
Metabolismo
Los inhibidores del metabolismo son compuestos que interfieren con las vías metabólicas, alterando la producción y utilización de energía dentro de las células. Estos inhibidores se utilizan para estudiar la regulación del metabolismo, el papel de las vías metabólicas en enfermedades como el cáncer y la diabetes, y para desarrollar nuevas estrategias terapéuticas. Los inhibidores del metabolismo pueden dirigirse a diversas enzimas y procesos involucrados en la glucólisis, la oxidación de ácidos grasos y otras funciones metabólicas. En CymitQuimica, ofrecemos una amplia gama de inhibidores del metabolismo de alta calidad para apoyar su investigación en bioquímica, trastornos metabólicos y desarrollo de fármacos.
Subcategorías de "Metabolismo"
- AhR(41 productos)
- Aminopeptidasa(67 productos)
- CETP(18 productos)
- Anhídrido carbónico(178 productos)
- Caseína quinasa(130 productos)
- DHFR(33 productos)
- Descarboxilasa(4 productos)
- Deshidrogenasa(269 productos)
- FAAH(64 productos)
- FXR(58 productos)
- Factor Xa(80 productos)
- Ácido graso sintasa(32 productos)
- Ferroptosis(215 productos)
- GR(3 productos)
- GSNOR(3 productos)
- Glucoquinasa(54 productos)
- HIF / HIF Prolilhidroxilasa(142 productos)
- HMG-CoA reductasa(33 productos)
- Hidroxilasa(30 productos)
- IDO(82 productos)
- LDL(8 productos)
- Lipasa(97 productos)
- Lípido(59 productos)
- Lipoxigenasa(124 productos)
- MAO(87 productos)
- MPO(2 productos)
- NAMPT(36 productos)
- P450(6 productos)
- PAI-1(25 productos)
- PDE(166 productos)
- PED(1 productos)
- PKM(15 productos)
- PPAR(164 productos)
- Fosfolipasa(82 productos)
- ROR(42 productos)
- Receptor de retinoides(29 productos)
- SGK(11 productos)
- Tiorredoxina(12 productos)
- Transferasa(30 productos)
- Transportador(42 productos)
- UGT(4 productos)
- Inhibidores de la xantina oxidasa (XO)(9 productos)
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Se han encontrado 8626 productos de "Metabolismo"
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ABL127
CAS:<p>ABL127 inhibits PME-1 with IC50s of 6.4 nM in HEK293T cells and 4.2 nM in MDA-MB-231 cells.</p>Fórmula:C17H20N2O5Pureza:98%Forma y color:SolidPeso molecular:332.35Butaperazine maleate
CAS:<p>Butaperazine maleate, a phenothiazine derivative, is an antipsychotic.</p>Fórmula:C32H39N3O9SPureza:98%Forma y color:SolidPeso molecular:641.73NPD7155
CAS:<p>NPD7155 is a competitive inhibitor of MTH1.</p>Fórmula:C15H21N5Pureza:98%Forma y color:SolidPeso molecular:271.36PD-34799-SA
CAS:<p>PD-34799-SA is an effective inhibitor of vasoconstrictor responses to sympathetic nerve stimulation.</p>Fórmula:C10H16N4O4Pureza:98%Forma y color:SolidPeso molecular:256.262Albifylline
CAS:<p>Albifylline: a xanthine derivative, anti-asthmatic, reduces leukocyte adhesion, enhances liver microcirculation post-hemorrhagic shock.</p>Fórmula:C13H20N4O3Forma y color:SolidPeso molecular:280.32AHR-activator-1023
CAS:<p>AHR-activator-1023 is the aryl hydrocarbon receptor activator. It is also a specific FGF2-induced branching morphogenesis modulator.</p>Fórmula:C14H8Cl2N2OForma y color:SolidPeso molecular:291.13SMP-028
CAS:<p>SMP-028 is a neutral cholesterol esterase (CEase) inhibitor(IC50 : 1.01 μM).</p>Fórmula:C23H26FN5O2SPureza:98%Forma y color:SolidPeso molecular:455.55BemPPOX
CAS:<p>BemPPOX is a potent inhibitor of DGL.</p>Fórmula:C23H20N2O5Forma y color:SolidPeso molecular:404.42N-(3-Oxooctanoyl)-DL-homoserine lactone
CAS:<p>N-(3-Oxooctanoyl)-DL-homoserine lactone with stereochemistry-dependent growth regulatory activity for roots .</p>Fórmula:C12H19NO4Pureza:98%Forma y color:SolidPeso molecular:241.28LY 79771
CAS:<p>LY-79771, a phenethanolamine antiobesity agent, can be effective in preventing fat regain following energy deprivation.</p>Fórmula:C18H24ClNO2Forma y color:SolidPeso molecular:321.84ML350
CAS:<p>ML350 (CYM-50202) is a potent KOR antagonist (IC50: 12.6 nM), selective over DOR/MOR, with high solubility and CNS penetration, lacking long-term effects.</p>Fórmula:C18H26BrN3O3Pureza:98%Forma y color:SolidPeso molecular:412.32L-693612
CAS:<p>L-693612 is an inhibitor of carbonic anhydrase.</p>Fórmula:C14H24N2O5S3Pureza:98%Forma y color:SolidPeso molecular:396.55RA 642
CAS:<p>RA 642 is used as a PDE-inhibitor.</p>Fórmula:C24H44N8O4Pureza:98%Forma y color:SolidPeso molecular:508.66NSC-79887
CAS:<p>NSC-79887 is a nucleoside hydrolase (NH) inhibitor.</p>Fórmula:C14H16ClNO4Pureza:98%Forma y color:SolidPeso molecular:297.73CL385319 HCl
CAS:<p>"CL385319: Inhibits H5N1 flu virus, blocks entry, low cytotoxicity, IC50=27.03μM in MDCK cells, ineffective on VSV-G pseudotypes."</p>Fórmula:C15H19ClF4N2OPureza:98%Forma y color:SolidPeso molecular:354.772-Methyldecanenitrile
CAS:<p>2-Methyldecanenitrile, intense peach scent with lactone notes, stable in all pH, effective at low concentration.</p>Fórmula:C11H21NPureza:98%Forma y color:Colourless Liquid LiquidPeso molecular:167.29GA11
CAS:<p>GA11is an inhibitor of ALDH1. It also displays anti-GBM effects in vitro and in vivo.</p>Fórmula:C19H14N2Pureza:98%Forma y color:SolidPeso molecular:270.33Chlorambucyl-proline
CAS:<p>Chlorambucyl-proline is a chlorambucil derivative of L-proline. It is an inhibitor of bovine lung angiotensin I-converting enzyme.</p>Fórmula:C19H26Cl2N2O3Pureza:98%Forma y color:SolidPeso molecular:401.33CP 99994 dihydrochloride
CAS:<p>High affinity NK1 antagonist</p>Fórmula:C19H26Cl2N2OPureza:98%Forma y color:SolidPeso molecular:369.33Lauroyl glutamic acid
CAS:<p>Lauroyl glutamic acid (N-Lauroyl-L-glutamic acid) exhibits antiasthmatic effects.</p>Fórmula:C17H31NO5Pureza:98.94%Forma y color:SolidPeso molecular:329.43WWL113
CAS:<p>WWL113 is a selective oral inhibitor for Ces3 and Ces1f, with IC50s of 120 nM and 100 nM, notably targeting the 60-kDa serine hydrolase.</p>Fórmula:C29H26N2O4Pureza:98%Forma y color:SolidPeso molecular:466.53Gemcabene
CAS:<p>Gemcabene (PD-72953) lowers LDL and triglycerides, boosts HDL, and reduces inflammation by decreasing C-reactive protein.</p>Fórmula:C16H30O5Pureza:≥98%Forma y color:SolidPeso molecular:302.41Fluasterone
CAS:<p>Fluasterone, an NF-κB activation inhibitor, is used potentially for the treatment of metabolic syndrome.</p>Fórmula:C19H27FOPureza:98%Forma y color:SolidPeso molecular:290.42Hydroxythiohomosildenafil
CAS:<p>Hydroxythiohomosildenafil, an analogue of sildenafil, is a phosphodiesterase-5 (PDE-5) inhibitor.</p>Fórmula:C23H32N6O4S2Pureza:99.45%Forma y color:SolidPeso molecular:520.67Tenuazonic acid
CAS:<p>Tenuazonic acid, a nonhost-selective mycotoxin from Alternaria alternate, inhibits PSII by blocking electron transport at D1 protein.</p>Fórmula:C10H15NO3Pureza:98%Forma y color:SolidPeso molecular:197.23(3S,5S)-Pitavastatin calcium
CAS:<p>(3S,5S)-Pitavastatin calcium is the 3-epimer of Pitavastatin which is a potent HMG-CoA reductase inhibitor.</p>Fórmula:C25H26CaFNO4Pureza:98%Forma y color:SolidPeso molecular:463.56212(S)-HpETE
CAS:<p>12(S)-HpETE activates human blood leukocyte 5-LOE and mediates induction of c-fos and c-jun, activation of AP-1, and endothelium-dependent vasoconstriction.</p>Fórmula:C20H32O4Forma y color:SolidPeso molecular:336.47Rev 6207
CAS:<p>Rev 6207 is a non-sulfhydryl ACE-inhibitor.</p>Fórmula:C21H31N3O5Forma y color:SolidPeso molecular:405.497ETMC
CAS:<p>7ETMC inhibits Human Cytochrome P450s 1A1/1A2 with IC50: 0.46/0.50 μM; not effective on P450s 2A6/2B1 even at 50 μM.</p>Fórmula:C14H12O2Pureza:98%Forma y color:SolidPeso molecular:212.24MAO-B Inhibitor 58
CAS:<p>MAO-B inhibitor 58 is an effective, selective, and reversible inhibitor of monoamine oxidase B.</p>Fórmula:C14H9Cl2N3Forma y color:SolidPeso molecular:290.15Muristerone A
CAS:<p>Muristerone A is a phytoecdysteroid analog of ecdysone and a potent ecdysteroid receptor agonist with a K d of 1 nM [1].</p>Fórmula:C27H44O8Forma y color:SolidPeso molecular:496.63AE0047 Hydrochloride
CAS:<p>AE0047 Hydrochloride is a blocker of calcium, and used in the research of the hypertensive disease.</p>Fórmula:C41H43ClN4O6Pureza:98%Forma y color:SolidPeso molecular:723.26SCH-51866
CAS:<p>SCH-51866 is a PDE1 and PDE5 phosphodiesterase inhibitor with IC50 value of 0.070 μM and IC50 0.060 μM respectively.</p>Fórmula:C19H18F3N5OPureza:98%Forma y color:SolidPeso molecular:389.37Benproperine
CAS:<p>Benproperine is a bioactive molecule with antineoplastic properties.</p>Fórmula:C21H27NOPureza:98%Forma y color:SolidPeso molecular:309.45Lucerastat
CAS:<p>Lucerastat(NBDGJ) is an orally available inhibitor of GCS for Fabry disease by reducing harmful substrates.. GCS is a key enzyme in sphingolipid synthesiss.</p>Fórmula:C10H21NO4Pureza:98%Forma y color:SolidPeso molecular:219.28WAY-213613
CAS:<p>WAY-213613: Potent GLT-1/EAAT2 inhibitor (IC50: 85 nM), selective over EAAT1/EAAT3; inactive at glutamate receptors.</p>Fórmula:C16H13BrF2N2O4Pureza:98%Forma y color:SolidPeso molecular:415.19Risarestat
CAS:<p>Risarestat (CT-112) is a potent aldose reductase inhibitor and thyroid hormone receptor (TR) antagonist for the treatment of hypoglycemia.</p>Fórmula:C16H21NO4SPureza:98.39%Forma y color:SolidPeso molecular:323.41Rentiapril racemate
CAS:<p>Rentiapril racemate (SA-446 racemate) is the racemate of Rentiapril.Rentiapril racemate has anti-inflammatory activity and may be used in glaucoma research.</p>Fórmula:C13H15NO4S2Pureza:98.96% - >99.99%Forma y color:SolidPeso molecular:313.39ACAT-IN-1 cis isomer
CAS:<p>ACAT-IN-1 cis isomer is a potent ACAT inhibitor (IC50: 100 nM) for the study of immune system-related diseases.</p>Fórmula:C29H25NO2Pureza:>99.99%Forma y color:SolidPeso molecular:419.51Peliglitazar racemate
CAS:<p>Peliglitazar racemate(BMS 426707-01 racemate) is the racemate of Peliglitazar.Peliglitazar racemate may be used as a potential antidiabetic and anti-obesity</p>Fórmula:C30H30N2O7Pureza:97.75%Forma y color:SolidPeso molecular:530.57PKM2 activator 5
CAS:<p>PKM2 activator 5 is a novel and potent PKM2 activator (AC50: 0.316 µM) with potential anticancer activity for the study of cancer metabolism-related diseases.</p>Fórmula:C18H19FN2O6S2Pureza:98%Forma y color:SolidPeso molecular:442.48IDO-IN-6
CAS:<p>IDO-IN-6 is an indoleamine 2,3-dioxygenase (IDO) inhibitor.</p>Fórmula:C18H21FN2O2Pureza:98%Forma y color:SolidPeso molecular:316.37Diaplasinin
CAS:<p>Diaplasinin (PAI-749) is a potent inhibitor of plasminogen activator inhibitor-1 (PAI-1) with antithrombotic activity, used in cardiovascular disease research.</p>Fórmula:C32H31N5OPureza:99.02%Forma y color:SolidPeso molecular:501.62Teglarinad chloride
CAS:<p>Teglarinad chloride (GMX-1777 chloride) is an inhibitor of NAMPT with antitumor activity that acts by interfering with DNA repair and inhibiting angiogenesis.</p>Fórmula:C30H43Cl2N5O8Pureza:98.09%Forma y color:SolidPeso molecular:672.6hCAIX-IN-5
CAS:<p>hCAIX-IN-5 was a selective hCAIX inhibitor, inhibiting hCAI, hCAII, hCAIV, and hCAIX with Ki values of >10000, >10000, 130.7, and 829.1 nM, respectively.</p>Fórmula:C18H12FNO3Pureza:99.26%Forma y color:SolidPeso molecular:309.2920(S)-Hydroxycholesterol
CAS:<p>20(S)-Hydroxycholesterol (20α-Hydroxycholesterol) is an allosteric activator of the oncoprotein smoothened (Smo).</p>Fórmula:C27H46O2Pureza:99.25% - 99.79%Forma y color:SolidPeso molecular:402.65Dehydronitrosonisoldipine
CAS:<p>Dehydronitrosonisoldipine blocks SARM1, slows axon decay & cADPR synthesis; useful in neurodegeneration research.</p>Fórmula:C20H22N2O5Pureza:99.68%Forma y color:SolidPeso molecular:370.4PDE5-IN-5
CAS:<p>PDE5-IN-5 is a selective inhibitor of phosphodiesterase 5 (PDE5) (IC50: 2.0 nM).</p>Fórmula:C23H20BrN3O4Forma y color:SolidPeso molecular:482.33D-Erythro-dihydrosphingosine
CAS:<p>D-Erythro-dihydrosphingosine (C18-Dihydrosphingosine) inhibits arachidonic acid release and cPLA2α activity.</p>Fórmula:C18H39NO2Pureza:99.50% - 99.88%Forma y color:SolidPeso molecular:301.51N-Acetylserine
CAS:<p>N-Acetylserine (N-Acetyl-L-serine) serves as the physiological inducer of cysteine biosynthesis by binding to the CysB apoprotein and stimulating cysJIH</p>Fórmula:C5H9NO4Pureza:99.28%Forma y color:SolidPeso molecular:147.13Autotaxin-IN-1
CAS:<p>Autotaxin-IN-1: strong inhibitor for osteoarthritis pain; IC50=2.2 nM; good PK and PK/PD.</p>Fórmula:C21H23N7O2Pureza:98%Forma y color:SolidPeso molecular:405.45Tralkoxydim
CAS:<p>Tralkoxydim (Tralkoxydime) is an alkyl ketone herbicide. Tralkoxydim works as an ACCase inhibitor.</p>Fórmula:C20H27NO3Pureza:97.44%Forma y color:SolidPeso molecular:329.43AN3199
CAS:<p>AN3199 is a selective inhibitor of PDE4 with an IC50 of 94.5 nM.</p>Fórmula:C17H18BNO5Pureza:99.45%Forma y color:SolidPeso molecular:327.14LGE-899
CAS:<p>LGE-899 (Sonidegib metabolite M48) is a main metabolite of Sonidegib which is an inhibitor of the hedgehog pathway.</p>Fórmula:C15H11F3O3Pureza:99.93%Forma y color:SolidPeso molecular:296.24Phytic acid dodecasodium salt hydrate
CAS:<p>Phytic acid salt hydrate: seed phosphorus compound, inhibits xanthine oxidase, IC50 6 mM, antioxidant, neuroprotective, anti-inflammatory.</p>Fórmula:C6H20NaO25P6Pureza:≥98%Forma y color:SolidPeso molecular:701.03311β-HSD1-IN-1
CAS:<p>11β-HSD1-IN-1 is an inhibitor of 11β-hydroxydehydrogenase 1 (11β-HSD1, IC50: 52 nM), and used for the treatment of pain.</p>Fórmula:C18H14ClF4N3OPureza:99.84%Forma y color:SolidPeso molecular:399.77PSB-1410
CAS:<p>PSB-1410 is a selective and highly efficient monoamine oxidase B (MAO-B) inhibitor, which can be used in research on neurological diseases.</p>Fórmula:C15H10Cl2N2OPureza:98.69%Forma y color:SolidPeso molecular:305.16(-)-Ketoconazole
CAS:<p>(-)-Ketoconazole is a potential mitochondrial CYP24A1 inhibitor and has antifungal activity against Aspergillus fumigatus.</p>Fórmula:C26H28Cl2N4O4Pureza:98%Forma y color:SolidPeso molecular:531.43Migoprotafib
CAS:<p>Migoprotafib (GDC-1971) is a potent and highly selective SHP2 (Src Homology-2 Domain-Containing Phosphatase 2) inhibitor for advanced solid tumours.</p>Fórmula:C25H26N8OForma y color:SolidPeso molecular:454.53Lirimilast
CAS:<p>Lirimilast: oral PDE4 inhibitor (IC50: 49 nM), anti-inflammatory, treats asthma/COPD.</p>Fórmula:C17H12Cl2N2O6SPureza:98%Forma y color:SolidPeso molecular:443.26UK51656
CAS:<p>UK51656 is an antagonist of calcium (IC50: 4 nM).</p>Fórmula:C22H28ClN3O6Pureza:98%Forma y color:SolidPeso molecular:465.93Palonidipine
CAS:<p>Palonidipine is an antagonist of calcium, is potential for the therapy of angina-pectoris and hypertension.</p>Fórmula:C29H34FN3O6Pureza:98%Forma y color:SolidPeso molecular:539.6Pparδ agonist 2
CAS:<p>Pparδ agonist 2 is an agonist of PPARδ.</p>Fórmula:C20H18F3N3O3SPureza:98%Forma y color:SolidPeso molecular:437.44IDO-IN-12
CAS:<p>IDO-IN-12 is an inhibitor of indoleamine 2,3-dioxygenase (IDO).</p>Fórmula:C13H11BrFN5O3SPureza:99.727%Forma y color:SolidPeso molecular:416.23(R)-Nepicastat HCl
CAS:<p>(R)-Nepicastat HCl (RS-25560-198 HCl), R-enantiomer, inhibits bovine/human dopamine-β-hydroxylase (IC50: 25.1/18.3 nM); not affecting other enzymes/receptors.</p>Fórmula:C14H15F2N3S·HClPureza:98%Forma y color:SolidPeso molecular:331.81BN82002
CAS:<p>BN82002 (CDC25 Phosphatase Inhibitor I) is a synthetic inhibitor of CDC25 phophatases</p>Fórmula:C19H25N3O4Pureza:98.24%Forma y color:SolidPeso molecular:359.42PSN-GK1
CAS:<p>PSN-GK1 is a potent activator of glucokinase (EC50: 0.13 μM).</p>Fórmula:C20H23FN2O4S2Pureza:98%Forma y color:SolidPeso molecular:438.54Endothelial lipase inhibitor-1
CAS:<p>Endothelial lipase inhibitor-1 is a potent endothelial lipase inhibitor with an IC50 of 49 nM.</p>Fórmula:C22H22N4O4Pureza:99.59%Forma y color:SolidPeso molecular:406.43Deltasonamide 2
CAS:<p>Deltasonamide 2 is a competitive, high affinity PDEδ inhibitor with a Kd of ~385 pM.</p>Fórmula:C30H39ClN6O4S2Pureza:98%Forma y color:SolidPeso molecular:647.25Enazadrem
CAS:<p>Enazadrem is a 5-lipoxygenase inhibitor with antiinflammatory activities.</p>Fórmula:C18H25N3OPureza:98%Forma y color:SolidPeso molecular:299.4113(S)-HOTrE(γ)
CAS:<p>13(S)-HOTrE(γ) is a metabolite and octadecatrienoic acid used as a metabolic marker, in the study of metabolic disorders and neurological diseases.</p>Fórmula:C18H30O3Forma y color:SolidPeso molecular:294.43SU 10603
CAS:<p>SU 10603 is a specific inhibitor of 17α-hydroxylase (also known as CYP17A1 and P450c17) used to study steroid hormone synthesis.</p>Fórmula:C15H12ClNOPureza:99.93% - 99.96%Forma y color:SolidPeso molecular:257.72AMPD2 inhibitor 1
CAS:<p>AMPD2 inhibitor 1 is an adenosine monophosphate deaminase 2 (AMPD2) inhibitor, useful for studying anorexia in the nervous system.</p>Fórmula:C25H22N2O2Forma y color:SolidPeso molecular:382.457-Ketolithocholic acid
CAS:<p>7-Ketolithocholic acid absorbs and reduces endogenous bile acid and cholesterol secretion.</p>Fórmula:C24H38O4Pureza:98.68% - 99.9%Forma y color:White - Almost White Solid PowderPeso molecular:390.56Seviteronel
CAS:<p>Seviteronel (VT-464) is a novel CYP17 cleavage enzyme inhibitor and androgen receptor antagonist for the study of breast and prostate cancer.</p>Fórmula:C18H17F4N3O3Pureza:99.67% - 99.98%Forma y color:SolidPeso molecular:399.34LYS006
CAS:<p>LYS006 is a highly efficient and selective LTA4H (leukotriene A4 hydrolase) inhibitor,for neutrophil-driven inflammatory diseases ulcerative colitis.</p>Fórmula:C16H14ClFN6O3Pureza:99.33%Forma y color:SoildPeso molecular:392.77PF-07208254
CAS:<p>PF-07208254, a potent BDK inhibitor, enhances cardiometabolic endpoints in mice [1].</p>Fórmula:C7H2ClFO2S2Pureza:98%Forma y color:SolidPeso molecular:236.67IDO1-IN-21
CAS:<p>IDO1-IN-21 (compound 10m), with an IC50 of 0.64 μM, acts as an IDO1 inhibitor and has demonstrated efficacy in suppressing tumor growth in murine models [1].</p>Fórmula:C21H19F2N3O6SPureza:98%Forma y color:SolidPeso molecular:479.45WES-1
CAS:<p>WES-1 (Compound 8g), a carbonic anhydrase IX inhibitor (Ki: 55.9 μM), exhibits broad-spectrum antiproliferative activity against various cancer cell lines,</p>Fórmula:C20H20N4O3SPureza:98%Forma y color:SolidPeso molecular:396.46Erythronic acid
CAS:<p>Erythronic acid, an endogenous carbohydrate metabolite, is instrumental for research into metabolism-associated disorders.</p>Fórmula:C4H8O5Pureza:98%Forma y color:SolidPeso molecular:136.117β-HSD10-IN-2
CAS:<p>17β-HSD10-IN-2 (compound 11), a benzothiazolylurea-based inhibitor, specifically targets 17β-hydroxysteroid dehydrogenase type 10 (17β-HSD10), avoiding</p>Fórmula:C15H10ClN3O4SPureza:98%Forma y color:SolidPeso molecular:363.78ASM-IN-1
CAS:<p>ASM-IN-1: Oral acid sphingomyelinase inhibitor, IC50 = 1.5 µM; reduces lipid plaques, plasma ceramide, Ox-LDL.</p>Fórmula:C16H12BrN3O4Pureza:98%Forma y color:SolidPeso molecular:390.19LZWL02003
CAS:<p>LZWL02003, an anti-neuroinflammatory agent, demonstrates a protective effect on MPP+-induced neuronal damage and reduces ROS expression.</p>Fórmula:C18H18N2O2Pureza:98%Forma y color:SolidPeso molecular:294.35IACS-8968
CAS:<p>IACS-8968 is a dual IDO and TDO inhibitor (pIC50s: 6.43 for IDO and <5 for TDO).</p>Fórmula:C17H18F3N5O2Pureza:98%Forma y color:SolidPeso molecular:381.35Calcium glycerophosphate
CAS:<p>CaGP inhibits intestinal alkaline phosphatase F3; used for calcium and phosphorus in parenteral nutrition.</p>Fórmula:C3H7CaO6PPureza:99.84%Forma y color:SolidPeso molecular:210.14(Z)-10-Hydroxynortriptyline
CAS:<p>(Z)-10-Hydroxynortriptyline ((Z)-10-Hydroxy Nortriptyline) is a norepinephrine reuptake inhibitor with antidepressant activity.</p>Fórmula:C19H21NOPureza:98%Forma y color:SolidPeso molecular:279.38EZ-482
CAS:<p>EZ-482 is an apolipoprotein (apoE) ligand used for Alzheimer's disease.</p>Fórmula:C23H19ClN4O5SPureza:97.29%Forma y color:SolidPeso molecular:498.941-Methyluric acid
CAS:<p>1-Methyluric acid (1-Methylurate) acts on the bladder mucosa and increases the levels of insulin, triglycerides, cholesterol, and blood glucose.</p>Fórmula:C6H6N4O3Pureza:98.05%Forma y color:SolidPeso molecular:182.14PDE7-IN-2
CAS:<p>PDE7-IN-2 is an inhibitor of phosphodiesterase 7 (IC50 = 2.1 µM) and can be used in Parkinson's disease studies.</p>Fórmula:C14H11ClN2O3SPureza:98%Forma y color:SolidPeso molecular:322.772'-Ethyl Simvastatin
CAS:<p>2'-Ethyl Simvastatin is a Mevinolin analog with HMG-CoA reductase inhibition.</p>Fórmula:C23H34O5Pureza:98%Forma y color:SolidPeso molecular:390.51Manitimus
CAS:<p>Manitimus is a potent immunosuppressive drug, and is an inhibitor of dehydroorotate dehydrogenase,.</p>Fórmula:C15H11F3N2O2Pureza:99.75% - 99.75%Forma y color:SolidPeso molecular:308.26PF-4191834
CAS:<p>PF-4191834: Non-iron, non-redox 5-LOX inhibitor, IC50 = 229 nM, 300x selective over 12/15-LOX, inactive on COX enzymes.</p>Fórmula:C22H23N3O2SPureza:99.83% - 99.98%Forma y color:SolidPeso molecular:393.5MAGL-IN-1
CAS:<p>MAGL-IN-1 is a selective and potent monoacylglycerol lipase (MAGL) inhibitor with an IC50 of 80 nM.</p>Fórmula:C22H24FNO3Pureza:98%Forma y color:SolidPeso molecular:369.43Reglitazar
CAS:<p>Reglitazar, a dual PPARα/γ agonist, enhances insulin signaling, reduces insulin resistance, and lowers hypertriglyceridemia in obese rats.</p>Fórmula:C22H20N2O5Pureza:97.07% - 98.72%Forma y color:SolidPeso molecular:392.4MK-4409
CAS:<p>MK-4409, a potent and selective fatty acid amide hydrolase (FAAH) inhibitor, is being investigated for the treatment of inflammatory and neuropathic pain.</p>Fórmula:C22H17ClFN3O2SPureza:99.80% - 99.87%Forma y color:SolidPeso molecular:441.91CYP11B2-IN-1
CAS:<p>CYP11B2-IN-1 是一种有效的选择性 CYP11B2 抑制剂,对 CYP11B2 和 CYP11B1 的 IC50 分别为 2.3 nM 和 142 nM。</p>Fórmula:C18H18FN3OPureza:99.79% - 99.89%Forma y color:SolidPeso molecular:311.352614W94
CAS:2614W94 is a selective inhibitor of MAO-A with IC50 of 5 nM and Ki of 1.6 nM.Fórmula:C15H11F3O4SPureza:99.6%Forma y color:SolidPeso molecular:344.31PAT-048
CAS:<p>PAT-048 is an effective and selective autotaxin inhibitor.</p>Fórmula:C22H18ClF2N3O2SPureza:98%Forma y color:SolidPeso molecular:461.91PDE9-IN-1
CAS:<p>PDE9-IN-1 is a selective and orally bioavailable Inhibitor of PDE9A(IC50 of 8.7 nM).</p>Fórmula:C17H23FN6O2Pureza:99.86%Forma y color:SolidPeso molecular:362.4IDO-IN-8
CAS:<p>IDO-IN-8 is an indoleamine 2,3-dioxygenase (IDO) inhibitor (IC50: 1-10 μM).</p>Fórmula:C18H21FN2O2Pureza:98%Forma y color:SolidPeso molecular:316.37Imazodan hydrochloride
CAS:<p>Imazodan hydrochloride (CI-914 HCl) is a potent and selective type III phosphodiesterase inhibitor used in the treatment of chronic congestive heart failure.</p>Fórmula:C13H13ClN4OPureza:98.97%Forma y color:SolidPeso molecular:276.72ML-148
CAS:<p>ML-148 is a selective inhibitor of 15-hydroxy prostaglandin dehydrogenase (15-PGDH, IC50 = 56 nM).</p>Fórmula:C20H21N3OPureza:99.88%Forma y color:SolidPeso molecular:319.4IDO1-IN-2
CAS:<p>IDO1-IN-2 is a potent and selective IDO1 inhibitor with IC50s of 81 nM, 59 nM (mouse), and 28 nM (rat), respectively. It has anti-cancer activity.</p>Fórmula:C15H17FN6O4Pureza:98%Forma y color:SolidPeso molecular:364.33Imazodan
CAS:<p>Imazodan is a compound with positive inotropic activity and is a type III phosphodiesterase inhibitor that can be used to study heart failure.</p>Fórmula:C13H12N4OPureza:98% - 98.31%Forma y color:SolidPeso molecular:240.26LP-533401
CAS:<p>LP-533401 is an inhibitor of Tryptophan hydroxylase 1. It is used for regulates serotonin production in the gut.</p>Fórmula:C27H22F4N4O3Pureza:98%Forma y color:SolidPeso molecular:526.48Ebaresdax hydrochloride
CAS:<p>Ebaresdax hydrochloride has analgesic activity and is used in the study of painful diabetic neuropathy caused by type I or type II diabetes.</p>Fórmula:C12H15ClN2O3SPureza:99.11% - 99.77%Forma y color:SolidPeso molecular:302.78CDC25B-IN-1
CAS:<p>CDC25B-IN-1 is an inhibitor of CDC25B with a Ki of 8.5 μM. CDC25B-IN-1 increases the G2/M phase by inhibiting cell proliferation and colony formation.</p>Fórmula:C20H19NO3Pureza:97.05%Forma y color:SolidPeso molecular:321.37(R)-Lercanidipine hydrochloride
CAS:<p>(R)-Lercanidipine hydrochloride is the R-enantiomer of Lercanidipine. (R)-lercanidipine hydrochloride is a blocker of calcium channel.</p>Fórmula:C36H42ClN3O6Pureza:98%Forma y color:SolidPeso molecular:648.2PPARα-MO-1
CAS:<p>PPARα-MO-1 is a potent modulator of PPARα.</p>Fórmula:C27H37NO5Pureza:98%Forma y color:SolidPeso molecular:455.59SC-22716
CAS:<p>SC-22716 is a LTA4 hydrolase inhibitor.SC-22716 has anti-inflammatory activity and may be used in the study of inflammatory bowel disease and psoriasis.</p>Fórmula:C18H21NOPureza:99.91%Forma y color:SolidPeso molecular:267.37Eribaxaban
CAS:<p>Eribaxaban (PD348292) is an orally available factor Xa inhibitor for the prevention and treatment of venous thromboembolism.</p>Fórmula:C24H22ClFN4O4Pureza:98.99% - 99.13%Forma y color:SolidPeso molecular:484.91Brofaromine
CAS:Brofaromine (CGP 11305A) is an MAO inhibitor (IC50: 0.2 μM for MAO-A).Fórmula:C14H16BrNO2Forma y color:SolidPeso molecular:310.19PGMI-004A
CAS:<p>PGMI-004A is an effective inhibitor of phosphoglycerate mutase 1 (IC50: 13.1 μM).</p>Fórmula:C21H12F3NO6SPureza:98%Forma y color:SolidPeso molecular:463.38SRPKIN-1
CAS:<p>SRPKIN-1 is a covalent and irreversible inhibitor of SRPK1/2 (IC50s: 35.6 and 98 nM, respectively).</p>Fórmula:C27H21FN2O3SPureza:98%Forma y color:SolidPeso molecular:472.53Rovazolac
CAS:<p>Rovazolac (ALX-101) is a liver x receptor (LXR) modulator used in the study of immune system disorders and atopic dermatitis.</p>Fórmula:C21H19F3N2O4SPureza:99.35%Forma y color:SolidPeso molecular:452.45ALDH1A1-IN-2
CAS:<p>ALDH1A1-IN-2 is an aldehyde dehydrogenase 1a1 inhibitor with anticancer activity.ALDH1A1-IN-2 may be used in the study of breast cancer, inflammation or obesity</p>Fórmula:C25H23ClN4O3SPureza:99.48%Forma y color:SolidPeso molecular:494.99BAY 73-6691
CAS:<p>BAY 73-6691 is an inhibitor of brain penetrant PDE9A.</p>Fórmula:C15H12ClF3N4OForma y color:SolidPeso molecular:356.73PDE4-IN-9
CAS:<p>PDE4-IN-9, a potent PDE4 inhibitor, has an IC50 of 1.4μM (better than rolipram) and is effective in LPS-induced asthma/COPD and sepsis models.</p>Fórmula:C15H12N4O3SForma y color:SolidPeso molecular:328.35Carbonic anhydrase inhibitor 14
CAS:<p>CA inhibitor 14 blocks hCA I/II/IX/XII (K i of 1203/99.7/9.4/27.7 nM) and CDK2 (IC50: 20.3 μM), showing antitumor effects.</p>Fórmula:C18H17N7O2SForma y color:SolidPeso molecular:395.44Acarbose sulfate
CAS:<p>Acarbose sulfate is an anti-diabetic drug and is an inhibitor of alpha-glucosidase.</p>Fórmula:C25H45NO22SPureza:98%Forma y color:SolidPeso molecular:743.68VP3.15
CAS:<p>VP3.15 is an orally bioavailable and CNS-penetrant dual inhibitor of phosphodiesterase (PDE)7- GSK3 (IC50s: 1.59 μM and 0.88 μM for PDE7 and GSK-3).</p>Fórmula:C20H22N4OSPureza:98%Forma y color:SolidPeso molecular:366.48Indoleacetyl phenylalanine
CAS:<p>Indoleacetyl phenylalanine is an indole-acetyl-amino acid involved in regulating auxin activity.</p>Fórmula:C19H18N2O3Pureza:98%Forma y color:SolidPeso molecular:322.36hCAXII-IN-5
CAS:<p>hCAXII-IN-5, or compound 6o, is a potent, selective hCAXII inhibitor with Ki values: hCAI & II >10000, hCAIX 286.1, hCAXII 1.0 nM.</p>Fórmula:C23H22N2O4Forma y color:SolidPeso molecular:390.43BDM14471
CAS:<p>BDM14471 is a selective inhibitor of hydroxamate PfAM1.</p>Fórmula:C17H15FN2O3Pureza:98%Forma y color:SolidPeso molecular:314.31ZM223
CAS:<p>ZM223 is an inhibitor of NEDD8 activating enzyme (NAE).</p>Fórmula:C23H17F3N4O2S2Pureza:99.73%Forma y color:SolidPeso molecular:502.5320-HC-Me-Pyrrolidine
<p>20-HC-Me-Pyrrolidine is a potent Aster protein inhibitor that blocks the ability of Aster proteins to bind and transfer cholesterol.</p>Fórmula:C28H47NO2Pureza:99.99%Forma y color:SolidPeso molecular:429.68NCX899
CAS:<p>NCX899 shows inhibitory activity against angiotensin-converting enzyme (ACE) activity.</p>Fórmula:C23H33N3O8Pureza:98%Forma y color:SolidPeso molecular:479.52HIF-1α inhibitor-1
CAS:<p>HIF-1α inhibitor-1 is a HIF-1 alpha inhibitor.</p>Fórmula:C15H11N3O4Forma y color:SolidPeso molecular:297.27HM-50316
CAS:<p>HM-50316 is a High affinity FABP4 inhibitor (Ki < 1 nM).</p>Fórmula:C29H23ClN2O3SPureza:98%Forma y color:SolidPeso molecular:515.02MMPX
CAS:<p>calmodulin-sensitive cyclic GMP phosphodiesterase inhibitor</p>Fórmula:C12H18N4O3Pureza:98%Forma y color:SolidPeso molecular:266.3TDP1 Inhibitor-1
CAS:<p>TDP1 Inhibitor-1 is a potent inhibitor of Tyrosyl-DNA Phosphodiesterase 1 (TDP1) (IC50 of 7 μM).</p>Fórmula:C26H26N2O5Pureza:98%Forma y color:SolidPeso molecular:446.49Lith-O-Asp
CAS:<p>Lith-O-Asp is a sialytransferase (ST) inhibitor,(IC50s:12-37 μM).</p>Fórmula:C28H45NO6Forma y color:SolidPeso molecular:491.66Quinaprilat
CAS:<p>Quinaprilat inhibits angiotensin converting enzyme.</p>Fórmula:C23H26N2O5Pureza:98%Forma y color:Crystalline SolidPeso molecular:410.46Ro-15-2041
CAS:<p>Ro 15-2041 is a selective inhibitor of platelet phosphodiesterase, with antithrombotic properties.</p>Fórmula:C12H12BrN3OPureza:98%Forma y color:SolidPeso molecular:294.15Afegostat D-Tartrate
CAS:<p>Afegostat D-Tartrate: pharmacological chaperone, reversibly binds acid-β-glucosidase in ER with high affinity.</p>Fórmula:C10H19NO9Pureza:98%Forma y color:SolidPeso molecular:297.26Palmostatin B
CAS:<p>Palmostatin B is a modulator of Ras-signaling that acts by targeting acyl protein thioesterase 1 (APT1) and 2 (APT2) in cells.</p>Fórmula:C23H36O4Pureza:98%Forma y color:SolidPeso molecular:376.53Safusidenib
CAS:<p>Safusidenib, oral mutant IDH1 inhibitor, selectively targets IDH1R132H/C mutations with IC50 of 15/130 nM; impairs chondrosarcoma growth.</p>Fórmula:C25H18Cl3FN2O4Forma y color:SolidPeso molecular:535.78Lipoxygenin
CAS:<p>Lipoxygenin: IC50 of 5 μM inhibits 5-LO, hedgehog, TGF-β, activin A, BMP, Wnt signaling, and boosts cardiac marker TnnT in iPSCs.</p>Fórmula:C24H22N2O4Forma y color:SolidPeso molecular:402.44Vilazodone carboxylic acid
CAS:<p>Vilazodone carboxylic acid is a vilazodone metabolite observed in both urine and plasma.</p>Fórmula:C26H26N4O3Pureza:98%Forma y color:SolidPeso molecular:442.51Soluble epoxide hydrolase inhibitor
CAS:<p>Soluble epoxide hydrolase inhibitor is a soluble epoxide hydrolase inhibitor (human soluble epoxide hydrolase (h-sEH) with pIC50 of 8.4).</p>Fórmula:C18H12F5N5O3Pureza:98%Forma y color:SolidPeso molecular:441.31ATX inhibitor 14
CAS:<p>ATX inhibitor 14, an indole carbamate, potently blocks self-adhesive proteins (IC50: 0.41 nM), aiding fibrosis research.</p>Fórmula:C26H26Cl2N4O3SForma y color:SolidPeso molecular:545.48L-(-)-threo-3-Hydroxyaspartic acid
CAS:<p>L-(-)-threo-3-Hydroxyaspartic acid is an EAAT1-4 inhibitor/non-transportable EAAT5 inhibitor.</p>Fórmula:C4H7NO5Pureza:98%Forma y color:SolidPeso molecular:149.1Sp-Cyclic AMPS (sodium salt)
CAS:<p>Sp-cAMPS Na salt activates PKA I/II and competitively inhibits PDE3A (Ki: 47.6 μM), also binds PDE10 GAF (EC50: 40 μM).</p>Fórmula:C10H12N5NaO5PSForma y color:SolidPeso molecular:367.25ROR Modulator I
CAS:<p>ROR Modulator I is the first potent inverse agonist of the retinoid-related orphan receptor. It also has dual selectivity for RORβ and RORγt.</p>Fórmula:C26H20Cl2N2O4S2Pureza:98%Forma y color:SolidPeso molecular:559.48Enpp-1-IN-9
CAS:<p>Enpp-1-IN-9 inhibits ENPP1, cleaves numerous bonds in nucleotides/sugars; may advance cancer/infectious disease research.</p>Fórmula:C17H24N4O5SForma y color:SolidPeso molecular:396.46Dibefurin
CAS:<p>Dibefurin blocks calcineurin, a calcium-dependent enzyme, reducing T lymphocyte activation.</p>Fórmula:C18H16O8Forma y color:SolidPeso molecular:360.317-Biopterin
CAS:<p>7-Biopterin, a 7-substituted pterin, forms non-enzymatically and elevates in urine of hyperphenylalaninemics with PCBD mutations.</p>Fórmula:C9H11N5O3Forma y color:SolidPeso molecular:237.224-Desmethyl Istradefylline
CAS:<p>4-Desmethyl Istradefylline: a metabolite of Istradefylline, a strong, selective oral adenosine A2A receptor blocker, Ki 2.2 nM, used in Parkinson's.</p>Fórmula:C19H22N4O4Pureza:98%Forma y color:SolidPeso molecular:370.40LY 269415
CAS:<p>LY 269415 is an anti-inflammatory agent with antioxidant properties in vitro and could be beneficial as therapeutic agents in inflammatory arthritis.</p>Fórmula:C19H28N2O2SForma y color:SolidPeso molecular:348.5Prolyl Endopeptidase Inhibitor 1
CAS:<p>Prolyl Endopeptidase Inhibitor 1 is a potent inhibitor of prolyl endopeptidase (PEP; PE)(Ki : 15 nM) , has anti-amnesic effect.</p>Fórmula:C15H24N2O4Pureza:98%Forma y color:SolidPeso molecular:296.36Utibapril
CAS:<p>Utibapril is an inhibitor of angiotensin-converting enzyme (ACE) with antihypertensive activities.</p>Fórmula:C22H31N3O5SPureza:98%Forma y color:SolidPeso molecular:449.56Cgp 8065
CAS:<p>Cgp 8065 is a filaricidal compound, a dithiocarbamate-derivative of amoscanate.</p>Fórmula:C16H15N3O4S2Forma y color:SolidPeso molecular:377.44β-Amino Acid Imagabalin Hydrochloride
CAS:<p>β-Amino Acid Imagabalin Hydrochloride is the voltage-dependent calcium channel ligand for the α2δ subunit.</p>Fórmula:C9H20ClNO2Pureza:98%Forma y color:SolidPeso molecular:209.71Pancreatic lipase/Carboxylesterase 1-IN-1
CAS:<p>Compound 39 is a dual inhibitor of PL (IC50: 2.13 μM) and hCES1A (IC50: 0.055 μM).</p>Fórmula:C30H44O4Forma y color:SolidPeso molecular:468.67SHP504
CAS:<p>SHP504 is an inhibitor of SHP2 phosphatase and acts on SHP21-525 (IC50: 21 μM).</p>Fórmula:C23H15ClN4O4Forma y color:SolidPeso molecular:446.84Glucokinase activator 1
CAS:<p>Glucokinase activator 1 is a liver-directed glucokinase activator (EC50: 34 nM).</p>Fórmula:C27H20F2N2O7S2Pureza:98%Forma y color:SolidPeso molecular:586.58Ro 41-0960
CAS:<p>Ro 41-0960 is used as a reversible and orally-active COMT-inhibitor.</p>Fórmula:C13H8FNO5Pureza:98%Forma y color:SolidPeso molecular:277.2DNS-8254
CAS:<p>DNS-8254: Potent, selective PDE2 inhibitor, enhances memory (IC50=8 nM), effective in rat memory tests.</p>Fórmula:C18H15BrF3N5OPureza:98%Forma y color:SolidPeso molecular:454.24Enpp-1-IN-10
CAS:<p>Enpp-1-IN-10 inhibits ENPP1 with 3.866 μM Ki, useful in cancer research.</p>Fórmula:C13H12N6OSForma y color:SolidPeso molecular:300.34(3S,5R)-Fluvastatin sodium
CAS:<p>(3S,5R)-Fluvastatin sodium: synthetic HMG-CoA reductase inhibitor, IC50 8 nM, boosts vascular cell antioxidant defense.</p>Fórmula:C24H26FNNaO4Pureza:98%Forma y color:SolidPeso molecular:434.463Adenosine 5'-phosphosulfate (sodium salt)
CAS:<p>Adenosine 5'-phosphosulfate (sodium salt) (APS) is a key intermediate in sulphur metabolism and a substrate for adenosine 5'-phosphosulfate kinase (APSK).</p>Fórmula:C10H12N5Na2O10PSForma y color:SolidPeso molecular:471.24PDE2/PDE10-IN-1
CAS:<p>PDE2/PDE10-IN-1 is a inhibitor of phosphodiesterase 2 (PDE2) and PDE10(IC50s of 29 and 480 nM, respectively).</p>Fórmula:C15H10ClN5Pureza:98%Forma y color:SolidPeso molecular:295.73ALRT 1550
CAS:<p>ALRT 1550, a retinoic acid agent (RAR) agonist, is used potentially for the treatment of cervical carcinoma.</p>Fórmula:C23H32O2Forma y color:SolidPeso molecular:340.5MMG-0358
CAS:<p>MMG-0358 is a novel potent IDO1 inhibitor, showing low cytotoxicity and higher selectivity for IDO1 over TDO enzyme.</p>Fórmula:C8H6ClN3OForma y color:SolidPeso molecular:195.61DSHN
CAS:<p>DSHN activates SHP, boosting its mRNA and protecting it from ubiquitination and degradation.</p>Fórmula:C15H17NO5SPureza:98%Forma y color:SolidPeso molecular:323.36Liarozole dihydrochloride
CAS:<p>Liarozole dihydrochloride, an oral CYP450 inhibitor, blocks estrogen and androgens, targeting prostate cancer and skin disorders.</p>Fórmula:C17H15Cl3N4Pureza:98%Forma y color:SolidPeso molecular:381.69NEP-IN-2
CAS:<p>NEP-IN-2 is an inhibitor of neutral endopeptidase. It also is used in the research of proliferation in atherosclerosis, restenosis.</p>Fórmula:C16H23NO3S2Pureza:98%Forma y color:SolidPeso molecular:341.49Cycloguanil
CAS:<p>Cycloguanil is an antimalarial.</p>Fórmula:C11H14ClN5Pureza:98%Forma y color:SolidPeso molecular:251.72AHR-5333
CAS:<p>AHR-5333 an antiallergy agent.</p>Fórmula:C30H33F2NO4Pureza:98%Forma y color:SolidPeso molecular:509.58Gemlapodect
CAS:<p>Gemlapodect (RO554965), a phosphodiesterase 10A (PDE10A) inhibitor, is utilized in schizophrenia research.</p>Fórmula:C22H21N7O3Forma y color:SolidPeso molecular:431.45Indolapril hydrochloride
CAS:<p>Indolapril hydrochloride is a nonsulfhydryl angiotensin converting enzyme (ACE) inhibitor with antihypertensive activity.</p>Fórmula:C24H35ClN2O5Forma y color:SolidPeso molecular:467ML368
CAS:<p>ML368 is a selective inhibitor of CYP3A4.</p>Fórmula:C26H18N6OPureza:98%Forma y color:SolidPeso molecular:430.46Prinoxodan
CAS:<p>Prinoxodan is an inhibitor of phosphodiesterase.</p>Fórmula:C13H14N4O2Pureza:98%Forma y color:SolidPeso molecular:258.28BI 689648
CAS:<p>BI 689648 is a highly selective inhibitor of aldosterone synthase(CYP11B1 and CYP11B2 with IC50s of 310 and 2.1 nM, respectively).</p>Fórmula:C16H18N4O2Forma y color:SolidPeso molecular:298.34Asterriquinol D dimethyl ether
CAS:<p>Asterriquinol D dimethyl ether inhibits mouse myeloma (IC50: 28 μg/mL) and Tritrichomonas foetus.</p>Fórmula:C26H24N2O4Forma y color:SolidPeso molecular:428.48Theodrenaline
CAS:<p>Theodrenaline is a cardiac stimulant, also acts as an agent of anti-hypotensive together with cafedrine.</p>Fórmula:C17H21N5O5Pureza:98%Forma y color:SolidPeso molecular:375.38OMDM-4
CAS:<p>OMDM-4 is a selective and metabolically stable anandamide cellular uptake (ACU)inhibitor(Ki of 17.7 μM).</p>Fórmula:C29H43NO3Pureza:98%Forma y color:SolidPeso molecular:453.66(1S,2S,3R)-DT-061
CAS:<p>(1S,2S,3R)-DT-061 is an enantiomer of DT-061 which is an orally bioavailable activator of PP2A.</p>Fórmula:C25H23F3N2O5SForma y color:SolidPeso molecular:520.52SWE101
CAS:<p>SWE101 is a potent human and rat soluble epoxide hydrolase (sEH)-P inhibitor(IC50s of 4 μM and 2.8 μM, respectively).</p>Fórmula:C19H15Cl2NO3Pureza:98%Forma y color:SolidPeso molecular:376.23PSB069
CAS:<p>NTPDase inhibitor</p>Fórmula:C20H13ClN2NaO5SPureza:98%Forma y color:SolidPeso molecular:451.84FCE 28654
CAS:<p>FCE 28654 is a water-soluble acyl-CoA inhibitor.</p>Fórmula:C25H35N2O7PForma y color:SolidPeso molecular:506.53IDO1-IN-18
CAS:<p>IDO1-IN-18 (Compound 14) is a potent inhibitor of IDO1. IDO1-IN-18 has potential for cancer disease research.</p>Fórmula:C23H18F4N2O3Forma y color:SolidPeso molecular:446.39RORγt/DHODH-IN-2
CAS:<p>RORγt/DHODH-IN-2 (compound 1) is a potent dual RORγt/DHODH inhibitor that can be used in the study of inflammatory bowel disease (IBD).</p>Fórmula:C25H30N4OSForma y color:SolidPeso molecular:434.6Glyoxalase I inhibitor 1
CAS:<p>Glyoxalase I inhibitor 1 is a potent inhibitor of glyoxalase I (GLO1) (IC50: 26 nM).</p>Fórmula:C30H27FN6O4SForma y color:SolidPeso molecular:586.64(+)-Cembrene A
CAS:<p>(+)-Cembrene A, a nontoxic α-glucosidase inhibitor to human normal hepatocyte (LO2) cells, exhibits an IC50 value of 30.31 μM.</p>Fórmula:C20H32Forma y color:SolidPeso molecular:272.47hCAXII-IN-3
CAS:<p>hCAXII-IN-3 (Compound 6o) is a selective inhibitor of human carbonic anhydrase XII (hCAXII) (Ki: 10.0 nM).</p>Fórmula:C26H20BrN5O3SForma y color:SolidPeso molecular:562.44Pimobendan hydrochloride
CAS:<p>Pimobendan hydrochloride is a selective inhibitor of PDE3 (IC50: 0.32 μM).</p>Fórmula:C19H19ClN4O2Pureza:98%Forma y color:SolidPeso molecular:370.83UK-371804 HCl
CAS:<p>UK-371804 is a potent and selective urokinase-type plasmogen activator (uPA) inhibitor with excellent enzyme potency (Ki=10 nM) and selectivity profile (2700-</p>Fórmula:C14H17Cl2N5O4SPureza:98%Forma y color:SolidPeso molecular:422.29IDO/TDO-IN-1
CAS:<p>IDO/TDO-IN-1 is an orally active dual indoleamine-2,3-dioxygenase (IDO) and tryptophan 2,3-dioxygenase (TDO) inhibitor (IC50s: 9.7 and 47 nM).</p>Fórmula:C25H24FN5Pureza:98%Forma y color:SolidPeso molecular:413.49hDHODH-IN-9
CAS:<p>hDHODH-IN-9 is a potent hDHODH inhibitor, IC50=0.34 μM, toxic to MCF-7/A375 cells, promising for cancer research.</p>Fórmula:C21H21NO4Forma y color:SolidPeso molecular:351.4SCD1 inhibitor-1
CAS:SCD1 inhibitor-1 is a potent and liver-selective inhibitor of stearoyl-CoA desaturase-1 (SCD1).Fórmula:C21H23N3NaO3S2Pureza:98%Forma y color:SolidPeso molecular:452.54SQ 27786
CAS:<p>SQ 27786 is an inhibitor of ACE.</p>Fórmula:C23H25ClN4O7S2Pureza:98%Forma y color:SolidPeso molecular:569.05Win 58237
CAS:<p>Win 58237 is an inhibitor of cyclic nucleotide phosphodiesterase (PDE) (Ki: 170 nM for PDE V), with vasorelaxant activity.</p>Fórmula:C16H17N5OPureza:98%Forma y color:SolidPeso molecular:295.34IHVR-19029
CAS:<p>IHVR-19029: ER α-glucosidases I/II inhibitor, IC50 0.48μM; halts Ebola, Dengue, Rift Valley fever virus replication.</p>Fórmula:C23H45N3O5Forma y color:SolidPeso molecular:443.62BMS 961
CAS:<p>BMS961 is a potent and selective retinoic acid receptor gamma (RARγ) agonist (IC50: 30 nM).</p>Fórmula:C23H26FNO4Pureza:98%Forma y color:SolidPeso molecular:399.46GSK360A
CAS:<p>GSK360A is a novel prolyl hydroxylase (PHD) domain-containing enzyme inhibitor.</p>Fórmula:C17H17FN2O5Pureza:98%Forma y color:SolidPeso molecular:348.33HS80
CAS:<p>HS-80, a Fasnall enantiomer, selectively inhibits FASN, blocking lipid synthesis (IC50: 7.13 μM).</p>Fórmula:C19H22N4SPureza:98%Forma y color:SolidPeso molecular:338.47Senazodan
CAS:<p>Senazodan is a sensitiser of Ca2+, and shows inhibition effect on PDE III.</p>Fórmula:C15H14N4OPureza:98%Forma y color:SolidPeso molecular:266.3CFG920
CAS:<p>CFG920 is an oral CYP17 inhibitor that may reduce androgen production and inhibit growth of androgen-dependent tumors.</p>Fórmula:C14H13ClN4OForma y color:SolidPeso molecular:288.73L-5-BromoTryptophan
CAS:<p>L-5-BromoTryptophan (5-BrW) is an analog of the tryptophan (Trp) effector and inhibits the gelation of hemoglobin S.</p>Fórmula:C11H11BrN2O2Pureza:99.86%Forma y color:SolidPeso molecular:283.12

