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Neurociencia

Neurociencia

Los inhibidores en neurociencia son compuestos diseñados para modular la actividad de proteínas, enzimas o receptores específicos dentro del sistema nervioso. Estos inhibidores son cruciales para estudiar los mecanismos moleculares subyacentes a la función neuronal, la transmisión sináptica y las enfermedades neurodegenerativas. Al dirigirse a los receptores de neurotransmisores, canales iónicos y vías de señalización, los inhibidores en neurociencia ayudan en la exploración de la función cerebral y en el desarrollo de estrategias terapéuticas para trastornos neurológicos como el Alzheimer, Parkinson y la epilepsia. En CymitQuimica, ofrecemos una amplia gama de inhibidores de neurociencia de alta calidad para apoyar su investigación en neurobiología, neurofarmacología y ciencias cognitivas.

Subcategorías de "Neurociencia"

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Se han encontrado 5532 productos de "Neurociencia"

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  • Afloqualone

    CAS:
    <p>Afloqualone (HQ-495) is a GABA Receptor agonist with sedative and muscle-relaxant properties.</p>
    Fórmula:C16H14FN3O
    Pureza:99.72%
    Forma y color:Solid
    Peso molecular:283.3
  • MK-3697

    CAS:
    <p>MK-3697, an isonicotinamide small molecule, acts as a potent and selective Orexin 2 receptor antagonist (Ki: 0.95 nM).</p>
    Fórmula:C23H21N5O3S
    Pureza:97.69% - 98.15%
    Forma y color:Solid
    Peso molecular:447.51
  • SB399885

    CAS:
    <p>SB399885 is a potent, brain-penetrant, oral SR-6 antagonist with 200-fold selectivity for SR-6 receptors.</p>
    Fórmula:C18H21Cl2N3O4S
    Pureza:98.94%
    Forma y color:Solid
    Peso molecular:446.35
  • VU0238441

    CAS:
    VU0238441 is agonist of Muscarinic acetylcholine receptor M5 (human) with EC50 of 2.1μM.
    Fórmula:C16H9ClF3NO2
    Pureza:100%
    Forma y color:Solid
    Peso molecular:339.7
  • CGP52432

    CAS:
    CGP52432 is a very potent antagonist of GABAB receptors (IC50 = 85 nM).
    Fórmula:C15H24Cl2NO4P
    Pureza:98.75%
    Forma y color:Solid
    Peso molecular:384.24
  • mAChR-IN-1 hydrochloride

    CAS:
    mAChR-IN-1 hydrochloride is a potent muscarinic cholinergic receptor (mAChR) antagonist, with an IC50 of 17 Nm.
    Fórmula:C23H26ClIN2O2
    Pureza:99.87%
    Forma y color:Solid
    Peso molecular:524.82
  • Loreclezole

    CAS:
    Loreclezole is a selective GABAA receptor modulator and acts as a positive allosteric modulator of β2 or β3-subunit-containing receptors.
    Fórmula:C10H6Cl3N3
    Pureza:99.78%
    Forma y color:Solid
    Peso molecular:274.53
  • PE859

    CAS:
    <p>PE859 is a potent inhibitor of both tau and Aβ aggregation.</p>
    Fórmula:C28H24N4O2
    Pureza:98.8% - 99.09%
    Forma y color:Solid
    Peso molecular:448.52
  • Bicuculline

    CAS:
    <p>Bicuculline, a plant-derived GABAA receptor antagonist, identified in 1932, reacts to light.</p>
    Fórmula:C20H17NO6
    Pureza:98% - 99.99%
    Forma y color:Light Yellow Powder
    Peso molecular:367.35
  • Atracurium besylate

    CAS:
    Atracurium besylate (51W89) is a short-acting, non-depolarizing muscle relaxant, not affecting the heart or reliant on kidneys.
    Fórmula:C65H82N2O18S2
    Pureza:98.94% - 99.71%
    Forma y color:Solid
    Peso molecular:1243.49
  • Renzapride hydrochloride

    CAS:
    Renzapride is a 5-HT3 antagonist and 5-HT4 agonist. Renzapride also functions as a 5-HT2B antagonist and has some affinity for the 5-HT2A and 5-HT2C receptors.
    Fórmula:C16H23Cl2N3O2
    Forma y color:Solid
    Peso molecular:360.28
  • KN-93

    CAS:
    <p>KN-93 is a selective inhibitor of Ca2+/calmodulin-dependent kinase II (CaMKII), competitively blocking CaM binding to the kinase.</p>
    Fórmula:C26H29ClN2O4S
    Pureza:99.56% - 99.86%
    Forma y color:White Solid
    Peso molecular:501.04
  • Solifenacin

    CAS:
    Solifenacin (YM905 free base) (YM905 free base) is a novel muscarinic receptor antagonist, its pKis for M1, M2 and M3 receptors is of 7.6, 6.9 and 8.0,
    Fórmula:C23H26N2O2
    Pureza:99.87%
    Forma y color:Solid
    Peso molecular:362.46
  • 5-Benzyloxygramine

    CAS:
    5-Benzyloxygramine blocks the Dopamin receptors and antagonizes the effects of 5-HT on the rat uterus and the rabbit ear.
    Fórmula:C18H20N2O
    Pureza:99.13%
    Forma y color:Solid
    Peso molecular:280.36
  • GSK2578215A

    CAS:
    GSK2578215A is a potent and selective LRRK2 kinase inhibitor.
    Fórmula:C24H18FN3O2
    Pureza:99.57% - 99.94%
    Forma y color:Solid
    Peso molecular:399.42
  • Indophagolin

    CAS:
    Indophagolin: autophagy inhibitor, IC50 140 nM; blocks P2X4, P2X1, P2X3 receptors, IC50s 2.71, 2.40, 3.49 μM.
    Fórmula:C19H15BrClF3N2O3S
    Pureza:99.76%
    Forma y color:Solid
    Peso molecular:523.75
  • Dihydroergotoxine mesylate

    CAS:
    Dihydroergotoxine mesylate (Ergoloid mesylates) is mainly used to improve symptoms and physical symptoms of mental degeneration related to aging.
    Fórmula:C20H29N3O5S
    Pureza:99.39% - ≥95%
    Forma y color:Solid
    Peso molecular:423.53
  • A-484954

    CAS:
    A-484954 (A 484954) is a highly specific eukaryotic elongation factor-2 (eEF2, IC50: 280 nM) inhibitor.
    Fórmula:C13H15N5O3
    Pureza:97.47% - 99.86%
    Forma y color:Solid
    Peso molecular:289.29
  • Imidafenacin

    CAS:
    Imidafenacin (KRP-197)(KRP-197; ONO-8025) is a potent and selective inhibitor of M3 receptors with Kb of 0.317 nM.
    Fórmula:C20H21N3O
    Pureza:99.17%
    Forma y color:Solid
    Peso molecular:319.4
  • PBD-150

    CAS:
    PBD-150 is an inhibitor of human glutaminyl cyclase (hQC) Y115E-Y117E variant( ki : 490 nM)
    Fórmula:C15H20N4O2S
    Pureza:99.68%
    Forma y color:Solid
    Peso molecular:320.41