
Metabolismo
Los inhibidores del metabolismo son compuestos que interfieren con las vías metabólicas, alterando la producción y utilización de energía dentro de las células. Estos inhibidores se utilizan para estudiar la regulación del metabolismo, el papel de las vías metabólicas en enfermedades como el cáncer y la diabetes, y para desarrollar nuevas estrategias terapéuticas. Los inhibidores del metabolismo pueden dirigirse a diversas enzimas y procesos involucrados en la glucólisis, la oxidación de ácidos grasos y otras funciones metabólicas. En CymitQuimica, ofrecemos una amplia gama de inhibidores del metabolismo de alta calidad para apoyar su investigación en bioquímica, trastornos metabólicos y desarrollo de fármacos.
Subcategorías de "Metabolismo"
- AhR(42 productos)
- Aminopeptidasa(76 productos)
- CETP(20 productos)
- Anhídrido carbónico(195 productos)
- Caseína quinasa(137 productos)
- DHFR(34 productos)
- Descarboxilasa(4 productos)
- Deshidrogenasa(302 productos)
- FAAH(66 productos)
- FXR(62 productos)
- Factor Xa(87 productos)
- Ácido graso sintasa(37 productos)
- Ferroptosis(226 productos)
- GR(3 productos)
- GSNOR(4 productos)
- Glucoquinasa(57 productos)
- HIF / HIF Prolilhidroxilasa(146 productos)
- HMG-CoA reductasa(33 productos)
- Hidroxilasa(35 productos)
- IDO(84 productos)
- LDL(8 productos)
- Lipasa(107 productos)
- Lípido(61 productos)
- Lipoxigenasa(134 productos)
- MAO(87 productos)
- MPO(2 productos)
- NAMPT(40 productos)
- P450(6 productos)
- PAI-1(26 productos)
- PDE(167 productos)
- PED(1 productos)
- PKM(17 productos)
- PPAR(169 productos)
- Fosfolipasa(83 productos)
- ROR(47 productos)
- Receptor de retinoides(28 productos)
- SGK(11 productos)
- Tiorredoxina(12 productos)
- Transferasa(29 productos)
- Transportador(46 productos)
- UGT(4 productos)
- Inhibidores de la xantina oxidasa (XO)(9 productos)
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Se han encontrado 9274 productos de "Metabolismo"
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LY-338979
CAS:LY-338979 is an impurity of pemetrexedone.Fórmula:C20H21N5O7Pureza:98%Forma y color:SolidPeso molecular:443.41ICMT-IN-43
CAS:ICMT-IN-43 (compound 22) acts as a potent inhibitor of the enzyme ICMT, exhibiting an inhibitory concentration (IC50) value of 0.04 μM [1].Fórmula:C23H31NOForma y color:SolidPeso molecular:337.5DPM-1001 trihydrochloride
DPM-1001 trihydrochloride: Potent PTP1B inhibitor, IC50 100 nM, oral, non-competitive, anti-diabetic.Fórmula:C35H60Cl3N3O3Forma y color:SolidPeso molecular:677.23VU0155069 hydrochloride
CAS:VU0155069 hydrochloride (CAY10593 hydrochloride) is a potent and selective inhibitor of phospholipase D (PLD), exhibiting IC50 values of 46 nM for PLD1 and 933 nM for PLD2. It effectively inhibits the migration of both human and mouse breast cancer cell lines [1] [2].Fórmula:C26H28Cl2N4O2Forma y color:SolidPeso molecular:499.4312-SAHSA
CAS:Branched fatty acid esters of hydroxy fatty acids (FAHFAs) are lipids recently discovered to be modulated by dietary influences such as fasting and high-fat feeding, and they play a role in enhancing insulin sensitivity. These compounds typically feature a carbon-16 or carbon-18 fatty acid (e.g., palmitoleic, palmitic, oleic, or stearic acid) esterified to a carbon-16 or carbon-18 hydroxy fatty acid. A specific example is 12-SAHSA, which consists of stearic acid linked to 12-hydroxy stearic acid. Notably, 12-SAHSA levels are found to be moderately increased in the serum of glucose tolerant AG4OX mice, a model characterized by adipose tissue-specific overexpression of the Glut4 glucose transporter.Fórmula:C36H70O4Forma y color:SolidPeso molecular:566.952C32 Ceramide (d18:1/32:0)
CAS:C32 Ceramide (d18:1/32:0) is a lipid molecule that can be used in life science related research. The CAS number of C32 Ceramide (d18:1/32:0) is 34227-73-1.Fórmula:C50H99NO3Forma y color:SolidPeso molecular:762.346MGAT2-IN-2
CAS:MGAT2-IN-2 is a potent inhibitor of acyl CoA:monoacylglycerol acyltransferase 2 (MGAT2) (IC50 of 3.4 nM).Fórmula:C26H21F5N4O4SPureza:98%Forma y color:SolidPeso molecular:580.53L-CCG-lll
CAS:inhibitor of both glial and neuronal uptake of glutamate, aspartate and cysteate.Fórmula:C6H9NO4Pureza:98%Forma y color:SolidPeso molecular:159.14Rosuvastatin zinc salt
CAS:Rosuvastatin zinc salt (Rosuvastatin zinc), a zinc-infused variant of Rosuvastatin, functions as an HMG-CoA reductase inhibitor, utilized primarily inFórmula:C44H54F2N6O12S2ZnForma y color:SolidPeso molecular:1026.47SREBP/SCAP-IN-1
CAS:SREBP/SCAP-IN-1 (compound 10b) serves as a selective inhibitor of SREBP/SCAP [1].Fórmula:C28H40F2N4OForma y color:SolidPeso molecular:486.64MR-2-93-3
CAS:MR-2-93-3, a long-chain fatty acid, functions as a carrier for polynucleotides [1].Fórmula:C89H150N2O8Forma y color:SolidPeso molecular:1376.15Iomazenil
CAS:Iomazenil is an antagonist and partial inverse agonist of benzodiazepine and potential therapy for alcohol abuse.Fórmula:C15H14IN3O3Pureza:98%Forma y color:SolidPeso molecular:411.19MK-8245 analog
CAS:<p>MK-8245 analog is an analog of MK-8245 which is a liver-targeted Inhibitor of Stearoyl-CoA Desaturase (SCD).</p>Fórmula:C16H15BrFN7O3SPureza:99.85%Forma y color:SolidPeso molecular:484.3Ref: TM-T20950
1mg87,00€2mg124,00€5mg187,00€10mg284,00€25mg452,00€50mg645,00€100mg867,00€200mg1.130,00€IDO1/2-IN-1 hydrochloride
CAS:IDO1/2-IN-1 hydrochloride: Dual IDO1/2 inhibitor, IC50 of 28/144 nM, oral, with antitumor properties.Fórmula:C16H19BrClFN8O4Forma y color:SolidPeso molecular:521.73GIV3727
CAS:GIV3727, a bitter taste receptor hTAS2R antagonist, inhibits the activation of hTAS2R31 by saccharin and acesulfame potassium, effectively diminishing theFórmula:C12H22O2Forma y color:SolidPeso molecular:198.3JTV-803 mesylate
CAS:JTV-803 inhibits factor Xa (K(i) 0.019 µM, IC(50) 0.081 µM), 100x more selective vs thrombin, extends clotting times dose-dependently.Fórmula:C23H31N5O6SPureza:98%Forma y color:SolidPeso molecular:505.599(Z),11(Z)-Octadecadienoic acid
CAS:9(Z),11(Z)-Octadecadienoic acid, an isomer of linoleic acid, demonstrates antitumor activity with an EC50 value of 446.1 µM [1].Fórmula:C18H32O2Forma y color:SolidPeso molecular:280.45Glycosidase-IN-1
CAS:Glycosidase-IN-1, a D-mannose-derived inhibitor, has hypoglycemic effects and aids in creating immunosuppressants and β-glucosidase blockers.Fórmula:C13H23NO5Pureza:98%Forma y color:SolidPeso molecular:273.338-Hydroxyguanine hydrochloride
CAS:8-Hydroxyguanine, generated through the oxidative degradation of DNA by the hydroxyl radical, serves as an indicator of oxidative stress in biological systems.Fórmula:C5H5N5O2HClForma y color:SolidPeso molecular:203.6S-Fcme
CAS:S-Fcme activates multidrug resistance transporter by boosting ATPase activity and competing for drug binding.Fórmula:C19H33NO2SForma y color:SolidPeso molecular:339.54
