
Transportador de membrana / canal de iones
Los inhibidores de transportadores de membrana y canales iónicos son compuestos que bloquean la función de proteínas responsables del transporte de iones, nutrientes y otras moléculas a través de las membranas celulares. Estos inhibidores son cruciales para estudiar la regulación de la homeostasis celular, la transducción de señales y la neurotransmisión. Los inhibidores de transportadores de membrana y canales iónicos también son importantes para desarrollar tratamientos para trastornos como la epilepsia, las enfermedades cardiovasculares y los síndromes metabólicos. En CymitQuimica, ofrecemos una amplia selección de inhibidores de alta calidad de transportadores de membrana y canales iónicos para apoyar su investigación en fisiología, neurociencia y farmacología.
Subcategorías de "Transportador de membrana / canal de iones"
- ABC(3 productos)
- ATPasa(93 productos)
- Receptor de adiponectina(5 productos)
- CFTR(66 productos)
- Receptor CGRP(55 productos)
- Canal de calcio(579 productos)
- Canal de cloruro(53 productos)
- Receptor GABA(367 productos)
- Transportador de monoamina(31 productos)
- Transportador de monocarboxilato(18 productos)
- NKCC(2 productos)
- NPC1L1(1 productos)
- Cotransportador de Na-K-Cl(9 productos)
- OAT(31 productos)
- OCT(7 productos)
- P-gp(64 productos)
- Canal de potasio(324 productos)
- Bomba de protones(42 productos)
- SGLT(32 productos)
- Canal de sodio(273 productos)
- Canal TRP / TRPV(99 productos)
Mostrar 13 subcategorías más
Se han encontrado 2714 productos para "Transportador de membrana / canal de iones".
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Flumazenil
CAS:Flumazenil (Ro 15-1788) antagonizes the benzodiazepine binding site of the gamma-aminobutyric acid (GABA)/benzodiazepine receptor complex in the central nervousFórmula:C15H14FN3O3Pureza:99.72% - 99.98%Forma y color:White SolidPeso molecular:303.29Trichlormethiazide
CAS:Trichlormethiazide (Naqua) is a short-acting, 3-dichloromethyl derivative of hydrochlorothiazide, belonging to the class of thiazide diuretics.Fórmula:C8H8Cl3N3O4S2Pureza:98.8% - 99.54%Forma y color:White SolidPeso molecular:380.66Fluxametamide
CAS:Fluxametamide, an isoxazoline insecticide, targets insect chloride channels with IC50s of 1.95 nM (GABA) and 225 nM (glutamate).Fórmula:C20H16Cl2F3N3O3Pureza:99.49%Forma y color:SolidPeso molecular:474.26Tocainide hydrochloride
CAS:Tocainide hydrochloride (2-amino-n-(2,6-dimethylphenyl)propanamide hydrochloride) is a sodium channel blocker.Fórmula:C11H17ClN2OPureza:97%Forma y color:SolidPeso molecular:228.72Nefiracetam
CAS:Nefiracetam (DM9384), in Phase 2 trials, enhances GABA, choline, monoamine systems, and treats Ro 5-4864 convulsions.Fórmula:C14H18N2O2Pureza:97.37%Forma y color:SolidPeso molecular:246.33,4,5-Trimethoxycinnamic acid
CAS:3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) (TMCA) is one of the constituents of Polygalae Radix and may exert anti-seizure activity by acting at theFórmula:C12H14O5Pureza:98.91%Forma y color:SolidPeso molecular:238.24Phenibut
CAS:Phenibut (Aminophenylbutyric acid) is a central depressant and derivative of the naturally occurring inhibitory neurotransmitter γ-aminobutyric acid (GABA).Fórmula:C10H13NO2Pureza:99.55%Forma y color:White SolidPeso molecular:179.22Prilocaine hydrochloride
CAS:Prilocaine HCl: local amino amide anesthetic, blocks voltage-gated sodium channels in neurons, inhibits Na+ permeability.Fórmula:C13H21ClN2OPureza:99.97%Forma y color:SolidPeso molecular:256.77Z433927330
CAS:Z433927330 is a potent and selective Aquaporin-7 (AQP7) inhibitor(IC50s of 0.2).Fórmula:C20H20N4O3Pureza:99.64%Forma y color:SolidPeso molecular:364.4Suloctidil
CAS:Suloctidil is a peripheral vasodilator that was formerly used in the management of peripheral and cerebral vascular disorders.Fórmula:C20H35NOSPureza:99.75% - >99.99%Forma y color:White SolidPeso molecular:337.56Carboxyamidotriazole Orotate
CAS:Carboxyamidotriazole Orotate (L-651582 Orotate) is a cytostatic inhibitor of non-voltage-operated calcium channels and calcium channel-mediated signalingFórmula:C22H16Cl3N7O6Pureza:99.37%Forma y color:SolidPeso molecular:580.76Bupivacaine hydrochloride
CAS:Bupivacaine hydrochloride (Vivacaine) is a long-lasting, amide local anesthetic that blocks sodium channels, inhibiting nerve impulses and sensation.Fórmula:C18H28N2O·HClPureza:99.89% - 99.9%Forma y color:White SolidPeso molecular:324.89Cycloleucine
CAS:Cycloleucine is an antagonist of NMDA receptor associated glycine receptor with a Ki of 600 μM.Fórmula:C6H11NO2Pureza:99.90%Forma y color:SolidPeso molecular:129.16Methocarbamol
CAS:Methocarbamol (AHR 85) is a centrally acting muscle relaxant whose mode of action has not been established.Fórmula:C11H15NO5Pureza:99.96%Forma y color:White SolidPeso molecular:241.24IK1 inhibitor PA-6
CAS:IK1 inhibitor PA-6 (PA-6) is a selective and potent inhibitor of IK1 (KIR2.x ion-channel-carried inward rectifier current)(IC50 of 12-15 nM for human and mouseFórmula:C31H32N4O2Pureza:98.9%Forma y color:SolidPeso molecular:492.61Bemegride
CAS:Bemegride (3-Ethyl-3-methylglutarimide), a central nervous system stimulant, serves as an antidote for barbiturate poisoning.Fórmula:C8H13NO2Pureza:99.89%Forma y color:SolidPeso molecular:155.19Ethaverine hydrochloride
CAS:Ethaverine hydrochloride is a homologue of papaverine and is used as a vasodilator and antispasmodic.Cost-effective and quality-assured.Fórmula:C24H30ClNO4Pureza:99.66% - 99.73%Forma y color:SolidPeso molecular:431.96Manidipine dihydrochloride
CAS:Manidipine dihydrochloride (Manidipine 2HCl) is a potent calcium channel blocker for Ca2+ current(IC50=2.6 nM).Fórmula:C35H40Cl2N4O6Pureza:99.76% - 99.86%Forma y color:SolidPeso molecular:683.62ML418
CAS:ML418 is a potent, selective and CNS penetrating Kir7.1 potassium channel blocker (IC50 = 310 nM), and also potently inhibits Kir6.2/SUR1.Fórmula:C19H24ClN3O3Pureza:99.3%Forma y color:SolidPeso molecular:377.87Ref: TM-T16110
1mg37,00€5mg79,00€1mL*10mM (DMSO)84,00€10mg111,00€25mg178,00€50mg288,00€100mg414,00€200mg583,00€Flavoxate hydrochloride
CAS:Flavoxate hydrochloride (DW61) , a muscarinic AChR antagonist, is used in the therapy of various urinary syndromes and as an antispasmodic.Fórmula:C24H26ClNO4Pureza:99.78%Forma y color:White SolidPeso molecular:427.92
