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Metabolismo

Metabolismo

Los inhibidores del metabolismo son compuestos que interfieren con las vías metabólicas, alterando la producción y utilización de energía dentro de las células. Estos inhibidores se utilizan para estudiar la regulación del metabolismo, el papel de las vías metabólicas en enfermedades como el cáncer y la diabetes, y para desarrollar nuevas estrategias terapéuticas. Los inhibidores del metabolismo pueden dirigirse a diversas enzimas y procesos involucrados en la glucólisis, la oxidación de ácidos grasos y otras funciones metabólicas. En CymitQuimica, ofrecemos una amplia gama de inhibidores del metabolismo de alta calidad para apoyar su investigación en bioquímica, trastornos metabólicos y desarrollo de fármacos.

Subcategorías de "Metabolismo"

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Se han encontrado 8626 productos de "Metabolismo"

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  • Clopidogrel-β-D-glucuronide
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    Clopidogrel-β-D-glucuronide

    CAS:
    <p>Clopidogrel-β-D-glucuronide is a metabolite of Clopidogrel. It directly interacts with the CYP2C8 enzyme and strongly inhibits the hepatic enzyme CYP2C8.</p>
    Fórmula:C21H22ClNO8S
    Forma y color:Solid
    Peso molecular:483.919

    Ref: TM-T206623

  • Logo de CymitQuimica
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    FXIa-IN-8

    <p>FXIa-IN-8: potent FXIa blocker (IC50: 14.2 nM), anti-thrombotic, low bleeding/toxicity risk.</p>
    Forma y color:Solid

    Ref: TM-T64257

  • Logo de CymitQuimica
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    AChE/PDE4-IN-1

    <p>AChE/PDE4-IN-1, compound 12c, dual inhibitor; IC50: 0.28μM for AChE, 1.88μM for PDE4D, may reduce Alzheimer's neuroinflammation.</p>
    Fórmula:C23H28N2O3
    Forma y color:Solid
    Peso molecular:380.48

    Ref: TM-T61620

  • Logo de CymitQuimica
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    RXR antagonist 2

    <p>RXR antagonist 2 is a potent antagonist of RXR (Ki: 0.391 μM, Kd: 0.281 μM). RXR antagonist 2 has shown research potential for RXR-related diseases.</p>
    Fórmula:C29H35F3N2O3
    Forma y color:Solid
    Peso molecular:516.6

    Ref: TM-T63597

  • CA IX-IN-3
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    CA IX-IN-3

    CAS:
    <p>CAIX-IN-3 (Compound 27) is a selective and potent inhibitor of carbonic anhydrase IX (CAIX), with an IC50 of 0.48 nM.</p>
    Fórmula:C21H19N5O4S2
    Forma y color:Solid
    Peso molecular:469.537

    Ref: TM-T204606

  • FXIa-IN-6
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    FXIa-IN-6

    CAS:
    <p>FXIa-IN-6: Potent, selective FXIa inhibitor (Ki=0.3 nM); strong PK with high oral bioavailability, low clearance preclinically.</p>
    Fórmula:C31H29ClF2N4O4
    Forma y color:Solid
    Peso molecular:595.04

    Ref: TM-T39035

  • (E)-10-Hydroxynortriptyline maleate
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    (E)-10-Hydroxynortriptyline maleate

    CAS:
    <p>(E)-10-Hydroxy Nortriptyline maleate, a derivative of antidepressant Nortriptyline, eases depression symptoms.</p>
    Fórmula:C23H25NO5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:395.455

    Ref: TM-T11135

  • Raloxifene N-Oxide
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    Raloxifene N-Oxide

    CAS:
    <p>Raloxifene N-Oxide is a Raloxifene oxidative degradation product.</p>
    Fórmula:C28H27NO5S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:489.58

    Ref: TM-T19545

  • Logo de CymitQuimica
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    Vimirogant hydrochloride

    <p>Vimirogant (VTP-43742) HCl: Oral, selective RORγt inhibitor (IC50: 17 nM, Ki: 3.5 nM), &gt;1000x selectivity over RORα/β, targets Th17, not Th1/2/Treg.</p>
    Fórmula:C27H36ClF3N4O3S
    Forma y color:Solid
    Peso molecular:588.21487

    Ref: TM-T64300

  • ZK168281
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    ZK168281

    CAS:
    <p>ZK168281 is a 1α,25(OH)2D3 analog, VDR antagonist with 0.1 nM Kd, and blocks receptor CoA interaction.</p>
    Fórmula:C32H46O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:510.70

    Ref: TM-T13404

  • 5-Carboxy-2′-deoxycytidine
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    5-Carboxy-2′-deoxycytidine

    CAS:
    <p>5-Carboxy-2′-deoxycytidine is a metabolite of Trifluridine.</p>
    Fórmula:C10H13N3O6
    Forma y color:Solid
    Peso molecular:271.227

    Ref: TM-TYD-02090

  • PRL3-CNNM4 interaction-IN-1
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    PRL3-CNNM4 interaction-IN-1

    CAS:
    <p>PRL3-CNNM4 interaction-IN-1 (Compound C28d52) is an inhibitor of the PRL3-CNNM4 interaction that also suppresses CNNM inhibition mediated by PRL. This compound exhibits favorable pharmacokinetic and drug metabolism properties.</p>
    Fórmula:C8H8O2S
    Forma y color:Solid
    Peso molecular:168.21

    Ref: TM-T200840

  • m-APTA
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    m-APTA

    CAS:
    <p>m-APTA (5'-S-(3-aminophenyl)-5'-thioadenosine) is a selective chemoprotective agent targeting methylthioadenosine phosphorylase (MTAP). It can be converted into adenine, which is a crucial step in shielding normal cells from the toxicity of nucleobase analogs (NBA). m-APTA holds potential for research in MTAP-deficient cancers.</p>
    Fórmula:C16H18N6O3S
    Forma y color:Solid
    Peso molecular:374.418

    Ref: TM-T206811

  • Buspirone N-oxide
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    Buspirone N-oxide

    CAS:
    <p>Buspirone N-oxide (Bu N-oxide) is a metabolite of Buspirone. Buspirone is an orally active 5-HT1A receptor agonist and a dopamine D2 (dopamine D2) autoreceptor antagonist. It is an anxiolytic agent used for research in generalized anxiety disorder.</p>
    Fórmula:C21H31N5O3
    Forma y color:Solid
    Peso molecular:401.503

    Ref: TM-TYD-01953

  • PF-07202954
    Targetmol
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    PF-07202954

    CAS:
    <p>PF-07202954, a weakly basic diacylglycerol O-acyltransferase 2 (DGAT2) inhibitor, exhibits an inhibition concentration half-maximum (IC50) of 10 nM against</p>
    Fórmula:C22H23FN6O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:438.45

    Ref: TM-T79764

  • OSI-413 free base
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    OSI-413 free base

    CAS:
    <p>OSI-413 (free base) (CP 373413) is the primary metabolite of Erlotinib. Erlotinib (CP-358774) acts as a direct EGFR tyrosine kinase inhibitor with an IC50 of 2 nM against human EGFR.</p>
    Fórmula:C21H21N3O4
    Forma y color:Solid
    Peso molecular:379.409

    Ref: TM-TYD-01898

  • hCAI/II/XII-IN-1
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    hCAI/II/XII-IN-1

    CAS:
    <p>hCAI/II/XII-IN-1 (compound 7) is an inhibitor of human carbonic anhydrases hCAI, hCAII, and hCAXII, with Ki values of 78.5 nM, 9.1 nM, 605 nM, 7.7 nM, and 3.7 nM.</p>
    Fórmula:C12H12N2O2S
    Forma y color:Solid
    Peso molecular:248.301

    Ref: TM-T204773

  • Logo de CymitQuimica
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    sEH inhibitor-4

    <p>Compound B15: potent sEH inhibitor (0.03 nm), reduces inflammation &amp; pain.</p>
    Fórmula:C27H28Cl2N4O3
    Forma y color:Solid
    Peso molecular:527.44

    Ref: TM-T63700

  • 11-trans Leukotriene E4
    Targetmol
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    11-trans Leukotriene E4

    CAS:
    <p>Slow isomerization of the C-11 double bond of LTE4 leads to the formation of 11-trans LTE4. 11-trans LTE4 is equipotent to LTE4 in contracting guinea pig ileum.</p>
    Fórmula:C23H37NO5S
    Forma y color:Solid
    Peso molecular:439.61

    Ref: TM-T37494

  • Logo de CymitQuimica
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    PHGDH-IN-2

    <p>PHGDH-IN-2: potent PHGDH inhibitor, IC50=5.2μM; hinders PHGDH cancer cell growth &amp; serine synthesis in MDA-MB-468.</p>
    Fórmula:C22H20N4O3S
    Forma y color:Solid
    Peso molecular:420.48

    Ref: TM-T62232