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Neurociencia

Neurociencia

Los inhibidores en neurociencia son compuestos diseñados para modular la actividad de proteínas, enzimas o receptores específicos dentro del sistema nervioso. Estos inhibidores son cruciales para estudiar los mecanismos moleculares subyacentes a la función neuronal, la transmisión sináptica y las enfermedades neurodegenerativas. Al dirigirse a los receptores de neurotransmisores, canales iónicos y vías de señalización, los inhibidores en neurociencia ayudan en la exploración de la función cerebral y en el desarrollo de estrategias terapéuticas para trastornos neurológicos como el Alzheimer, Parkinson y la epilepsia. En CymitQuimica, ofrecemos una amplia gama de inhibidores de neurociencia de alta calidad para apoyar su investigación en neurobiología, neurofarmacología y ciencias cognitivas.

Subcategorías de "Neurociencia"

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Se han encontrado 5516 productos de "Neurociencia"

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  • Almotriptan Malate

    CAS:
    <p>Almotriptan Malate (PNU180638), a selective 5-HT1B/1D receptor agonist, is used in the therapy of Migraine attacks in adults.</p>
    Fórmula:C17H25N3O2S·C4H6O5
    Pureza:99.95%
    Forma y color:Pale Yellow Solid
    Peso molecular:469.55
  • Rivanicline hemioxalate


    <p>Rivanicline hemioxalate is a selective α4β2 nicotinic receptor agonist (K i =26 nM), over 1,000x preference to α7 (K i =3.6 μM), with limited side effects.</p>
    Fórmula:C12H16N2O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:207.23
  • JI130

    CAS:
    JI130 hinders Hes1 transcription repression; notably shrinks pancreatic tumor volume in mice.
    Fórmula:C23H24N2O3
    Pureza:99.61%
    Forma y color:Solid
    Peso molecular:376.45
  • CRANAD 2

    CAS:
    <p>CRANAD-2, a near-infrared probe, detects amyloid-beta in vivo, increasing fluorescence 70x and shifting blue 90 nm upon binding.</p>
    Fórmula:C23H25BF2N2O2
    Pureza:99.44%
    Forma y color:Dark Blue To Black Powder
    Peso molecular:410.27
  • Piboserod hydrochloride

    CAS:
    Piboserod HCl is a selective antagonist of 5-HT4 and muscarinic receptor.
    Fórmula:C22H32ClN3O2
    Forma y color:Solid
    Peso molecular:405.96
  • Cyclopiazonic acid

    CAS:
    <p>Cyclopiazonic acid (CPA) is a neurotoxic secondary metabolite (SM) made by A.</p>
    Fórmula:C20H20N2O3
    Pureza:99.27% - 99.80%
    Forma y color:Solid
    Peso molecular:336.38
  • LY 2886721 Hydrochloride

    CAS:
    Potent, selective BACE inhibitor; IC50 of 10.2 nM (BACE2) & 20.3 nM (BACE1). >5000x selectivity vs. other proteases. Lowers Aβ & sAPPβ in Alzheimer's mice.
    Fórmula:C18H17ClF2N4O2S
    Forma y color:Solid
    Peso molecular:426.87
  • Propantheline

    CAS:
    Propantheline: oral muscarinic receptor blocker for smooth muscle issues, hyperhidrosis, and bladder control.
    Fórmula:C23H30NO3
    Forma y color:Solid
    Peso molecular:368.49
  • SAX-187 hydrochloride

    CAS:
    WAY-181187 is a potent, selective 5-HT6 agonist with high affinity (2.2-4.8 nM), and increases GABA in rat cortex at 3-30 mg/kg s.c.
    Fórmula:C15H14Cl2N4O2S2
    Forma y color:Solid
    Peso molecular:417.33
  • VU0357017 hydrochloride

    CAS:
    VU0357017 hydrochloride (ML071 hydrochloride) is highly selective M1 agonists act at an allosteric site to activate the receptor (EC50: 477 ± 172 nM; Pec50: 6.
    Fórmula:C18H28ClN3O3
    Pureza:99% - 99.97%
    Forma y color:Solid
    Peso molecular:369.89
  • Propiverine

    CAS:
    Propiverine reduces muscle spasms by limiting calcium influx, targeting bladder smooth muscles, aiding OAB research.
    Fórmula:C23H29NO3
    Forma y color:Solid
    Peso molecular:367.48
  • Solifenacin hydrochloride

    CAS:
    Solifenacin Hcl is a muscarinic receptor antagonist.
    Fórmula:C23H27ClN2O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:398.93
  • GSK163090

    CAS:
    <p>GSK163090 is a specific and orally active 5-HT1A/B/D receptor antagonist (pKis: 9.4/8.5/9.7, and 6.3/6.7 for 5-HT1A/B/D, and dopamine D2/D3).</p>
    Fórmula:C25H29N5O
    Pureza:99.2%
    Forma y color:Solid
    Peso molecular:415.53
  • 1,1'-Methylenedi-2-naphthol

    CAS:
    <p>1,1'-Methylenedi-2-naphthol target CYP2C19 - cytochrome P450 family 2 subfamily C member 19 (human).</p>
    Fórmula:C21H16O2
    Pureza:98.91%
    Forma y color:Light Pink To Light Brown Crystalline Powder
    Peso molecular:300.35
  • CL 218872

    CAS:
    CL 218872: selective α1 GABAA receptor agonist, anxiolytic, and anticonvulsant; Ki=130 nM for α1, less potent for α2-α6.
    Fórmula:C13H9F3N4
    Pureza:99.92%
    Forma y color:Solid
    Peso molecular:278.23
  • Pipamperone HCl

    CAS:
    <p>Pipamperone blocks 5-HT2A/B/C, D2/D3/D4, α1/α2 receptors; favors 5-HT2A/D4 over D2; negligible affinity for H1, mACh. Highly selective at low doses.</p>
    Fórmula:C21H31ClFN3O2
    Forma y color:Solid
    Peso molecular:411.95
  • AZD-8529

    CAS:
    AZD-8529: selective, oral mGluR2 modulator, EC50 285 nM; inactive on mGluR1,3-8 at 20-25 M.
    Fórmula:C24H24F3N5O3
    Forma y color:Solid
    Peso molecular:487.47
  • Syk Inhibitor II dihydrochloride

    CAS:
    Syk inhibitor II selectively blocks Syk (IC50 = 41 nM), impacting platelet function and inflammation, with lower potency against other kinases.
    Fórmula:C14H17Cl2F3N6O
    Pureza:98.53%
    Forma y color:Solid
    Peso molecular:413.22
  • γ-Acetylenic GABA

    CAS:
    <p>γ-Acetylenic GABA (4-Aminohex-5-ynoic acid) is a potent, irreversible inhibitor of GABA-transaminase.</p>
    Fórmula:C6H9NO2
    Forma y color:Solid
    Peso molecular:127.143
  • Piperidolate hydrochloride

    CAS:
    Piperidolate hydrochloride, an antimuscarinic, reduces acetylcholine-induced intestinal spasms in rats and dogs.
    Fórmula:C21H26ClNO2
    Pureza:99.5%
    Forma y color:Solid
    Peso molecular:359.89