
Transportador de membrana / canal de iones
Los inhibidores de transportadores de membrana y canales iónicos son compuestos que bloquean la función de proteínas responsables del transporte de iones, nutrientes y otras moléculas a través de las membranas celulares. Estos inhibidores son cruciales para estudiar la regulación de la homeostasis celular, la transducción de señales y la neurotransmisión. Los inhibidores de transportadores de membrana y canales iónicos también son importantes para desarrollar tratamientos para trastornos como la epilepsia, las enfermedades cardiovasculares y los síndromes metabólicos. En CymitQuimica, ofrecemos una amplia selección de inhibidores de alta calidad de transportadores de membrana y canales iónicos para apoyar su investigación en fisiología, neurociencia y farmacología.
Subcategorías de "Transportador de membrana / canal de iones"
- ABC(3 productos)
- ATPasa(101 productos)
- Receptor de adiponectina(5 productos)
- CFTR(65 productos)
- Receptor CGRP(54 productos)
- Canal de calcio(543 productos)
- Canal de cloruro(53 productos)
- Receptor GABA(366 productos)
- Transportador de monoamina(30 productos)
- Transportador de monocarboxilato(18 productos)
- NKCC(2 productos)
- NPC1L1(3 productos)
- Cotransportador de Na-K-Cl(10 productos)
- OAT(32 productos)
- OCT(7 productos)
- P-gp(55 productos)
- Canal de potasio(280 productos)
- Bomba de protones(42 productos)
- SGLT(31 productos)
- Canal de sodio(210 productos)
- Canal TRP / TRPV(96 productos)
Mostrar 13 subcategorías más
Se han encontrado 2534 productos de "Transportador de membrana / canal de iones"
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Penicillin G sodium salt
CAS:<p>Penicillin G sodium(Benzylpenicillin sodium) salt is a penicillin derivative commonly used in the form of its sodium or potassium salts in the treatment of a</p>Fórmula:C16H17N2NaO4SPureza:98.11%Forma y color:White To Off-White Crystalline PowderPeso molecular:356.37Pramocaine hydrochloride
CAS:Pramocaine hydrochloride (Pramoxine HCl), a topical anesthetic, is served as an antipruritic.Fórmula:C17H27NO3·HClPureza:99.15% - 99.61%Forma y color:Crystals White Or Off White Crystalline PowderPeso molecular:329.86NaV1.7 inhibitor-1
CAS:NaV1.7 inhibitor-1, an efficacious inhibitor of voltage-gated sodium channel (NaV) 1.7 (IC50 of 0.6 nM for hNaV1.7).Fórmula:C23H30FNO4SPureza:99.89%Forma y color:SolidPeso molecular:435.55Ref: TM-T12181
1mg104,00€5mg255,00€10mg406,00€25mg700,00€50mg938,00€100mg1.378,00€1mL*10mM (DMSO)280,00€Tocainide hydrochloride
CAS:<p>Tocainide hydrochloride (2-amino-n-(2,6-dimethylphenyl)propanamide hydrochloride) is a sodium channel blocker.</p>Fórmula:C11H17ClN2OPureza:97%Forma y color:SolidPeso molecular:228.72ML418
CAS:ML418 is a potent, selective and CNS penetrating Kir7.1 potassium channel blocker (IC50 = 310 nM), and also potently inhibits Kir6.2/SUR1.Fórmula:C19H24ClN3O3Pureza:99.3%Forma y color:SolidPeso molecular:377.87Ref: TM-T16110
1mg37,00€5mg79,00€10mg111,00€25mg178,00€50mg288,00€100mg414,00€200mg583,00€1mL*10mM (DMSO)88,00€EN6
CAS:EN6, a small molecule, activates autophagy by modifying ATP6V1A, inhibiting mTORC1 and enhancing lysosomal function to clear TDP-43 aggregates.Fórmula:C19H14F2N4O2Pureza:95.74% - 97.04%Forma y color:SolidPeso molecular:368.34Ref: TM-T11191
1mg47,00€5mg88,00€10mg137,00€25mg205,00€50mg264,00€100mg400,00€500mg909,00€1mL*10mM (DMSO)70,00€Fluxametamide
CAS:Fluxametamide, an isoxazoline insecticide, targets insect chloride channels with IC50s of 1.95 nM (GABA) and 225 nM (glutamate).Fórmula:C20H16Cl2F3N3O3Pureza:99.49%Forma y color:SolidPeso molecular:474.26Dooku1
CAS:Dooku1, Yoda1 analog, blocks Piezo1 channels, halting Ca2+ entry. IC50: 1.3μM in HEK 293, 1.5μM in HUVEC, stops Yoda1's aortic relaxation.Fórmula:C13H9Cl2N3OSPureza:98.87% - 99.74%Forma y color:SolidPeso molecular:326.2Ref: TM-T11076
1mg46,00€2mg59,00€5mg87,00€10mg140,00€25mg274,00€50mg510,00€100mg735,00€1mL*10mM (DMSO)96,00€MRZ 2-514
CAS:MRZ 2-514 (8-bromo-4,5-dihydroxypyridazino[4,5-b]quinolin-1-one) is a strychnine-insensitive modulatory site of the NMDA receptor (glycineB)antagonist with KiFórmula:C11H6BrN3O3Pureza:98.459%Forma y color:SolidPeso molecular:308.09Ref: TM-T12110
1mg96,00€5mg202,00€10mg329,00€25mg655,00€50mg1.103,00€100mg1.483,00€1mL*10mM (DMSO)224,00€Indapamide
CAS:Indapamide (Noranat) is a non-thiazide sulphonamide diuretic compound, generally used in the treatment of hypertension, as well as decompensated cardiac failure.Fórmula:C16H16ClN3O3SPureza:98.97% - 99.83%Forma y color:SolidPeso molecular:365.83Ciclopirox olamine
CAS:Ciclopirox olamine is a broad-spectrum antifungal agent with additional antibacterial and anti-inflammatory activities.Fórmula:C14H24N2O3Pureza:99.16% - >99.99%Forma y color:White To Yellow Solid Solid Particulate/PowderPeso molecular:268.35Methocarbamol
CAS:Methocarbamol (AHR 85) is a centrally acting muscle relaxant whose mode of action has not been established.Fórmula:C11H15NO5Pureza:99.96%Forma y color:Crystals From Benzene SolidPeso molecular:241.24Prilocaine hydrochloride
CAS:Prilocaine HCl: local amino amide anesthetic, blocks voltage-gated sodium channels in neurons, inhibits Na+ permeability.Fórmula:C13H21ClN2OPureza:99.97%Forma y color:Needles White Or Off White Crystalline PowderPeso molecular:256.77NS13001
CAS:NS13001, an oral SK channel modulator, shows promise for SCA2 therapy; EC50: 1.8 µM (SK2), 0.14 µM (SK3).Fórmula:C17H16ClN7Pureza:99.55%Forma y color:SolidPeso molecular:353.81Lotilaner
CAS:Lotilaner is a parasiticide.Fórmula:C20H14Cl3F6N3O3SPureza:99.56%Forma y color:SolidPeso molecular:596.76Ref: TM-T15775
1mg44,00€2mg58,00€5mg94,00€10mg144,00€25mg335,00€50mg550,00€100mg882,00€200mg1.188,00€1mL*10mM (DMSO)111,00€Bupivacaine hydrochloride
CAS:Bupivacaine hydrochloride (Vivacaine) is a long-lasting, amide local anesthetic that blocks sodium channels, inhibiting nerve impulses and sensation.Fórmula:C18H28N2O·HClPureza:99.89% - 99.9%Forma y color:SolidPeso molecular:324.89Phenibut
CAS:Phenibut (Aminophenylbutyric acid) is a central depressant and derivative of the naturally occurring inhibitory neurotransmitter γ-aminobutyric acid (GABA).Fórmula:C10H13NO2Pureza:99.55%Forma y color:SolidPeso molecular:179.22VU6036720
<p>VU6036720 is a potent and selective inhibitor of the isomeric Kir4.1/5.1.VU6036720 inhibits Kir4.1/5.1 activity by decreasing the channel open-circuit</p>Fórmula:C20H22ClFN4O2SPureza:98.1%Forma y color:SoildPeso molecular:436.93VU0134992 hydrochloride
CAS:VU0134992 hydrochloride is the first subtype-preferring, orally active and selective blocker of Kir4.1 potassium channel pore(IC50 : 0.97 μM).Fórmula:C20H32BrClN2O2Pureza:>99.99%Forma y color:SolidPeso molecular:447.84Ref: TM-T13316
5mg37,00€10mg59,00€25mg104,00€50mg170,00€100mg283,00€200mg437,00€1mL*10mM (DMSO)42,00€5,5-Dimethyloxazolidine-2,4-dione
CAS:5,5-Dimethyloxazolidine-2,4-dione (Dimethadione) is an anticonvulsant that is the active metabolite of TRIMETHADIONE.Fórmula:C5H7NO3Pureza:99.12%Forma y color:Drypowder PelletslargecrystalsPeso molecular:129.11
