Metabolismo
Los inhibidores del metabolismo son compuestos que interfieren con las vías metabólicas, alterando la producción y utilización de energía dentro de las células. Estos inhibidores se utilizan para estudiar la regulación del metabolismo, el papel de las vías metabólicas en enfermedades como el cáncer y la diabetes, y para desarrollar nuevas estrategias terapéuticas. Los inhibidores del metabolismo pueden dirigirse a diversas enzimas y procesos involucrados en la glucólisis, la oxidación de ácidos grasos y otras funciones metabólicas. En CymitQuimica, ofrecemos una amplia gama de inhibidores del metabolismo de alta calidad para apoyar su investigación en bioquímica, trastornos metabólicos y desarrollo de fármacos.
Subcategorías de "Metabolismo"
- AhR(41 productos)
- Aminopeptidasa(67 productos)
- CETP(18 productos)
- Anhídrido carbónico(177 productos)
- Caseína quinasa(130 productos)
- DHFR(32 productos)
- Descarboxilasa(4 productos)
- Deshidrogenasa(267 productos)
- FAAH(63 productos)
- FXR(58 productos)
- Factor Xa(80 productos)
- Ácido graso sintasa(32 productos)
- Ferroptosis(215 productos)
- GR(3 productos)
- GSNOR(3 productos)
- Glucoquinasa(53 productos)
- HIF / HIF Prolilhidroxilasa(142 productos)
- HMG-CoA reductasa(32 productos)
- Hidroxilasa(30 productos)
- IDO(82 productos)
- LDL(8 productos)
- Lipasa(96 productos)
- Lípido(59 productos)
- Lipoxigenasa(124 productos)
- MAO(87 productos)
- MPO(2 productos)
- NAMPT(36 productos)
- P450(6 productos)
- PAI-1(25 productos)
- PDE(166 productos)
- PED(1 productos)
- PKM(15 productos)
- PPAR(164 productos)
- Fosfolipasa(82 productos)
- ROR(42 productos)
- Receptor de retinoides(29 productos)
- SGK(11 productos)
- Tiorredoxina(12 productos)
- Transferasa(30 productos)
- Transportador(42 productos)
- UGT(4 productos)
- Inhibidores de la xantina oxidasa (XO)(9 productos)
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Se han encontrado 8595 productos de "Metabolismo"
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CCR1/5/8 activator 1
CAS:<p>CCR1/5/8 activator 1 is a cytoplasmic phospholipase A inhibitor with antifungal activity.</p>Fórmula:C10H9NOPureza:>99.99%Forma y color:SolidPeso molecular:159.18Norfenfluramine hydrochloride
CAS:<p>Norfenfluramine hydrochloride ((±)-Norfenfluramine hydrochloride) is the primary metabolite of Fenfluramine, resulting from its N-dealkylation. It serves as a potent anorectic agent and can modulate serotonin neurotransmission. In addition, Norfenfluramine hydrochloride exhibits sedative effects following acute administration.</p>Fórmula:C10H13ClF3NForma y color:SolidPeso molecular:239.67ChAT IN-1
<p>ChAT IN-1 is a selective inhibitor of Choline Acetyltransferase (ChAT) that is utilized in studying mechanisms related to non-neuronal ChAT overexpression in cancers such as colon cancer and lung cancer, as well as in research concerning Alzheimer's disease (AD).</p>Fórmula:C21H15N3O2Forma y color:SolidPeso molecular:341.36PKM2 activator 6
<p>Compound Z10 (PKM2 activator 6) serves as both a PKM2 activator and a PDK1 inhibitor, exhibiting dissociation constants (K D ) of 121 μM and 19.6 μM,</p>Forma y color:Odour SolidAcyl coenzyme A synthetase
CAS:<p>ACS activates fatty acids for lipid metabolism and the TCA cycle.</p>Forma y color:SolidRubratoxin A
CAS:<p>Rubratoxin A is a classical mycotoxin used as a PP2A-specific inhibitor.</p>Fórmula:C26H32O11Pureza:98%Forma y color:SolidPeso molecular:520.531EDDA
CAS:<p>Ethylenediaminediacetic acid is derived from two molecules of glycine linked by amines.</p>Fórmula:C6H12N2O4Forma y color:SolidPeso molecular:176.1718:0,18:1 PS sodium
CAS:<p>18:0,18:1 PS sodium, a lipid found in synaptic vesicles and cholesterol, serves a role in metabolic research [1].</p>Fórmula:C42H79NNaO10PForma y color:SolidPeso molecular:812.04cMCoFx1
CAS:<p>cMCoFx1 is an effective and selective FXIIa cyclic peptide inhibitor. It exhibits high binding affinity for FXIIa (KD: 900 pM) and potent inhibitory activity (Ki: 370 pM). cMCoFx1 effectively suppresses the intrinsic coagulation pathway, demonstrates high stability in serum, and shows no cytotoxicity.</p>Fórmula:C146H232N52O44S6Forma y color:SolidPeso molecular:3612.12FXR agonist 11
CAS:<p>FXR agonist11 (Compound 14) is an FXR activator with an EC50 of 1.2 μM and a maximal effect of 73.7%. It significantly increases GSH levels in the liver and is used to study drug-induced liver injury.</p>Fórmula:C18H16N2O5Forma y color:SolidPeso molecular:340.33Tetracosanoyl-sulfatide
CAS:<p>C24 3'-sulfo Galactosylceramide is a key myelin sulfatide, high in leukodystrophy patients, non-immunogenic compared to C24:1 variant.</p>Fórmula:C48H93NO11SForma y color:SolidPeso molecular:892.32LH10
<p>LH10 is an FXR agonist based on fexaramine, with an EC50 of 0.14 μM. It offers hepatoprotective effects, mitigating conditions such as cholestasis induced by alpha naphthylisothiocyanate (ANIT), acute liver injury caused by APAP, and non-alcoholic steatohepatitis (NASH).</p>Fórmula:C34H33N3O2Forma y color:SolidPeso molecular:515.642-(2',3',4'-Trihydroxybutyl)quinoxaline
CAS:<p>2-(2',3',4'-Trihydroxybutyl)quinoxaline is a food metabolite.</p>Fórmula:C12H14N2O3Pureza:98%Forma y color:SolidPeso molecular:234.25Anticancer agent 260
CAS:<p>Anticanceragent 260 (Compound 3g/4d) is an orally effective anticancer agent that inhibits the proliferation of cancer cells HCT-116, MIA-PaCa2, and MDA-MB231, with IC50 values of 98.7, 81.0, and 77.2 µg/mL, respectively. It also promotes ulcer formation and lipid peroxidation, and exhibits anti-inflammatory and analgesic activities.</p>Fórmula:C14H11N3OForma y color:SolidPeso molecular:237.26TSPO/Carbonic Anhydrase Modulator 1
<p>TSPO/Carbonic Anhydrase Modulator 1 (Compound 3) acts as a dual modulator of mitochondrial translocator protein and carbonic anhydrase, with a TSPOKi of 1.340 μM and a CAVII KA of 10.7 μM. It enhances neurosteroid production, increases BDNF gene expression, and demonstrates neuroprotective activity.</p>Fórmula:C35H51N3O3Forma y color:SolidPeso molecular:561.798LZ-007
CAS:<p>LZ-007 is an agonist of the Farnesoid X receptor (FXR), with an EC50 of 51 nM as determined by TR-FRET assay, and an EC50 of 76 nM in HepG2 cells. It exhibits favorable pharmacokinetic properties in SD rats and can improve metabolic dysfunction-associated steatohepatitis induced by high-fat diets and CCl4 in mice.</p>Fórmula:C27H29F3N2O5Forma y color:SolidPeso molecular:518.535(S)-HPETE
CAS:<p>5(S)-HpETE is a PUFA made by 5-LO from arachidonic acid, metabolized into LTA4, a key leukotriene precursor.</p>Fórmula:C20H32O4Forma y color:SolidPeso molecular:336.4725β-Androstan-3β-ol-17-one
CAS:<p>5β-Androstan-3β-ol-17-one (3β-Etiocholanolone; 5β-Epiandrosterone), a 5β-reduced steroid and a significant metabolic derivative of dehydroepiandrosterone (DHEA</p>Fórmula:C19H30O2Forma y color:SolidPeso molecular:290.44DSPE-PEG1000-R6H4
<p>DSPE-PEG1000-R6H4 is a PEG compound comprised of DSPE and pH-responsive cell-penetrating peptide (R6H4), designed for pH-sensitive anti-cancer drug delivery. It is utilized in drug delivery applications.</p>Forma y color:Odour Solidα-Glucosidase-IN-76
<p>α-Glucosidase-IN-76 (Compound 4r) is an inhibitor of α-glucosidase, with an IC50 of 5.44 μM. It can clear ABTS+ free radicals, with a TEAC value of 0.49. Additionally, α-Glucosidase-IN-76 inhibits the proliferation of T24 bladder cancer cells, with an IC50 of 1.74 μM.</p>Fórmula:C21H24N4O10Forma y color:SolidPeso molecular:492.44PROTAC NAMPT Degrader-1
<p>PROTACNAMPT Degrader-1 is an effective NAMPT-targeting PROTAC with a DC50 value of 217 nM. It exhibits antiproliferative activity, with an IC50 value of 0.12 μM against A2780 cells.</p>Fórmula:C57H69N13O8S2Peso molecular:1127.48335GF 109
CAS:<p>GF 109 is an inhibitor of ACE.</p>Fórmula:C53H74N14O13Pureza:98%Forma y color:SolidPeso molecular:1115.24APOL1-IN-2
CAS:<p>APOL1-IN-2 (Compound 467) acts as an inhibitor of apolipoprotein L1 (APOL1). It effectively reduces HEK293 cell death induced by APOL1 G2/G1, with EC50 values of 4.74 nM and 14.3 nM, respectively. Additionally, APOL1-IN-2 decreases the mortality of trypanosomes triggered by APOL1 G2/G1/G0, with EC50 values of 2.24, 6.03, and 3.72 nM, respectively.</p>Fórmula:C28H30ClF3N4O5Forma y color:SolidPeso molecular:595.01Fumonisin B2
CAS:<p>Fumonisin B2, from Fusarium moniliforme in grains, blocks ceramide synthase, disrupting sphingolipid biosynthesis.</p>Fórmula:C34H59NO14Pureza:98%Forma y color:SolidPeso molecular:705.83Lexacalcitol
CAS:<p>Lexacalcitol is a potent compound, 100x more effective than 1alpha,25-(OH)2D3 in antiproliferation and cell differentiation tests.</p>Fórmula:C29H48O4Pureza:98%Forma y color:SolidPeso molecular:460.69Norpropranolol hydrochloride
CAS:<p>Norpropranolol hydrochloride is the active metabolite of Propranolol.</p>Fórmula:C13H16ClNO2Forma y color:SolidPeso molecular:253.73Etavopivat
CAS:<p>Etavopivat activates PKR in RBCs; taken orally, prevents sickling.</p>Fórmula:C22H23N3O6SForma y color:SolidPeso molecular:457.5Terpendole C
CAS:<p>Terpendole C, an indole diterpene from A. yamanashiensis, inhibits ACAT with IC50 of 2.1 μM in rats, 0.46 μM in J774 cells, non-toxic.</p>Fórmula:C32H41NO5Forma y color:SolidPeso molecular:519.682Secaubryenol
CAS:<p>Secaubryenol is a 3,4-secocycloartane triterpenes isolated from Coussarea macrophylla.</p>Fórmula:C30H48O3Pureza:98%Forma y color:SolidPeso molecular:456.74-Hydroxybenzoic acid-d4
CAS:<p>4-Hydroxybenzoicacid-d4 is a deuterated form of 4-Hydroxybenzoicacid, which is a phenolic derivative of benzoic acid. It is effective in inhibiting most Gram-positive bacteria and some Gram-negative bacteria with an IC50 of 160 μg/mL.</p>Fórmula:C7H6O3Forma y color:SolidPeso molecular:142.15Purpactin A
CAS:<p>Purpactin A is a useful organic compound for research related to life sciences. The catalog number is T126026 and the CAS number is 133806-59-4.</p>Fórmula:C23H26O7Forma y color:SolidPeso molecular:414.4543α-Hydroxysteroid dehydrogenase
CAS:<p>3α-Hydroxysteroid dehydrogenase (3α-HSD), encoded by the AKR1C4 gene, is responsible for catalyzing the transformation of 3-ketosteroids into 3α-hydroxy</p>Forma y color:SolidDSPE-PEG2000-R8
<p>DSPE-PEG2000-R8 is a PEGylated compound composed of DSPE and the cell-penetrating peptide (R8). It can be applied in drug delivery.</p>Forma y color:Odour Solidα-Glucosidase-IN-44
<p>α-Glucosidase-IN-44 (compound IT4) is an α-glucosidase inhibitor with an IC50 value of 2.35 μM. This compound is orally active and has the ability to reduce fasting blood glucose levels in diabetic mice.</p>Fórmula:C23H21N3O3SPeso molecular:419.13036PAPA NONOate
CAS:<p>PAPA NONOate is a pH-regulated NO donor.PAPA NONOate has potential antitumor activity and can be used to study diabetic wound healing disorders.</p>Fórmula:C6H16N4O2Pureza:98%Forma y color:SolidPeso molecular:176.22POPG sodium salt
CAS:<p>POPG sodium salt is a phospholipid and a component of biological membranes and can be used to study the function of biological membranes.</p>Fórmula:C40H76NaO10PPureza:98.21%Forma y color:SolidPeso molecular:770.99Dorzolamide
CAS:<p>Dorzolamide is an anti-glaucoma agent and is a carbonic anhydrase inhibitor.</p>Fórmula:C10H16N2O4S3Pureza:98%Forma y color:White Or Almost White Crystalline PowderPeso molecular:324.44α-Glucosidase-IN-48
<p>α-Glucosidase-IN-48 (compound 9) is a potent inhibitor of α-Glucosidase, with an IC50 of 1.30 μM.</p>Fórmula:C15H9Cl2N5O3SPeso molecular:408.98032PDE4-IN-13
<p>PDE4-IN-13 is a phosphodiesterase 4 (PDE4) inhibitor exhibiting anti-inflammatory and antioxidant activities, with an half maximal inhibitory concentration (</p>Fórmula:C20H20O5Forma y color:SolidPeso molecular:340.37β-Tetralone
CAS:<p>β-Tetralone (2-Tetralone) is a vital drug synthesis precursor with complex pharmacological properties in combating neurological disorders. Cost-effective and quality-assured.</p>Fórmula:C10H10OPureza:97.26% - 99.18%Forma y color:Clear To Yellow LiquidPeso molecular:146.19TDI-11055
<p>TDI-11055 is a chromatin reader 11-19 leukemia inhibitor and can be used to study acute myeloid leukemia (AML).</p>Fórmula:C22H24N6OPureza:98.48%Forma y color:SolidPeso molecular:388.472-(Isopentylamino)naphthalene-1,4-dione
CAS:<p>2-(Isopentylamino)naphthalene-1,4-dione: a vitamin K analog inhibiting spasms and seizures in mice with various ED50 values.</p>Fórmula:C15H17NO2Forma y color:SolidPeso molecular:243.306Saccharopine
CAS:<p>L-Saccharopine is a product of the breakdown of essential amino acid Lysine.</p>Fórmula:C11H20N2O6Forma y color:SolidPeso molecular:276.29Allotetrahydrocortisol
CAS:<p>Allotetrahydrocortisol (5a-Tetrahydrocortisol) is a metabolite of Cortisol. Cortisol is the main glucocorticoid in human.</p>Fórmula:C21H34O5Pureza:98%Forma y color:SolidPeso molecular:366.491,1,3-Tribromoacetone
CAS:<p>1,1,3-Tribromoacetone (1,1,3-tribromo-2-propanone) is an impurity of methotrexate.</p>Fórmula:C3H3Br3OPureza:98%Forma y color:SolidPeso molecular:294.77α-2,6-Sialyltransferase (Pd26ST)
CAS:<p>Alpha-2,6-Sialyltransferase (Pd26ST) efficiently catalyzes the sialylation of both terminal and internal galactose and N-acetylgalactosamine residues, resulting</p>Forma y color:SolidPorfimer Sodium
CAS:<p>Porfimer sodium, a sodium salt with photodynamic properties, targets tumor cells and induces cytotoxicity with 630 nm laser activation.</p>Fórmula:C68H74N8O11Forma y color:SolidPeso molecular:1179.385DSPE-PEG2000-CCK8
<p>DSPE-PEG2000-CCK8 is a PEG compound comprising DSPE and Cholecystokinin-8 (CCK8). Cholecystokinin-8 exhibits peptide activity responsible for regulating gallbladder contractions and digestive system functions. DSPE-PEG2000-CCK8 is applicable for drug delivery.</p>Forma y color:Odour SolidSKI2852
CAS:<p>SKI2852 is an 11β-HSD1 inhibitor that improves metabolic syndrome in diabetic mouse models.</p>Fórmula:C27H34FN5O4SPureza:99.89%Forma y color:SolidPeso molecular:543.65NoxA1ds
CAS:<p>Selective NOX1 inhibitor; IC50 at 20 nM; spares NOX2/4/5 and xanthine oxidase; reduces HT-29 O2- and hinders VEGF-induced cell migration.</p>Fórmula:C50H88N14O15Pureza:98%Forma y color:SolidPeso molecular:1125.33
