
Metabolismo
Los inhibidores del metabolismo son compuestos que interfieren con las vías metabólicas, alterando la producción y utilización de energía dentro de las células. Estos inhibidores se utilizan para estudiar la regulación del metabolismo, el papel de las vías metabólicas en enfermedades como el cáncer y la diabetes, y para desarrollar nuevas estrategias terapéuticas. Los inhibidores del metabolismo pueden dirigirse a diversas enzimas y procesos involucrados en la glucólisis, la oxidación de ácidos grasos y otras funciones metabólicas. En CymitQuimica, ofrecemos una amplia gama de inhibidores del metabolismo de alta calidad para apoyar su investigación en bioquímica, trastornos metabólicos y desarrollo de fármacos.
Subcategorías de "Metabolismo"
- AhR(41 productos)
- Aminopeptidasa(67 productos)
- CETP(18 productos)
- Anhídrido carbónico(177 productos)
- Caseína quinasa(130 productos)
- DHFR(32 productos)
- Descarboxilasa(4 productos)
- Deshidrogenasa(267 productos)
- FAAH(63 productos)
- FXR(58 productos)
- Factor Xa(80 productos)
- Ácido graso sintasa(32 productos)
- Ferroptosis(215 productos)
- GR(3 productos)
- GSNOR(3 productos)
- Glucoquinasa(53 productos)
- HIF / HIF Prolilhidroxilasa(142 productos)
- HMG-CoA reductasa(32 productos)
- Hidroxilasa(30 productos)
- IDO(82 productos)
- LDL(8 productos)
- Lipasa(96 productos)
- Lípido(59 productos)
- Lipoxigenasa(124 productos)
- MAO(87 productos)
- MPO(2 productos)
- NAMPT(36 productos)
- P450(6 productos)
- PAI-1(25 productos)
- PDE(165 productos)
- PED(1 productos)
- PKM(15 productos)
- PPAR(164 productos)
- Fosfolipasa(82 productos)
- ROR(42 productos)
- Receptor de retinoides(29 productos)
- SGK(11 productos)
- Tiorredoxina(12 productos)
- Transferasa(30 productos)
- Transportador(42 productos)
- UGT(4 productos)
- Inhibidores de la xantina oxidasa (XO)(9 productos)
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Se han encontrado 8597 productos de "Metabolismo"
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Quizalofop
CAS:<p>Quizalofop (Xylafop) is a reagent of biochemical.</p>Fórmula:C17H13ClN2O4Pureza:97.14%Forma y color:SolidPeso molecular:344.75ICMT-IN-52
CAS:<p>ICMT-IN-52 (compound 44) serves as an ICMT inhibitor with an IC50 value of 0.052 μM [1].</p>Fórmula:C21H26FNOForma y color:SolidPeso molecular:327.44CAY10435
CAS:<p>CAY10435, a β-ketooxazapyridine and selective FAAH inhibitor, exhibits antimicrobial properties. It binds non-competitively to the FAAH of Dictyostelium discoideum, demonstrating a Kd value of 0.57 nM [1] [2].</p>Fórmula:C18H26N2O2Forma y color:SolidPeso molecular:302.41LNP Lipid-8
CAS:<p>LNP Lipid-8 (11-A-M), an ionizable lipid, is utilized in lipid nanoparticles (LNP) for siRNA delivery to T cells without ligand targeting. When loaded with GFP siRNA (siGFP), it significantly silences the GFP gene in a mouse model [1].</p>Fórmula:C42H71NO7Forma y color:SolidPeso molecular:702.02DHODH-IN-22
CAS:<p>DHODH-IN-22: potent, selective DHODH inhibitor, orally active, IC50: 0.3 nM, for AML research.</p>Fórmula:C21H21ClF4N6O5Forma y color:SolidPeso molecular:548.88Eucalyptacid A
CAS:<p>Eucalyptacid A, a metabolite with antifungal properties, demonstrates efficacy against Alternaria solani, displaying minimum inhibitory concentrations (MIC)</p>Fórmula:C17H32O5Forma y color:SolidPeso molecular:316.43GPX4-IN-2
CAS:<p>GPX4-IN-2 is a potent inhibitor of GPX4, exhibiting antiproliferative activity. It holds potential for cancer research applications.</p>Fórmula:C30H40N2OForma y color:SolidPeso molecular:444.65OSMI-1
CAS:<p>OSMI-1: cell-permeable OGT inhibitor, blocks O-GlcNAcylation (IC50: 2.7 μM), no effect on other cell glycans.</p>Fórmula:C28H25N3O6S2Pureza:96.79% - 99.39%Forma y color:SolidPeso molecular:563.64JTT 551
CAS:<p>JTT 551: Selective PTP1B inhibitor for type 2 diabetes research; Ki=0.22μM for PTP1B, 9.3μM for TCPTP.</p>Fórmula:C34H43N3O3S2Pureza:98%Forma y color:SolidPeso molecular:605.85CYP17-IN-1
CAS:<p>CYP17-IN-1 is an effective oral inhibitor of CYP17 that can inhibit CYP17 in rats and humans with IC50 of 15.8 and 20.1 nM.</p>Fórmula:C18H17FN2SPureza:99.14% - 99.83%Forma y color:SolidPeso molecular:312.4Anticancer agent 121
CAS:<p>Anticancer agent 121, a human lactate dehydrogenase A (hLDHA) inhibitor, exhibits potent anticancer activities, suitable for use in anticancer research [1].</p>Fórmula:C19H18N2O3SForma y color:SolidPeso molecular:354.42Yonkenafil
CAS:<p>Yonkenafil, a PDE5 inhibitor, may reduce stroke damage and aid in Alzheimer's treatment.</p>Fórmula:C24H33N5O4SForma y color:SolidPeso molecular:487.61N-Stearoyl Taurine
CAS:<p>N-Arachidonoyl dopamine (NADA) and N-Arachidonoyl serine (ARA-S), among various arachidonoyl amino acids, have been extracted from bovine brain, while a novel series of fatty acyl amides of taurine were unearthed in rat brain through mass spectral lipidomic analysis, indicating the discovery of a new class of compounds also located in the kidney. These compounds are known to activate members of the transient receptor potential (TRP) family of calcium channels. Notably, N-Stearoyl taurine emerges as a significant amino-acyl endocannabinoid identified in rat brain lipidomics profiling.</p>Fórmula:C20H41NO4SForma y color:SolidPeso molecular:391.61GSK3987
CAS:<p>GSK3987 is an LXR ligand. GSK3987 recruits the steroid receptor coactivator-1 to human LXRalpha and LXRbeta with EC50s of 40 nM.</p>Fórmula:C24H20N2O3Pureza:99.92%Forma y color:SolidPeso molecular:384.43ICMT-IN-53
CAS:<p>ICMT-IN-53 (compound 12) is an ICMT inhibitor exhibiting an IC50 of 0.96 μM, alongside favorable PAMPA permeability and antiproliferative properties.</p>Fórmula:C26H36FN3Forma y color:SolidPeso molecular:409.58PF-04937319
CAS:<p>PF-04937319 activates glucokinase (EC50=154.4μM) with low hypoglycemia risk, researched for type 2 diabetes treatment.</p>Fórmula:C22H20N6O4Pureza:99.89%Forma y color:SolidPeso molecular:432.43BMS-795311
CAS:<p>Potent CETP inhibitor, boosts HDL-C levels, orally active; IC50=4nM.</p>Fórmula:C33H23F10NO3Forma y color:SolidPeso molecular:671.52VT-1598 tosylate
CAS:<p>VT-1598 tosylate is a selective, orally active antifungal compound that targets CYP51. It demonstrates efficacy against C. auris.</p>Fórmula:C38H28F4N6O5SForma y color:SolidPeso molecular:756.72ICMT-IN-39
CAS:<p>ICMT-IN-39, also known as compound 18, functions as an inhibitor of ICMT with an IC50 value of 0.031 µM [1].</p>Fórmula:C22H29NOForma y color:SolidPeso molecular:323.47ICMT-IN-44
CAS:<p>ICMT-IN-44 (compound 23) serves as an ICMT inhibitor with an IC50 value of 0.167 μM [1].</p>Fórmula:C24H33NOForma y color:SolidPeso molecular:351.52

