
Neurociencia
Los inhibidores en neurociencia son compuestos diseñados para modular la actividad de proteínas, enzimas o receptores específicos dentro del sistema nervioso. Estos inhibidores son cruciales para estudiar los mecanismos moleculares subyacentes a la función neuronal, la transmisión sináptica y las enfermedades neurodegenerativas. Al dirigirse a los receptores de neurotransmisores, canales iónicos y vías de señalización, los inhibidores en neurociencia ayudan en la exploración de la función cerebral y en el desarrollo de estrategias terapéuticas para trastornos neurológicos como el Alzheimer, Parkinson y la epilepsia. En CymitQuimica, ofrecemos una amplia gama de inhibidores de neurociencia de alta calidad para apoyar su investigación en neurobiología, neurofarmacología y ciencias cognitivas.
Subcategorías de "Neurociencia"
- Receptor 5-HT(993 productos)
- ACK(1 productos)
- AChR(612 productos)
- ATP Citrato Liasa(17 productos)
- Receptor adrenérgico(3.004 productos)
- BACE(36 productos)
- Beta amiloide(216 productos)
- CAMK(71 productos)
- Inhibidores de ciclooxigenasa (COX)(592 productos)
- Receptor de dopamina(433 productos)
- Receptor GABA(355 productos)
- Gamma-secretasa(63 productos)
- GluR(261 productos)
- GlyT(24 productos)
- Receptor de histamina(381 productos)
- LRRK2(41 productos)
- Receptor de melatonina(26 productos)
- NMDAR(15 productos)
- Receptor de OX(41 productos)
- Receptor de opioides(310 productos)
Mostrar 12 subcategorías más
Se han encontrado 5516 productos de "Neurociencia"
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Almotriptan Malate
CAS:<p>Almotriptan Malate (PNU180638), a selective 5-HT1B/1D receptor agonist, is used in the therapy of Migraine attacks in adults.</p>Fórmula:C17H25N3O2S·C4H6O5Pureza:99.95%Forma y color:Pale Yellow SolidPeso molecular:469.55Rivanicline hemioxalate
<p>Rivanicline hemioxalate is a selective α4β2 nicotinic receptor agonist (K i =26 nM), over 1,000x preference to α7 (K i =3.6 μM), with limited side effects.</p>Fórmula:C12H16N2O4Pureza:98%Forma y color:SolidPeso molecular:207.23JI130
CAS:JI130 hinders Hes1 transcription repression; notably shrinks pancreatic tumor volume in mice.Fórmula:C23H24N2O3Pureza:99.61%Forma y color:SolidPeso molecular:376.45CRANAD 2
CAS:<p>CRANAD-2, a near-infrared probe, detects amyloid-beta in vivo, increasing fluorescence 70x and shifting blue 90 nm upon binding.</p>Fórmula:C23H25BF2N2O2Pureza:99.44%Forma y color:Dark Blue To Black PowderPeso molecular:410.27Piboserod hydrochloride
CAS:Piboserod HCl is a selective antagonist of 5-HT4 and muscarinic receptor.Fórmula:C22H32ClN3O2Forma y color:SolidPeso molecular:405.96Cyclopiazonic acid
CAS:<p>Cyclopiazonic acid (CPA) is a neurotoxic secondary metabolite (SM) made by A.</p>Fórmula:C20H20N2O3Pureza:99.27% - 99.80%Forma y color:SolidPeso molecular:336.38LY 2886721 Hydrochloride
CAS:Potent, selective BACE inhibitor; IC50 of 10.2 nM (BACE2) & 20.3 nM (BACE1). >5000x selectivity vs. other proteases. Lowers Aβ & sAPPβ in Alzheimer's mice.Fórmula:C18H17ClF2N4O2SForma y color:SolidPeso molecular:426.87Propantheline
CAS:Propantheline: oral muscarinic receptor blocker for smooth muscle issues, hyperhidrosis, and bladder control.Fórmula:C23H30NO3Forma y color:SolidPeso molecular:368.49SAX-187 hydrochloride
CAS:WAY-181187 is a potent, selective 5-HT6 agonist with high affinity (2.2-4.8 nM), and increases GABA in rat cortex at 3-30 mg/kg s.c.Fórmula:C15H14Cl2N4O2S2Forma y color:SolidPeso molecular:417.33VU0357017 hydrochloride
CAS:VU0357017 hydrochloride (ML071 hydrochloride) is highly selective M1 agonists act at an allosteric site to activate the receptor (EC50: 477 ± 172 nM; Pec50: 6.Fórmula:C18H28ClN3O3Pureza:99% - 99.97%Forma y color:SolidPeso molecular:369.89Propiverine
CAS:Propiverine reduces muscle spasms by limiting calcium influx, targeting bladder smooth muscles, aiding OAB research.Fórmula:C23H29NO3Forma y color:SolidPeso molecular:367.48Solifenacin hydrochloride
CAS:Solifenacin Hcl is a muscarinic receptor antagonist.Fórmula:C23H27ClN2O2Pureza:98%Forma y color:SolidPeso molecular:398.93GSK163090
CAS:<p>GSK163090 is a specific and orally active 5-HT1A/B/D receptor antagonist (pKis: 9.4/8.5/9.7, and 6.3/6.7 for 5-HT1A/B/D, and dopamine D2/D3).</p>Fórmula:C25H29N5OPureza:99.2%Forma y color:SolidPeso molecular:415.531,1'-Methylenedi-2-naphthol
CAS:<p>1,1'-Methylenedi-2-naphthol target CYP2C19 - cytochrome P450 family 2 subfamily C member 19 (human).</p>Fórmula:C21H16O2Pureza:98.91%Forma y color:Light Pink To Light Brown Crystalline PowderPeso molecular:300.35CL 218872
CAS:CL 218872: selective α1 GABAA receptor agonist, anxiolytic, and anticonvulsant; Ki=130 nM for α1, less potent for α2-α6.Fórmula:C13H9F3N4Pureza:99.92%Forma y color:SolidPeso molecular:278.23Pipamperone HCl
CAS:<p>Pipamperone blocks 5-HT2A/B/C, D2/D3/D4, α1/α2 receptors; favors 5-HT2A/D4 over D2; negligible affinity for H1, mACh. Highly selective at low doses.</p>Fórmula:C21H31ClFN3O2Forma y color:SolidPeso molecular:411.95AZD-8529
CAS:AZD-8529: selective, oral mGluR2 modulator, EC50 285 nM; inactive on mGluR1,3-8 at 20-25 M.Fórmula:C24H24F3N5O3Forma y color:SolidPeso molecular:487.47Syk Inhibitor II dihydrochloride
CAS:Syk inhibitor II selectively blocks Syk (IC50 = 41 nM), impacting platelet function and inflammation, with lower potency against other kinases.Fórmula:C14H17Cl2F3N6OPureza:98.53%Forma y color:SolidPeso molecular:413.22γ-Acetylenic GABA
CAS:<p>γ-Acetylenic GABA (4-Aminohex-5-ynoic acid) is a potent, irreversible inhibitor of GABA-transaminase.</p>Fórmula:C6H9NO2Forma y color:SolidPeso molecular:127.143Piperidolate hydrochloride
CAS:Piperidolate hydrochloride, an antimuscarinic, reduces acetylcholine-induced intestinal spasms in rats and dogs.Fórmula:C21H26ClNO2Pureza:99.5%Forma y color:SolidPeso molecular:359.89
