Metabolismo
Los inhibidores del metabolismo son compuestos que interfieren con las vías metabólicas, alterando la producción y utilización de energía dentro de las células. Estos inhibidores se utilizan para estudiar la regulación del metabolismo, el papel de las vías metabólicas en enfermedades como el cáncer y la diabetes, y para desarrollar nuevas estrategias terapéuticas. Los inhibidores del metabolismo pueden dirigirse a diversas enzimas y procesos involucrados en la glucólisis, la oxidación de ácidos grasos y otras funciones metabólicas. En CymitQuimica, ofrecemos una amplia gama de inhibidores del metabolismo de alta calidad para apoyar su investigación en bioquímica, trastornos metabólicos y desarrollo de fármacos.
Subcategorías de "Metabolismo"
- AhR(41 productos)
- Aminopeptidasa(67 productos)
- CETP(18 productos)
- Anhídrido carbónico(178 productos)
- Caseína quinasa(130 productos)
- DHFR(33 productos)
- Descarboxilasa(4 productos)
- Deshidrogenasa(270 productos)
- FAAH(64 productos)
- FXR(58 productos)
- Factor Xa(80 productos)
- Ácido graso sintasa(33 productos)
- Ferroptosis(215 productos)
- GR(3 productos)
- GSNOR(3 productos)
- Glucoquinasa(54 productos)
- HIF / HIF Prolilhidroxilasa(142 productos)
- HMG-CoA reductasa(33 productos)
- Hidroxilasa(30 productos)
- IDO(82 productos)
- LDL(8 productos)
- Lipasa(97 productos)
- Lípido(59 productos)
- Lipoxigenasa(125 productos)
- MAO(87 productos)
- MPO(2 productos)
- NAMPT(36 productos)
- P450(6 productos)
- PAI-1(25 productos)
- PDE(166 productos)
- PED(1 productos)
- PKM(15 productos)
- PPAR(164 productos)
- Fosfolipasa(82 productos)
- ROR(42 productos)
- Receptor de retinoides(29 productos)
- SGK(11 productos)
- Tiorredoxina(12 productos)
- Transferasa(30 productos)
- Transportador(42 productos)
- UGT(4 productos)
- Inhibidores de la xantina oxidasa (XO)(9 productos)
Mostrar 34 subcategorías más
Se han encontrado 8625 productos de "Metabolismo"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
4-Desmethyl Istradefylline
CAS:<p>4-Desmethyl Istradefylline: a metabolite of Istradefylline, a strong, selective oral adenosine A2A receptor blocker, Ki 2.2 nM, used in Parkinson's.</p>Fórmula:C19H22N4O4Pureza:98%Forma y color:SolidPeso molecular:370.40Quinalizarin
CAS:<p>Quinalizarin, the most selective CK2 inhibitor, is superior to CX-4945 which is the first-in-class CK2 inhibitor.</p>Fórmula:C14H8O6Pureza:98%Forma y color:SolidPeso molecular:272.21SHP836
CAS:<p>SHP836 is an inhibitor of SHP2 allosteric (IC50: 12 μM for the full-length SHP2).</p>Fórmula:C16H19Cl2N5Pureza:98%Forma y color:SolidPeso molecular:352.26Mesopram
CAS:<p>PDE4 inhibitor, orally active</p>Fórmula:C14H19NO4Pureza:98%Forma y color:SolidPeso molecular:265.3β-Amino Acid Imagabalin Hydrochloride
CAS:<p>β-Amino Acid Imagabalin Hydrochloride is the voltage-dependent calcium channel ligand for the α2δ subunit.</p>Fórmula:C9H20ClNO2Pureza:98%Forma y color:SolidPeso molecular:209.71IHVR-11029
CAS:<p>IHVR-11029 inhibits ER α-glucosidase, combats hemorrhagic fever viruses, and hinders enveloped virus morphogenesis.</p>Fórmula:C18H27F2NO5Forma y color:SolidPeso molecular:375.41Ro 41-0960
CAS:<p>Ro 41-0960 is used as a reversible and orally-active COMT-inhibitor.</p>Fórmula:C13H8FNO5Pureza:98%Forma y color:SolidPeso molecular:277.2Adenosine 5'-phosphosulfate (sodium salt)
CAS:<p>Adenosine 5'-phosphosulfate (sodium salt) (APS) is a key intermediate in sulphur metabolism and a substrate for adenosine 5'-phosphosulfate kinase (APSK).</p>Fórmula:C10H12N5Na2O10PSForma y color:SolidPeso molecular:471.24PDE2/PDE10-IN-1
CAS:<p>PDE2/PDE10-IN-1 is a inhibitor of phosphodiesterase 2 (PDE2) and PDE10(IC50s of 29 and 480 nM, respectively).</p>Fórmula:C15H10ClN5Pureza:98%Forma y color:SolidPeso molecular:295.73Rosuvastatin lactone
CAS:<p>Tilavonemab (ABBV-8E12) is a monoclonal antibody that binds to the N-terminus of the human microtubule-associated protein tau.</p>Fórmula:C22H26FN3O5SForma y color:SolidPeso molecular:463.52L 669262
CAS:<p>L 669262 is a potent inhibitor of HMG-CoA reductase.</p>Fórmula:C25H36O6Forma y color:SolidPeso molecular:432.55ALRT 1550
CAS:<p>ALRT 1550, a retinoic acid agent (RAR) agonist, is used potentially for the treatment of cervical carcinoma.</p>Fórmula:C23H32O2Forma y color:SolidPeso molecular:340.5DSHN
CAS:<p>DSHN activates SHP, boosting its mRNA and protecting it from ubiquitination and degradation.</p>Fórmula:C15H17NO5SPureza:98%Forma y color:SolidPeso molecular:323.36Abiraterone metabolite 1
CAS:<p>Abiraterone metabolite 1, a derivative of abiraterone, inhibits CYP17A1, halts androgen formation, aiding in prostate cancer treatment.</p>Fórmula:C24H33NOPureza:98%Forma y color:SolidPeso molecular:351.52EP6
CAS:<p>EP6 blocks 5-LO, key in the AA cascade, reducing leukotrienes to curb inflammation and allergies.</p>Fórmula:C24H30N4OPureza:98%Forma y color:SolidPeso molecular:390.52BML-111
CAS:<p>inhibits leukotriene B4 (LTB4)-induced polymorphonuclear neutrophils (PMN) chemotaxis</p>Fórmula:C8H16O5Forma y color:SolidPeso molecular:192.21RG 6866
CAS:RG 6866 is a inhibitor of 5-lipoxygenase.Fórmula:C16H17NO3Pureza:98%Forma y color:SolidPeso molecular:271.31Prinoxodan
CAS:<p>Prinoxodan is an inhibitor of phosphodiesterase.</p>Fórmula:C13H14N4O2Pureza:98%Forma y color:SolidPeso molecular:258.28SCH 42495 racemate
CAS:<p>SCH 42495 racemate is the racemate of SCH 42495. SCH 42495 is an orally active neutral inhibitor of metalloendopeptidase (NEP), with antihypertensive effect.</p>Fórmula:C20H29NO4S2Pureza:98%Forma y color:SolidPeso molecular:411.58Theodrenaline
CAS:<p>Theodrenaline is a cardiac stimulant, also acts as an agent of anti-hypotensive together with cafedrine.</p>Fórmula:C17H21N5O5Pureza:98%Forma y color:SolidPeso molecular:375.38(1S,2S,3R)-DT-061
CAS:<p>(1S,2S,3R)-DT-061 is an enantiomer of DT-061 which is an orally bioavailable activator of PP2A.</p>Fórmula:C25H23F3N2O5SForma y color:SolidPeso molecular:520.52SWE101
CAS:<p>SWE101 is a potent human and rat soluble epoxide hydrolase (sEH)-P inhibitor(IC50s of 4 μM and 2.8 μM, respectively).</p>Fórmula:C19H15Cl2NO3Pureza:98%Forma y color:SolidPeso molecular:376.23N-Methylmoranoline
CAS:<p>N-Methylmoranoline is an inhibitor of α-glucosidase.</p>Fórmula:C7H15NO4Pureza:98%Forma y color:SolidPeso molecular:177.2Antitumor agent-87
CAS:<p>Antitumor agent-87: potent, high CYP1A1 affinity (Ki 0.23µM), antiproliferative, arrests G2/M cell cycle.</p>Fórmula:C22H28N2O6SPureza:99.48%Forma y color:SolidPeso molecular:448.53Glyoxalase I inhibitor 1
CAS:<p>Glyoxalase I inhibitor 1 is a potent inhibitor of glyoxalase I (GLO1) (IC50: 26 nM).</p>Fórmula:C30H27FN6O4SForma y color:SolidPeso molecular:586.64(+)-Cembrene A
CAS:<p>(+)-Cembrene A, a nontoxic α-glucosidase inhibitor to human normal hepatocyte (LO2) cells, exhibits an IC50 value of 30.31 μM.</p>Fórmula:C20H32Forma y color:SolidPeso molecular:272.47IDO/TDO-IN-1
CAS:<p>IDO/TDO-IN-1 is an orally active dual indoleamine-2,3-dioxygenase (IDO) and tryptophan 2,3-dioxygenase (TDO) inhibitor (IC50s: 9.7 and 47 nM).</p>Fórmula:C25H24FN5Pureza:98%Forma y color:SolidPeso molecular:413.49SCD1 inhibitor-1
CAS:SCD1 inhibitor-1 is a potent and liver-selective inhibitor of stearoyl-CoA desaturase-1 (SCD1).Fórmula:C21H23N3NaO3S2Pureza:98%Forma y color:SolidPeso molecular:452.54CR4056
CAS:<p>CR4056 (6-(1H-imidazol-1-yl)-2-phenylquinazoline) is a selective inhibitor of MAO-A with IC50 of 202.7 nM and a ligand of I2-imidazoline receptor with IC50 of</p>Fórmula:C17H12N4Pureza:98.73%Forma y color:SolidPeso molecular:272.3BMS 961
CAS:<p>BMS961 is a potent and selective retinoic acid receptor gamma (RARγ) agonist (IC50: 30 nM).</p>Fórmula:C23H26FNO4Pureza:98%Forma y color:SolidPeso molecular:399.46Senazodan
CAS:<p>Senazodan is a sensitiser of Ca2+, and shows inhibition effect on PDE III.</p>Fórmula:C15H14N4OPureza:98%Forma y color:SolidPeso molecular:266.3CFG920
CAS:<p>CFG920 is an oral CYP17 inhibitor that may reduce androgen production and inhibit growth of androgen-dependent tumors.</p>Fórmula:C14H13ClN4OForma y color:SolidPeso molecular:288.73L-5-BromoTryptophan
CAS:<p>L-5-BromoTryptophan (5-BrW) is an analog of the tryptophan (Trp) effector and inhibits the gelation of hemoglobin S.</p>Fórmula:C11H11BrN2O2Pureza:99.86%Forma y color:SolidPeso molecular:283.12Razaxaban hydrochloride
CAS:<p>Razaxaban hydrochloride is a highly potent, selective and orally active inhibitor of factor Xa(Ki of 0.19 nM),has strongly antithrombotic activity.</p>Fórmula:C24H21ClF4N8O2Pureza:98%Forma y color:SolidPeso molecular:564.92Entacapone sodium salt
CAS:<p>Entacapone sodium salt, a potent peripheral COMT inhibitor (IC50=151 nM), hinders α-syn/β-amyloid aggregation and protects PC12 cells.</p>Fórmula:C14H15N3NaO5Pureza:98%Forma y color:SolidPeso molecular:328.28Allylglycine
CAS:<p>Allylglycine is a glutamate decarboxylase inhibitor and a GAMMA-AMINOBUTYRIC ACID antagonist. It is used to induce convulsions in experimental animals.</p>Fórmula:C5H9NO2Pureza:98%Forma y color:SolidPeso molecular:115.13p-Synephrine
CAS:<p>p-Synephrine is a natural product for research related to life sciences. The catalog number is T8265 and the CAS number is 614-35-7.</p>Fórmula:C9H13NO2Pureza:98%Forma y color:SolidPeso molecular:167.21Pulixin
CAS:<p>Pulixin blocks FREP1 from P. falciparum, hinders parasite spread (EC50: 11µM), and stops its growth (EC50: 47nM).</p>Fórmula:C14H11NO4Forma y color:SolidPeso molecular:257.24Incadronate Disodium
CAS:<p>Incadronate Disodium: halts bone loss, limits macrophage migration and inflammation, and induces cancer cell apoptosis in vitro.</p>Fórmula:C8H19NNaO6P2Pureza:98%Forma y color:SolidPeso molecular:310.178S 12340
CAS:<p>S 12340 is a potent inhibitor of the oxidative modification of low-density lipoprotein.</p>Fórmula:C24H38N2O3SForma y color:SolidPeso molecular:434.64MSPG
CAS:<p>mGlu receptor antagonist</p>Fórmula:C9H11NO5SPureza:98%Forma y color:SolidPeso molecular:245.25GSK2945
CAS:<p>GSK2945, a specific Rev-erbα antagonist, boosts CYP7A1 and cholesterol metabolism. EC50: 21.5 μM (mouse), 20.8 μM (human).</p>Fórmula:C20H18Cl2N2O2SPureza:98%Forma y color:SolidPeso molecular:421.34hACC2-IN-1
CAS:<p>hACC2-IN-1 is a potent inhibitor of acetyl coenzyme A carboxylase 2 (ACC2) with an IC50 value of 2.5 μM for hACC2. hACC2-IN-1 has potential for obesity studies.</p>Fórmula:C23H32N2O4SForma y color:SolidPeso molecular:432.58Succinyladenosine
CAS:<p>Succinyladenosine, a marker for ASL deficiency, is made by dephosphorylating S-AMP with 5-nucleotidase.</p>Fórmula:C14H17N5O8Forma y color:SolidPeso molecular:383.317S32826 disodium
CAS:<p>autotaxin inhibitor</p>Fórmula:C21H36NNa2O4PPureza:98%Forma y color:SolidPeso molecular:443.47SCH-351591
CAS:<p>SCH-351591 is an orally active inhibitor of phosphodiesterase 4.</p>Fórmula:C17H10Cl2F3N3O3Pureza:98%Forma y color:SolidPeso molecular:432.18Nebicapone
CAS:<p>Nebicapone, a reversible COMT inhibitor, reduces L-DOPA breakdown, aiding Parkinson's treatment.</p>Fórmula:C14H11NO5Pureza:98%Forma y color:SolidPeso molecular:273.24CAY10487
CAS:<p>CAY10487 reduces aortic fatty streaks in high-cholesterol rabbits by 37.4% and inhibits LDL oxidation by 75% at 2μM, without altering lipids or ACAT activity.</p>Fórmula:C13H15NO5Forma y color:SolidPeso molecular:265.26PGAM1-IN-2
CAS:<p>PGAM1-IN-2 is an inhibitor of phosphoglycerate mutase 1 ( PGAM1 ) with an IC 50 of 2.1 μM [1].</p>Fórmula:C25H16N2O7SPureza:98%Forma y color:SolidPeso molecular:488.47OMDM-2
CAS:<p>OMDM-2 is a metabolically stable and selective inhibitor of anandamide cellular uptake (ACU), exhibiting a Ki value of 3.0 μM in RBL-2H3 cells.</p>Fórmula:C27H45NO3Pureza:98%Forma y color:SolidPeso molecular:431.65Enpp-1-IN-13
CAS:<p>Enpp-1-IN-13 inhibits ENPP1 (IC50: 1.29 μM) & ENPP3 (IC50: 20.2 μM) with anticancer properties.</p>Fórmula:C28H22ClN5OSForma y color:SolidPeso molecular:512.03Spiraprilat
CAS:<p>Spiraprilat is an ACE inhibitor. It also is an active metabolite of spirapril.</p>Fórmula:C20H26N2O5S2Pureza:98%Forma y color:SolidPeso molecular:438.56sPLA2-X Inhibitor 31
CAS:<p>sPLA2-X Inhibitor 31 targets sPLA2-X with IC50: 26 nM; less effective on sPLA2-IIa (310 nM), sPLA2-V (2230 nM).</p>Fórmula:C19H15F3N2O4Pureza:98%Forma y color:SolidPeso molecular:392.33AGN 191701
CAS:<p>AGN 191701 is an agonist of the Retinoid X receptor.</p>Fórmula:C23H28O2SPureza:98%Forma y color:SolidPeso molecular:368.532'-O-Methyladenosine
CAS:<p>2'-O-Methyladenosine, a methylated adenine residue is found in the urine of normals and adenosine deaminase deficient patients.</p>Fórmula:C11H15N5O4Pureza:99.89%Forma y color:White SolidPeso molecular:281.2793-O17O
CAS:<p>93-O17O is a cationic lipidoid used in lipid nanoparticles for spleen-targeted delivery and genome editing in mice.</p>Fórmula:C44H83N3O6Forma y color:SolidPeso molecular:750.15Isospaglumate sodium
CAS:<p>Isospaglumate sodium is the sodium salt of isospaglumate which is an antiallergic agent.</p>Fórmula:C11H16N2NaO8Forma y color:SolidPeso molecular:327.245JNJ-42314415
CAS:<p>JNJ-42314415 is a potent, specific, and centrally active inhibitor of PDE10A.</p>Fórmula:C19H23N5O2Pureza:98%Forma y color:SolidPeso molecular:353.42ARN19874
CAS:<p>ARN19874 is a selective, reversible uncompetitive N-acylphosphatidylethanolamine phospholipase D (NAPE-PLD) activity inhibitor. With an IC50 of ~34 μM[1].</p>Fórmula:C19H14N4O4SPureza:98%Forma y color:SolidPeso molecular:394.4OL-135
CAS:<p>OL-135: CNS-accessible, potent, selective FAAH inhibitor with analgesic effects in animals, no motor impairment.</p>Fórmula:C21H22N2O2Forma y color:SolidPeso molecular:334.41POP-IN-2
CAS:<p>Compound 7k (POP-IN-2) is a potent POP inhibitor with Ki of 6 nM, useful in neurodegenerative and cancer studies.</p>Fórmula:C24H33BN2O5Forma y color:SolidPeso molecular:440.34IDO1/TDO-IN-3
CAS:<p>IDO1/TDO-IN-3 inhibits IDO1 (IC50: 0.005 μM) and TDO (IC50: 0.004 μM) with strong anti-tumor activity and low toxicity.</p>Fórmula:C16H6ClF2N3O2Forma y color:SolidPeso molecular:345.69M8891
CAS:<p>M8891: Oral, reversible MetAP-2 inhibitor, brain-penetrant (IC50: 54nM; Ki: 4.33nM), hinders endothelial & tumor cell growth, antiangiogenic & antitumor.</p>Fórmula:C20H17F2N3O3Forma y color:SolidPeso molecular:385.36GW844520
CAS:<p>GW844520 is a potent and selective inhibitor of the cytochrome bc1 complex of mitochondrial electron transport in P. falciparum.</p>Fórmula:C20H15ClF3NO3Forma y color:SolidPeso molecular:409.79PF-06471553
CAS:<p>PF-06471553 is an effective and selective inhibitor of monoacylglycerol acyltransferase 3 (IC50: 92 nM).</p>Fórmula:C23H25N5O4SPureza:98%Forma y color:SolidPeso molecular:467.54Oosponol
CAS:<p>Oosponol is a dopamine beta-hydroxylase inhibitor exhibiting hypotensive effects.</p>Fórmula:C11H8O5Pureza:98%Forma y color:SolidPeso molecular:220.18α-Glucosidase-IN-3
CAS:<p>α-Glucosidase-IN-3 is an oleanolic acid oxime ester derivative targeting α-glucosidase and α-amylase with an IC50 value of 0.35 μM for α-glucosidase.</p>Fórmula:C39H53NO4Forma y color:SolidPeso molecular:599.84T-1095A
CAS:<p>T-1095A, a T-1095 metabolite, inhibits SGLTs, lowers blood glucose, improves glucose intolerance in mice, and prevents neuropathy in diabetic rats.</p>Fórmula:C24H26O9Pureza:98%Forma y color:SolidPeso molecular:458.46Crilvastatin
CAS:<p>Crilvastatin (PMD 387) is an HMGCR inhibitor with cholesterol-lowering activity that inhibits cholesterol uptake in rats with hereditary hypercholesterolemia.</p>Fórmula:C14H23NO3Pureza:98.69% - 99.54%Forma y color:SolidPeso molecular:253.34Tanogitran
CAS:<p>Tanogitran, a coagulation factor Xa inhibitor, is used potentially for the treatment of septic shock.</p>Fórmula:C25H31N7O3Pureza:98%Forma y color:SolidPeso molecular:477.56KT109
CAS:<p>KT109 is a DAGLβ inhibitor (IC50=42nM), lessens LPS allodynia in mice without tolerance, and has no major side effects.</p>Fórmula:C27H26N4OPureza:98%Forma y color:SolidPeso molecular:422.521E7-03
CAS:<p>1E7-03 is an inhibitor of HIV-1 transcription, by targeting host Protein Phosphatase-1 (PP1).</p>Fórmula:C28H29N3O6Forma y color:SolidPeso molecular:503.55ML299
CAS:<p>ML299 (VU0463568) is a dual PLD1/2 inhibitor (PLD1 and PLD2, IC50 of 6 nM, 20 nM, respectively).</p>Fórmula:C23H26BrFN4O2Pureza:98%Forma y color:SolidPeso molecular:489.38Aldophosphamide
CAS:<p>Aldophosphamide possesses apoptotic antitumor activity.</p>Fórmula:C7H15Cl2N2O3PPureza:98%Forma y color:SolidPeso molecular:277.09NPD-001
CAS:<p>NPD-001 is an effective inhibitor of TbrPDEB1. NPD-001 is 10-fold more potent on hPDE4 (hPDE4B1 IC50 = 0.6 nM) than on TbrPDEB1 (IC50 = 4 nM).</p>Fórmula:C33H40N6O4Pureza:98%Forma y color:SolidPeso molecular:584.71AK-106
CAS:<p>AK-106, or AK106-001616, selectively inhibits cPLA2 and has NSAID-like analgesic effects.</p>Fórmula:C26H25N3O3Forma y color:SolidPeso molecular:427.49Abiraterone decanoate
CAS:<p>Abiraterone decanoate is a prodrug of Abiraterone that provides controlled release and prolonged inhibition of the enzyme CYP17 through intramuscular.</p>Fórmula:C34H49NO2Pureza:99.69%Forma y color:SolidPeso molecular:503.76PGAM1-IN-1
CAS:<p>PGAM1-IN-1 is an inhibitor of phosphoglycerate mutase 1 ( PGAM1 ) with an IC 50 of 6.4 μM [1].</p>Fórmula:C19H11ClFNO6SPureza:98%Forma y color:SolidPeso molecular:435.81Dacisteine
CAS:<p>Dacisteine (N,S-Diacetyl-L-cysteine) is an inhibitor of New Delhi metallo-beta-lactamase-1 (NDM-1, IC50 = 1000 μM).</p>Fórmula:C7H11NO4SPureza:99.57%Forma y color:SolidPeso molecular:205.23Win-62005
CAS:<p>Win-62005 is an inhibitor of cyclic AMP phosphodiesterase III (PDE III)(Kis: 25 and 26 nM for rat heart and canine aorta).</p>Fórmula:C12H10N4OPureza:98%Forma y color:SolidPeso molecular:226.23BN-82685
CAS:<p>BN-82685, a quinone-based CDC25 inhibitor, shows in vitro and in vivo efficacy, suggesting potential as an anticancer therapy.</p>Fórmula:C12H15N3O2SPureza:98%Forma y color:SolidPeso molecular:265.33L 656224
CAS:<p>L 656224 is a 5-LO inhibitor.</p>Fórmula:C20H21ClO3Pureza:98%Forma y color:SolidPeso molecular:344.83Fenleuton
CAS:<p>Fenleuton is a 5-lipoxygenase inhibitor.</p>Fórmula:C17H15FN2O3Pureza:98%Forma y color:SolidPeso molecular:314.31Glucosylceramide synthase-IN-2
CAS:<p>T-690: Potent, BBB-permeable, oral GCS inhibitor; human IC50: 15 nM, mouse IC50: 190 nM; non-competitive with C8 ceramide/UDP glucose.</p>Fórmula:C22H20F3N3O4Forma y color:SolidPeso molecular:447.41HCAIX-IN-2
CAS:<p>HCAIX-IN-2 (compound 9d) is a selective inhibitor of carbonic anhydrase and acts on hCA IX (Ki: 24.6 nM) and hCA XII (Ki: 45.3 nM).</p>Fórmula:C19H16N8O4SForma y color:SolidPeso molecular:452.45Mevalonic acid
CAS:<p>Mevalonic acid is essential for cell growth and proliferation,Mevalonic acid is a precursor in the mevalonate pathway.</p>Fórmula:C6H12O4Pureza:98%Forma y color:SolidPeso molecular:148.16γ-Methylleucine
CAS:<p>Gamma-Methylleucine (2-Amino-3-tert-butylpropionic acid) is an auxiliary for copper-catalyzed asymmetric Michael reactions.</p>Fórmula:C7H15NO2Pureza:≥98%Forma y color:SolidPeso molecular:145.2ZSET-845
CAS:<p>ZSET-845 is an enhancer of cognitive which enhances choline acetyltransferase activity in the hippocampus in the rat.</p>Fórmula:C21H18N2OPureza:98%Forma y color:SolidPeso molecular:314.38Piragliatin
CAS:<p>Piragliatin (RO4389620) activates glucokinase, boosts insulin, and lowers glucose in type 2 diabetes.</p>Fórmula:C19H20ClN3O4SForma y color:SolidPeso molecular:421.9Seviteronel racemate
CAS:<p>Seviteronel racemate is the racemate form of Seviteronel and is a potent inhibitor of CYP17 lyase.</p>Fórmula:C18H17F4N3O3Pureza:98%Forma y color:SolidPeso molecular:399.34Seviteronel R enantiomer
CAS:<p>Seviteronel R enantiomer (VT-464 R enantiomer) is a Seviteronel isomer produced during the manufacturing process.</p>Fórmula:C18H17F4N3O3Pureza:97.97% - >99.99%Forma y color:SolidPeso molecular:399.34ARL-67156 trisodium salt hydrate
CAS:<p>ARL-67156 trisodium salt hydrate is an ecto-ATPase inhibitor that prevents metabolism of P2 purinoceptor agonists.</p>Fórmula:C15H24Br2N5O12P3Forma y color:SolidPeso molecular:719.11(Rac)-Etavopivat
CAS:<p>(Rac)-Etavopivat, an oral PKR activator, targets sickle cell disease and haemoglobinopathies.</p>Fórmula:C22H23N3O6SForma y color:SolidPeso molecular:457.5Mufemilast
CAS:<p>Mufemilast is an inhibitor of phosphodiesterase 4 (PDE4).</p>Fórmula:C20H22N2O7S2Forma y color:SolidPeso molecular:466.53GS 389
CAS:<p>GS 389, a tetrahydroisoquinoline, relaxes blood vessels by inhibiting brain PDE and raising aorta cGMP.</p>Fórmula:C19H23NO3Pureza:98%Forma y color:SolidPeso molecular:313.39SAR629
CAS:<p>SAR-629 is an MGL inhibitor or 2-AG degradation inhibitor.</p>Fórmula:C20H19F2N5OForma y color:SolidPeso molecular:383.39hCAIX-IN-11
CAS:<p>hCAIX-IN-11 inhibits carbonic anhydrases IX & XII with Ki of 32.7 nM & 623.5 nM, respectively.</p>Fórmula:C21H15ClN4O3Forma y color:SolidPeso molecular:406.82ONO-1603
CAS:<p>ONO-1603, a prolyl endopeptidase inhibitor, is used potentially for the treatment of Alzheimer's disease.</p>Fórmula:C16H19ClN2O3Pureza:98%Forma y color:SolidPeso molecular:322.79CD 2314
CAS:<p>CD2314 is a potent and subtype-selective RARβ receptor agonist with a Kd of 195 nM in S91 melanoma cells [1].</p>Fórmula:C23H24O2SForma y color:SolidPeso molecular:364.5Fodipir
CAS:<p>Fodipir, the active metabolite of mangafodipir, plays a crucial role in the mechanism of mangafodipir-mediated cytoprotection, specifically mitigating cell</p>Fórmula:C22H32N4O14P2Pureza:98%Forma y color:SolidPeso molecular:638.46Carbazomycin B
CAS:<p>Carbazomycin B, a Streptomyces metabolite, combats fungi, bacteria, P. falciparum, C. albicans, and some cancer cells; inhibits 5-LO (IC50=1.5µM).</p>Fórmula:C15H15NO2Forma y color:SolidPeso molecular:241.29Enpp-1-IN-6
CAS:<p>Enpp-1-IN-6, a potent enpp-1 inhibitor, may aid cancer and infectious disease studies (WO2021203772A1, compound 51).</p>Fórmula:C22H28N4O5SForma y color:SolidPeso molecular:460.55TFB-TBOA
CAS:<p>glial glutamate transporter EAAT1 and EAAT2 inhibitor</p>Fórmula:C19H17F3N2O6Pureza:98%Forma y color:SolidPeso molecular:426.34hCAI/II-IN-1
CAS:<p>hCAI/II-IN-1 (Compound 3h) is a human carbonic anhydrase I and II (hCA I/II) inhibitor that acts on hCA I (IC50: 0.047 μM) and hCA II (IC50: 0.024 μM).</p>Fórmula:C18H29N5O3S3Forma y color:SolidPeso molecular:459.65IDH-C227
CAS:<p>IDH-C227 is a selective and potent inhibitor of IDH1R132H that exhibits anticancer activity.</p>Fórmula:C30H31FN4O2Forma y color:SolidPeso molecular:498.59UK-500001
CAS:<p>UK-500001 is a potent PDE4 inhibitor with robust anti-inflammatory activity.</p>Fórmula:C26H24F3N3O4Pureza:98%Forma y color:SolidPeso molecular:499.48LY367385
CAS:<p>LY367385 is a highly effective and selective mGluR1a antagonist.</p>Fórmula:C10H11NO4Pureza:98%Forma y color:SolidPeso molecular:209.2Semotiadil recemate fumarate
CAS:<p>Semotiadil recemate fumarate is the recemate of Semotiadil fumarate. Semotiadil fumarate is a novel antagonist of vasoselective Ca2+ channel.</p>Fórmula:C33H36N2O10SPureza:98%Forma y color:SolidPeso molecular:652.71SHP2 inhibitor LY6
CAS:<p>SHP2 inhibitor LY6 (LY6) is a potent and selective SHP2 inhibitor (IC50: 9.8 μM) that blocks SHP2-mediated cell signaling and proliferation.</p>Fórmula:C30H27Cl2N3O4Forma y color:SolidPeso molecular:564.46PKM2 activator 3
CAS:<p>PKM2 activator 3, with 90 nM AC50, enhances PKM2. It has good Caco-2 permeability, stable, and aids cancer research.</p>Fórmula:C15H11ClF2N2O3SForma y color:SolidPeso molecular:372.77LB42908
CAS:<p>LB42908 is a highly potent Ras farnesyltransferase inhibitor(IC(50)=0.9 nM against H-Ras and 2.4 nM against K-Ras) with potential anticancer activity.</p>Fórmula:C32H31N5O3Forma y color:SolidPeso molecular:533.62N-Oleoyl Leucine
CAS:<p>N-Oleoyl Leucine (Oleoyl-L-leucine) is an N-fatty acyl amino acid present in plasma.</p>Fórmula:C24H45NO3Pureza:98.25%Forma y color:SolidPeso molecular:395.62MEDS433
CAS:<p>MEDS433 inhibits dihydroorotate dehydrogenase (IC50 1.2 nM) and blocks replication of hCoV-OC43, hCoV-229E, SARS-CoV-2 at nanomolar levels.</p>Fórmula:C20H11F4N3O2Forma y color:SolidPeso molecular:401.31Loxoprofenol-SRS
CAS:<p>Loxoprofenol-SRS, a potent metabolite of Loxoprofen, is an IV NSAID with enhanced anti-inflammatory and pain relief properties.</p>Fórmula:C15H20O3Forma y color:SolidPeso molecular:248.32DNJNAc
CAS:<p>DNJNAc (2-Acetamido-1,2-dideoxynojirimycin) is a potent β-hexosaminidase inhibitor, reducing cartilage matrix degradation, relevant in glycoconjugate studies.</p>Fórmula:C8H16N2O4Pureza:98.65% - 99.37%Forma y color:SolidPeso molecular:204.22GlcN-6-P Synthase-IN-1
CAS:<p>'GlcN-6-P Synthase-IN-1, IC50 3.47 μM, inhibits GlcN-6-P synthase & CYP3A4. Has antimicrobial activity and CNS penetration.'</p>Fórmula:C20H21N7SForma y color:SolidPeso molecular:391.4914-dehydro Zymostenol
CAS:<p>14-dehydro Zymostenol, a cholesterol precursor, boosts MBP+ oligodendrocytes from precursors at 5.8-17 μM.</p>Fórmula:C27H44OForma y color:SolidPeso molecular:384.64hCAI/II-IN-2
CAS:<p>hCAI/II-IN-2 (2b) inhibits hCA I/II (Ki: 40.97 nM, 15.15 nM) and IX (61.88 nM), fights AMS with anti-hypoxic effects, but has low cellular activity.</p>Fórmula:C12H12N4O5S2Forma y color:SolidPeso molecular:356.38103D5R
CAS:<p>103D5R selectively inhibits hif-1α, reducing its levels in hypoxia or with cobalt ions, dose- and time-dependently.</p>Fórmula:C20H21N3O2Forma y color:SolidPeso molecular:335.4IQA
CAS:<p>IQA is a casein kinase 2 (CK2) inhibitor.</p>Fórmula:C17H12N2O3Forma y color:SolidPeso molecular:292.29SCD1 Inhibitor
CAS:<p>SCD1 Inhibitor is a novel stearoyl-CoA desaturase1 (SCD1) inhibitor.</p>Fórmula:C21H20F3N3O3Forma y color:SolidPeso molecular:419.4Kurasoin B
CAS:<p>Kurasoin B is an inhibitor of protein farnesyltransferase.</p>Fórmula:C18H17NO2Forma y color:SolidPeso molecular:279.33JBP485
CAS:<p>JBP485 is an inhibitor of renal transporters OAT1 and OAT3. JBP485 is an antihepatitis agent as a substrate for intestinal PEPT1.</p>Fórmula:C8H12N2O4Forma y color:SolidPeso molecular:200.19Anserinone B
CAS:<p>Anserinone B: Antifungal, antibacterial; inhibits S.fimicola (50%), A. furfuraceus (37%); cytotoxic to human tumor cells (GI50=4.4 µg/mL).</p>Fórmula:C11H14O4Forma y color:SolidPeso molecular:210.23EDP-305
CAS:<p>EDP-305, an oral FXR agonist, has EC50s of 34 nM/8 nM in CHO/HEK cells, aids in PBC and NASH research with antifibrotic properties.</p>Fórmula:C36H58N2O5SForma y color:SolidPeso molecular:630.92Trandolaprilate hydrate
CAS:<p>Trandolaprilate hydrate, a powerful ACE inhibitor and Trandolapril's main metabolite, is lipophilic with partial c-fos blocking.</p>Fórmula:C22H32N2O6Forma y color:SolidPeso molecular:420.5ASP3662
CAS:<p>ASP3662/SPI-62: Potent, selective CNS-penetrable 11β-HSD1 inhibitor; potential neuropathic pain treatment.</p>Fórmula:C19H16ClF3N4O2Forma y color:SolidPeso molecular:424.8TM-1
CAS:<p>TM-1: PDHK inhibitor, IC50 - PDHK1: 2.97μM, PDHK2: 5.2μM, prevents PDHC phosphorylation, inhibits cancer cell growth.</p>Fórmula:C26H32N2O6Forma y color:SolidPeso molecular:468.54CAY10486
CAS:<p>CAY10486 blocks ACAT-1/2, which form cholesterol esters, potentially reducing atherosclerosis; inhibits LDL oxidation. IC50 ~60μM; 28% effect at 3μM.</p>Fórmula:C19H19NO4Forma y color:SolidPeso molecular:325.36Valibose
CAS:<p>Valibose, α-glucosidase inhibitor, improves glucose/lipid metabolism, lowers serum BUN/NAG, reduces kidney weight index.</p>Fórmula:C10H21NO6Forma y color:SolidPeso molecular:251.28(R)-Irsenontrine
CAS:<p>(R)-Irsenontrine (R-E2027), R-enantiomer, is a potent PDE9 inhibitor, IC50 = 0.041 μM, for neurological disease research.</p>Fórmula:C22H22N4O3Forma y color:SolidPeso molecular:390.44sEH inhibitor-6
CAS:<p>sEH inhibitor-6 (Compound 3g) is a highly potent soluble epoxide hydrolase (sEH) inhibitor, exhibiting an IC 50 value of 0.5 nM [1].</p>Fórmula:C21H14ClN3O2Forma y color:SolidPeso molecular:375.81Kojibiose
CAS:<p>Kojibiose (Kojibiose) is a disaccharide in honey. Kojibiose is a product of the caramelization of glucose.</p>Fórmula:C12H22O11Pureza:99.933%Forma y color:SolidPeso molecular:342.3SAR127303
CAS:<p>SAR127303 is an effective covalent inhibitor of MAGL. SAR127303 behaves as a selective and competitive inhibitor of mouse and human MAGL.</p>Fórmula:C16H17ClF6N2O4SPureza:98%Forma y color:SolidPeso molecular:482.83(E/Z)-Ensifentrine
CAS:<p>RPL-554 (LS-193,855) is a dual PDE3/4 inhibitor with bronchodilator and anti-inflammatory properties, in trials for asthma and hay fever by Verona Pharma.</p>Fórmula:C26H31N5O4Forma y color:SolidPeso molecular:477.56Y-29794
CAS:<p>Y-29794, a covalent POP inhibitor with a Ki of 0.95 nM, holds research potential for neurodegenerative diseases and cancer.</p>Fórmula:C22H32N2OS2Forma y color:SolidPeso molecular:404.63YC-001
CAS:<p>YC-001: inverse agonist/antagonist for rod opsin, prevents light-induced retinal degeneration.</p>Fórmula:C12H7ClO2S2Forma y color:SolidPeso molecular:282.77YM 26734
CAS:<p>Competitive inhibitor of secretory phospholipase A2 (sPLA2)</p>Fórmula:C45H62O8Pureza:98%Forma y color:SolidPeso molecular:730.97Imidazoleacetic acid
CAS:<p>Imidazoleacetic acid, an endogenous ligand, stimulates imidazole receptors.</p>Fórmula:C5H6N2O2Pureza:98%Forma y color:SolidPeso molecular:126.11LAS-31180
CAS:<p>LAS-31180 is a phosphodiesterase 3 inhibitor. It also has positive inotropic and vasodilator properties.</p>Fórmula:C11H12N2O3SPureza:98%Forma y color:SolidPeso molecular:252.29DMPAC-Chol
CAS:<p>DMPAC-Chol, a cationic cholesterol, aids gene transfection, DNA protection, binds DNA, and lowers HepG2 viability at 37.5 μg/ml.</p>Fórmula:C33H58N2O2Forma y color:SolidPeso molecular:514.83hCAIX-IN-7
CAS:<p>hCAIX-IN-7 (6c) selectively inhibits tumor-related isoform hCAIX (KI: 410.6 nM) and weakly affects hCAI/II (KI: >10000 nM).</p>Fórmula:C18H12FNO3Forma y color:SolidPeso molecular:309.29ML202
CAS:<p>ML202 activates human pyruvate kinase M2, affecting PEP cooperativity with minimal impact on ADP binding.</p>Fórmula:C18H17N3O3S2Forma y color:SolidPeso molecular:387.48SQ 28853
CAS:<p>SQ 28853 is an inhibitor of ACE with diuretic properties.</p>Fórmula:C19H25ClN4NaO6S3Forma y color:SolidPeso molecular:560.05HX-600
CAS:<p>HX-600 is a synthetic agonist for the RXR-Nurr1 heterodimer complex. HX-600 prevents ischemia-induced neuronal damage.</p>Fórmula:C29H30N2O2Forma y color:SolidPeso molecular:438.56(Rac)-3′-Hydroxy simvastatin
CAS:<p>(Rac)-3′-Hydroxy Simvastatin, a metabolite of Simvastatin, acts as a competitive inhibitor of HMG-CoA reductase, demonstrating a K i value of 0.2 nM.</p>Fórmula:C25H38O6Forma y color:SolidPeso molecular:434.57BMS 740808
CAS:<p>BMS-740808 is a highly effective and selective factor X inhibitor.</p>Fórmula:C31H27F3N6O3Forma y color:SolidPeso molecular:588.58TMCB
CAS:<p>CK2 and ERK8 inhibitor</p>Fórmula:C11H9Br4N3O2Pureza:98%Forma y color:SolidPeso molecular:534.82α-Glucosidase-IN-20
CAS:<p>α-Glucosidase-IN-20 (Compound 3B) is a highly effective and orally active inhibitor of α-glucosidase.</p>Fórmula:C23H21NOSForma y color:SolidPeso molecular:359.48Chaetomellic acid A
CAS:<p>Chaetomellic acid A inhibits farnesyltransferase (IC50=55nM), not active in cells, and selective over geranylgeranyltransferases (IC50: 92µM, 34µM).</p>Fórmula:C19H34O4Forma y color:SolidPeso molecular:326.47LEO-29102
CAS:<p>LEO-29102: Potent, selective PDE4 inhibitor, promising for treating skin diseases, phase 2 efficacy in atopic dermatitis.</p>Fórmula:C20H22Cl2N2O5Forma y color:SolidPeso molecular:441.31HIF-PHD-IN-2
CAS:<p>HIF-PHD-IN-2 (compound 25) is a highly effective PHD inhibitor, displaying IC50 values below 100 nM for PHD1, PHD2, and PHD3 [1].</p>Fórmula:C17H15N5O3SForma y color:SolidPeso molecular:369.4α-Amylase-IN-2
CAS:<p>α-Glucosidase-IN-3, an oxime ester derivative of oleanolic acid (OA), exhibits inhibitory activity against α-glucosidase (IC50 = 1.28 µM) and α-amylase (IC50 =</p>Fórmula:C39H52BrNO4Forma y color:SolidPeso molecular:678.74Glucosylceramide synthase-IN-1
CAS:<p>Potent oral GCS inhibitor T-036, crosses BBB, targets human (IC50: 31 nM) and mouse GCS (IC50: 51 nM), for Gaucher disease research.</p>Fórmula:C24H20F4N2O3Forma y color:SolidPeso molecular:460.42α-Glycosidase-IN-1
CAS:<p>α-Glycosidase-IN-1 (compound MZ7) is a potent inhibitor of α-GLY (α-glycosidase) (IC50: 44.72 nM, Ki: 44.74 nM).</p>Fórmula:C21H19N9O6S2Forma y color:SolidPeso molecular:557.56Agn 190727
CAS:<p>Agn 190727 is a retonoic acid receptor that can induce retinoid-induced hypertriglyceridemia.</p>Fórmula:C20H22O2Forma y color:SolidPeso molecular:294.39HIF-1α-IN-3
CAS:<p>HIF-1α-IN-3, also known as Compound (S)-3f, is a hypoxia-selective inhibitor of HIF-1α. It exhibits potent antiestrogenic activity [1].</p>Fórmula:C19H17N5O2Forma y color:SolidPeso molecular:347.37Delapril
CAS:<p>Delapril is an ACE inhibitor. It blocks the conversion of angiotensin I to angiotensin II.</p>Fórmula:C26H32N2O5Pureza:98%Forma y color:SolidPeso molecular:452.54MDK-4823
CAS:<p>MDK-4823 (LMPTP inhibitor1) blocks LMPTP, fighting insulin resistance and diabetes in obesity.</p>Fórmula:C28H36N4OForma y color:SolidPeso molecular:444.61Enpp-1-IN-8
CAS:<p>Enpp-1-IN-8: potent inhibitor of enpp-1, an enzyme breaking down various nucleotide bonds; potential in cancer/infectious disease research.</p>Fórmula:C19H26N6O4SForma y color:SolidPeso molecular:434.51FAAH-IN-7
<p>FAAH-IN-7: Reversible FAAH inhibitor, IC50=8.29 nM, reduces oxidative stress, neuroprotective in neuroinflammation.</p>Fórmula:C26H29N3O4Forma y color:SolidPeso molecular:447.53SYN20028567
CAS:<p>SYN20028567, an aromatase (CYP19) inhibitor, exhibits an IC50 value of 9.4 nM. It has potential applications in breast cancer research [1].</p>Fórmula:C20H29N3O3SForma y color:SolidPeso molecular:391.53mEH-IN-1
CAS:<p>mEH-IN-1 (Compound 62) is a potent mEH enzyme inhibitor with an IC50 of 2.2 nM, relevant in preeclampsia, hypercholanemia, and cancer research.</p>Fórmula:C16H17F6NOSForma y color:SolidPeso molecular:385.37hCAIX-IN-3
CAS:<p>hCAII-IN-3 (7e) selectively inhibits CA II/IX with Kis of 124.2/30.5 nM, showing promise for cancer treatment.</p>Fórmula:C21H21BrN6O4SForma y color:SolidPeso molecular:533.4Fmoc-5-aminopentanoic acid
CAS:<p>Fmoc-5-aminopentanoic acid: alkane, Fmoc-protected amine, carboxyl group, PROTAC linker, deprotects to free amine, forms amides with activators.</p>Fórmula:C20H21NO4Forma y color:SolidPeso molecular:339.39Antitumor agent-88
CAS:<p>Antitumor agent-88, a potent antimitotic, arrests G2/M phase, disrupts microtubules in breast cancer, and inhibits CYP1A1 (Ki: 1.4 μM).</p>Fórmula:C23H30N2O7SForma y color:SolidPeso molecular:478.56α-Glucosidase-IN-21
CAS:<p>α-Glucosidase-IN-21 (Compound 2B) is a highly potent and orally bioavailable inhibitor of α-glucosidase.</p>Fórmula:C24H23NO2SForma y color:SolidPeso molecular:389.513,3-Dimethyl-1-butanol
CAS:<p>3,3-Dimethyl-1-butanol (DMB) inhibits TMA/TMAO and affects p65 NF-κB, TGF-β1/Smad3 signaling; potential for CVD treatment.</p>Fórmula:C6H14OForma y color:SolidPeso molecular:102.17hCA IX-IN-2
<p>hCA IX-IN-2 is a highly potent and selective inhibitor of hCA IX, exhibiting an inhibition constant (K I) value of 32.1 nM and demonstrating anti-proliferative</p>Fórmula:C23H24N2O4STeForma y color:SolidPeso molecular:552.11Arasertaconazole
CAS:<p>Arasertaconazole, a sterol-14-alpha demethylation inhibitor, is used potentially for the treatment of vulvovaginal candcanidiasis.</p>Fórmula:C20H15Cl3N2OSForma y color:SolidPeso molecular:437.77A-908292
CAS:<p>A-908292: potent ACC2 inhibitor with 38 nM IC50, useful for studying fatty acid metabolism.</p>Fórmula:C18H20N2O4SForma y color:SolidPeso molecular:360.43FABP-IN-2
CAS:<p>FABP-IN-2, a novel ligand for FABP3, demonstrates inhibition of both FABP3 and FABP4 with IC50 values of 1.16 μM and 4.27 μM, respectively.</p>Fórmula:C25H21ClN2O3Forma y color:SolidPeso molecular:432.9hCAXII-IN-1
CAS:<p>hCAXII-IN-1 selectively inhibits HCA IX/XII, promising for new cancer drug development.</p>Fórmula:C20H17NO5Forma y color:SolidPeso molecular:351.35ENPP1 inhibitor 43
CAS:<p>ENPP1 inhibitor 43 is a novel small molecule for cancer immunotherapy.</p>Fórmula:C16H18N6O3SForma y color:SolidPeso molecular:374.42DP00477
CAS:<p>DP00477, a potent inhibitor of indoleamine 2,3-dioxygenase 1 (IDO1), exhibits an inhibitory concentration (IC50) of 7.0 µM.</p>Fórmula:C17H11ClF3N3OSForma y color:SolidPeso molecular:397.8Xanthine oxidase-IN-4
CAS:<p>Xanthine oxidase-IN-4: an oral XO inhibitor with 0.039 μM IC50, useful for hyperuricemia/gout research.</p>Fórmula:C15H13N5O2Forma y color:SolidPeso molecular:295.3PRRSV/CD163-IN-1
CAS:<p>PRRSV/CD163-IN-1 blocks PRRSV GP2a/GP4 and CD163-SRCR5, aiding PRRS research.</p>Fórmula:C25H24FN5O5S2Forma y color:SolidPeso molecular:557.62hCAIX-IN-8
CAS:<p>hCAIX-IN-8, a selective hCAIX inhibitor, IC50: 0.024 μM. Also affects CAII, CAVA (IC50s: 1.99, 1.10 μM), limits cell migration, and induces apoptosis.</p>Fórmula:C19H16N4O6Forma y color:SolidPeso molecular:396.35D-threo-PPMP hydrochloride
CAS:<p>D-threo-PPMP inhibits GlyCer synthetase; active enantiomer; reduces MDCK cell growth by 70% at 20 μM.</p>Fórmula:C29H51ClN2O3Forma y color:SolidPeso molecular:511.19NPD-1335
CAS:<p>NPD1335: potent TbrPDEB1 inhibitor, submicromolar efficacy, low toxicity, raises cAMP, disrupts cell cycle, kills T. brucei.</p>Fórmula:C28H29N3O3Pureza:98%Forma y color:SolidPeso molecular:455.55Sch 34826
CAS:<p>Sch 34826 is a potent, selective neutral endopeptidase inhibitor.</p>Fórmula:C27H34N2O7Pureza:98%Forma y color:SolidPeso molecular:498.57Boc-Glu(OBzl)-OSu
CAS:<p>Boc-Glu(OBzl)-OSu can be used for the synthesis of solid phase peptides containing benzyl glutamate residues.</p>Fórmula:C21H26N2O8Forma y color:SolidPeso molecular:434.44AMG-221
CAS:<p>AMG-221: potent 11β-HSD1 inhibitor, lowers glucose & insulin, reduces obesity in mice.</p>Fórmula:C14H22N2OSPureza:98%Forma y color:SolidPeso molecular:266.4JTP-4819
CAS:<p>JTP-4819: potent PEP inhibitor, may treat Alzheimer's, boosts brain peptides and acetylcholine, aiding memory.</p>Fórmula:C19H25N3O4Forma y color:SolidPeso molecular:359.42Andolast
CAS:<p>Andolast (CR-2039) is an anti-allergic for asthma and COPD, inhibiting IgE synthesis and improving airflow.</p>Fórmula:C15H11N9OForma y color:SolidPeso molecular:333.31sEH inhibitor-14
CAS:<p>sEH inhibitor-14, a benzoxazolone-5-urea analogue, acts as an efficient soluble Epoxide Hydrolase (sEH) inhibitor, demonstrating significant activity with an</p>Fórmula:C16H12F3N3O4Forma y color:SoildPeso molecular:367.28Deltazinone
CAS:<p>Deltazinone selectively inhibits PDEδ with low cytotoxicity, mimicking PDEδ knockdown in human pancreatic cancer cells.</p>Fórmula:C27H31N5O2Pureza:98%Forma y color:SolidPeso molecular:457.57SGK1 inhibitor
CAS:<p>SGK1 inhibitor targets SGK1/2 over SGK3, blocks GSK3β phosphorylation, lowers HCC1954 cell viability with BYL719, and reduces tumor growth in mice.</p>Fórmula:C17H12Cl2N6O2SForma y color:SolidPeso molecular:435.29CAY10485
CAS:<p>CAY10485 blocks human ACAT-1 & ACAT-2 (IC50: 95 & 81 μM) and hinders oxidation of LDL by 91% at 2 μM, possibly impacting atherosclerosis development.</p>Fórmula:C27H27NO7Forma y color:SolidPeso molecular:477.51Enpp-1-IN-5
CAS:<p>Enpp-1-IN-5 is a potent enpp-1 inhibitor with potential in cancer and infectious disease research.</p>Fórmula:C17H26N6O4SForma y color:SolidPeso molecular:410.49mIDH1-IN-1
CAS:<p>mIDH1-IN-1 is a selective mIDH1 inhibitor (IC50: 961.5 nM), blocks 2-HG production, and hinders IDH1 mutant cell growth (IC50: 41.8 nM).</p>Fórmula:C25H27N3O5Forma y color:SolidPeso molecular:449.5UK-414,495
CAS:<p>UK-414,495 is a potent, selective inhibitor of the neutral endopeptidase, the enzyme normally serves to break down the neuropeptide VIP.</p>Fórmula:C16H25N3O3SForma y color:SolidPeso molecular:339.45AMG-7980
CAS:<p>AMG-7980 is a highly specific phosphodiesterase 10A ligand. It shows a good uptake in the striatum.</p>Fórmula:C19H22N4O2Pureza:98%Forma y color:SolidPeso molecular:338.4Xanthine oxidoreductase-IN-2
CAS:<p>Xanthine oxidoreductase-IN-2 inhibits XOR with 7.2 nM IC50 and shows hypouricemic effects in mice.</p>Fórmula:C21H19N3O2Forma y color:SolidPeso molecular:345.39α-Glucosidase-IN-8
CAS:<p>α-Glucosidase-IN-8 (Compound 4k) is a potent, competitive inhibitor of α-glucosidase. It displays an impressive IC50 value of 0.18 μg/mL [1].</p>Fórmula:C19H20FN3O2Forma y color:SolidPeso molecular:341.38Eggmanone
CAS:<p>EGM1: potent PDE4D3 inhibitor, IC50=72 nM, 40-50x selectivity over other PDEs, activates PKA, blocks Hh.</p>Fórmula:C20H20N2O2S3Forma y color:SolidPeso molecular:416.58hCAIX-IN-6
CAS:<p>6B and 14g inhibit tumor-associated HCA IX with low nanomolar potency; 6K targets HCA XII. All are potential cancer drug leads.</p>Fórmula:C18H12N2O4SForma y color:SolidPeso molecular:352.36Carbonic anhydrase inhibitor 13
CAS:<p>Carbonic anhydrase inhibitor 13 (compound 7) is a potent inhibitor of carbonic anhydrase (CA).</p>Fórmula:C17H15N5O3S2Forma y color:SolidPeso molecular:401.46IDO1-IN-17
CAS:<p>IDO1-IN-17 (I-4) is an IDO1 inhibitor, with an IC 50 of 0.44 μM in hela cells .</p>Fórmula:C28H32BrClFN5O2Forma y color:SolidPeso molecular:604.94FAAH-IN-5
CAS:<p>FAAH-IN-5 (Compound 7) selectively, irreversibly inhibits FAAH (IC50: 10.5 nM) with low PAMPA permeability.</p>Fórmula:C21H19N3O6SForma y color:SolidPeso molecular:441.46
