
Neurociencia
Los inhibidores en neurociencia son compuestos diseñados para modular la actividad de proteínas, enzimas o receptores específicos dentro del sistema nervioso. Estos inhibidores son cruciales para estudiar los mecanismos moleculares subyacentes a la función neuronal, la transmisión sináptica y las enfermedades neurodegenerativas. Al dirigirse a los receptores de neurotransmisores, canales iónicos y vías de señalización, los inhibidores en neurociencia ayudan en la exploración de la función cerebral y en el desarrollo de estrategias terapéuticas para trastornos neurológicos como el Alzheimer, Parkinson y la epilepsia. En CymitQuimica, ofrecemos una amplia gama de inhibidores de neurociencia de alta calidad para apoyar su investigación en neurobiología, neurofarmacología y ciencias cognitivas.
Subcategorías de "Neurociencia"
- Receptor 5-HT(993 productos)
- ACK(1 productos)
- AChR(612 productos)
- ATP Citrato Liasa(17 productos)
- Receptor adrenérgico(3.004 productos)
- BACE(36 productos)
- Beta amiloide(216 productos)
- CAMK(71 productos)
- Inhibidores de ciclooxigenasa (COX)(592 productos)
- Receptor de dopamina(433 productos)
- Receptor GABA(355 productos)
- Gamma-secretasa(63 productos)
- GluR(261 productos)
- GlyT(24 productos)
- Receptor de histamina(381 productos)
- LRRK2(41 productos)
- Receptor de melatonina(26 productos)
- NMDAR(15 productos)
- Receptor de OX(41 productos)
- Receptor de opioides(310 productos)
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Se han encontrado 5516 productos de "Neurociencia"
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PNU-282987
CAS:PNU-282987 is a selective α7 nicotinic acetylcholine receptor(α7 nAChR) agonist with Ki of 26 nM; no affinity for α1β1γδ and α3β4 nAChRs (IC50 ≥ 60 μM).Fórmula:C14H18Cl2N2OPureza:99% - >99.99%Forma y color:SolidPeso molecular:301.21CCMI
CAS:<p>CCMI (AVL-3288) is a potent and selective modulator of α7 nAChR-positive allosteric.</p>Fórmula:C19H15Cl2N3O2Pureza:>99.99%Forma y color:SolidPeso molecular:388.25MTEP hydrochloride
CAS:<p>MTEP hydrochloride (MTEP) is non-competitive mGlu5 antagonist (IC50 and Ki of 5 nM and 16 nM, respectively)</p>Fórmula:C11H9ClN2SPureza:99.58%Forma y color:SolidPeso molecular:236.72IPSU
CAS:<p>IPSU is an antagonist of OX2 receptor. IPSU Exhibits approximately six-fold selectivity for OX2 versus OX1 receptors.</p>Fórmula:C23H27N5O2Pureza:97.05%Forma y color:SolidPeso molecular:405.49Nor-benzetimide
CAS:Norbenzetimide, an organic compound, is prepared from benzetimide by catalytic transfer hydrogenolysis.Fórmula:C16H20N2O2Pureza:98.63%Forma y color:SolidPeso molecular:272.34DMAB-anabaseine dihydrochloride
CAS:<p>DMAB-anabaseine dihydrochloride (N,N-dimethyl-4-[(E)-(6-pyridin-3-yl-3,4-dihydro-2H-pyridin-5-ylidene)methyl]aniline;dihydrochloride) is an α7-containing</p>Fórmula:C19H23Cl2N3Pureza:99.91%Forma y color:SolidPeso molecular:364.31Rotigotine-
CAS:Rotigotine (N-0923) is a non-ergot dopamine receptor agonist used in the therapy of Parkinson disease and restless leg syndrome.Fórmula:C19H25NOSPureza:98.08% - 99.59%Forma y color:SolidPeso molecular:315.47SEN12333
CAS:<p>SEN12333 is an α7 nicotinic acetylcholine receptor (nAChR) agonist</p>Fórmula:C20H25N3O2Pureza:99.02%Forma y color:SolidPeso molecular:339.43Cinitapride
CAS:Cinitapride (Blaston) treats acid reflux and gastric issues, targeting 5-HT2, 5-HT1, and 5-HT4 receptors.Fórmula:C21H30N4O4Pureza:99.52%Forma y color:SolidPeso molecular:402.49AF-353
CAS:AF-353 (Ro-4), an effective and orally bioavailable antagonist of the P2X3/P2X2/3 receptor, inhibits human and rat P2X3 (pIC50= 8.0).Fórmula:C14H17IN4O2Pureza:92.98% - 99.356%Forma y color:SolidPeso molecular:400.21Eliapixant
CAS:Eliapixant (BAY 1817080) is a selective P2X3 antagonist with an 8 nM IC50, used for refractory chronic cough research.Fórmula:C22H21F3N4O3SPureza:99.86%Forma y color:SolidPeso molecular:478.49KN-93
CAS:<p>KN-93 is a selective inhibitor of Ca2+/calmodulin-dependent kinase II (CaMKII), competitively blocking CaM binding to the kinase.</p>Fórmula:C26H29ClN2O4SPureza:99.56% - 99.86%Forma y color:White SolidPeso molecular:501.04Solifenacin
CAS:Solifenacin (YM905 free base) (YM905 free base) is a novel muscarinic receptor antagonist, its pKis for M1, M2 and M3 receptors is of 7.6, 6.9 and 8.0,Fórmula:C23H26N2O2Pureza:99.87%Forma y color:SolidPeso molecular:362.46Lerisetron
CAS:Lerisetron is an antagonist of serotonin type 3 (5-HT3) receptor, with antiemetic activity.Fórmula:C18H20N4Pureza:99.15% - 99.82%Forma y color:SolidPeso molecular:292.38Tropisetron
CAS:Tropisetron (ICS 205-930) is an α7-nicotinic receptor agonist and 5-HT3 receptor antagonist with Kis of 6.9 nM and 5.3 nM, respectively.Fórmula:C17H20N2O2Pureza:99.68%Forma y color:White SolidPeso molecular:284.35Tasimelteon
CAS:<p>Tasimelteon (BMS-214778) is a melatonin receptor agonist that is used for the treatment of non-24 hour sleep-wake disorder in blind individuals.</p>Fórmula:C15H19NO2Pureza:98.93% - 99.93%Forma y color:SolidPeso molecular:245.32VU 0357121
CAS:VU0357121, a positive allosteric modulator of mGlu5 (EC50: 33 nM), is inactive or very weakly antagonizing at other mGlu receptor subtypes.Fórmula:C17H17F2NO2Pureza:99% - >99.99%Forma y color:SolidPeso molecular:305.32Basmisanil
CAS:Basmisanil (RG1662) is a negative allosteric modulator/inverse agonist of GABAAα5 receptors.Formulations containing basmisanil are in clinical trials for theFórmula:C21H20FN3O5SPureza:99.21% - 99.42%Forma y color:SolidPeso molecular:445.46Pardoprunox hydrochloride
CAS:Pardoprunox hydrochloride (SLV-308 hydrochloride) is a novel partial dopamine D2 and D3 receptor agonist and serotonin 5-HT1A receptor agonist, D2 (pKi = 8.1)Fórmula:C12H16ClN3O2Pureza:98.95% - 99.13%Forma y color:SolidPeso molecular:269.73trans-ACPD
CAS:trans-ACPD ((±)-trans-ACPD) is an equimolecular mixture of (1S, 3R)- and (1R, 3S)-ACPD.Fórmula:C7H11NO4Pureza:99.53%Forma y color:SolidPeso molecular:173.17
