
Metabolismo
Los inhibidores del metabolismo son compuestos que interfieren con las vías metabólicas, alterando la producción y utilización de energía dentro de las células. Estos inhibidores se utilizan para estudiar la regulación del metabolismo, el papel de las vías metabólicas en enfermedades como el cáncer y la diabetes, y para desarrollar nuevas estrategias terapéuticas. Los inhibidores del metabolismo pueden dirigirse a diversas enzimas y procesos involucrados en la glucólisis, la oxidación de ácidos grasos y otras funciones metabólicas. En CymitQuimica, ofrecemos una amplia gama de inhibidores del metabolismo de alta calidad para apoyar su investigación en bioquímica, trastornos metabólicos y desarrollo de fármacos.
Subcategorías de "Metabolismo"
- AhR(42 productos)
- Aminopeptidasa(76 productos)
- CETP(20 productos)
- Anhídrido carbónico(196 productos)
- Caseína quinasa(138 productos)
- DHFR(32 productos)
- Descarboxilasa(4 productos)
- Deshidrogenasa(301 productos)
- FAAH(64 productos)
- FXR(62 productos)
- Factor Xa(85 productos)
- Ácido graso sintasa(37 productos)
- Ferroptosis(226 productos)
- GR(3 productos)
- GSNOR(3 productos)
- Glucoquinasa(57 productos)
- HIF / HIF Prolilhidroxilasa(146 productos)
- HMG-CoA reductasa(34 productos)
- Hidroxilasa(36 productos)
- IDO(84 productos)
- LDL(7 productos)
- Lipasa(107 productos)
- Lípido(61 productos)
- Lipoxigenasa(133 productos)
- MAO(87 productos)
- MPO(2 productos)
- NAMPT(40 productos)
- P450(6 productos)
- PAI-1(26 productos)
- PDE(169 productos)
- PED(1 productos)
- PKM(17 productos)
- PPAR(170 productos)
- Fosfolipasa(86 productos)
- ROR(47 productos)
- Receptor de retinoides(21 productos)
- SGK(10 productos)
- Tiorredoxina(12 productos)
- Transferasa(29 productos)
- Transportador(44 productos)
- UGT(4 productos)
- Inhibidores de la xantina oxidasa (XO)(9 productos)
Mostrar 34 subcategorías más
Se han encontrado 9161 productos de "Metabolismo"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
13(R)-HODE
CAS:13(R)-HODE, produced from linoleic acid, inhibits platelet aggregation (IC50=2.7μM) and is found in bovine endothelial cells.Fórmula:C18H32O3Forma y color:SolidPeso molecular:296.44CHI3L1-IN-2
CAS:CHI3L1-IN-2 (Compound 36), a potent inhibitor of CHI3L1 (YKL-40), effectively blocks the interaction between CHI3L1 and heparan sulfate (CHI3L1:HSIII), demonstrating an IC 50 of 26 nM [1].Fórmula:C26H37ClN4Peso molecular:441.05Carbonic anhydrase inhibitor 10
CA inhibitor 10 targets MCF-7 cells, IC50: 11.9 μM; potent h CA IX inhibitor, Ki: 6.2 nM. Anti-cancer research.Fórmula:C14H17N5O3SForma y color:SolidPeso molecular:335.389(S)-HEPE
CAS:9(S)-HEPE is a monohydroxy fatty acid derived from EPA. The biological activity of 9(S)-HEPE has not been documented.Fórmula:C20H30O3Forma y color:SolidPeso molecular:318.45HSD17B13-IN-17
CAS:HSD17B13-IN-17 (compound 9) serves as a potent inhibitor of hydroxysteroid 17β-dehydrogenase 13 (HSD17B13). It demonstrates inhibitory efficacy with IC50 values of <0.1 μM for estradiol and <1 μM for Leukotriene B3 as substrates. This compound is significant in the management of nonalcoholic fatty liver diseases (NAFLDs), including nonalcoholic steatohepatitis (NASH) [1].Fórmula:C20H16ClFN2O3SForma y color:SolidPeso molecular:418.8722-HDHA
CAS:22-HDHA is an oxidation product of docosahexaenoic acid .Fórmula:C22H32O3Forma y color:SolidPeso molecular:344.49Hcyb1
Hcyb1 specifically inhibits PDE2A with 0.57 μM IC50, over 250x selective, and has neuroprotective and antidepressant effects.Fórmula:C24H20N4OForma y color:SolidPeso molecular:380.44hDHODH-IN-10
hDHODH-IN-10: selective oral inhibitor of hDHODH (IC50: 10.9 nM); blocks cancer cell growth, aids cancer research.Fórmula:C21H15ClF4N2O4Forma y color:SolidPeso molecular:470.8IDO1-IN-14
IDO1-IN-14 is an IDO1 enzyme inhibitor with an IC50 of 396.9 nM and suppresses HeLa cell activity with an EC50 of 3393 nM.Fórmula:C18H12Cl2FN3O2Forma y color:SolidPeso molecular:392.21Complex III-IN-1
Complex III-IN-1 inhibits complex III, has antifungal properties, and an EC50 of 18.53 mg/L against S. sclerotiorum.Fórmula:C14H20ClNO2S2Forma y color:SolidPeso molecular:333.99(Z),12(E)-Octadecadienoic Acid
CAS:9(Z),12(E)-Octadecadienoic Acid (C18:2(9E,12Z); C18:2 n-6), an isomer of linoleic acid, is a type of ω-6 polyunsaturated fatty acid containing a trans double bond at the C9 position. It is identified as a minor component in milk fat and partially hydrogenated vegetable oils. The concentration of 9(Z),12(E)-Octadecadienoic Acid in rabbit meat increases following supplementation with heated sunflower seed oil, α-tocopherol acetate, and zinc.Fórmula:C18H32O2Peso molecular:280.45DC360
CAS:DC360 is a synthetic analog of all-trans retinoic acid (ATRA) that can induce the expression of RARβ. It is useful for studies characterizing the retinoic acid signaling pathway.
Fórmula:C23H23NO2Forma y color:SolidPeso molecular:345.434T-3764518
CAS:T-3764518 is a novel and potent inhibitor of stearoyl coenzyme A desaturase (SCD)(IC50 of 4.7 nM).Fórmula:C20H17F6N5O2Pureza:98%Forma y color:SolidPeso molecular:473.37Casein kinase 1δ-IN-16
CAS:Casein kinase1δ-IN-16 (compound 506) is an inhibitor of casein kinase 1δ (CK1δ). This compound is applicable in research related to neurodegenerative diseases.Fórmula:C17H12N4S2Forma y color:SolidPeso molecular:336.434BRD2879
CAS:BRD2879 is a potent and cell-active inhibitor of IDH1-R132H (IC50 = 50 nM).Fórmula:C30H38FN3O5SPureza:98%Forma y color:SolidPeso molecular:571.70AZD 4407
CAS:AZD 4407 is a potent inhibitor of 5-lipoxygenase.Fórmula:C19H21NO3S2Pureza:98%Forma y color:SolidPeso molecular:375.5hCAII-IN-4
CAS:hCAII-IN-4 (Compound 12j) is a potent inhibitor of human carbonic anhydrase II (hCA II), exhibiting an inhibitory concentration (IC50) of 7.78 μM.Fórmula:C31H23NO9Forma y color:SolidPeso molecular:553.52GNTI TFA
CAS:GNTI TFA is a selective kappa opioid receptor antagonist.Fórmula:C31H31F6N5O7Forma y color:SolidPeso molecular:699.60CP 524515
CAS:CP 524515 is a potent inhibitor of cholesterol ester transfer protein (CETP), which results in increased levels of high-density lipoprotein cholesterol.
Fórmula:C27H27F9N2O4Forma y color:SolidPeso molecular:614.5hCAII-IN-3
hCAII-IN-3 inhibits key hCA isoforms with Ki: hCA I (403.8 nM), hCA II (5.1 nM), hCA IX (10.2 nM), hCA XII (5.2 nM); shows anticancer potential.
Fórmula:C17H21N3O3SForma y color:SolidPeso molecular:347.43

