
Neurociencia
Los inhibidores en neurociencia son compuestos diseñados para modular la actividad de proteínas, enzimas o receptores específicos dentro del sistema nervioso. Estos inhibidores son cruciales para estudiar los mecanismos moleculares subyacentes a la función neuronal, la transmisión sináptica y las enfermedades neurodegenerativas. Al dirigirse a los receptores de neurotransmisores, canales iónicos y vías de señalización, los inhibidores en neurociencia ayudan en la exploración de la función cerebral y en el desarrollo de estrategias terapéuticas para trastornos neurológicos como el Alzheimer, Parkinson y la epilepsia. En CymitQuimica, ofrecemos una amplia gama de inhibidores de neurociencia de alta calidad para apoyar su investigación en neurobiología, neurofarmacología y ciencias cognitivas.
Subcategorías de "Neurociencia"
- Receptor 5-HT(1.003 productos)
- ACK(1 productos)
- AChR(616 productos)
- ATP Citrato Liasa(17 productos)
- Receptor adrenérgico(3.010 productos)
- BACE(36 productos)
- Beta amiloide(218 productos)
- CAMK(72 productos)
- Inhibidores de ciclooxigenasa (COX)(592 productos)
- Receptor de dopamina(435 productos)
- Receptor GABA(360 productos)
- Gamma-secretasa(63 productos)
- GluR(262 productos)
- GlyT(25 productos)
- Receptor de histamina(381 productos)
- LRRK2(41 productos)
- Receptor de melatonina(26 productos)
- NMDAR(14 productos)
- Receptor de OX(41 productos)
- Receptor de opioides(321 productos)
Mostrar 12 subcategorías más
Se han encontrado 5532 productos de "Neurociencia"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Afloqualone
CAS:<p>Afloqualone (HQ-495) is a GABA Receptor agonist with sedative and muscle-relaxant properties.</p>Fórmula:C16H14FN3OPureza:99.72%Forma y color:SolidPeso molecular:283.3MK-3697
CAS:<p>MK-3697, an isonicotinamide small molecule, acts as a potent and selective Orexin 2 receptor antagonist (Ki: 0.95 nM).</p>Fórmula:C23H21N5O3SPureza:97.69% - 98.15%Forma y color:SolidPeso molecular:447.51SB399885
CAS:<p>SB399885 is a potent, brain-penetrant, oral SR-6 antagonist with 200-fold selectivity for SR-6 receptors.</p>Fórmula:C18H21Cl2N3O4SPureza:98.94%Forma y color:SolidPeso molecular:446.35VU0238441
CAS:VU0238441 is agonist of Muscarinic acetylcholine receptor M5 (human) with EC50 of 2.1μM.Fórmula:C16H9ClF3NO2Pureza:100%Forma y color:SolidPeso molecular:339.7CGP52432
CAS:CGP52432 is a very potent antagonist of GABAB receptors (IC50 = 85 nM).Fórmula:C15H24Cl2NO4PPureza:98.75%Forma y color:SolidPeso molecular:384.24mAChR-IN-1 hydrochloride
CAS:mAChR-IN-1 hydrochloride is a potent muscarinic cholinergic receptor (mAChR) antagonist, with an IC50 of 17 Nm.Fórmula:C23H26ClIN2O2Pureza:99.87%Forma y color:SolidPeso molecular:524.82Loreclezole
CAS:Loreclezole is a selective GABAA receptor modulator and acts as a positive allosteric modulator of β2 or β3-subunit-containing receptors.Fórmula:C10H6Cl3N3Pureza:99.78%Forma y color:SolidPeso molecular:274.53PE859
CAS:<p>PE859 is a potent inhibitor of both tau and Aβ aggregation.</p>Fórmula:C28H24N4O2Pureza:98.8% - 99.09%Forma y color:SolidPeso molecular:448.52Bicuculline
CAS:<p>Bicuculline, a plant-derived GABAA receptor antagonist, identified in 1932, reacts to light.</p>Fórmula:C20H17NO6Pureza:98% - 99.99%Forma y color:Light Yellow PowderPeso molecular:367.35Atracurium besylate
CAS:Atracurium besylate (51W89) is a short-acting, non-depolarizing muscle relaxant, not affecting the heart or reliant on kidneys.Fórmula:C65H82N2O18S2Pureza:98.94% - 99.71%Forma y color:SolidPeso molecular:1243.49Renzapride hydrochloride
CAS:Renzapride is a 5-HT3 antagonist and 5-HT4 agonist. Renzapride also functions as a 5-HT2B antagonist and has some affinity for the 5-HT2A and 5-HT2C receptors.Fórmula:C16H23Cl2N3O2Forma y color:SolidPeso molecular:360.28KN-93
CAS:<p>KN-93 is a selective inhibitor of Ca2+/calmodulin-dependent kinase II (CaMKII), competitively blocking CaM binding to the kinase.</p>Fórmula:C26H29ClN2O4SPureza:99.56% - 99.86%Forma y color:White SolidPeso molecular:501.04Solifenacin
CAS:Solifenacin (YM905 free base) (YM905 free base) is a novel muscarinic receptor antagonist, its pKis for M1, M2 and M3 receptors is of 7.6, 6.9 and 8.0,Fórmula:C23H26N2O2Pureza:99.87%Forma y color:SolidPeso molecular:362.465-Benzyloxygramine
CAS:5-Benzyloxygramine blocks the Dopamin receptors and antagonizes the effects of 5-HT on the rat uterus and the rabbit ear.Fórmula:C18H20N2OPureza:99.13%Forma y color:SolidPeso molecular:280.36GSK2578215A
CAS:GSK2578215A is a potent and selective LRRK2 kinase inhibitor.Fórmula:C24H18FN3O2Pureza:99.57% - 99.94%Forma y color:SolidPeso molecular:399.42Indophagolin
CAS:Indophagolin: autophagy inhibitor, IC50 140 nM; blocks P2X4, P2X1, P2X3 receptors, IC50s 2.71, 2.40, 3.49 μM.Fórmula:C19H15BrClF3N2O3SPureza:99.76%Forma y color:SolidPeso molecular:523.75Dihydroergotoxine mesylate
CAS:Dihydroergotoxine mesylate (Ergoloid mesylates) is mainly used to improve symptoms and physical symptoms of mental degeneration related to aging.Fórmula:C20H29N3O5SPureza:99.39% - ≥95%Forma y color:SolidPeso molecular:423.53A-484954
CAS:A-484954 (A 484954) is a highly specific eukaryotic elongation factor-2 (eEF2, IC50: 280 nM) inhibitor.Fórmula:C13H15N5O3Pureza:97.47% - 99.86%Forma y color:SolidPeso molecular:289.29Imidafenacin
CAS:Imidafenacin (KRP-197)(KRP-197; ONO-8025) is a potent and selective inhibitor of M3 receptors with Kb of 0.317 nM.Fórmula:C20H21N3OPureza:99.17%Forma y color:SolidPeso molecular:319.4PBD-150
CAS:PBD-150 is an inhibitor of human glutaminyl cyclase (hQC) Y115E-Y117E variant( ki : 490 nM)Fórmula:C15H20N4O2SPureza:99.68%Forma y color:SolidPeso molecular:320.41
