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Metabolismo

Metabolismo

Los inhibidores del metabolismo son compuestos que interfieren con las vías metabólicas, alterando la producción y utilización de energía dentro de las células. Estos inhibidores se utilizan para estudiar la regulación del metabolismo, el papel de las vías metabólicas en enfermedades como el cáncer y la diabetes, y para desarrollar nuevas estrategias terapéuticas. Los inhibidores del metabolismo pueden dirigirse a diversas enzimas y procesos involucrados en la glucólisis, la oxidación de ácidos grasos y otras funciones metabólicas. En CymitQuimica, ofrecemos una amplia gama de inhibidores del metabolismo de alta calidad para apoyar su investigación en bioquímica, trastornos metabólicos y desarrollo de fármacos.

Subcategorías de "Metabolismo"

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Se han encontrado 8597 productos de "Metabolismo"

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  • Ch55

    CAS:
    <p>Ch55, a potent HL60 cell differentiator (EC50=200nM), binds well to RAR-α/β, useful for cancer research.</p>
    Fórmula:C24H28O3
    Pureza:99.55%
    Forma y color:Solid
    Peso molecular:364.48
  • Nanterinone

    CAS:
    <p>Nanterinone: oral phosphodiesterase inhibitor, improves acute heart failure hemodynamics.</p>
    Fórmula:C15H15N3O
    Pureza:99.53%
    Forma y color:Solid
    Peso molecular:253.3
  • L-Threonine derivative-1

    CAS:
    <p>L-Threonine derivative-1 is acetylsalicylic acid-L-threonine ester with potential analgesic activity.</p>
    Fórmula:C13H15NO6
    Pureza:97.03% - 98.91%
    Forma y color:Solid
    Peso molecular:281.26
  • ARRY-403

    CAS:
    <p>ARRY-403 is a novel glucokinase activator that reduces fasting and postprandial blood glucose in patients with type 2 diabetes.</p>
    Fórmula:C20H18N6O3S2
    Pureza:98.80%
    Forma y color:Solid
    Peso molecular:454.52
  • PKUMDL-LC-101-D04

    CAS:
    <p>PKUMDL-LC-101-D04 enhances GPX4, curbs iron death, boosts enzyme activity 150% at 20 μM, effective in wild-type MEF, reduces lipid peroxide toxicity.</p>
    Fórmula:C14H23ClN4O2S2
    Pureza:98.71%
    Forma y color:Solid
    Peso molecular:378.94
  • NCGC 607

    CAS:
    <p>NCGC 607 is a a noninhibitory chaperone of glucocerebrosidase (GCase).</p>
    Fórmula:C24H22IN3O4
    Pureza:99.69%
    Forma y color:Solid
    Peso molecular:543.35
  • G6PD activator AG1

    CAS:
    <p>G6PD activator AG1 is a G6PD agonist that promotes G6PD oligomerization to a catalytically competent form.</p>
    Fórmula:C24H30N4S2
    Pureza:98.38% - 99.51%
    Forma y color:Solid
    Peso molecular:438.65
  • S-2474

    CAS:
    <p>S-2474, an inhibitor of COX-2 and 5-lipoxygenase, has anti-inflammatory and neuroprotective activities, and inhibits cell death.</p>
    Fórmula:C20H31NO3S
    Pureza:99.03%
    Forma y color:Solid
    Peso molecular:365.53
  • Autotaxin-IN-3

    CAS:
    <p>Autotaxin-IN-3 is an inhibitor of Autotaxin (IC50 = 2.4 nM) which is responsible for the increase in lysophosphatidic acid in ascites and plasma.</p>
    Fórmula:C22H21N9O2
    Pureza:99.54% - 99.79%
    Forma y color:Solid
    Peso molecular:443.46
  • A-69412

    CAS:
    <p>A-69412 is a reversible 5-lipoxygenase inhibitor, potentially treating ulcerative colitis and asthma.</p>
    Fórmula:C7H10N2O3
    Pureza:99.54%
    Forma y color:Solid
    Peso molecular:170.17
  • AWD 12-281

    CAS:
    <p>AWD 12-281 is a PDE4 inhibitor with anti-inflammatory activity and bronchodilator activity for the study of chronic obstructive pulmonary disease (COPD).</p>
    Fórmula:C22H14Cl2FN3O3
    Pureza:99.25% - 99.85%
    Forma y color:Solid
    Peso molecular:458.27
  • Tofimilast

    CAS:
    <p>Tofimilast (CP-325366), a PDE4 inhibitor, is used potentially for the treatment of asthma and chronic obstructive pulmonary disease.</p>
    Fórmula:C18H21N5S
    Pureza:99.55%
    Forma y color:Solid
    Peso molecular:339.46
  • AC-261066

    CAS:
    <p>AC-261066 is an orally available and isoform-selective agonist of RARβ2 with a pEC50 of 8.0.</p>
    Fórmula:C17H20FNO4S
    Pureza:99.64%
    Forma y color:Solid
    Peso molecular:353.41
  • Pradefovir

    CAS:
    <p>Pradefovir (Remofovir) is a prodrug for chronic HBV, converting to PMEA in the liver with a Km of 60 μM and clearance of 359 ml/min.</p>
    Fórmula:C17H19ClN5O4P
    Pureza:97.50%
    Forma y color:Solid
    Peso molecular:423.79
  • Esuprone

    CAS:
    <p>Esuprone (LU-43839) is a novel reversible and highly selective MAO-A inhibitor with anticonvulsant activity for the treatment of depression.</p>
    Fórmula:C13H14O5S
    Pureza:99.45%
    Forma y color:Solid
    Peso molecular:282.31
  • Phosphatase-IN-1

    CAS:
    <p>Phosphatase-IN-1 is a phosphatidic acid phosphatase (Pah) inhibitor with antifungal activity for the study of rice blast and ruderalia.</p>
    Fórmula:C16H16Cl2FNO2
    Pureza:99.88%
    Forma y color:Solid
    Peso molecular:344.21
  • Salnacedin

    CAS:
    <p>Salnacedin (G-201) treats immune, skin, and musculoskeletal issues, suitable for acne, dermatitis, and psoriasis research.</p>
    Fórmula:C12H13NO5S
    Pureza:99.13%
    Forma y color:Solid
    Peso molecular:283.3
  • Bupicomide

    CAS:
    <p>Bupicomide is a dopamine β-hydroxylase inhibitor with antihypertensive and vasodilatory activity and may be used in the study of hypertension.</p>
    Fórmula:C10H14N2O
    Pureza:99.84% - >99.99%
    Forma y color:Solid
    Peso molecular:178.23
  • PDE4B-IN-2

    CAS:
    <p>PDE4B-IN-2 (A 33), an oral PDE4B inhibitor, IC50: 15 nM; less potent on PDE4D (IC50: 1.7 µM), has anti-inflammatory properties.</p>
    Fórmula:C19H18ClN3O2S
    Pureza:99.32%
    Forma y color:Solid
    Peso molecular:387.88
  • SBI-425

    CAS:
    <p>SBI-425: orally available TNAP inhibitor, enhances cardiovascular health &amp; survival, no bone impact.</p>
    Fórmula:C13H12ClN3O4S
    Pureza:99.88%
    Forma y color:Solid
    Peso molecular:341.77