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Neurociencia

Neurociencia

Los inhibidores en neurociencia son compuestos diseñados para modular la actividad de proteínas, enzimas o receptores específicos dentro del sistema nervioso. Estos inhibidores son cruciales para estudiar los mecanismos moleculares subyacentes a la función neuronal, la transmisión sináptica y las enfermedades neurodegenerativas. Al dirigirse a los receptores de neurotransmisores, canales iónicos y vías de señalización, los inhibidores en neurociencia ayudan en la exploración de la función cerebral y en el desarrollo de estrategias terapéuticas para trastornos neurológicos como el Alzheimer, Parkinson y la epilepsia. En CymitQuimica, ofrecemos una amplia gama de inhibidores de neurociencia de alta calidad para apoyar su investigación en neurobiología, neurofarmacología y ciencias cognitivas.

Subcategorías de "Neurociencia"

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Se han encontrado 5557 productos de "Neurociencia"

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  • Desvenlafaxine succinate hydrate

    CAS:
    Desvenlafaxine succinate hydrate (WY 45233 Succinate) is an antidepressant of the serotonin-norepinephrine reuptake inhibitor (SNRI).
    Fórmula:C20H33NO7
    Pureza:99.26%
    Forma y color:White Crystalline Powde
    Peso molecular:399.48
  • Myristicin

    CAS:
    <p>Myristicin is a natural spice extract with antibacterial, anti-inflammatory, and hepatoprotective properties, and can induce apoptosis.</p>
    Fórmula:C11H12O3
    Pureza:99.828%
    Forma y color:Liquid
    Peso molecular:192.21
  • Vortioxetine

    CAS:
    Vortioxetine (Lu AA 21004) is a serotonergic antidepressant used for major depression disorders.
    Fórmula:C18H22N2S
    Pureza:99.34% - 99.34%
    Forma y color:Solid
    Peso molecular:298.45
  • RU 24969 succinate

    CAS:
    <p>RU 24969 succinate, a 5-HT receptor agonist, exhibits K i values of 0.38 nM for 5-HT 1B and 2.5 nM for 5-HT 1A, indicating its affinity towards these receptors. It reduces fluid consumption and enhances forward locomotion. This compound is utilized in neurological disease research.</p>
    Fórmula:C18H22N2O5
    Forma y color:Solid
    Peso molecular:346.38
  • MK-1064

    CAS:
    MK-1064 (Urokinase inhibitor 1) is a selective orexin 2 receptor antagonist (2-SORA).
    Fórmula:C24H20ClN5O3
    Pureza:99.19% - 99.82%
    Forma y color:Solid
    Peso molecular:461.9
  • Vortioxetine hydrobromide

    CAS:
    Vortioxetine hydrobromide (Lu AA21004 hydrobromide) is a serotonin (5-HT) modulator and stimulator (SMS), inhibits 5-HT1A/1B/3A/7 receptor and SERT (IC50: 15/33
    Fórmula:C18H22N2S·HBr
    Pureza:98.85% - 99.98%
    Forma y color:Solid
    Peso molecular:379.36
  • Acotiamide hydrochloride

    CAS:
    Acotiamide hydrochloride, an oral AChE inhibitor (IC50: 1.79 μM), boosts gastric movement and treats functional dyspepsia.
    Fórmula:C21H31ClN4O5S
    Forma y color:Solid
    Peso molecular:487.01
  • Ramosetron

    CAS:
    Ramosetron 是一种血清素 5-HT3 受体拮抗剂,用于治疗恶心和呕吐。它被认为比其他一代 5-HT3 拮抗剂如昂丹司琼具有更高的效力和更长的止吐作用。它还适用于治疗“男性以腹泻为主的肠易激综合征”。它仅获准在日本和选定的东南亚国家使用。
    Fórmula:C17H17N3O
    Pureza:98.84%
    Forma y color:Solid
    Peso molecular:279.34
  • Eltoprazine dihydrochloride

    CAS:
    Eltoprazine dihydrochloride, a drug developed for aggression, is now studied for L-DOPA-induced dyskinesia in Parkinson's.
    Fórmula:C12H18Cl2N2O2
    Pureza:99.64%
    Forma y color:Solid
    Peso molecular:293.19
  • MK-3697

    CAS:
    <p>MK-3697, an isonicotinamide small molecule, acts as a potent and selective Orexin 2 receptor antagonist (Ki: 0.95 nM).</p>
    Fórmula:C23H21N5O3S
    Pureza:97.69% - 98.15%
    Forma y color:Solid
    Peso molecular:447.51
  • Pozanicline dihydrochloride

    CAS:
    Pozanicline dihydrochloride (ABT-089 dihydrochloride) is an orally bioavailable agonist of nicotinic acetylcholine receptor (nAChR) (Ki = 16.7 nM)
    Fórmula:C11H18Cl2N2O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:265.18
  • SKF89976A HCl

    CAS:
    SKF89976A: GABA uptake inhibitor, selective for GAT-1, passes blood-brain barrier, active in vivo (IC50: 0.13 μM hGAT-1).
    Fórmula:C22H25NO2
    Forma y color:Solid
    Peso molecular:335.44
  • suvn-911

    CAS:
    suvn-911 is a potent and selective antagonist of neuronal nicotinic acetylcholine α4β2 receptor (Ki = 1.5 nM) with antidepressant activity.
    Fórmula:C11H14Cl2N2O
    Pureza:98.88%
    Forma y color:Solid
    Peso molecular:261.15
  • Encequidar

    CAS:
    <p>Encequidar (HM30181A) is a potent and selective P-glycoprotein inhibitor.</p>
    Fórmula:C38H36N6O7
    Pureza:99.93%
    Forma y color:Solid
    Peso molecular:688.73
  • MPEP

    CAS:
    MPEP is a selective mGlu5 receptor antagonist with IC50 of 36 nM, exhibits no appreciable activity at mGlu1b/2/3/4a/7b/8a/6 receptors.
    Fórmula:C14H11N
    Pureza:99.54%
    Forma y color:Solid
    Peso molecular:193.24
  • Hypidone hydrochloride

    CAS:
    Hypidone hydrochloride (YL0919) is a novel antidepressant candidate with dual activity as a 5-HT1A receptor agonist and a selective serotonin reuptake inhibitor
    Fórmula:C18H23ClN2O2
    Pureza:99.82% - 99.93%
    Forma y color:Solid
    Peso molecular:334.84
  • Omberacetam

    CAS:
    Omberacetam (Noopept), a synthetic dipeptide, enhances cognition similarly to racetams.
    Fórmula:C17H22N2O4
    Pureza:≥95%
    Forma y color:White Powder
    Peso molecular:318.37
  • NMDAR antagonist 1

    CAS:
    <p>NMDAR antagonist 1 is an orally active, NR2B-selective NMDAR antagonist.</p>
    Fórmula:C20H20BrN3O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:414.3
  • CTEP

    CAS:
    CTEP (RO 4956371) (RO4956371) is a novel, long-acting, orally bioavailable allosteric antagonist of mGlu5 receptor with IC50 of 2.2 nM, shows >1000-fold
    Fórmula:C19H13ClF3N3O
    Pureza:99.17%
    Forma y color:Solid
    Peso molecular:391.77
  • Serotonin hydrochloride

    CAS:
    Serotonin hydrochloride (Serotonin HCl) is an endogenous 5-HT receptor agonist, a monoamine neurotransmitter in the CNS, and a catechol O-methyltransferase (
    Fórmula:C10H13ClN2O
    Pureza:98.05% - 99.93%
    Forma y color:White To Cream Powder
    Peso molecular:212.676