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Neurociencia

Neurociencia

Los inhibidores en neurociencia son compuestos diseñados para modular la actividad de proteínas, enzimas o receptores específicos dentro del sistema nervioso. Estos inhibidores son cruciales para estudiar los mecanismos moleculares subyacentes a la función neuronal, la transmisión sináptica y las enfermedades neurodegenerativas. Al dirigirse a los receptores de neurotransmisores, canales iónicos y vías de señalización, los inhibidores en neurociencia ayudan en la exploración de la función cerebral y en el desarrollo de estrategias terapéuticas para trastornos neurológicos como el Alzheimer, Parkinson y la epilepsia. En CymitQuimica, ofrecemos una amplia gama de inhibidores de neurociencia de alta calidad para apoyar su investigación en neurobiología, neurofarmacología y ciencias cognitivas.

Subcategorías de "Neurociencia"

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Se han encontrado 5398 productos de "Neurociencia"

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  • S1RA hydrochloride

    CAS:
    <p>S1RA hydrochloride (E-52862 hydrochloride) is an effective and specific sigma-1 receptor(σ1R, Ki: 17 nM) antagonist, and has good selectivity against σ2R (Ki &gt;</p>
    Fórmula:C20H24ClN3O2
    Pureza:98% - 99.84%
    Forma y color:Solid
    Peso molecular:373.87
  • Indomethacin heptyl ester

    CAS:
    <p>Indomethacin heptyl ester is a non-selective inhibitor of both COX-1 and COX-2</p>
    Fórmula:C26H30ClNO4
    Pureza:99.86%
    Forma y color:Solid
    Peso molecular:455.97
  • Oxyphencyclimine

    CAS:
    <p>Oxyphencyclimine is a muscarinic receptor antagonist (MRA) anticholinergic drug used to treat peptic ulcers.</p>
    Fórmula:C20H28N2O3
    Forma y color:Solid
    Peso molecular:344.45
  • Teriflunomide impurity 3

    CAS:
    <p>Teriflunomide impurity 3 (4-Amino-N-(4-trifluoromethylphenyl)benzamide) is a selective COX-1 inhibitor(IC50 of 30 μM).</p>
    Fórmula:C14H11F3N2O
    Pureza:99.62%
    Forma y color:Solid
    Peso molecular:280.25
  • Urapidil

    CAS:
    <p>Urapidil (Ebrantil), a sympatholytic antihypertensive drug, acts as a 5-HT1A receptor agonist and as an α1-adrenoceptor antagonist.</p>
    Fórmula:C20H29N5O3
    Pureza:99.85% - >99.99%
    Forma y color:Solid
    Peso molecular:387.48
  • β-Amyloid (31-35)

    CAS:
    <p>β-Amyloid (31-35) (β-Amyloid 31-35) is the shortest sequence of native Amyloid-β peptide.</p>
    Fórmula:C25H47N5O6S
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:545.74
  • γ-secretase modulator 1 hydrochloride

    CAS:
    <p>gamma-secretase inhibitior-1 is a gamma-secretase modulator that is useful to Alzheimer's disease [1].</p>
    Fórmula:C24H25ClN4OS
    Pureza:98%
    Forma y color:Solid
    Peso molecular:453
  • TCS 1102

    CAS:
    <p>TCS 1102 is an effective, dual orexin receptor antagonist (Ki: 0.2/3 nM for OX2/1 receptors).</p>
    Fórmula:C27H26N4O2S
    Pureza:99.35% - 99.52%
    Forma y color:Solid
    Peso molecular:470.59
  • Jatrorrhizine

    CAS:
    <p>Jatrorrhizine (neprotin) is a protoberberine alkaloid isolated from Enantia chlorantha (Annonaceae) and other species.</p>
    Fórmula:C20H20NO4
    Pureza:97.18% - 99.06%
    Forma y color:Solid
    Peso molecular:338.38
  • PRX-07034 hydrochloride

    CAS:
    <p>PRX-07034 hydrochloride is a selective antagonist of 5-HT6 receptor. It has cognition and memory-enhancing properties and decreases body weight in rodents.</p>
    Fórmula:C21H29Cl2N3O4S
    Pureza:98.5%
    Forma y color:Solid
    Peso molecular:490.44
  • Ilmetropium iodide

    CAS:
    <p>Ilmetropium iodide is a bronchodilator.</p>
    Fórmula:C20H30INO3
    Pureza:98.45%
    Forma y color:Solid
    Peso molecular:459.36
  • AZ 11645373

    CAS:
    <p>AZ 11645373 (3-[1-[[(3'-NITRO[1,1'-BIPHENYL]-4-YL)OXY]METHYL]-3-(4-PYRIDINYL)PROPYL]-2,4-THIAZOLIDINEDIONE) is a highly selective and potent human P2X7 receptor</p>
    Fórmula:C24H21N3O5S
    Pureza:99.47%
    Forma y color:Solid
    Peso molecular:463.51
  • Gabazine free base

    CAS:
    <p>Gabazine free base is a specific antagonist of the GABA receptor. It does not affect GABA-transaminase or glutamate-decarboxylase activities.</p>
    Fórmula:C15H17N3O3
    Forma y color:Solid
    Peso molecular:287.31
  • Naluzotan

    CAS:
    <p>Naluzotan(PRX 00023) is a novel and potent 5-HT1A agonist with IC50 and Ki values of approximately 20 nM and 5.1 nM, respectively.Naluzotan is a potent hERG K+</p>
    Fórmula:C23H38N4O3S
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:450.64
  • Cinitapride

    CAS:
    <p>Cinitapride (Blaston) treats acid reflux and gastric issues, targeting 5-HT2, 5-HT1, and 5-HT4 receptors.</p>
    Fórmula:C21H30N4O4
    Pureza:99.52%
    Forma y color:Solid
    Peso molecular:402.49
  • SB 242084 dihydrochloride

    CAS:
    <p>SB 242084 hydrochloride is a 5-HT2C receptor antagonist(pKi=9.0) that displays 158- and 100-fold selectivity over 5-HT2A and 5-HT2B receptors respectively.</p>
    Fórmula:C21H21Cl3N4O2
    Forma y color:Solid
    Peso molecular:467.78
  • 1-(1-Naphthyl) piperazine hydrochloride

    CAS:
    <p>1-(1-Naphthyl) piperazine hydrochloride (1-naphthalen-1-ylpiperazine hydrochloride) is a serotonergic ligand which could bind nonselectively with multiple</p>
    Fórmula:C14H17ClN2
    Pureza:98.27%
    Forma y color:Solid
    Peso molecular:248.75
  • lavendustin C

    CAS:
    <p>lavendustin C (NSC 666251) is a potent inhibitor of epidermal growth factor (EGF) receptor-associated tyrosine kinase.</p>
    Fórmula:C14H13NO5
    Pureza:98.06%
    Forma y color:Yellow To Tan Powder
    Peso molecular:275.26
  • Zacopride hydrochloride

    CAS:
    <p>Zacopride is a highly potent 5-HT3 receptor antagonist (Kd = 0.38 nM) and 5-HT4 receptor agonist (Ki = 373 nM). It also is a selective IK1 channel agonist.</p>
    Fórmula:C15H20ClN3O2·HCl
    Pureza:98.32%
    Forma y color:Solid
    Peso molecular:346.26
  • Acetoxyvalerensre

    CAS:
    <p>Acetoxyvalerensre (acetylvalerenolic acid) (acetylvalerenolic acid) is a derivative of valerenic acid, which is a a GABAA receptor modulator.</p>
    Fórmula:C17H24O4
    Pureza:98.22%
    Forma y color:Solid
    Peso molecular:292.37
  • Amentoflavone

    CAS:
    <p>Amentoflavone (3',8''-Biapigenin), as a potent inhibitor of CYP3A4 and CYP2C9, can interact with many other medications.</p>
    Fórmula:C30H18O10
    Pureza:98.21% - 99.22%
    Forma y color:Odourless Whitish Solid
    Peso molecular:538.46
  • 5-HT1A modulator 2 hydrochloride

    CAS:
    <p>5-HT1A modulator 2 hydrochloride is a modulator of 5-HT1A showing an affinity of 53 nM for 5-HT1A binding.</p>
    Fórmula:C11H16ClNO
    Pureza:98.5%
    Forma y color:Solid
    Peso molecular:213.7
  • pep2-SVKI acetate


    <p>Pep2-SVKI acetate(pep2-SVKI acetate (328944-75-8 free base)) is a synthetic peptide salt that prevents internalization of AMPA-type glutamate receptor.</p>
    Fórmula:C62H97N13O20
    Pureza:97.14%
    Forma y color:Solid
    Peso molecular:1344.51
  • Piperazine citrate

    CAS:
    <p>Piperazine citrate, an organic compound, consists of a six-membered ring, containing two nitrogen atoms at opposite positions in the ring.</p>
    Fórmula:C24H46N6O14
    Pureza:99.8%
    Forma y color:Crystals Indication
    Peso molecular:642.65
  • EUK-134

    CAS:
    <p>EUK-134, a synthetic SOD/catalase mimetic, exhibits potent antioxidant activities, and inhibits the formation of β-amyloid and related amyloid fibril.</p>
    Fórmula:C18H18ClMnN2O4
    Pureza:98.39%
    Forma y color:Solid
    Peso molecular:416.74
  • SEN12333

    CAS:
    <p>SEN12333 is an α7 nicotinic acetylcholine receptor (nAChR) agonist</p>
    Fórmula:C20H25N3O2
    Pureza:99.02%
    Forma y color:Solid
    Peso molecular:339.43
  • LY310762

    CAS:
    <p>LY310762 is a 5-HT1D receptor antagonist with Ki of 249 nM.</p>
    Fórmula:C24H27FN2O2·HCl
    Pureza:99.8%
    Forma y color:Solid
    Peso molecular:430.94
  • MK-3697

    CAS:
    <p>MK-3697, an isonicotinamide small molecule, acts as a potent and selective Orexin 2 receptor antagonist (Ki: 0.95 nM).</p>
    Fórmula:C23H21N5O3S
    Pureza:97.69% - 98.15%
    Forma y color:Solid
    Peso molecular:447.51
  • Frentizole

    CAS:
    <p>Frentizole, an immunosuppressive agent, is an inhibitor of the Aβ-ABAD interaction</p>
    Fórmula:C15H13N3O2S
    Pureza:99.82%
    Forma y color:Solid
    Peso molecular:299.35
  • RS-67333

    CAS:
    <p>RS-67333 is a partial agonist of 5-HT4R with neuroprotective effects.</p>
    Fórmula:C19H29ClN2O2
    Pureza:99.24%
    Forma y color:Solid
    Peso molecular:352.9
  • Umibecestat HCl

    CAS:
    <p>Umibecestat HCl (CNP520 HCl) is an efficient β-secretase (BACE1/BACE2) inhibitor that reduces Aβ levels in mice and rats.</p>
    Fórmula:C19H16Cl2F7N5O2
    Pureza:99.92%
    Forma y color:Solid
    Peso molecular:550.26
  • CALP1 acetate


    <p>CALP1 acetate is a calmodulin (CaM) agonist (Kd of 88 µM) that binds to the CaM EF-hand/Ca2+-binding site.</p>
    Fórmula:C42H79N9O12
    Pureza:99.63%
    Forma y color:Solid
    Peso molecular:902.13
  • (-)-(S)-B-973B

    CAS:
    <p>(-)-(S)-B-973B is an effective allosteric agonist and a positive allosteric modulator of α7 nAChR.</p>
    Fórmula:C24H26F2N6O
    Pureza:99.52%
    Forma y color:Solid
    Peso molecular:452.5
  • Trihexyphenidyl hydrochloride

    CAS:
    <p>Trihexyphenidyl hydrochloride (Benzhexol hydrochloride) is an antiparkinsonian agent of the antimuscarinic class.</p>
    Fórmula:C20H32ClNO
    Pureza:99.65%
    Forma y color:Solid
    Peso molecular:337.927
  • BRL-15572 dihydrochloride

    CAS:
    <p>BRL-15572 dihydrochloride: 5-HT1D antagonist, pKi 7.9, also binds 5-HT1A/2B, 60x selective over 5-HT1B.</p>
    Fórmula:C25H27ClN2O·2HCl
    Pureza:99.74%
    Forma y color:Solid
    Peso molecular:479.87
  • Dicyclomine

    CAS:
    <p>Dicyclomine: oral muscarinic antagonist, eases GI muscle spasms, high affinity for M1/M2 receptors, Ki of 5.1 nM/54.6 nM.</p>
    Fórmula:C19H35NO2
    Forma y color:Solid
    Peso molecular:309.49
  • Azaphen dihydrochloride monohydrate

    CAS:
    <p>Azaphen dihydrochloride monohydrate is a 5-hydroxytryptamine reabsorption inhibitor with antidepressant activity and can be used to study neurological diseases.</p>
    Fórmula:C16H23Cl2N5O2
    Pureza:99.85%
    Forma y color:Solid
    Peso molecular:388.29
  • Acamprosate calcium

    CAS:
    <p>Acamprosate calcium (Campral EC) is a GABA receptor agonist and modulator of glutamatergic systems, used for treating alcohol dependence.</p>
    Fórmula:C10H20CaN2O8S2
    Pureza:98% - 99.93%
    Forma y color:White Odorless Or Nearly Odorless Powder
    Peso molecular:400.48
  • PF-06447475

    CAS:
    <p>PF-06447475 is a highly effective, specific, brain penetrant LRRK2 inhibitor with IC0 of 3/11 nM for wild type LRRK2 and G2019S LRRK2 respectively.</p>
    Fórmula:C17H15N5O
    Pureza:98.61% - 99.62%
    Forma y color:Solid
    Peso molecular:305.33
  • Piperidolate hydrochloride

    CAS:
    <p>Piperidolate hydrochloride, an antimuscarinic, reduces acetylcholine-induced intestinal spasms in rats and dogs.</p>
    Fórmula:C21H26ClNO2
    Pureza:99.5%
    Forma y color:Solid
    Peso molecular:359.89
  • Vortioxetine hydrobromide

    CAS:
    <p>Vortioxetine hydrobromide (Lu AA21004 hydrobromide) is a serotonin (5-HT) modulator and stimulator (SMS), inhibits 5-HT1A/1B/3A/7 receptor and SERT (IC50: 15/33</p>
    Fórmula:C18H22N2S·HBr
    Pureza:98.85% - 99.98%
    Forma y color:Solid
    Peso molecular:379.36
  • MK-1064

    CAS:
    <p>MK-1064 (Urokinase inhibitor 1) is a selective orexin 2 receptor antagonist (2-SORA).</p>
    Fórmula:C24H20ClN5O3
    Pureza:99.19% - 99.82%
    Forma y color:Solid
    Peso molecular:461.9
  • β-Amyloid 15-21 acetate


    <p>β-Amyloid 15-21 acetate (Beta-Amyloid (15-21) acetate) is a fragment of Amyloid-β peptide, maybe used in the research of neurological disease.</p>
    Fórmula:C45H69N9O11
    Pureza:99.62%
    Forma y color:Solid
    Peso molecular:912.1
  • Donepezil

    CAS:
    <p>Donepezil (Aricept) is a piperidine-based, potent, specific, and reversible inhibitor of acetylcholinesterase (AChE).</p>
    Fórmula:C24H29NO3
    Pureza:99.69%
    Forma y color:White Or Almost White Crystal Powder
    Peso molecular:379.49
  • Loreclezole

    CAS:
    <p>Loreclezole is a selective GABAA receptor modulator and acts as a positive allosteric modulator of β2 or β3-subunit-containing receptors.</p>
    Fórmula:C10H6Cl3N3
    Pureza:99.78%
    Forma y color:Solid
    Peso molecular:274.53
  • PE859

    CAS:
    <p>PE859 is a potent inhibitor of both tau and Aβ aggregation.</p>
    Fórmula:C28H24N4O2
    Pureza:98.8% - 99.09%
    Forma y color:Solid
    Peso molecular:448.52
  • Metoclopramide hydrochloride hydrate

    CAS:
    <p>Metoclopramide hydrochloride hydrate (Metoclopramide monohydrochloride monohydrate) is a dopamine D2 antagonist that is a drug used for digestive dysfunction.</p>
    Fórmula:C14H25Cl2N3O3
    Pureza:99.33%
    Forma y color:Solid
    Peso molecular:354.27
  • VU-1545

    CAS:
    <p>VU-1545 is mGlu5 positive allosteric modulator.</p>
    Fórmula:C22H15FN4O3
    Pureza:98.8%
    Forma y color:Solid
    Peso molecular:402.38
  • Eltoprazine hydrochloride

    CAS:
    <p>Eltoprazine hydrochloride (DU 28853 hydrochloride) is a partial agonist at serotonin 5-HT1A, 5-HT1B, and 5-HT2B receptors (Ki value of 40, 52, and 81 nM,</p>
    Fórmula:C12H17ClN2O2
    Pureza:99.35%
    Forma y color:Solid
    Peso molecular:256.73
  • FK 3311

    CAS:
    <p>FK 3311 (COX-2 Inhibitor V) is a cell permeable and orally available sulfonanilide that acts as a COX-2 inhibitor and non-steroidal anti-inflammatory drug (</p>
    Fórmula:C15H13F2NO4S
    Pureza:97.98%
    Forma y color:Solid
    Peso molecular:341.33