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Metabolismo

Metabolismo

Los inhibidores del metabolismo son compuestos que interfieren con las vías metabólicas, alterando la producción y utilización de energía dentro de las células. Estos inhibidores se utilizan para estudiar la regulación del metabolismo, el papel de las vías metabólicas en enfermedades como el cáncer y la diabetes, y para desarrollar nuevas estrategias terapéuticas. Los inhibidores del metabolismo pueden dirigirse a diversas enzimas y procesos involucrados en la glucólisis, la oxidación de ácidos grasos y otras funciones metabólicas. En CymitQuimica, ofrecemos una amplia gama de inhibidores del metabolismo de alta calidad para apoyar su investigación en bioquímica, trastornos metabólicos y desarrollo de fármacos.

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Se han encontrado 8625 productos de "Metabolismo"

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  • Incadronate Disodium

    CAS:
    <p>Incadronate Disodium: halts bone loss, limits macrophage migration and inflammation, and induces cancer cell apoptosis in vitro.</p>
    Fórmula:C8H19NNaO6P2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:310.178
  • K103 Hydrochloride

    CAS:
    <p>K103 Hydrochloride, an inhibitor of peptidoglycan synthesis, targets the lipid II precursor.</p>
    Fórmula:C19H22Cl2N2S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:381.36
  • JCP-170

    CAS:
    <p>JCP-170 is an ABHD6 inhibitor.</p>
    Fórmula:C24H18ClNO4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:419.86
  • GNF7686

    CAS:
    <p>GNF7686 is a novel Trypanosoma cruzi inhibitor.</p>
    Fórmula:C15H13N3O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:251.28
  • Succinyladenosine

    CAS:
    <p>Succinyladenosine, a marker for ASL deficiency, is made by dephosphorylating S-AMP with 5-nucleotidase.</p>
    Fórmula:C14H17N5O8
    Forma y color:Solid
    Peso molecular:383.317
  • RA 642

    CAS:
    <p>RA 642 is used as a PDE-inhibitor.</p>
    Fórmula:C24H44N8O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:508.66
  • Emiglitate

    CAS:
    <p>Emiglitate is a selective and competitive α-glucoside hydrolase inhibitor.</p>
    Fórmula:C17H25NO7
    Pureza:98%
    Forma y color:Solid
    Peso molecular:355.38
  • NSC-79887

    CAS:
    <p>NSC-79887 is a nucleoside hydrolase (NH) inhibitor.</p>
    Fórmula:C14H16ClNO4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:297.73
  • CL385319 HCl

    CAS:
    "CL385319: Inhibits H5N1 flu virus, blocks entry, low cytotoxicity, IC50=27.03μM in MDCK cells, ineffective on VSV-G pseudotypes."
    Fórmula:C15H19ClF4N2O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:354.77
  • Adenosine 5'-phosphosulfate (sodium salt)

    CAS:
    <p>Adenosine 5'-phosphosulfate (sodium salt) (APS) is a key intermediate in sulphur metabolism and a substrate for adenosine 5'-phosphosulfate kinase (APSK).</p>
    Fórmula:C10H12N5Na2O10PS
    Forma y color:Solid
    Peso molecular:471.24
  • URB-694

    CAS:
    <p>URB-694 is a fatty acid amide hydrolase (FAAH) inhibitor.</p>
    Fórmula:C19H21NO3
    Forma y color:Solid
    Peso molecular:311.37
  • Hexazinone

    CAS:
    <p>Hexazinone: a triazine herbicide blocks photosynthesis by binding to D-1 protein in photosystem II.</p>
    Fórmula:C12H20N4O2
    Pureza:99.99%
    Forma y color:Solid
    Peso molecular:252.31
  • 14(S)-HDHA

    CAS:
    <p>DHA is an ω-3 important for development and therapy for inflammation and cancer; its derivative, 14(S)-HDHA, aids in reducing inflammation.</p>
    Fórmula:C22H32O3
    Forma y color:Solid
    Peso molecular:344.49
  • Hydroxythiohomosildenafil

    CAS:
    <p>Hydroxythiohomosildenafil, an analogue of sildenafil, is a phosphodiesterase-5 (PDE-5) inhibitor.</p>
    Fórmula:C23H32N6O4S2
    Pureza:99.45%
    Forma y color:Solid
    Peso molecular:520.67
  • ATX inhibitor 5

    CAS:
    <p>ATX inhibitor 5: potent, oral autotaxin blocker, IC50 15.3 nM, curbs CCl4 liver fibrosis.</p>
    Fórmula:C22H18ClF3N6O
    Pureza:98.77%
    Forma y color:Solid
    Peso molecular:474.87
  • 11β-HSD1-IN-6

    CAS:
    <p>11β-HSD1-IN-6 is a potent inhibitor of 11β hydroxysteroid dehydrogenase enzymes (11β-HSDs).</p>
    Fórmula:C21H19ClN4O
    Forma y color:Solid
    Peso molecular:378.86
  • Fluasterone

    CAS:
    <p>Fluasterone, an NF-κB activation inhibitor, is used potentially for the treatment of metabolic syndrome.</p>
    Fórmula:C19H27FO
    Pureza:98%
    Forma y color:Solid
    Peso molecular:290.42
  • ACAT-IN-1 cis isomer

    CAS:
    <p>ACAT-IN-1 cis isomer is a potent ACAT inhibitor (IC50: 100 nM) for the study of immune system-related diseases.</p>
    Fórmula:C29H25NO2
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:419.51
  • 2'-Ethyl Simvastatin

    CAS:
    <p>2'-Ethyl Simvastatin is a Mevinolin analog with HMG-CoA reductase inhibition.</p>
    Fórmula:C23H34O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:390.51
  • Brofaromine

    CAS:
    Brofaromine (CGP 11305A) is an MAO inhibitor (IC50: 0.2 μM for MAO-A).
    Fórmula:C14H16BrNO2
    Forma y color:Solid
    Peso molecular:310.19
  • Quinapril-d5

    CAS:
    <p>Quinapril-d5: An internal standard for quinapril quantification via GC/LC-MS; a prodrug ACE inhibitor for hypertension and heart failure.</p>
    Fórmula:C25H25D5N2O5
    Forma y color:Solid
    Peso molecular:443.55
  • CL 242817

    CAS:
    <p>CL 242817 is an inhibitor of angiotensin converting enzyme (ACE).</p>
    Fórmula:C18H21NO5S
    Forma y color:Solid
    Peso molecular:363.43
  • 11β-HSD1-IN-9

    CAS:
    <p>11β-HSD1-IN-9 is a potent inhibitor of 11β-HSD1, displaying IC50 values of 0.48 µM for human and 1.3 µM for murine variants, respectively.</p>
    Fórmula:C13H9F3N2O
    Forma y color:Solid
    Peso molecular:266.22
  • Benserazide

    CAS:
    <p>Benserazide blocks dopa decarboxylase; paired with levodopa for Parkinson's to boost CNS dopamine levels and lower dosage.</p>
    Fórmula:C10H15N3O5
    Forma y color:Solid
    Peso molecular:257.24
  • GK187

    CAS:
    <p>GK187 is a selective and potent Group VIA calcium-independent phospholipase A2 (GVIA iPLA2) inhibitor, used in the study of neurological disorders.</p>
    Fórmula:C14H15F5O2
    Forma y color:Solid
    Peso molecular:310.26
  • ML-148

    CAS:
    <p>ML-148 is a selective inhibitor of 15-hydroxy prostaglandin dehydrogenase (15-PGDH, IC50 = 56 nM).</p>
    Fórmula:C20H21N3O
    Pureza:99.88%
    Forma y color:Solid
    Peso molecular:319.4
  • CDK2-IN-11

    CAS:
    <p>CDK2-IN-11 inhibits CDK2 (IC50: 6.4 μM) and targets hCA II, IX, XII (Ki: 23.4-56.3 nM); suited for cancer research.</p>
    Fórmula:C18H14ClN7O2S
    Forma y color:Solid
    Peso molecular:427.87
  • KD-027

    CAS:
    <p>KD-027 is a novel and long-acting PDE5A(phosphodiesterase 5A) inhibitor with potential antihypertensive activity.</p>
    Fórmula:C25H35N7O6S
    Pureza:99.55%
    Forma y color:Solid
    Peso molecular:561.65
  • AVE5688

    CAS:
    <p>AVE5688 is an inhibitor of glycogen phosphorylase (GP, IC50s: 430 nM and 915 nM; Kds: 170 nM and 530 nM for rmGPb and rmGPa).</p>
    Fórmula:C16H8ClF5N2O5
    Pureza:99.65%
    Forma y color:Solid
    Peso molecular:438.69
  • FASN-IN-4

    CAS:
    <p>FAS-IN-1 is a potent inhibitor of Fatty acid synthase (FAS) wtih IC50 of 10 nM.</p>
    Fórmula:C26H27N3O4S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:477.58
  • RO-28-1675

    CAS:
    <p>RO-28-1675 is a direct and selective glucokinase activator, the GK/GKRP complex,insulin secretion and type 2 diabetes.</p>
    Fórmula:C18H22N2O3S2
    Pureza:98.13%
    Forma y color:Solid
    Peso molecular:378.51
  • Glucocerebrosidase-IN-1

    CAS:
    <p>Glucocerebrosidase-IN-1 inhibits GCase with IC50 of 29.3 μM, Ki 18.5 μM, useful for Gaucher's and Parkinson's research.</p>
    Fórmula:C13H27NO3
    Forma y color:Solid
    Peso molecular:245.36
  • AGI-026

    CAS:
    <p>AGI-026 (AGI-12026) is a novel and potent dual inhibitor of the mutant isocitrate dehydrogenase mIDH1/2 blood-brain barrier, reduce d-2-hydroxyglutarate (2-HG).</p>
    Fórmula:C18H15F6N7
    Pureza:99.79% - 99.86%
    Forma y color:Solid
    Peso molecular:443.35
  • IDO-IN-4

    CAS:
    <p>IDO-IN-4 is an indoleamine 2,3-dioxygenase 1 (IDO-1) inhibitor.</p>
    Fórmula:C26H35N3O3
    Forma y color:Solid
    Peso molecular:437.57
  • TDP1 Inhibitor-1

    CAS:
    <p>TDP1 Inhibitor-1 is a potent inhibitor of Tyrosyl-DNA Phosphodiesterase 1 (TDP1) (IC50 of 7 μM).</p>
    Fórmula:C26H26N2O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:446.49
  • Calcium glycerophosphate

    CAS:
    <p>CaGP inhibits intestinal alkaline phosphatase F3; used for calcium and phosphorus in parenteral nutrition.</p>
    Fórmula:C3H7CaO6P
    Pureza:99.84%
    Forma y color:Solid
    Peso molecular:210.14
  • PGMI-004A

    CAS:
    <p>PGMI-004A is an effective inhibitor of phosphoglycerate mutase 1 (IC50: 13.1 μM).</p>
    Fórmula:C21H12F3NO6S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:463.38
  • LEO 39652

    CAS:
    <p>LEO 39652: Dual-soft PDE4 inhibitor, IC50s: PDE4A/B: 1.2 nM, PDE4C: 3.0 nM, PDE4D: 3.8 nM; TNF-α IC50: 6.0 nM; for Atopic dermatitis research.</p>
    Fórmula:C23H23N3O5
    Forma y color:Solid
    Peso molecular:421.45
  • 3-Oxo-hop-22(29)-ene

    CAS:
    <p>3-Oxo-hop-22(29)-ene inhibits yeast α-glucosidase, moderately affects T. cruzi and L. mexicana, and has slight anti-inflammatory activity.</p>
    Fórmula:C30H48O
    Forma y color:Solid
    Peso molecular:424.7
  • Ro 41-0960

    CAS:
    <p>Ro 41-0960 is used as a reversible and orally-active COMT-inhibitor.</p>
    Fórmula:C13H8FNO5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:277.2
  • LGE-899

    CAS:
    <p>LGE-899 (Sonidegib metabolite M48) is a main metabolite of Sonidegib which is an inhibitor of the hedgehog pathway.</p>
    Fórmula:C15H11F3O3
    Pureza:99.93%
    Forma y color:Solid
    Peso molecular:296.24
  • Vorozole

    CAS:
    <p>Vorozole (R83842) is an orally active, potent, and selective nonsteroidal aromatase inhibitor.Vorozole exhibits antitumor activity in vivo and may be used in</p>
    Fórmula:C16H13ClN6
    Pureza:99.65% - 99.94%
    Forma y color:Solid
    Peso molecular:324.77
  • Lombricine

    CAS:
    <p>Lombricine, as a phosphodiester of 2-guanidinoethanol and D-serine in structure, is a phosphagen that is unique to earthworms.</p>
    Fórmula:C6H15N4O6P
    Forma y color:Solid
    Peso molecular:270.18
  • IACS-8968

    CAS:
    <p>IACS-8968 is a dual IDO and TDO inhibitor (pIC50s: 6.43 for IDO and &lt;5 for TDO).</p>
    Fórmula:C17H18F3N5O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:381.35
  • Inolitazone dihydrochloride

    CAS:
    <p>Inolitazone dihydrochloride is an effective, high-affinity PPARγ agonist; its biological activity is dependent on PPARγ (IC50:0.8 nM) to inhibit cell growth.</p>
    Fórmula:C27H28Cl2N4O4S
    Forma y color:Solid
    Peso molecular:575.51
  • OMDM-2

    CAS:
    <p>OMDM-2 is a metabolically stable and selective inhibitor of anandamide cellular uptake (ACU), exhibiting a Ki value of 3.0 μM in RBL-2H3 cells.</p>
    Fórmula:C27H45NO3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:431.65
  • Ambuphylline

    CAS:
    <p>Ambuphylline (Bufylline) is a theophylline derivative and bronchodilator for asthma and lung disease research.</p>
    Fórmula:C11H19N5O3
    Forma y color:Solid
    Peso molecular:269.305
  • PDE9-IN-1

    CAS:
    <p>PDE9-IN-1 is a selective and orally bioavailable Inhibitor of PDE9A(IC50 of 8.7 nM).</p>
    Fórmula:C17H23FN6O2
    Pureza:99.86%
    Forma y color:Solid
    Peso molecular:362.4
  • Talarozole (R enantiomer)

    CAS:
    <p>Talarozole R enantiomer is a potent and selective inhibitor of cytochrome P450 26-mediated breakdown of endogenous all-trans retinoic acid.</p>
    Fórmula:C21H23N5S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:377.51
  • MK-4409

    CAS:
    <p>MK-4409, a potent and selective fatty acid amide hydrolase (FAAH) inhibitor, is being investigated for the treatment of inflammatory and neuropathic pain.</p>
    Fórmula:C22H17ClFN3O2S
    Pureza:99.80% - 99.87%
    Forma y color:Solid
    Peso molecular:441.91
  • sPLA2-X Inhibitor 31

    CAS:
    <p>sPLA2-X Inhibitor 31 targets sPLA2-X with IC50: 26 nM; less effective on sPLA2-IIa (310 nM), sPLA2-V (2230 nM).</p>
    Fórmula:C19H15F3N2O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:392.33
  • AGN 191701

    CAS:
    <p>AGN 191701 is an agonist of the Retinoid X receptor.</p>
    Fórmula:C23H28O2S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:368.53
  • IM176OUT05

    CAS:
    <p>IM176OUT05 activates stem cell metabolism with hair regrowth-promoting effects.</p>
    Fórmula:C11H17N5
    Forma y color:Solid
    Peso molecular:219.29
  • LY 113174

    CAS:
    <p>LY 113174, a novel nonsteroidal aromatase inhibitor, may prove useful in the treatment of estrogen-dependent diseases.</p>
    Fórmula:C17H10Cl2N2
    Forma y color:Solid
    Peso molecular:313.18
  • FC11409B

    CAS:
    <p>FC11409B is a CAIX inhibitor, inhibiting breast cancer invasion and metastasis.</p>
    Fórmula:C29H23BF4N2O3S
    Forma y color:Solid
    Peso molecular:566.38
  • 7-Ketolithocholic acid

    CAS:
    <p>7-Ketolithocholic acid absorbs and reduces endogenous bile acid and cholesterol secretion.</p>
    Fórmula:C24H38O4
    Pureza:98.68% - 99.9%
    Forma y color:White - Almost White Solid Powder
    Peso molecular:390.56
  • Manitimus

    CAS:
    <p>Manitimus is a potent immunosuppressive drug, and is an inhibitor of dehydroorotate dehydrogenase,.</p>
    Fórmula:C15H11F3N2O2
    Pureza:99.75% - 99.75%
    Forma y color:Solid
    Peso molecular:308.26
  • Cholesteryl Palmitoleate

    CAS:
    <p>Cholesteryl palmitoleate, a cholesterol ester, exhibits elevated plasma levels in ApoE-/- mice following exposure to cigarette smoke and in pediatric patients diagnosed with biliary atresia. It serves as a standard for identifying cholesterol esters in human meibomian gland secretions.</p>
    Fórmula:C43H74O2
    Forma y color:Solid
    Peso molecular:623.1
  • 11β-HSD1-IN-1

    CAS:
    <p>11β-HSD1-IN-1 is an inhibitor of 11β-hydroxydehydrogenase 1 (11β-HSD1, IC50: 52 nM), and used for the treatment of pain.</p>
    Fórmula:C18H14ClF4N3O
    Pureza:99.84%
    Forma y color:Solid
    Peso molecular:399.77
  • TF-S14

    CAS:
    <p>TF-S14 is an inverse agonist of RORγt. It functions by binding to RORγt and inhibiting its activity, leading to a reduction in Th17 cell-associated cytokine production, including IL-17A, IL-21, and IL-22. TF-S14 is applicable in research related to autoimmune diseases and allogeneic transplant rejection.</p>
    Fórmula:C22H27N3O2S
    Forma y color:Solid
    Peso molecular:397.53
  • 93-O17O

    CAS:
    <p>93-O17O is a cationic lipidoid used in lipid nanoparticles for spleen-targeted delivery and genome editing in mice.</p>
    Fórmula:C44H83N3O6
    Forma y color:Solid
    Peso molecular:750.15
  • p-Valerylphenol

    CAS:
    p-Valerylphenol (NSC-49186) can be used to synthesize acylphenoxyacetic acid compounds.
    Fórmula:C11H14O2
    Pureza:99.87%
    Forma y color:White To Light Beige Powder
    Peso molecular:178.23
  • SRPKIN-1

    CAS:
    <p>SRPKIN-1 is a covalent and irreversible inhibitor of SRPK1/2 (IC50s: 35.6 and 98 nM, respectively).</p>
    Fórmula:C27H21FN2O3S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:472.53
  • Rev 5975

    CAS:
    <p>Rev 5975 is a non-sulfhydryl ACE-inhibitor.</p>
    Fórmula:C24H30N2O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:426.51
  • OSMI-3

    CAS:
    <p>OSMI-3 is a potent and cell-permeable inhibitor of O-GlcNAc transferase (OGT) for the study of cancer and cardiovascular disease.</p>
    Fórmula:C32H35N3O9S2
    Pureza:99.03% - 99.08%
    Forma y color:Solid
    Peso molecular:669.77
  • BI-L 357

    CAS:
    <p>BI-L 357, a prodrug of BL-L 226, is a selective, orally active inhibitor of 5-lipoxygenase.</p>
    Fórmula:C18H18O4S
    Forma y color:Solid
    Peso molecular:330.4
  • IDO-IN-3

    CAS:
    <p>IDO-IN-3 is a potent indoleamine 2,3-dioxygenase (IDO) inhibitor (IC50: 290 nM).</p>
    Fórmula:C11H12BrFN6O2
    Forma y color:Solid
    Peso molecular:359.15
  • IHVR-11029

    CAS:
    <p>IHVR-11029 inhibits ER α-glucosidase, combats hemorrhagic fever viruses, and hinders enveloped virus morphogenesis.</p>
    Fórmula:C18H27F2NO5
    Forma y color:Solid
    Peso molecular:375.41
  • LZWL02003

    CAS:
    <p>LZWL02003, an anti-neuroinflammatory agent, demonstrates a protective effect on MPP+-induced neuronal damage and reduces ROS expression.</p>
    Fórmula:C18H18N2O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:294.35
  • 2614W94

    CAS:
    2614W94 is a selective inhibitor of MAO-A with IC50 of 5 nM and Ki of 1.6 nM.
    Fórmula:C15H11F3O4S
    Pureza:99.6%
    Forma y color:Solid
    Peso molecular:344.31
  • JZP-MA-13


    <p>JZP-MA-13: selective α/β-hydrolase domain 6 inhibitor, IC 50 392 nM, doesn't inhibit MAGL/ABHD12/FAAH, used in PET imaging.</p>
    Fórmula:C14H15FN4O3S
    Forma y color:Solid
    Peso molecular:338.36
  • NCT-506

    CAS:
    <p>NCT-506 is an orally bioavailable inhibitors of aldehyde dehydrogenase 1A1 (ALDH1A1) (IC50 of 7 nM).</p>
    Fórmula:C25H23FN4O3S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:478.54
  • BRD9500

    CAS:
    <p>BRD9500 is an oral PDE3 inhibitor, IC50: 10 nM (PDE3A), 27 nM (PDE3B); effective in SK-MEL-3 cancer model.</p>
    Fórmula:C15H18FN3O2
    Forma y color:Solid
    Peso molecular:291.32
  • PF-07208254

    CAS:
    <p>PF-07208254, a potent BDK inhibitor, enhances cardiometabolic endpoints in mice [1].</p>
    Fórmula:C7H2ClFO2S2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:236.67
  • hCA I-IN-1

    CAS:
    <p>hCA I-IN-1 inhibits hCA I (Ki: 38.3 nM), II (Ki: 716.4 nM), IX (Ki: 940.1 nM), XII (Ki: 192.8 nM).</p>
    Fórmula:C27H23N5O4S
    Forma y color:Solid
    Peso molecular:513.57
  • Tebuconazole-d9

    CAS:
    <p>Tebuconazole-d9 is a GC/LC-MS standard for quantifying the triazole fungicide tebuconazole, affecting seed/foliar fungi and androgen receptors.</p>
    Fórmula:C16H13ClD9N3O
    Forma y color:Solid
    Peso molecular:316.87
  • Enpp-1-IN-17

    CAS:
    <p>Enpp-1-IN-17 (example 274) is a potent inhibitor of ENPP1, exhibiting inhibition constants (Ki values) of 100 nM-1 μM for cGAMP hydrolysis and &gt;1 μM for ATP</p>
    Fórmula:C18H24N4O2
    Forma y color:Solid
    Peso molecular:328.41
  • HFI-437

    CAS:
    <p>HFI-437 is a potent, non-peptidic, insulin-regulated aminopeptidase (IRAP) inhibitor with a K i of 20 nM and functions as a cognitive enhancer [1].</p>
    Fórmula:C23H20N2O5
    Forma y color:Solid
    Peso molecular:404.42
  • 17β-HSD10-IN-2

    CAS:
    <p>17β-HSD10-IN-2 (compound 11), a benzothiazolylurea-based inhibitor, specifically targets 17β-hydroxysteroid dehydrogenase type 10 (17β-HSD10), avoiding</p>
    Fórmula:C15H10ClN3O4S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:363.78
  • AVX-001

    CAS:
    <p>AVX-001, a cytosolic phospholipase A2 (cPLA2) inhibitor, is used potentially for the treatment of psoriasis.</p>
    Fórmula:C21H29F3OS
    Forma y color:Solid
    Peso molecular:386.51
  • Moperone Hydrochloride

    CAS:
    <p>Moperone Hydrochloride, a dopamine D2-receptor antagonist, is used for the treatment of psychiatric disorders.</p>
    Fórmula:C22H27ClFNO2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:391.91
  • Glyoxalase I inhibitor 7

    CAS:
    <p>Glyoxalase I inhibitor 7 (Compound 6) is a potent inhibitor of glyoxalase I (Glo-I) with an IC50 of 3.65 μM. It exhibits potential as an anticancer agent [1].</p>
    Fórmula:C17H16N4O3S
    Forma y color:Solid
    Peso molecular:356.4
  • BTX161

    CAS:
    <p>BTX161: potent CKIα degrader, surpasses Lenalidomide in AML, triggers DDR + p53, stabilizes MDM2.</p>
    Fórmula:C15H16N2O3
    Forma y color:Solid
    Peso molecular:272.3
  • RP 73163 Racemate

    CAS:
    <p>RP 73163 Racemate is the racemate of RP 73163. RP 73163 is a potent inhibitor of ACAT, shows cholesterol lowering activity.</p>
    Fórmula:C25H28N4OS
    Pureza:98%
    Forma y color:Solid
    Peso molecular:432.58
  • Safusidenib

    CAS:
    <p>Safusidenib, oral mutant IDH1 inhibitor, selectively targets IDH1R132H/C mutations with IC50 of 15/130 nM; impairs chondrosarcoma growth.</p>
    Fórmula:C25H18Cl3FN2O4
    Forma y color:Solid
    Peso molecular:535.78
  • L 652343

    CAS:
    <p>L 652343 is an inhibitor of cyclooxygenase and 5-lipoxygenase in vitro. It also inhibits the synthesis of the products of both these pathways in whole cells.</p>
    Fórmula:C22H14F3NO2S2
    Forma y color:Solid
    Peso molecular:445.48
  • trans-Ned 19

    CAS:
    <p>trans-Ned 19 blocks NAADP and TPC, hindering calcium signaling and aorta relaxation at low histamine levels.</p>
    Fórmula:C30H31FN4O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:514.59
  • JTP 103237

    CAS:
    <p>JTP 103237 is a potent and selective monoacyglycerol acyltransferase 2 (MOGAT2) inhibitor.</p>
    Fórmula:C24H29F3N6O
    Forma y color:Solid
    Peso molecular:474.52
  • FTase-IN-1

    CAS:
    <p>FTase-IN-1, a potent FTase inhibitor, has an IC50 of 0.35 μM with strong antitumor activity and cytotoxicity.</p>
    Fórmula:C23H16N2O2S
    Forma y color:Solid
    Peso molecular:384.45
  • Niraparib metabolite M1

    CAS:
    <p>Niraparib metabolite M1 (Niraparib carboxylic acid metabolite M1) is the carboxylic acid metabolite of niraparib.</p>
    Fórmula:C19H19N3O2
    Pureza:99.65%
    Forma y color:Solid
    Peso molecular:321.37
  • SQ-31765

    CAS:
    <p>SQ-31765 is a blocker of benzazepine calcium channel.</p>
    Fórmula:C24H27F3N2O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:464.48
  • Erythronic acid

    CAS:
    <p>Erythronic acid, an endogenous carbohydrate metabolite, is instrumental for research into metabolism-associated disorders.</p>
    Fórmula:C4H8O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:136.1
  • Lauroyl glutamic acid

    CAS:
    <p>Lauroyl glutamic acid (N-Lauroyl-L-glutamic acid) exhibits antiasthmatic effects.</p>
    Fórmula:C17H31NO5
    Pureza:98.94%
    Forma y color:Solid
    Peso molecular:329.43
  • IDO1-IN-21

    CAS:
    <p>IDO1-IN-21 (compound 10m), with an IC50 of 0.64 μM, acts as an IDO1 inhibitor and has demonstrated efficacy in suppressing tumor growth in murine models [1].</p>
    Fórmula:C21H19F2N3O6S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:479.45
  • SHP2-IN-5

    CAS:
    <p>SHP2-IN-5 (compound 1) is a non-receptor protein tyrosine phosphatase inhibitor targeting SHP2 with an IC50 value of 97 nM, associated with regulating cell</p>
    Fórmula:C12H8O6
    Forma y color:Solid
    Peso molecular:248.19
  • ONO-6126

    CAS:
    <p>ONO-6126 has anti-inflammatory activity and can inhibit Phosphodiesterase and PDE4 in the treatment of respiratory diseases.</p>
    Fórmula:C20H27N3O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:373.45
  • WES-1

    CAS:
    <p>WES-1 (Compound 8g), a carbonic anhydrase IX inhibitor (Ki: 55.9 μM), exhibits broad-spectrum antiproliferative activity against various cancer cell lines,</p>
    Fórmula:C20H20N4O3S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:396.46
  • CP 99994 dihydrochloride

    CAS:
    <p>High affinity NK1 antagonist</p>
    Fórmula:C19H26Cl2N2O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:369.33
  • Oleyl Anilide

    CAS:
    <p>"Oleyl analide (OA) inhibits ACAT (IC50 26 μM), linked to toxic oil syndrome (TOS) with eosinophilia, T-cell activation, and high IL-4, IL-2R, IL-5."</p>
    Fórmula:C24H39NO
    Forma y color:Solid
    Peso molecular:357.57
  • OL-135

    CAS:
    <p>OL-135: CNS-accessible, potent, selective FAAH inhibitor with analgesic effects in animals, no motor impairment.</p>
    Fórmula:C21H22N2O2
    Forma y color:Solid
    Peso molecular:334.41
  • Levophencynonate HCl

    CAS:
    <p>Levophencynonate HCl is a muscarinic receptor antagonist.</p>
    Fórmula:C22H32ClNO3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:393.95
  • UK-371804 HCl

    CAS:
    <p>UK-371804 is a potent and selective urokinase-type plasmogen activator (uPA) inhibitor with excellent enzyme potency (Ki=10 nM) and selectivity profile (2700-</p>
    Fórmula:C14H17Cl2N5O4S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:422.29
  • M8891

    CAS:
    <p>M8891: Oral, reversible MetAP-2 inhibitor, brain-penetrant (IC50: 54nM; Ki: 4.33nM), hinders endothelial &amp; tumor cell growth, antiangiogenic &amp; antitumor.</p>
    Fórmula:C20H17F2N3O3
    Forma y color:Solid
    Peso molecular:385.36
  • GSK 264220A

    CAS:
    <p>endothelial lipase and lipoprotein lipase inhibitor</p>
    Fórmula:C17H21N3O4S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:363.43
  • IHMT-PI3Kδ-372

    CAS:
    <p>IHMT-PI3Kδ-372 is a selective inhibitor of PI3Kδ with an IC50 of 14 nM and can be used in studies about chronic obstructive pulmonary disease.</p>
    Fórmula:C26H23F2N7O2
    Pureza:99.77%
    Forma y color:Solid
    Peso molecular:503.5
  • Ciraparantag

    CAS:
    <p>Ciraparantag inhibits thrombin, factor Xa, and reverses various anticoagulants.</p>
    Fórmula:C22H48N12O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:512.7
  • LG 101506

    CAS:
    <p>RXR modulator</p>
    Fórmula:C25H34F2O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:420.53
  • Oosponol

    CAS:
    <p>Oosponol is a dopamine beta-hydroxylase inhibitor exhibiting hypotensive effects.</p>
    Fórmula:C11H8O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:220.18
  • BML-111

    CAS:
    <p>inhibits leukotriene B4 (LTB4)-induced polymorphonuclear neutrophils (PMN) chemotaxis</p>
    Fórmula:C8H16O5
    Forma y color:Solid
    Peso molecular:192.21
  • Spirapril

    CAS:
    <p>Spiropril is an ACE inhibitor antihypertensive drug, which belongs to the bicarboxyl group of ACE inhibitors and is used in the treatment of hypertension.</p>
    Fórmula:C22H30N2O5S2
    Forma y color:Solid
    Peso molecular:466.61
  • BMS270394

    CAS:
    <p>BMS270394 is a RARγ agonist used in the study of breast cancer and skin diseases.</p>
    Fórmula:C23H26FNO4
    Forma y color:Solid
    Peso molecular:399.46
  • RORγt/DHODH-IN-2

    CAS:
    <p>RORγt/DHODH-IN-2 (compound 1) is a potent dual RORγt/DHODH inhibitor that can be used in the study of inflammatory bowel disease (IBD).</p>
    Fórmula:C25H30N4OS
    Forma y color:Solid
    Peso molecular:434.6
  • Carbonic anhydrase inhibitor 7

    CAS:
    <p>Potent hCA inhibitor; targets hCA IX, II, XII, I with Ki: 6.5, 7.1, 72.1, 255.8 nM respectively.</p>
    Fórmula:C23H17N3O5S
    Forma y color:Solid
    Peso molecular:447.46
  • Choline theophyllinate

    CAS:
    <p>Choline theophyllinate (Oxtriphylline) is the choline salt of theophylline, a small molecule PDE inhibitor that can be used to treat immune system disorders and</p>
    Fórmula:C12H21N5O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:283.33
  • Arasertaconazole

    CAS:
    <p>Arasertaconazole, a sterol-14-alpha demethylation inhibitor, is used potentially for the treatment of vulvovaginal candcanidiasis.</p>
    Fórmula:C20H15Cl3N2OS
    Forma y color:Solid
    Peso molecular:437.77
  • A-908292

    CAS:
    <p>A-908292: potent ACC2 inhibitor with 38 nM IC50, useful for studying fatty acid metabolism.</p>
    Fórmula:C18H20N2O4S
    Forma y color:Solid
    Peso molecular:360.43
  • FABP-IN-2

    CAS:
    <p>FABP-IN-2, a novel ligand for FABP3, demonstrates inhibition of both FABP3 and FABP4 with IC50 values of 1.16 μM and 4.27 μM, respectively.</p>
    Fórmula:C25H21ClN2O3
    Forma y color:Solid
    Peso molecular:432.9
  • Seviteronel

    CAS:
    <p>Seviteronel (VT-464) is a novel CYP17 cleavage enzyme inhibitor and androgen receptor antagonist for the study of breast and prostate cancer.</p>
    Fórmula:C18H17F4N3O3
    Pureza:99.67% - 99.98%
    Forma y color:Solid
    Peso molecular:399.34
  • NEP-IN-2

    CAS:
    <p>NEP-IN-2 is an inhibitor of neutral endopeptidase. It also is used in the research of proliferation in atherosclerosis, restenosis.</p>
    Fórmula:C16H23NO3S2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:341.49
  • MY33-3 hydrochloride

    CAS:
    <p>MY33-3 HCl: Inhibits RPTPβ/ζ (IC50~0.1μM), PTP-1B (IC50~0.7μM), curbs alcohol intake, fights neuroinflammation and memory issues.</p>
    Fórmula:C16H14ClF6NS2
    Forma y color:Solid
    Peso molecular:433.86
  • BN82002

    CAS:
    <p>BN82002 (CDC25 Phosphatase Inhibitor I) is a synthetic inhibitor of CDC25 phophatases</p>
    Fórmula:C19H25N3O4
    Pureza:98.24%
    Forma y color:Solid
    Peso molecular:359.42
  • α-Amylase/α-Glucosidase-IN-1

    CAS:
    <p>α-Amylase/α-Glucosidase-IN-1 (compound 33) is an effective inhibitor of α-amylase/α-glucosidase with IC 50 s of 2.01, 2.09 μM for α-amylase and α-glucosidase,</p>
    Fórmula:C11H9N5
    Forma y color:Solid
    Peso molecular:211.22
  • XY101

    CAS:
    <p>XY101 is a selective, metabolically stable and orally available agonist of RORγ inverse(IC50 of 30 nM and a Kd of 380 nM).</p>
    Fórmula:C25H20F7NO4S
    Pureza:99.83%
    Forma y color:Solid
    Peso molecular:563.48
  • AZD8329

    CAS:
    <p>AZD8329 is an 11β-HSD1 inhibitor that inhibits 11β-HSD2, 17β-HSD1, 17β-HSD3, and can be used to study allergic reactions in humans.</p>
    Fórmula:C25H31N3O3
    Pureza:99.31%
    Forma y color:Solid
    Peso molecular:421.53
  • BKIDC-1553

    CAS:
    <p>BKIDC-1553, an orally active antiglycolytic agent and bumped kinase inhibitor-derived compound, has a predicted half-life of approximately 17 hours in humans. It inhibits CYP2C8 and Angiotensin Converting Enzyme, making it suitable for cancer research [1].</p>
    Fórmula:C22H23N5O2
    Forma y color:Solid
    Peso molecular:389.45
  • PDE4-IN-11

    CAS:
    <p>PDE4-IN-11: Potent PDE4 inhibitor with strong bronchodilatory and anti-inflammatory effects for airway disease research.</p>
    Fórmula:C21H19FN2O2
    Forma y color:Solid
    Peso molecular:350.39
  • L-693612 HCl

    CAS:
    <p>L-693612 HCl is an inhibitor of carbonic anhydrase.</p>
    Fórmula:C14H25ClN2O5S3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:433.01
  • TK-642

    CAS:
    <p>TK-642 is a potent and selective SHP2 inhibitor with oral activity, based on pyrazole and pyrazine structures (IC50 = 2.7 nmol/L). It effectively inhibits the proliferation of esophageal carcinoma cells and induces apoptosis, making it useful for studying esophageal cancer.</p>
    Fórmula:C17H20ClN7S
    Forma y color:Solid
    Peso molecular:389.91
  • BMS-593214

    CAS:
    <p>BMS-593214 is an inhibitor of active site-directed factor VIIa and a non-competitive inhibitor of the VIIa-activated substrate FX.</p>
    Fórmula:C31H27N3O4
    Pureza:96.63% - 98.04%
    Forma y color:Solid
    Peso molecular:505.56
  • α-Amylase/α-Glucosidase-IN-2

    CAS:
    α-Amylase/α-Glucosidase-IN-2 (compound 5) exhibits strong inhibition activity towards both α-amylase and α-glucosidase enzymes, with IC 50 values of 13.02 μM
    Fórmula:C22H16ClN5
    Forma y color:Solid
    Peso molecular:385.85
  • NPD-1335

    CAS:
    <p>NPD1335: potent TbrPDEB1 inhibitor, submicromolar efficacy, low toxicity, raises cAMP, disrupts cell cycle, kills T. brucei.</p>
    Fórmula:C28H29N3O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:455.55
  • GSK376501A

    CAS:
    <p>GSK376501A is a selective and effective modulator of peroxisome proliferator-activated receptor γ (PPARγ) for the study of type 2 diabetes.</p>
    Fórmula:C32H37NO6
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:531.64
  • Sch 34826

    CAS:
    <p>Sch 34826 is a potent, selective neutral endopeptidase inhibitor.</p>
    Fórmula:C27H34N2O7
    Pureza:98%
    Forma y color:Solid
    Peso molecular:498.57
  • Boc-Glu(OBzl)-OSu

    CAS:
    <p>Boc-Glu(OBzl)-OSu can be used for the synthesis of solid phase peptides containing benzyl glutamate residues.</p>
    Fórmula:C21H26N2O8
    Forma y color:Solid
    Peso molecular:434.44
  • PDE5-IN-4

    CAS:
    <p>PDE5-IN-4, a phosphodiesterase 5 (PDE5) inhibitor, is utilized in research concerning acute myocardial infarction and reperfusion-related damage,</p>
    Fórmula:C21H27N5O5S
    Forma y color:Solid
    Peso molecular:461.53
  • 5β-​Dutasteride

    CAS:
    <p>5β-Dutasteride is the S configuration of Dutasteride. It is a potent inhibitor of both 5 alpha-reductase isozymes.</p>
    Fórmula:C27H30F6N2O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:528.53
  • Glutamamide

    CAS:
    <p>Glutamamide is an anticancer drug.</p>
    Fórmula:C5H11N3O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:145.16
  • Oxagrelate

    CAS:
    <p>Oxagrelate inhibits cAMP phosphodiesterase and reduces platelet aggregation by collagen and ADP.</p>
    Fórmula:C14H16N2O4
    Forma y color:Solid
    Peso molecular:276.29
  • Quinethazone

    CAS:
    <p>Quinethazone is a thiazide diuretic used to treat hypertension. Common side effects include dizziness, dry mouth, nausea, and low potassium levels.</p>
    Fórmula:C10H12ClN3O3S
    Forma y color:Fibrous Crystals From 50% Acetone Physical Description Fibrous Crystals Or White Powder (Ntp 1992)
    Peso molecular:289.74
  • Deltazinone

    CAS:
    <p>Deltazinone selectively inhibits PDEδ with low cytotoxicity, mimicking PDEδ knockdown in human pancreatic cancer cells.</p>
    Fórmula:C27H31N5O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:457.57
  • Acetyl-CoA Carboxylase-IN-1

    CAS:
    Acetyl-CoA Carboxylase-IN-1 (ACC-IN-1) is a potent acetyl-CoA carboxylase (ACC) inhibitor with antibacterial activity, used in metabolic disease research.
    Fórmula:C13H9Br2N5
    Pureza:98.73%
    Forma y color:Solid
    Peso molecular:395.05
  • MitoTEMPO hydrate

    CAS:
    <p>MitoTEMPO, a mitochondria-targeted antioxidant, scavenges superoxide and alkyl radicals supporting potential therapy for mitochondrial dysfunction.</p>
    Fórmula:C29H35N2O2P·Cl·H2O
    Forma y color:Solid
    Peso molecular:528.04
  • GT 949

    CAS:
    <p>GT 949 is a selective excitatory positive allosteric modulator of amino acid transporter-2 (EAAT2) (EC50: 0.26 nM).</p>
    Fórmula:C30H37N7O2
    Pureza:99.95%
    Forma y color:Solid
    Peso molecular:527.66
  • JMS-053

    CAS:
    <p>JMS-053 is a phosphatase DUSP3 inhibitor that inhibits CDC25B and prevents VEGF from disrupting the microvascular endothelial barrier.</p>
    Fórmula:C13H8N2O2S
    Pureza:≥98.0%
    Forma y color:Solid
    Peso molecular:256.28
  • GNF362

    CAS:
    <p>GNF362 is an ITPKB inhibitor that inhibits Itpka and Itpkc and reverses the migratory stimulatory effect of ITPKA overexpression.</p>
    Fórmula:C22H21F3N6
    Pureza:99.63%
    Forma y color:Solid
    Peso molecular:426.44
  • RORγt inverse agonist 30

    CAS:
    <p>RORγt inverse agonist 30 (Compound 1) is a potent RORγt inverse agonist (IC50: 46 nM).</p>
    Fórmula:C24H31N3O3S
    Forma y color:Solid
    Peso molecular:441.59
  • ATX inhibitor 11

    CAS:
    <p>ATX inhibitor 11 blocks autotaxin (IC50: 2.7 nM), reduces fibrosis and α-SMA in mice. Useful for lung fibrosis studies.</p>
    Fórmula:C32H35N5O6
    Forma y color:Solid
    Peso molecular:585.65
  • S07-2010

    CAS:
    <p>S07-2010 is a pan-Aldo-Keto Reductase 1C3 (AKR1C3) inhibitor with potential anti-cancer activity, inducing apoptosis in A549/DDP cells.</p>
    Fórmula:C19H21N3O3S
    Pureza:98.13%
    Forma y color:Solid
    Peso molecular:371.45
  • CD 1530

    CAS:
    <p>CD 1530 is an ARγ agonist (Kd:150 nM) with potential anticancer activity for the study of oral carcinogenesis.</p>
    Fórmula:C27H26O3
    Pureza:98.13%
    Forma y color:Solid
    Peso molecular:398.49
  • Cefetrizole

    CAS:
    <p>Ceftezole is an α-Glucosidase inhibitor (IC50: 2.1 μM; Ki: 0.578 μM).</p>
    Fórmula:C16H15N5O4S3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:437.52
  • Dopropidil

    CAS:
    <p>Dopropidil: anti-angina calcium regulator with anti-ischemic properties in animal models.</p>
    Fórmula:C20H35NO2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:321.5
  • SA57

    CAS:
    <p>SA57 is a potent, selective inhibitor of FAAH(IC50s of 3.2 nM and 1.9 nM for mouse and human FAAH).</p>
    Fórmula:C17H23ClN2O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:338.83
  • Xanthine oxidoreductase-IN-2

    CAS:
    <p>Xanthine oxidoreductase-IN-2 inhibits XOR with 7.2 nM IC50 and shows hypouricemic effects in mice.</p>
    Fórmula:C21H19N3O2
    Forma y color:Solid
    Peso molecular:345.39
  • Glucokinase activator 3

    CAS:
    <p>Glucokinase activator 3: potent GK activator, AC50=38 nM, potential for type 2 diabetes research.</p>
    Fórmula:C26H33N2O9PS2
    Forma y color:Solid
    Peso molecular:612.65
  • FSG67

    CAS:
    <p>FSG67 is an inhibitor of glycerol 3-phosphate acyltransferase (IC 50 =24 μM) [1].</p>
    Fórmula:C16H25NO4S
    Pureza:99.76%
    Forma y color:Solid
    Peso molecular:327.44
  • α-Glucosidase-IN-8

    CAS:
    <p>α-Glucosidase-IN-8 (Compound 4k) is a potent, competitive inhibitor of α-glucosidase. It displays an impressive IC50 value of 0.18 μg/mL [1].</p>
    Fórmula:C19H20FN3O2
    Forma y color:Solid
    Peso molecular:341.38
  • hCAIX-IN-6

    CAS:
    <p>6B and 14g inhibit tumor-associated HCA IX with low nanomolar potency; 6K targets HCA XII. All are potential cancer drug leads.</p>
    Fórmula:C18H12N2O4S
    Forma y color:Solid
    Peso molecular:352.36
  • Carbonic anhydrase inhibitor 13

    CAS:
    <p>Carbonic anhydrase inhibitor 13 (compound 7) is a potent inhibitor of carbonic anhydrase (CA).</p>
    Fórmula:C17H15N5O3S2
    Forma y color:Solid
    Peso molecular:401.46
  • α-2,3-sialyltransferase-IN-1

    CAS:
    <p>α-2,3-sialyltransferase-IN-1 is a noncompetitive inhibitor of α-2,3-sialyltransferase(IC50 of 6 μM).</p>
    Fórmula:C28H45NO6
    Pureza:98% - 98%
    Forma y color:Solid
    Peso molecular:491.66
  • IDO1-IN-17

    CAS:
    <p>IDO1-IN-17 (I-4) is an IDO1 inhibitor, with an IC 50 of 0.44 μM in hela cells .</p>
    Fórmula:C28H32BrClFN5O2
    Forma y color:Solid
    Peso molecular:604.94
  • FAAH-IN-5

    CAS:
    <p>FAAH-IN-5 (Compound 7) selectively, irreversibly inhibits FAAH (IC50: 10.5 nM) with low PAMPA permeability.</p>
    Fórmula:C21H19N3O6S
    Forma y color:Solid
    Peso molecular:441.46
  • IDH2R140Q-IN-1

    CAS:
    <p>IDH2R140Q-IN-1 is a potent inhibitor of IDH2R140Q (IC50: 6.1 nM) and can be used in studies of acute myeloid leukemia.</p>
    Fórmula:C22H20F6N6
    Forma y color:Solid
    Peso molecular:482.42
  • Piritrexim

    CAS:
    <p>Piritrexim (BW 301U) is an orally available fat-soluble dihydrofolate reductase inhibitor with pulmonary toxicity used in the study of uroepithelial carcinoma</p>
    Fórmula:C17H19N5O2
    Pureza:98.50% - >99.99%
    Forma y color:Solid
    Peso molecular:325.37
  • IDO1-IN-2

    CAS:
    <p>IDO1-IN-2 is a potent and selective IDO1 inhibitor with IC50s of 81 nM, 59 nM (mouse), and 28 nM (rat), respectively. It has anti-cancer activity.</p>
    Fórmula:C15H17FN6O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:364.33
  • ALRT 1550

    CAS:
    <p>ALRT 1550, a retinoic acid agent (RAR) agonist, is used potentially for the treatment of cervical carcinoma.</p>
    Fórmula:C23H32O2
    Forma y color:Solid
    Peso molecular:340.5
  • S32826 disodium

    CAS:
    <p>autotaxin inhibitor</p>
    Fórmula:C21H36NNa2O4P
    Pureza:98%
    Forma y color:Solid
    Peso molecular:443.47
  • Aminopeptidase-IN-1

    CAS:
    <p>Aminopeptidase-IN-1: potent IRAP blocker, Ki 7.7 μM, useful for cognitive/memory disorder research.</p>
    Fórmula:C18H16N2O6
    Pureza:98.37%
    Forma y color:Solid
    Peso molecular:356.33
  • PKR activator 2

    CAS:
    PKR activator 2 is a potent activator of pyruvate kinase-R (PKR).
    Fórmula:C18H16N8OS
    Pureza:98%
    Forma y color:Solid
    Peso molecular:392.44
  • TTA-A8

    CAS:
    <p>TTA-A8 is an antagonist of T-type calcium channel.</p>
    Fórmula:C22H21F3N4O2
    Pureza:99.22%
    Forma y color:Solid
    Peso molecular:430.42
  • FXR agonist 4


    <p>FXR agonist 4: EC50 of 1.05μM, treats hyperlipidemia, steatosis, insulin resistance, inflammation in DIO mice, for NAFLD research.</p>
    Fórmula:C21H28ClN3O
    Forma y color:Solid
    Peso molecular:373.92
  • Albaconazole

    CAS:
    <p>Albaconazole, a small fungal CYP51A1 inhibitor, treats fungal infections and some musculoskeletal disorders.</p>
    Fórmula:C20H16ClF2N5O2
    Pureza:99.27%
    Forma y color:Solid
    Peso molecular:431.82
  • DHODH-IN-17

    CAS:
    <p>DHODH-IN-17 is a human DHODH inhibitor with an IC50 of 0.40 μM.</p>
    Fórmula:C12H9ClN2O2
    Pureza:99.41% - 99.52%
    Forma y color:Solid
    Peso molecular:248.67
  • KCN1

    CAS:
    <p>KCN1: a synthetic sulfonamide, nanomolar HIF inhibitor with preclinical anti-glioma and anti-pancreatic cancer effects.</p>
    Fórmula:C26H27NO5S
    Forma y color:Solid
    Peso molecular:465.56
  • F-1394

    CAS:
    <p>F-1394 is an ACAT inhibitor that reduces atherosclerosis and neointimal thickening without changing serum cholesterol.</p>
    Fórmula:C33H61N3O6
    Forma y color:Solid
    Peso molecular:595.85
  • SCH-42354

    CAS:
    <p>SCH-42354: potent oral NEP inhibitor, activates ANP &amp; leu-enkephalin, has anti-hypertensive properties, IC50s of 8.3 &amp; 10.0 nM.</p>
    Fórmula:C16H23NO3S2
    Forma y color:Solid
    Peso molecular:341.49
  • BDM14471

    CAS:
    <p>BDM14471 is a selective inhibitor of hydroxamate PfAM1.</p>
    Fórmula:C17H15FN2O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:314.31
  • ICI 211965

    CAS:
    <p>ICI 211965 is a selective and orally potent of 5-Lipoxygenase (5-LPO).</p>
    Fórmula:C24H23NO2S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:389.51
  • SQ28603

    CAS:
    <p>SQ28603 is a potent and selective neutral endopeptidase 3.4.24.11 (NEP) inhibitor.</p>
    Fórmula:C13H17NO3S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:267.34
  • CM39

    CAS:
    <p>CM39 inhibits ALDH, linked to cancer stem-like cells &amp; chemoresistance.</p>
    Fórmula:C19H15FN4OS
    Forma y color:Solid
    Peso molecular:366.41
  • Oxythiamine diphosphate

    CAS:
    <p>Oxythiamine diphosphate is a competitivethiamine pyrophosphate inhibitor(Ki of 30 nM).</p>
    Fórmula:C12H17N3O8P2S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:425.29
  • DTP348

    CAS:
    <p>DTP348: Oral carbonic anhydrase IX inhibitor &amp; hypoxic cell radiosensitizer with sulfamide &amp; 5-nitroimidazole components.</p>
    Fórmula:C6H11N5O4S
    Forma y color:Solid
    Peso molecular:249.25
  • PDE2/PDE10-IN-1

    CAS:
    <p>PDE2/PDE10-IN-1 is a inhibitor of phosphodiesterase 2 (PDE2) and PDE10(IC50s of 29 and 480 nM, respectively).</p>
    Fórmula:C15H10ClN5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:295.73
  • Nitrefazole

    CAS:
    <p>Nitrefazole: a 4-nitroimidazole, inhibits ALDH enzyme crucial for alcohol metabolism, has potent, durable effects.</p>
    Fórmula:C10H8N4O4
    Forma y color:Solid
    Peso molecular:248.19
  • Tenuazonic acid

    CAS:
    <p>Tenuazonic acid, a nonhost-selective mycotoxin from Alternaria alternate, inhibits PSII by blocking electron transport at D1 protein.</p>
    Fórmula:C10H15NO3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:197.23
  • P-3FAX-Neu5Ac

    CAS:
    <p>P-3FAX-Neu5Ac is a sialic acid analog and a sialyltransferase inhibitor.</p>
    Fórmula:C22H30FNO14
    Pureza:97.08%
    Forma y color:Solid
    Peso molecular:551.47
  • Pirbuterol hydrochloride

    CAS:
    <p>Pirbuterol hydrochloride is a bronchodilator.</p>
    Fórmula:C12H21ClN2O3
    Forma y color:Solid
    Peso molecular:276.76
  • Manninotrionate

    CAS:
    <p>Manninotrionate, an antitumor agent, linked to BSA; rabbit antiserum made, doesn't agglutinate Ehrlich tumor cells with alpha-D-galactosyl groups.</p>
    Fórmula:C18H32KO17
    Pureza:98%
    Forma y color:Solid
    Peso molecular:559.535
  • CYP3A4-IN-3

    CAS:
    <p>CYP3A4-IN-3, a ritonavir analogue, is a potent CYP3A4 inhibitor with an IC50 of 0.075 μM, used as an antiviral and immunosuppressant.</p>
    Fórmula:C34H39N3O3S
    Forma y color:Solid
    Peso molecular:569.76
  • Rev 6207

    CAS:
    <p>Rev 6207 is a non-sulfhydryl ACE-inhibitor.</p>
    Fórmula:C21H31N3O5
    Forma y color:Solid
    Peso molecular:405.49
  • Cholesteryl behenate

    CAS:
    <p>Cholesteryl behenate is a standard in electrospray ionization tandem mass spectrometry for the analysis of cholesteryl esters and cholesterol.</p>
    Fórmula:C49H88O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:709.22
  • (R)-Lercanidipine hydrochloride

    CAS:
    <p>(R)-Lercanidipine hydrochloride is the R-enantiomer of Lercanidipine. (R)-lercanidipine hydrochloride is a blocker of calcium channel.</p>
    Fórmula:C36H42ClN3O6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:648.2
  • CAY10486

    CAS:
    <p>CAY10486 blocks ACAT-1/2, which form cholesterol esters, potentially reducing atherosclerosis; inhibits LDL oxidation. IC50 ~60μM; 28% effect at 3μM.</p>
    Fórmula:C19H19NO4
    Forma y color:Solid
    Peso molecular:325.36
  • Valibose

    CAS:
    <p>Valibose, α-glucosidase inhibitor, improves glucose/lipid metabolism, lowers serum BUN/NAG, reduces kidney weight index.</p>
    Fórmula:C10H21NO6
    Forma y color:Solid
    Peso molecular:251.28
  • (R)-Irsenontrine

    CAS:
    <p>(R)-Irsenontrine (R-E2027), R-enantiomer, is a potent PDE9 inhibitor, IC50 = 0.041 μM, for neurological disease research.</p>
    Fórmula:C22H22N4O3
    Forma y color:Solid
    Peso molecular:390.44
  • PPARα-MO-1

    CAS:
    <p>PPARα-MO-1 is a potent modulator of PPARα.</p>
    Fórmula:C27H37NO5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:455.59
  • IDO1-IN-18

    CAS:
    <p>IDO1-IN-18 (Compound 14) is a potent inhibitor of IDO1. IDO1-IN-18 has potential for cancer disease research.</p>
    Fórmula:C23H18F4N2O3
    Forma y color:Solid
    Peso molecular:446.39
  • PSN-GK1

    CAS:
    <p>PSN-GK1 is a potent activator of glucokinase (EC50: 0.13 μM).</p>
    Fórmula:C20H23FN2O4S2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:438.54
  • sEH inhibitor-6

    CAS:
    <p>sEH inhibitor-6 (Compound 3g) is a highly potent soluble epoxide hydrolase (sEH) inhibitor, exhibiting an IC 50 value of 0.5 nM [1].</p>
    Fórmula:C21H14ClN3O2
    Forma y color:Solid
    Peso molecular:375.81
  • LH65.3

    CAS:
    <p>LH65.3 is an inhibitor of S. typhimurium infection on the activity of DUSP3, DUSP11, and DUSP27.</p>
    Fórmula:C21H20N2O5S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:412.46
  • hCAXII-IN-2

    CAS:
    <p>hCAXII-IN-2 is a potent inhibitor of hCA XII (Ki: 84.2 nM) and hCA IX (Ki: 268.5 nM), with low activity on hCA I/II.</p>
    Fórmula:C21H18ClN3O4
    Forma y color:Solid
    Peso molecular:411.84