- OAT(27 productos)
- OCT(7 productos)
- P-gp(53 productos)
- Canal de potasio(276 productos)
- Bomba de protones(39 productos)
- SGLT(30 productos)
- Canal de sodio(202 productos)
- Canal TRP / TRPV(92 productos)
Mostrar 13 subcategorías más
Se han encontrado 2270 productos de "Transportador de membrana / canal de iones"
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17β-Estradiol sulfate sodium
CAS:<p>17β-Estradiol sulfate sodium (17β-Estradiol 3-sulfate sodium) is a neuroactive estrogen with vasoprotective properties that inhibits the growth of Neisseria brasiliensis and disrupts aquatic ecosystems.</p>Fórmula:C18H23NaO5SPureza:99%Forma y color:SolidPeso molecular:374.43Phenazopyridine
CAS:<p>Phenazopyridine is an orally administered azo dye with local analgesic effects on urinary tract infections,. against SARM1 and TRPM8.</p>Fórmula:C11H11N5Pureza:99.98%Forma y color:SolidPeso molecular:213.24Dipropofol
CAS:<p>Dipropofol (4,4-Bis(2,6-di-isopropylphenol)) is a small molecule GABAA receptor agonist that can be used to study epilepsy.</p>Fórmula:C24H34O2Pureza:99.51%Forma y color:SolidPeso molecular:354.53NS 383
CAS:<p>ASIC blocker with varying IC50: 0.12 μM in hASIC1a, and ineffective on hASIC2a/3; <5 μM on rASIC1a/2a/3; alleviates pain in inflamed/CCI rats.</p>Fórmula:C19H19N3O2Forma y color:SolidPeso molecular:321.37Flecainide
CAS:<p>Flecainide is an orally administered antiarrhythmic agent acting as a sodium channel blocker and IKr inhibitor,PSVT.</p>Fórmula:C17H20F6N2O3Pureza:99.896%Forma y color:SolidPeso molecular:414.34KCNQ1 activator-1
CAS:<p>N-[4-(4-Methoxyphenyl)-2-thiazolyl]-2-piperidinecarboxamide is a potent KCNQ1 activator for LQTS research.</p>Fórmula:C22H23N3O4S2Pureza:99.71%Forma y color:SolidPeso molecular:457.57Norverapamil-d7
CAS:<p>Norverapamil D7 is a deuterium labeled Norverapamil . Norverapamil is a blocker of L-type calcium channel and an inhibitor of P-glycoprotein (P-gp) function .</p>Fórmula:C26H36N2O4Pureza:98%Forma y color:SolidPeso molecular:447.62Ethacizine hydrochloride
CAS:<p>Ethacizine hydrochloride (NIK-244) has antiarrhythmic activity and can be used to study arrhythmias and myocardial infarction.</p>Fórmula:C22H28ClN3O3SPureza:98.08% - 98.08%Forma y color:SolidPeso molecular:449.99MRK-016
CAS:<p>MRK-016 is a selective GABAA α5 receptor inverse agonist/ negative allosteric modulator, orally available and penetrating the BBB. MRK-016 is antidepressant.</p>Fórmula:C17H20N8O2Pureza:99.76%Forma y color:SolidPeso molecular:368.39GYKI 52466 dihydrochloride
CAS:<p>GYKI 52466 dihydrochloride is an AMPA/Kainate receptor antagonist with anticonvulsant activity and can be used to study neurological diseases.</p>Fórmula:C17H17Cl2N3O2Pureza:99.38%Forma y color:SolidPeso molecular:366.24(R)-3-Amino-4-hydroxybutanoic acid
CAS:<p>(R)-3-Amino-4-hydroxybutanoic acid,L-beta-Homoserine, is a full agonist at the human recombinant rho1 GABAC receptor, a modulator of GABAA and GABAB receptors.</p>Fórmula:C4H9NO3Pureza:99.92%Forma y color:SolidPeso molecular:119.12BTD
CAS:<p>BTD is a TRPC5 activator that activates heteromeric channel complexes composed of TRPC5 and its closest relatives TRPC1 or TRPC4.</p>Fórmula:C24H33N3O4SForma y color:SolidPeso molecular:459.6AM-2099
CAS:<p>AM-2099 is a selective voltage-gated sodium channel Nav1.7 inhibitor used in pain research.</p>Fórmula:C19H13F3N4O3S2Forma y color:SolidPeso molecular:466.46Valnoctamide
CAS:<p>Valnoctamide (Valmethamide) has antiepileptic and anticonvulsant activity and may be used in the study of neurological disorders.</p>Fórmula:C8H17NOPureza:98%Forma y color:SolidPeso molecular:143.23Bamaquimast
CAS:<p>Bamaquimast (L 0042) is a proton pump inhibitor for the study of asthma-like immune system disorders and respiratory diseases.</p>Fórmula:C16H21N3O3Pureza:98.47%Forma y color:SolidPeso molecular:303.36Fanapanel hydrate
CAS:<p>Fanapanel hydrate selectively blocks AMPA/kainate over NMDA; Ki: 3.2 nM (quisqualate), 100 nM (kainate), 8.5 μM (NMDA).</p>Fórmula:C14H17F3N3O7PForma y color:SolidPeso molecular:427.27Neosolaniol
CAS:<p>Neosolaniol, a type A trichothecene mycotoxin produced by Fusarium species, strongly induces an anorectic (loss of appetite) response.</p>Fórmula:C19H26O8Pureza:98%Forma y color:SolidPeso molecular:382.4Vigabatrin Hydrochloride
CAS:<p>Vigabatrin Hydrochloride (γ-Vinyl-GABA hydrochloride) is a structural analog of the GABA, irreversibly inhibiting the catabolism of GABA by GABA transaminase.</p>Fórmula:C6H11NO2·HClPureza:98%Forma y color:SolidPeso molecular:165.62Mepivacaine
CAS:<p>Mepivacaine (Carbocaine) is an amide local anesthetic, blocking sodium channels for nerve blocks and epidurals.</p>Fórmula:C15H22N2OPureza:99.35%Forma y color:SolidPeso molecular:246.35Lubiprostone hemiketal
CAS:<p>Lubiprostone (hemiketal) (RU-0211 (hemiketal)), a selective activator of the chloride channel 2 (CLCN2), facilitates the treatment of chronic idiopathic constipation and opioid-induced constipation. It functions by enhancing CLCN2 channel activity, which boosts chloride ion secretion in the intestines, subsequently increasing fluid secretion and improving intestinal peristalsis. Additionally, Lubiprostone (hemiketal) may be utilized in research related to chronic constipation and cancer.</p>Fórmula:C20H32F2O5Forma y color:SolidPeso molecular:390.46CGP 36742
CAS:<p>CGP 36742 blocks GABAB receptor, crosses blood-brain barrier, aids depression treatment (IC50: 32 μM).</p>Fórmula:C7H18NO2PForma y color:SolidPeso molecular:179.2γ-DGG
CAS:<p>gamma-DGG is a competitive blocker of AMPA receptor.</p>Fórmula:C7H12N2O5Pureza:98%Forma y color:SolidPeso molecular:204.18Furosemide-d5
CAS:<p>Furosemide-d5 is a deuterium marker for Furosemide and used in isotope tracer experiments. orally active inhibitor of Na+/K+/2Cl- (NKCC) diuretic reagent.</p>Fórmula:C12H11ClN2O5SForma y color:SolidPeso molecular:335.78(+)-SJ733
CAS:<p>(+)-SJ733 (SJ000557733) is a potent Na+-ATPase PfATP4 inhibitor with antimalarial activity for the study of malaria.</p>Fórmula:C24H16F4N4O2Pureza:99.21%Forma y color:SolidPeso molecular:468.4(R)-BPO-27
CAS:<p>(R)-BPO-27 is an orally active and potent ATP-competitive CFTR inhibitor (IC50: 4 nM) for the study of diarrhoea and polycystic kidney.</p>Fórmula:C26H18BrN3O6Pureza:99.1%Forma y color:SolidPeso molecular:548.34MDL 105519
CAS:<p>MDL 105519 is a selective, non-competitive antagonist of NMDA receptors. It inhibits cyclic GMP accumulation in brain slices, anxiolytic in rat models.</p>Fórmula:C18H11Cl2NO4Forma y color:SolidPeso molecular:376.19Crinecerfont hydrochloride
CAS:<p>SSR-125543, a potent CRF1 receptor non-peptide antagonist, effective in CAH research, taken orally.</p>Fórmula:C27H29Cl2FN2OSForma y color:SolidPeso molecular:519.5Etifoxine
CAS:<p>Etifoxine targets β2/β3 GABAA receptors, is anxiolytic in humans/rodents, boosts GABAA, binds TSPO, aids axon regeneration, no sedative effects.</p>Fórmula:C17H17ClN2OPureza:98%Forma y color:SolidPeso molecular:300.78L-Palmitoylcarnitine
CAS:<p>L-Palmitoylcarnitine (L-PC) inhibits Na/K ATPase activity and potentiates fibrinolytic enzymes and tPA to inhibit thrombosis.</p>Fórmula:C23H45NO4Pureza:97% - 99.81%Forma y color:SolidPeso molecular:399.61Clamikalant sodium
CAS:<p>Clamikalant sodium (HMR 1098) is an ATP-dependent potassium channel (KATP) cardiac-selective blocker, used in the study of arrhythmias.</p>Fórmula:C19H21ClN3NaO5S2Pureza:99.95%Forma y color:SolidPeso molecular:493.96L-655708
CAS:<p>L-655708 is a selective and highly potent GABAA receptor reverse agonist with a Ki value of 0.45 nM.</p>Fórmula:C18H19N3O4Pureza:98.41%Forma y color:PowderPeso molecular:341.36MRS1845
CAS:<p>MRS1845 is a selective inhibitor of store-operated calcium (SOC) channel (IC50 of 1.7 μM).</p>Fórmula:C21H22N2O6Pureza:99.69%Forma y color:SolidPeso molecular:398.41Pirmenol hydrochloride
CAS:<p>Pirmenol hydrochloride functions by inhibiting I_K.ACh through the blockade of muscarinic receptors, demonstrating a potent effect with an IC_50 value of 0.1 μM</p>Fórmula:C22H31ClN2OForma y color:SolidPeso molecular:374.95QO-58
CAS:<p>QO-58 is a novel Kv7 activator (opener) that activates neuronal Kv7/KCNQ/M channels, danti-nociceptive effects on inflammatory pain</p>Fórmula:C18H8Cl2F4N4OPureza:99.17%Forma y color:SolidPeso molecular:443.18(-)-α-Pinene
CAS:<p>(-)-α-Pinene ((1S)-(-)-Alpha-Pinene) enhances the quantity of NREMS without affecting the intensity of NREMS by prolonging GABAergic synaptic transmission,</p>Fórmula:C10H16Pureza:98.02% - 98.60%Forma y color:Colourless LiquidPeso molecular:136.23GI-530159
CAS:<p>TREK1/2 activator, selective over TRAAK/TASK3; hyperpolarizes neurons, depresses activity (EC50 = 0.76 μM).</p>Fórmula:C27H20F6N2O2Forma y color:White CrystalsPeso molecular:518.45Poneratoxin acetate
<p>Poneratoxin acetate is a neurotoxic peptide and modulator of NaV1.6/NaV1.7, lowering the activation threshold of voltage-gated sodium channels and causing pain.</p>Fórmula:C129H215N33O31S·xC2H4O2Forma y color:SolidPeso molecular:2756.35 (free base)Tetramethrin
CAS:<p>Tetramethrin is a type I pyrethroid insecticide that affects the inactivation process of sodium channels in insect neurons, prolonged sodium currents.</p>Fórmula:C19H25NO4Pureza:98.85%Forma y color:White Crystals Or PowderPeso molecular:331.41Benzocaine hydrochloride
CAS:<p>Benzocaine hydrochloride (Ethyl 4-aminobenzoate hydrochloride) is a surface anesthetic that acts by preventing transmission of impulses along nerve fibers and</p>Fórmula:C9H11NO2·HClPureza:98%Forma y color:SolidPeso molecular:201.65Ethyl tosylcarbamate
CAS:<p>Gliclazide blocks beta-cell ATP-sensitive K+ currents, IC50: 184 nM. Ethyl tosylcarbamate is a synthesis intermediate.</p>Fórmula:C10H13NO4SForma y color:SolidPeso molecular:243.28H-D-Allo-Ile-OH
CAS:<p>H-D-Allo-Ile-OH inhibits 3[H] gabapentin binding/voltage-dependent L-type calcium channels and can be used for studying neurological and psychiatric disorders.</p>Fórmula:C6H13NO2Pureza:99.92%Forma y color:SolidPeso molecular:131.17Dibucaine hydrochloride
CAS:<p>Dibucaine hydrochloride (Cinchocaine hydrochloride), a long-acting local amide anestheticsis, is usually used for surface anesthesia.</p>Fórmula:C20H30ClN3O2Pureza:99.66%Forma y color:White PowderPeso molecular:379.92Lesinurad sodium
CAS:<p>Lesinurad sodium (RDEA594 sodium) is a selective inhibitor of uric acid reabsorption and is used in the study of cardiovascular diseases.</p>Fórmula:C17H13BrN3NaO2SPureza:99.97%Forma y color:SolidPeso molecular:426.26β-Cyfluthrin
CAS:<p>β-Cyfluthrin is a type II synthetic pyrethroid compound commonly utilized as an active ingredient in agricultural insecticide products.</p>Fórmula:C22H18Cl2FNO3Forma y color:SolidPeso molecular:434.29BI-9627 hydrochloride
CAS:<p>BIX HCl is a sodium-hydrogen exchange type 1 inhibitor.</p>Fórmula:C16H20ClF3N4O2Forma y color:SolidPeso molecular:392.8Flumazenil acid
CAS:<p>Flumazenil is an antagonist of GABAA receptor. Flumazenil acid is a metabolite of Flumazenil.</p>Fórmula:C13H10FN3O3Forma y color:SolidPeso molecular:275.24Tetrabenazine-d6
CAS:<p>Tetrabenazine D6 is the deuterium-labeled Tetrabenazine. Tetrabenazine is a VMAT-inhibitor used for the treatment of hyperkinetic movement disorder.</p>Fórmula:C19H27NO3Pureza:98%Forma y color:SolidPeso molecular:323.46VU041
CAS:<p>VU041 inhibits mosquito Kir1 channels (IC50: An. gambiae 2.5μM, Ae. aegypti 1.7μM), less on mammalian Kir2.1 (12.7μM), and minimally on other Kir channels.</p>Fórmula:C19H20F3N3OPureza:98%Forma y color:SolidPeso molecular:363.38(R)-Tegoprazan
CAS:<p>(R)-Tegoprazan, a benzimidazole derivative, inhibits kidney H+/K+-ATPase (IC50: 98 nM). Potential in GI disease research.</p>Fórmula:C20H19F2N3O3Forma y color:SolidPeso molecular:387.38PF-04856264
CAS:<p>PF-04856264 is a Nav1.7 blocker.,modulates intracellular Ca 2+ signaling and chondrocyte secretome, raises the threshold of mechanical pain analgesic.</p>Fórmula:C20H15N5O3S2Pureza:97.43%Forma y color:SolidPeso molecular:437.5
