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Metabolismo

Metabolismo

Los inhibidores del metabolismo son compuestos que interfieren con las vías metabólicas, alterando la producción y utilización de energía dentro de las células. Estos inhibidores se utilizan para estudiar la regulación del metabolismo, el papel de las vías metabólicas en enfermedades como el cáncer y la diabetes, y para desarrollar nuevas estrategias terapéuticas. Los inhibidores del metabolismo pueden dirigirse a diversas enzimas y procesos involucrados en la glucólisis, la oxidación de ácidos grasos y otras funciones metabólicas. En CymitQuimica, ofrecemos una amplia gama de inhibidores del metabolismo de alta calidad para apoyar su investigación en bioquímica, trastornos metabólicos y desarrollo de fármacos.

Subcategorías de "Metabolismo"

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Se han encontrado 8625 productos de "Metabolismo"

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  • DH376
    Targetmol
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    DH376

    CAS:
    <p>DH376 inhibits DAGLα in a time and dose dependent manner in mouse brain. DH376 shows picomolar activity.</p>
    Fórmula:C31H28F2N4O3
    Forma y color:Solid
    Peso molecular:542.58

    Ref: TM-T27161

  • Calcipotriol Impurity C
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    Calcipotriol Impurity C

    CAS:
    <p>Calcipotriol Impurity C is the impurity of Calcipotriol. Calcipotriol is a VDR-like receptors ligand.</p>
    Fórmula:C27H40O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:412.614

    Ref: TM-T13590

  • AChE/hCA I-IN-1
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    AChE/hCA I-IN-1

    CAS:
    <p>AChE/hCA I-IN-1 (Compound L3) is an inhibitor of acetylcholinesterase (AChE) and carbonic anhydrase (CA), effectively inhibiting AChE, hCA I, and hCA II with IC50 values of 302 nM, 265 nM, and 283 nM, respectively.</p>
    Fórmula:C13H9BrNNaO4S
    Forma y color:Solid
    Peso molecular:378.174

    Ref: TM-T204128

  • LXRβ agonist-3
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    LXRβ agonist-3

    CAS:
    <p>LXRβ agonist-3 is a potent and selective LXRβ (liver X receptor β) agonist (EC50: 0.095 μM).</p>
    Fórmula:C30H33N3O6S
    Forma y color:Solid
    Peso molecular:563.66

    Ref: TM-T63989

  • Logo de CymitQuimica
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    PDE4-IN-12

    <p>PDE4-IN-12 is a potent and safe PDE4 ubiquitous inhibitor that acts on PDE4 (IC50: 3.5 nM, SI: 2.71) and PDE7 (IC50: 15 nM, SI: 4.27).</p>
    Fórmula:C34H35NO6
    Forma y color:Solid
    Peso molecular:553.64

    Ref: TM-T63912

  • Darlifarnib
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    Darlifarnib

    CAS:
    <p>Darlifarnib (Compound (S)-058) is an inhibitor of farnesyl transferase and geranylgeranyltransferase, with IC50 values of ≤ 10 nM and &gt; 1000 nM, respectively. It exhibits high metabolic stability in human and mouse liver microsomes, with a half-life of over 100 minutes.</p>
    Fórmula:C29H20N6O
    Forma y color:Solid
    Peso molecular:468.509

    Ref: TM-T206317

  • FXR agonist 12
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    FXR agonist 12

    CAS:
    <p>FXR agonist12 (Compound C7) is an orally active FXR agonist. It downregulates bile acid synthesis-related genes and upregulates bile acid transport-related genes in HepG2 cells. FXR agonist12 alleviates ANIT-induced cholestasis and reduces liver damage and fibrosis in a mouse model of NASH.</p>
    Fórmula:C26H44O3
    Forma y color:Solid
    Peso molecular:404.626

    Ref: TM-T205709

  • Logo de CymitQuimica
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    L-690330 hydrate

    <p>L-690330 hydrate inhibits IMPase; Ki: 0.30 μM (human), 0.42 μM (bovine cortex); 0.27 μM (recom. human), 0.19 μM (bovine).</p>
    Fórmula:C8H14O9P2
    Forma y color:Solid
    Peso molecular:316.14

    Ref: TM-T60820

  • Logo de CymitQuimica
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    EB-0156

    <p>EB-0156: potent ER α-glucosidase inhibitor, IC50 of 0.0479/ &lt;0.001 μM, N-substituted valerian, broad-spectrum antiviral potential.</p>
    Fórmula:C21H32N6O7
    Forma y color:Solid
    Peso molecular:480.51

    Ref: TM-T63170

  • Retezorogant
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    Retezorogant

    CAS:
    <p>Retezorogant is a retinoic acid receptor-related orphan receptor gamma (RORγ) antagonist.</p>
    Fórmula:C23H33ClN2O3
    Forma y color:Solid
    Peso molecular:420.97

    Ref: TM-T62242

  • Nomelidine
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    Nomelidine

    CAS:
    Nomelidine, the active N-demethylated metabolite of zimelidine, has been used as an antidepressant and analgesic.
    Fórmula:C15H15BrN2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:303.20

    Ref: TM-T28186

  • (-)-Mesembrine
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    (-)-Mesembrine

    CAS:
    <p>Mesembrine is a serotonin reuptake inhibitor and is also a weak inhibitor of the enzyme phosphodiesterase 4 (PDE4).</p>
    Fórmula:C17H23NO3
    Forma y color:Solid
    Peso molecular:289.37

    Ref: TM-T28019

  • Logo de CymitQuimica
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    CYP2C1/CYP2C19-IN-2

    <p>CYP2C1/CYP2C19-IN-2 is a potent inhibitor of CYP2C9/CYP2C19 without liver toxicity or genotoxicity and can be used to study Zika virus (ZIKV) infection.</p>
    Fórmula:C27H28N2O6S
    Forma y color:Solid
    Peso molecular:508.59

    Ref: TM-T63495

  • Zaragozic acid C
    Targetmol
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    Zaragozic acid C

    CAS:
    <p>Zaragozic acid C is an effective inhibitor of squalene synthase.</p>
    Fórmula:C40H50O14
    Pureza:98%
    Forma y color:Solid
    Peso molecular:754.82

    Ref: TM-T24710

  • Nampt-IN-15
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    Nampt-IN-15

    CAS:
    Nampt-IN-15 (Example 3) is a Nampt inhibitor that exhibits cytotoxic effects on various cell lines, including BxPC-3, HepG2, L540cy, and MOLM-13. The respective IC50 values for these cell lines are 38.5 nM, 8 nM, 8.5 nM, and 7 nM.
    Fórmula:C24H30N4O2
    Forma y color:Solid
    Peso molecular:406.52

    Ref: TM-T201167

  • SAL-0010042
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    SAL-0010042

    CAS:
    <p>SAL-0010042 is an inhibitor of Plasmodium phosphodiesterase β (PDEβ), effectively blocking the hydrolysis of cAMP and cGMP in gametocytes with an IC50 of 48.9 nM, thereby activating PKG and inhibiting the growth and development of Plasmodium (IC50s for 3D7 and Dd2 are 142 nM and 218 nM, respectively). It also inhibits hPDE5 and hPDE6 with IC50 values of 632 nM and 73 nM, respectively.</p>
    Fórmula:C15H15FN4O
    Forma y color:Solid
    Peso molecular:286.304

    Ref: TM-T204533

  • FXR/CES2 modulator 1
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    FXR/CES2 modulator 1

    CAS:
    <p>Compound LE-77, known as FXR/CES2 modulator 1, functions as a dual regulator that activates FXR and inhibits CES2. It effectively mitigates the intestinal toxicity of irinotecan.</p>
    Fórmula:C27H21Cl2NO5
    Forma y color:Solid
    Peso molecular:510.36

    Ref: TM-T200901

  • ABD957
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    ABD957

    CAS:
    <p>ABD957: covalent ABHD17 depalmitoylases inhibitor, IC50 0.21µM for ABHD17B, blocks N-Ras, halts NRAS-mutant AML cell growth.</p>
    Fórmula:C27H36F3N7O5S
    Forma y color:Solid
    Peso molecular:627.68

    Ref: TM-T73481

  • Logo de CymitQuimica
    Targetmol
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    α-Glucosidase-IN-13

    <p>α-Glucosidase-IN-13 is an inhibitor of α-glucosidase (IC50: 5.69 μM).</p>
    Fórmula:C25H28N4O3S2
    Forma y color:Solid
    Peso molecular:496.64

    Ref: TM-T63361

  • Logo de CymitQuimica
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    HIF-1α-IN-4

    <p>HIF-1α-IN-4 is an inhibitor of HIF-1α with IC50 of 24 nM in HEK293T cells which has potential antitumor effects.</p>
    Fórmula:C16H12N2O3
    Forma y color:Solid
    Peso molecular:280.28

    Ref: TM-T60524