Transportador de membrana / canal de iones
Los inhibidores de transportadores de membrana y canales iónicos son compuestos que bloquean la función de proteínas responsables del transporte de iones, nutrientes y otras moléculas a través de las membranas celulares. Estos inhibidores son cruciales para estudiar la regulación de la homeostasis celular, la transducción de señales y la neurotransmisión. Los inhibidores de transportadores de membrana y canales iónicos también son importantes para desarrollar tratamientos para trastornos como la epilepsia, las enfermedades cardiovasculares y los síndromes metabólicos. En CymitQuimica, ofrecemos una amplia selección de inhibidores de alta calidad de transportadores de membrana y canales iónicos para apoyar su investigación en fisiología, neurociencia y farmacología.
Subcategorías de "Transportador de membrana / canal de iones"
- ABC(3 productos)
- ATPasa(98 productos)
- Receptor de adiponectina(5 productos)
- CFTR(66 productos)
- Receptor CGRP(54 productos)
- Canal de calcio(528 productos)
- Canal de cloruro(52 productos)
- Receptor GABA(360 productos)
- Transportador de monoamina(28 productos)
- Transportador de monocarboxilato(18 productos)
- NKCC(2 productos)
- NPC1L1(3 productos)
- Cotransportador de Na-K-Cl(9 productos)
- OAT(31 productos)
- OCT(7 productos)
- P-gp(54 productos)
- Canal de potasio(280 productos)
- Bomba de protones(42 productos)
- SGLT(31 productos)
- Canal de sodio(206 productos)
- Canal TRP / TRPV(94 productos)
Mostrar 13 subcategorías más
Se han encontrado 2460 productos de "Transportador de membrana / canal de iones"
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Tirofiban hydrochloride monohydrate
CAS:<p>Tirofiban（MK383） hydrochloride monohydrate is a non-peptide glycoprotein IIb/IIIa antagonist. Cost-effective and quality-assured.</p>Fórmula:C22H39ClN2O6SPureza:98.81% - >99.99%Forma y color:White SolidPeso molecular:495.07Chloroprocaine hydrochloride
CAS:Chloroprocaine hydrochloride (Chloroprocaine HCl) is a local anesthetic during surgical procedures.Fórmula:C13H20Cl2N2O2Pureza:99.65%Forma y color:White Crystalline PowderPeso molecular:307.22CTP disodium dihydrate
CAS:<p>CTP disodium dihydrate is an agonist of P2X4 purinergic receptor</p>Fórmula:C9H18N3Na2O16P3Pureza:98.51%Forma y color:White Crystalline PowderPeso molecular:563.15Vonoprazan hydrochloride
CAS:<p>Vonoprazan hydrochloride is a potent PPI and P-CAB for treating acid-related diseases and H. pylori infection.</p>Fórmula:C17H17ClFN3O2SForma y color:SolidPeso molecular:381.85Songorine
CAS:Songorine (Napellonine) shows anti-tumor activity in preliminary pharmacological verification trials including cell proliferation and molecular docking assays.Fórmula:C22H31NO3Pureza:98% - 99.92%Forma y color:SolidPeso molecular:357.49KM11060
CAS:KM11060 is a novel corrector of the F508del-CFTR trafficking defect, Correcting F508del-CFTR trafficking, increasing the amount of functional CFTR at the plasmaFórmula:C19H17Cl2N3O2SPureza:98.86%Forma y color:SolidPeso molecular:422.33Delucemine Free Base
CAS:Delucemine Free Base is an NMDA Receptor AntagonistFórmula:C16H17F2NForma y color:SolidPeso molecular:261.31Nisoxetine
CAS:Nisoxetine is a selective NET (noradrenaline transporter) inhibitor (Kd=0.76 nM) capable of blocking voltage-gated sodium channels.Fórmula:C17H21NO2Pureza:98.71%Forma y color:SolidPeso molecular:271.35VU590 HCl
CAS:VU590 is a small molecule inhibitor of KCNJ1 (IC50 = 294 nM).Fórmula:C24H34Cl2N4O7Forma y color:SolidPeso molecular:561.457Chembridge-5861528
CAS:Chembridge-5861528 (TCS 5861528) is a TRPA1 channel blocker that antagonizes AITC- and 4-HNE-evoked calcium influx with IC50 values of 14.3 and 18.7 μM.Fórmula:C19H23N5O3Pureza:99.97%Forma y color:SolidPeso molecular:369.42CFTR(inh)-172
CAS:<p>CFTR(inh)-172 (CFTR Inhibitor-172) is a voltage-independent, selective CFTR inhibitor.</p>Fórmula:C18H10F3NO3S2Pureza:98% - 99.72%Forma y color:SolidPeso molecular:409.4Phe-Met-Arg-Phe, amide acetate
Phe-Met-Arg-Phe amide acetate (ED50=23 nM) triggers K+ current in caudodorsal neurons, co-localizes with neuropeptide Y in brain areas.Fórmula:C31H46N8O6SPureza:99.4%Forma y color:SolidPeso molecular:658.82KB-R7943 mesylate
CAS:<p>KB-R7943 mesylate is a widely used inhibitor of the reverse Na+/Ca2+ exchanger (NCXrev) with IC50 of 5.7±2.1 μM.</p>Fórmula:C17H21N3O6S2Pureza:99.88% - ≥95%Forma y color:SolidPeso molecular:427.5TGN-020
CAS:<p>TGN-020 is an inhibitor of Aquaporin 4 (AQP4, IC50: 3.1 μM), the most abundant water channel in the brain.</p>Fórmula:C8H6N4OSPureza:99.54% - 99.99%Forma y color:SolidPeso molecular:206.22VU0071063
CAS:VU0071063 is a Kir6.2/SUR1 activator.Fórmula:C18H22N4O2Pureza:99.33%Forma y color:SolidPeso molecular:326.39Esomeprazole Magnesium trihydrate
CAS:<p>Esomeprazole Magnesium trihydrate ((S)-Omeprazole magnesium trihydrate) is a proton pump inhibitor indicated for the short-term treatment of gastroesophageal</p>Fórmula:C34H42MgN6O9S2Pureza:98.52%Forma y color:Off-White PowderPeso molecular:767.17OAC2
CAS:<p>OAC2, an Oct4 activator, boosts iPSC creation from embryonic fibroblasts, similar to OAC1.</p>Fórmula:C15H12N2OPureza:99.58% - ≥95%Forma y color:SolidPeso molecular:236.27Cyclothiazide
CAS:<p>Cyclothiazide enhances AMPA receptors, prevents desensitization, and boosts glutamic acid response (EC50 = 3.8µM).</p>Fórmula:C14H16ClN3O4S2Pureza:98.23% - 99.49%Forma y color:Crystals From Dilute Alcohol SolidPeso molecular:389.88Vanilloid receptor antagonist 1
CAS:Vanilloid receptor antagonist 1 (4-(7-Hydroxy-2-isopropyl-4-oxoquinazolin-3(4H)-yl)benzonitrile) is a potent vanilloid receptor TRPV1 antagonist.Fórmula:C18H15N3O2Pureza:98.14%Forma y color:SolidPeso molecular:305.33SKA-31
CAS:SKA-31 (Naphtho[1,2-d]thiazol-2-ylamine) is an activator of KCa3.1 and KCa2 channels (EC50s: 260, 2900, 2900 nM for KCa3.1, KCa2.1 and KCa2.2 respectively).Fórmula:C11H8N2SPureza:99.38%Forma y color:SolidPeso molecular:200.26MDR-652
CAS:MDR-652 is a highly specific and efficacious agonist of nonpungent transient receptor potential vanilloid 1 (TRPV1) with Ki value of 11.4 nM and 23.8 nM forFórmula:C22H23ClFN3O2SPureza:99.96%Forma y color:SolidPeso molecular:447.95ICILIN
CAS:<p>ICILIN (AG-3-5) is a synthetic TRPM8 ion channel super-agonist.</p>Fórmula:C16H13N3O4Pureza:98.45% - ≥95%Forma y color:Light Yellow SolidPeso molecular:311.29VU6036720 hydrochloride
VU6036720 hydrochloride inhibits Kir4.1/5.1. channels with 0.24 μM IC50; used in brain and kidney research.Fórmula:C20H23Cl2FN4O2SForma y color:SolidPeso molecular:473.39SN 2
CAS:SN 2 is a novel and potent TRPML3 ion channel activator(EC50 = 1.13 μM). SN 2 also shares a similar antiviral effect against DENV2 and ZIKV.Fórmula:C17H21NOPureza:99.86%Forma y color:SolidPeso molecular:255.35Blebbistatin
CAS:Blebbistatin ((±)-Blebbistatin) is a non-muscle myosin II (NMII)-selective and non-muscle myosin heavy chain 9 (MYH9)-specific inhibitor.Cost-effective and quality-assured.Fórmula:C18H16N2O2Pureza:99.88% - 99.97%Forma y color:Bright Yellow SolidPeso molecular:292.33Flupirtine
CAS:<p>Flupirtine(D 9998) is a selective neuronal potassium channel opener as well as shows properties of NMDA receptor antagonist.</p>Fórmula:C15H17FN4O2Forma y color:SolidPeso molecular:304.32Acamprosate calcium
CAS:Acamprosate calcium (Campral EC) is a GABA receptor agonist and modulator of glutamatergic systems, used for treating alcohol dependence.Fórmula:C10H20CaN2O8S2Pureza:98% - 99.93%Forma y color:White Odorless Or Nearly Odorless PowderPeso molecular:400.48Arecaidine hydrochloride
CAS:Arecaidine hydrochloride may have carcinogenesis.Fórmula:C7H12ClNO2Pureza:99.69% - ≥95%Forma y color:SolidPeso molecular:177.63Metaflumizone
CAS:Metaflumizone (BAS-320I) is a sodium channel blocker insecticide.Fórmula:C24H16F6N4O2Pureza:98.73%Forma y color:SolidPeso molecular:506.40(-)-Securinine
CAS:<p>(-)-Securinine (Securinine) is plant-derived alkaloid and also a GABAA receptor antagonist.</p>Fórmula:C13H15NO2Pureza:99.58% - 99.87%Forma y color:SolidPeso molecular:217.26Tenapanor
CAS:Tenapanor (RDX 5791), an NHE3 inhibitor, regulates sodium in the gut and kidney with a strong preclinical safety record and minimal side effects.Fórmula:C50H66Cl4N8O10S2Pureza:99.49% - 99.85%Forma y color:SolidPeso molecular:1145.05Mitiglinide
CAS:Mitiglinide (KAD-1229), an insulinotropic ATP-sensitive K+ channel antagonist, targets Kir6.2/SUR1; used in type 2 diabetes research.Fórmula:C19H25NO3Forma y color:SolidPeso molecular:315.41A2764 dihydrochloride
CAS:A2764 dihydrochloride is a highly selective inhibitor of TRESK.Fórmula:C15H21Cl3N2OPureza:99.05%Forma y color:SolidPeso molecular:351.7Mirogabalin besylate
CAS:Mirogabalin besylate is an oral α2δ ligand for voltage-gated calcium channels, with Kd values of 13.5-47.6 nM across species.Fórmula:C18H25NO5SForma y color:SolidPeso molecular:367.46Verinurad
CAS:Verinurad (RDEA3170) (RDEA3170) is an organic anion transporter URAT1 (SLC22A12) inhibitor for the treatment of gout and hyperuricemia.Fórmula:C20H16N2O2SPureza:97.36% - 99.22%Forma y color:SolidPeso molecular:348.42Pyr6
CAS:Pyr6 (N-[4-[3,5-Bis(trifluoromethyl)-1H-pyrazol-1-yl]phenyl]-3-fluoro-4-pyridinecarboxamide) is a selective TRPC3 inhibitor with IC50 of 0.49 uM(Ca2+ influxFórmula:C17H9F7N4OPureza:98.89%Forma y color:SolidPeso molecular:418.27SB 452533
CAS:<p>SB 452533 is an antagonist of the vanilloid receptor 1(pKb: 7.8).</p>Fórmula:C18H22BrN3OPureza:99.87%Forma y color:SolidPeso molecular:376.29Levolansoprazole
CAS:<p>Levolansoprazole ((S)-Lansoprazole), a proton pump inhibitor, irreversibly inhibits H+/K+-stimulated ATPase pumps in parietal cells (IC50: 5.2 μM).</p>Fórmula:C16H14F3N3O2SPureza:98.629%Forma y color:SolidPeso molecular:369.36U93631
CAS:GABAA antagonist; binds picrotoxin site, stabilizes inactive channel. Speeds GABA-induced Cl- decay, minor peak effect. Inhibits 5-HT3A receptors.Fórmula:C17H21N3O2Pureza:99.65% - 99.76%Forma y color:SolidPeso molecular:299.37Doxapram
CAS:Doxapram (Dopram) is a respiratory stimulant that inhibits TASK-1, TASK-3, and TASK-1/TASK-3 heterodimer channels.Fórmula:C24H30N2O2Pureza:99.42%Forma y color:SolidPeso molecular:378.51N-Methyl-L-leucin
CAS:N-Methyl-L-leucine ((S)-4-Methyl-2-(methylamino)pentanoic acid) is a novel calcium channel antagonist used in pain research.Fórmula:C7H15NO2Pureza:99.87%Forma y color:SolidPeso molecular:145.2Riluzole
CAS:<p>Riluzole (RP-54274) is an anticonvulsant, glutamate antagonist, and prolongs ALS patient survival.</p>Fórmula:C8H5F3N2OSPureza:99.71% - 99.88%Forma y color:PowderPeso molecular:234.2SRI-41315
CAS:SRI-41315 is an eRF1 degrader that acts as a molecular glue at the ribosomal decoding center.SRI-41315 induces extended pauses at the termination codon.Fórmula:C22H19N3O2Pureza:99.87%Forma y color:SolidPeso molecular:357.41Dimiracetam
CAS:<p>Dimiracetam, a NMDA-receptor antagonist, is used potentially for the treatment of neuropathic pain.</p>Fórmula:C6H8N2O2Pureza:>99.99% - >99.99%Forma y color:SolidPeso molecular:140.14Propoxycaine hydrochloride
CAS:Propoxycaine hydrochloride is an ester local anesthetic that inhibits voltage-gated sodium channels, modulates nerve impulses, and induces loss of sensation.Fórmula:C16H27ClN2O3Pureza:97.25%Forma y color:SolidPeso molecular:330.85Safinamide
CAS:<p>Safinamide: reversible MAO-B inhibitor, enhances dopamine, blocks glutamate release, sodium, calcium channels; may treat Parkinson's, RLS, epilepsy.</p>Fórmula:C17H19FN2O2Pureza:99.92%Forma y color:SolidPeso molecular:302.34VU590
CAS:VU590 is an inhibitor of extrarenal medullary potassium ROMK.VU590 inhibits Kir7.1 and modulates uterine myometrial contractility and melanocortin signalling.Fórmula:C24H32N4O7Pureza:98.06%Forma y color:SolidPeso molecular:488.53CX717
CAS:<p>CX 717 is a positive allosteric modulator of AMPA receptor which has an antidepressant-like effect.</p>Fórmula:C11H11N3O3Pureza:99.81%Forma y color:SoildPeso molecular:233.23JNJ-28583113
CAS:JNJ-28583113 is a TRPM2 antagonist, inducing phosphorylation of GSK3α and β subunits, protecting cells from oxidative stress-induced cell death.Fórmula:C19H21F3N2O2Pureza:98.57%Forma y color:SolidPeso molecular:366.38VB124
CAS:VB124 is an orally active, potent and selective MCT4 inhibitor. VB124 blocked lactate importand expor in MDA-MB-231 cells.Cost-effective and quality-assured.Fórmula:C23H23ClN2O4Pureza:99.21% - 99.57%Forma y color:SoildPeso molecular:426.89
