
Metabolismo
Los inhibidores del metabolismo son compuestos que interfieren con las vías metabólicas, alterando la producción y utilización de energía dentro de las células. Estos inhibidores se utilizan para estudiar la regulación del metabolismo, el papel de las vías metabólicas en enfermedades como el cáncer y la diabetes, y para desarrollar nuevas estrategias terapéuticas. Los inhibidores del metabolismo pueden dirigirse a diversas enzimas y procesos involucrados en la glucólisis, la oxidación de ácidos grasos y otras funciones metabólicas. En CymitQuimica, ofrecemos una amplia gama de inhibidores del metabolismo de alta calidad para apoyar su investigación en bioquímica, trastornos metabólicos y desarrollo de fármacos.
Subcategorías de "Metabolismo"
- AhR(42 productos)
- Aminopeptidasa(76 productos)
- CETP(20 productos)
- Anhídrido carbónico(196 productos)
- Caseína quinasa(138 productos)
- DHFR(32 productos)
- Descarboxilasa(4 productos)
- Deshidrogenasa(302 productos)
- FAAH(64 productos)
- FXR(62 productos)
- Factor Xa(85 productos)
- Ácido graso sintasa(37 productos)
- Ferroptosis(226 productos)
- GR(3 productos)
- GSNOR(3 productos)
- Glucoquinasa(57 productos)
- HIF / HIF Prolilhidroxilasa(146 productos)
- HMG-CoA reductasa(34 productos)
- Hidroxilasa(36 productos)
- IDO(84 productos)
- LDL(7 productos)
- Lipasa(107 productos)
- Lípido(61 productos)
- Lipoxigenasa(134 productos)
- MAO(87 productos)
- MPO(2 productos)
- NAMPT(40 productos)
- P450(6 productos)
- PAI-1(26 productos)
- PDE(169 productos)
- PED(1 productos)
- PKM(17 productos)
- PPAR(170 productos)
- Fosfolipasa(86 productos)
- ROR(47 productos)
- Receptor de retinoides(22 productos)
- SGK(10 productos)
- Tiorredoxina(12 productos)
- Transferasa(29 productos)
- Transportador(45 productos)
- UGT(4 productos)
- Inhibidores de la xantina oxidasa (XO)(9 productos)
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Se han encontrado 9181 productos de "Metabolismo"
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Mitiperstat
CAS:Mitiperstat, a strong MPO inhibitor, helps prevent heart failure and coronary artery disease.Fórmula:C15H15ClN4OSPureza:98.36%Forma y color:SolidPeso molecular:334.82Ref: TM-T61028
1mg147,00€5mg356,00€10mg432,00€25mg700,00€50mg888,00€100mg1.243,00€1mL*10mM (DMSO)393,00€ER 50891
CAS:ER-50891 is a potent RARα antagonist, countering retinoic acid inhibition and aiding BMP2-induced osteoblast differentiation.Fórmula:C29H24N2O2Pureza:99.43%Forma y color:SolidPeso molecular:432.51Dechloro Rivaroxaban
CAS:Dechloro Rivaroxaban is a Factor Xa inhibitor that inhibits free FXa and plasminogen and fibrin-associated FXa activity in humans.Fórmula:C19H19N3O5SPureza:98.63%Forma y color:SolidPeso molecular:401.44Ref: TM-T78215
5mg40,00€10mg63,00€25mg107,00€50mg170,00€100mg264,00€200mg418,00€1mL*10mM (DMSO)44,00€PDE9-IN-(S)-C33
CAS:PDE9-IN-(S)-C33: potent PDE9 inhibitor with 11 nM IC50, for CNS diseases and diabetes study.Fórmula:C18H20ClN5OPureza:98.75%Forma y color:SolidPeso molecular:357.84Ref: TM-T28352
1mg37,00€5mg70,00€10mg88,00€25mg144,00€50mg207,00€100mg309,00€200mg440,00€1mL*10mM (DMSO)79,00€OGT 2115
CAS:OGT 2115 blocks heparanase (IC50=0.4µM), cleaving heparan sulfate; antiangiogenic (IC50=1µM).
Fórmula:C24H16BrFN2O4Pureza:97.17%Forma y color:SolidPeso molecular:495.3TP-10
CAS:TP-10 is a selective inhibitor of PDE10A against other PDEs with IC50 of 0.8 nM.Fórmula:C26H19F3N4OPureza:99.21%Forma y color:SolidPeso molecular:460.45Ref: TM-T13189
1mg87,00€2mg114,00€5mg177,00€10mg264,00€25mg460,00€50mg668,00€100mg945,00€500mg1.783,00€1mL*10mM (DMSO)178,00€KB-74935
CAS:KB-74935: enzyme inhibitor, mineralocorticoid blocker, treats cholesterol, hypolipidemia, neurological issues, Alzheimer's.Fórmula:C19H18ClF4N3O3SPureza:99.4%Forma y color:SolidPeso molecular:479.88h-NTPDase-IN-2
CAS:h-NTPDase-IN-2 is a broad-spectrum NTPDase inhibitor that inhibits multiple h-NTPDas isoforms.Fórmula:C19H16N4SPureza:99.58%Forma y color:SolidPeso molecular:332.42Enpp-1-IN-16
CAS:Enpp-1-IN-16 is an ENPP1 inhibitor, yo anti-cancer activity.Enpp-1-IN-16 can be used to study insulin resistance and chondrocalcinosis.Fórmula:C23H32N4O4Pureza:99.87%Forma y color:SolidPeso molecular:428.52Varespladib methyl
CAS:Varespladib methyl (LY333013), a bioavailable prodrug of Varespladib, is a selective group II secretory phospholipase A2 inhibitor.Fórmula:C22H22N2O5Pureza:99.42% - 99.97%Forma y color:SolidPeso molecular:394.42Ref: TM-T17218
1mg93,00€2mg123,00€5mg200,00€10mg319,00€25mg528,00€50mg730,00€100mg999,00€200mg1.333,00€1mL*10mM (DMSO)220,00€ML400
CAS:ML400 (CID73050863) is an allosteric inhibitor of LMPTP with an EC50 of 1μM. ML400 displays good cell-based activity and rodent pharmacokinetics.Fórmula:C24H29N3OPureza:99.95%Forma y color:SolidPeso molecular:375.51Ref: TM-T25824
1mg92,00€5mg172,00€10mg281,00€25mg447,00€50mg618,00€100mg853,00€500mg1.701,00€1mL*10mM (DMSO)222,00€Fluspirilene
CAS:Fluspirilene is a long-acting antipsychotic for schizophrenia, inhibiting L-type calcium channels (IC50: 0.03 μM).Fórmula:C29H31F2N3OPureza:99.59%Forma y color:SolidPeso molecular:475.57NPAS3-IN-1
CAS:NPAS3-IN-1 is an NPAS3-ARNT heterodimerization inhibitor that regulates NPAS3 transcription by modulating the heterodimerization of NPAS3 with ARNT.Fórmula:C10H5N3O2S3Pureza:99.56%Forma y color:SolidPeso molecular:295.36PDDC inhibitor
CAS:PDDC inhibitor (Phenyl (R)-(1-(3-(3,4-dimethoxyphenyl)-2,6-dimethylimidazo[1,2-b]pyridazin-8-yl)pyrrolidin-3-yl)carbamate) is an nSMase2 inhibitor.Fórmula:C27H29N5O4Pureza:96.09% - 99.39%Forma y color:SolidPeso molecular:487.55Cudetaxestat
CAS:Cudetaxestat (BLD-0409) is a potent inhibitor of orally active autotaxin.Fórmula:C21H15Cl2F2N3O2SPureza:99.9%Forma y color:SolidPeso molecular:482.33Ref: TM-T63190
1mg77,00€5mg170,00€10mg248,00€25mg444,00€50mg662,00€100mg929,00€200mg1.225,00€1mL*10mM (DMSO)170,00€RS 8359
CAS:RS 8359 is a selective MAO-A reversible inhibitor with a 2200:1 A:B ratio, exhibiting antidepressant effects.Fórmula:C14H12N4OPureza:99.3%Forma y color:SolidPeso molecular:252.27Ref: TM-T16803
1mg81,00€5mg170,00€10mg274,00€25mg550,00€50mg885,00€100mg1.415,00€1mL*10mM (DMSO)188,00€7-BIA
CAS:7-BIA is a receptor-type protein tyrosine phosphatase D (PTPRD) inhibitor with anti-addictive properties and can be used in the study of neuropathic pain.Fórmula:C15H18O6Pureza:≥98% - ≥98%Forma y color:SolidPeso molecular:294.3Ref: TM-T10190
1mg145,00€5mg354,00€10mg612,00€25mg1.130,00€50mg1.786,00€100mg2.832,00€1mL*10mM (DMSO)378,00€CB29
CAS:CB29 is a specific inhibitor of aldehyde dehydrogenase 3A1 (ALDH3A1).
Fórmula:C15H15N3O5SPureza:99.36%Forma y color:SolidPeso molecular:349.36Mutant IDH1-IN-2
CAS:Mutant IDH1-IN-2 is a inhibitor of mutant Isocitrate dehydrogenase (IDH) proteins, with IC50 of 16.6 nM in Fluorescence biochemical assay, IC50 of <22 nM in LS-Fórmula:C24H31F2N5O2Pureza:99.88%Forma y color:SolidPeso molecular:459.53Ref: TM-T12128
1mg60,00€5mg138,00€10mg224,00€25mg374,00€50mg532,00€100mg718,00€200mg964,00€1mL*10mM (DMSO)137,00€Monometacrine
CAS:Monometacrine, a cholesterol esterase inhibitor, exhibits antidepressant effects [1].Fórmula:C19H24N2Forma y color:SolidPeso molecular:280.41
