
Neurociencia
Los inhibidores en neurociencia son compuestos diseñados para modular la actividad de proteínas, enzimas o receptores específicos dentro del sistema nervioso. Estos inhibidores son cruciales para estudiar los mecanismos moleculares subyacentes a la función neuronal, la transmisión sináptica y las enfermedades neurodegenerativas. Al dirigirse a los receptores de neurotransmisores, canales iónicos y vías de señalización, los inhibidores en neurociencia ayudan en la exploración de la función cerebral y en el desarrollo de estrategias terapéuticas para trastornos neurológicos como el Alzheimer, Parkinson y la epilepsia. En CymitQuimica, ofrecemos una amplia gama de inhibidores de neurociencia de alta calidad para apoyar su investigación en neurobiología, neurofarmacología y ciencias cognitivas.
Subcategorías de "Neurociencia"
- Receptor 5-HT(1.025 productos)
- ACK(1 productos)
- AChR(630 productos)
- ATP Citrato Liasa(17 productos)
- Receptor adrenérgico(3.030 productos)
- BACE(36 productos)
- Beta amiloide(227 productos)
- CAMK(73 productos)
- Inhibidores de ciclooxigenasa (COX)(602 productos)
- Receptor de dopamina(444 productos)
- Receptor GABA(369 productos)
- Gamma-secretasa(62 productos)
- GluR(264 productos)
- GlyT(26 productos)
- Receptor de histamina(385 productos)
- LRRK2(42 productos)
- Receptor de melatonina(26 productos)
- NMDAR(10 productos)
- Receptor de OX(42 productos)
- Receptor de opioides(325 productos)
Mostrar 12 subcategorías más
Se han encontrado 5518 productos de "Neurociencia"
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LB-102
CAS:LB-102 is an orally active inhibitor of dopamine D2, D3, and serotonin 5-HT7 receptors, utilized in the study of schizophrenia and other psychiatric disorders.Fórmula:C18H29N3O4SForma y color:SolidPeso molecular:383.51(E)-CHBO4
CAS:(E)-CHBO4 is an MAO-B inhibitor with an IC50 value of 0.023 μM, making it a potential candidate for research into Parkinson's disease treatment.Fórmula:C15H10BrFOForma y color:SolidPeso molecular:305.1425-HT7R antagonist 3
CAS:Compound 6.4, also known as 5-HT7R antagonist 3, is a selective antagonist of the 5-HT7R with a Ki of 8 nM. It exhibits significantly less affinity towards D2R, 5-HT1AR, and 5-HT2AR with Ki values of 511 nM, 8930 nM, and 5786 nM, respectively. In mice, 5-HT7R antagonist 3 demonstrates anti-depressant and anti-anxiety activities.Fórmula:C30H33FN4O3Forma y color:SolidPeso molecular:516.611,9-Dideoxyforskolin
CAS:The compound is an inactive analog of forskolin(an adenylyl cyclase activator).Fórmula:C22H34O5Pureza:98%Forma y color:SolidPeso molecular:378.5VU6007496
CAS:VU6007496 is a highly selective and CNS-penetrating M1 positive allosteric modulator (PAM) that exhibits good pharmacokinetics (PK).Fórmula:C25H27N5O2Forma y color:SolidPeso molecular:429.51RO-1-5237
CAS:RO-1-5237, a cholinergic compound and a metabolic product of Pyridostigmine Bromide, is utilized in research for myasthenia gravis.Fórmula:C6H8BrNOForma y color:SolidPeso molecular:190.04BRD0418
CAS:BRD0418 acts as an upregulator of TRIB1 expression by leading to reprogramming of hepatic lipoprotein metabolism from adipogenesis to clearance it.Fórmula:C29H32N2O5Pureza:99.57%Forma y color:SolidPeso molecular:488.57YM 202074
CAS:metabotropic glutamate receptor type 1 (mGlu1) antagonistFórmula:C56H72N8O16S2Pureza:98%Forma y color:SolidPeso molecular:1177.34LY593093
CAS:LY593093 is a selective partial orthosteric agonist of M1 muscarinic acetylcholine receptor.Fórmula:C32H30FN3O2Pureza:98%Forma y color:SolidPeso molecular:507.6NB-360
CAS:NB-360: potent, brain-penetrant BACE1/2 inhibitor; IC50s: 5-6 nM; high selectivity vs pepsin, cathepsin E/D.Fórmula:C21H19F4N5O2Pureza:99.72%Forma y color:SolidPeso molecular:449.4Ref: TM-T12188
1mg104,00€5mg215,00€10mg318,00€25mg510,00€50mg692,00€100mg888,00€500mg1.783,00€1mL*10mM (DMSO)235,00€BDZ-g
CAS:BDZ-g: potent, selective AMPA receptor antagonist; useful for researching neurological disorders.Fórmula:C21H21N5O2SPureza:99.97%Forma y color:SolidPeso molecular:407.49BMS 299897
CAS:<p>BMS 299897, a sulfonamide γ-secretase inhibitor, inhibits Aβ production with an IC50 of 7 nM in HEK293 cells overexpressing APP.</p>Fórmula:C24H21ClF3NO4SPureza:99.82%Forma y color:SolidPeso molecular:511.94AChE-IN-26
CAS:<p>AChE-IN-26 (compound 4a) is an AChE (acetylcholinesterase) inhibitor (IC50: 0.42 μM).</p>Fórmula:C21H21BrN2O3Pureza:99.24% - 99.85%Forma y color:SoildPeso molecular:429.31Iclepertin
CAS:Iclepertin (BI-425809) is a GlyT1 inhibitor.Iclepertin is used for the treatment of Alzheimer;s disease and other CNS disorders.Fórmula:C20H18F6N2O5SPureza:98.89% - 98.93%Forma y color:SolidPeso molecular:512.42Ref: TM-T37089
1mg96,00€2mg120,00€5mg169,00€10mg224,00€25mg368,00€50mg552,00€100mg827,00€200mg1.111,00€1mL*10mM (DMSO)183,00€AChE/BChE-IN-10
CAS:<p>AChE/BChE-IN-10 inhibits AChE/BChE (IC50: 0.176/0.47 μM), crosses the blood-brain barrier, and prevents Aβ-aggregation.</p>Fórmula:C26H30N2O2Pureza:99.55% - 99.88%Forma y color:SoildPeso molecular:402.53LY2979165
CAS:LY2979165 (mGlu2 agonist) is an orthosteric agonist of mGluR2 and can be used in studies about serving as an anti-depressant.Fórmula:C13H22N6O6SPureza:98.41%Forma y color:SolidPeso molecular:390.42Umibecestat
CAS:Umibecestat inhibits human and mouse BACE-1 (IC50: 11 nM & 10 nM), potentially for Alzheimer's research.Fórmula:C19H15ClF7N5O2Pureza:99.88%Forma y color:SolidPeso molecular:513.8Ref: TM-T13253
1mg172,00€5mg354,00€10mg512,00€25mg852,00€50mg1.159,00€100mg1.568,00€1mL*10mM (DMSO)398,00€SB-224289 hydrochloride
CAS:SB-224289 hydrochloride (SB-224289A) is a selective antagonist of 5-HT1B receptor, with anxiolytic effect.Fórmula:C32H33ClN4O3Pureza:98.99% - 99.96%Forma y color:SolidPeso molecular:557.084-Amino-6-hydroxypyrazolo[3,4-d]pyrimidine
CAS:Fórmula:C5H5N5OPureza:>93.0%(HPLC)Forma y color:White to Light yellow to Light orange powder to crystallinePeso molecular:151.13BF 227
CAS:BF 227 is a candidate for an amyloid imaging probe for PET [Ki: 4.3 nM for Aβ1-42 fibrils].Fórmula:C16H16FN3O2SForma y color:SolidPeso molecular:333.38

