
Neurociencia
Los inhibidores en neurociencia son compuestos diseñados para modular la actividad de proteínas, enzimas o receptores específicos dentro del sistema nervioso. Estos inhibidores son cruciales para estudiar los mecanismos moleculares subyacentes a la función neuronal, la transmisión sináptica y las enfermedades neurodegenerativas. Al dirigirse a los receptores de neurotransmisores, canales iónicos y vías de señalización, los inhibidores en neurociencia ayudan en la exploración de la función cerebral y en el desarrollo de estrategias terapéuticas para trastornos neurológicos como el Alzheimer, Parkinson y la epilepsia. En CymitQuimica, ofrecemos una amplia gama de inhibidores de neurociencia de alta calidad para apoyar su investigación en neurobiología, neurofarmacología y ciencias cognitivas.
Subcategorías de "Neurociencia"
- Receptor 5-HT(1.020 productos)
- ACK(1 productos)
- AChR(619 productos)
- ATP Citrato Liasa(17 productos)
- Receptor adrenérgico(3.022 productos)
- BACE(36 productos)
- Beta amiloide(222 productos)
- CAMK(72 productos)
- Inhibidores de ciclooxigenasa (COX)(599 productos)
- Receptor de dopamina(442 productos)
- Receptor GABA(365 productos)
- Gamma-secretasa(62 productos)
- GluR(262 productos)
- GlyT(26 productos)
- Receptor de histamina(385 productos)
- LRRK2(42 productos)
- Receptor de melatonina(26 productos)
- NMDAR(13 productos)
- Receptor de OX(41 productos)
- Receptor de opioides(322 productos)
Mostrar 12 subcategorías más
Se han encontrado 5557 productos de "Neurociencia"
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Aβ42 agonist-1
CAS:<p>Aβ42 agonist-1 is a small molecule compound with anti-cancer activity and NF-κB inhibitory properties, inducing Aβ42 aggregation.</p>Fórmula:C15H11NO2Pureza:99.77%Forma y color:SolidPeso molecular:237.25DA-8031
CAS:<p>DA-8031 is a selective and orally active serotonin reuptake inhibitor. It is utilized in research related to premature ejaculation (PE).</p>Fórmula:C21H24N2O2Forma y color:SolidPeso molecular:336.43AAK1-IN-3 TFA
AAK1-IN-3 TFA, an AAK1 inhibitor with IC50 of 11 nM, crosses the blood-brain barrier, is a quinoline analogue, and may aid neuropathic pain research.Fórmula:C24H22F6N4O4Forma y color:SolidPeso molecular:544.45Sulamserod hydrochloride
CAS:<p>Sulamserod hydrochloride is a 5-HT4 receptor antagonist. It is utilized in research related to gastrointestinal disorders.</p>Fórmula:C19H29Cl2N3O5SForma y color:SolidPeso molecular:482.425-HT7R antagonist 3
CAS:Compound 6.4, also known as 5-HT7R antagonist 3, is a selective antagonist of the 5-HT7R with a Ki of 8 nM. It exhibits significantly less affinity towards D2R, 5-HT1AR, and 5-HT2AR with Ki values of 511 nM, 8930 nM, and 5786 nM, respectively. In mice, 5-HT7R antagonist 3 demonstrates anti-depressant and anti-anxiety activities.Fórmula:C30H33FN4O3Forma y color:SolidPeso molecular:516.61BChE-IN-5
BChE-IN-5: potent, selective BChE inhibitor (IC50: 2.8 nM), more effective on hBChE, potential in Alzheimer's research.Fórmula:C30H42N4OForma y color:SolidPeso molecular:474.68(+)-Cevimeline hydrochloride hemihydrate
(+)-Cevimeline HCl hemihydrate is a muscarinic agonist for dry mouth in Sjogren's with rapid absorption, differing metabolism in species.Fórmula:C10H19ClNO1·5SPureza:98%Forma y color:SolidPeso molecular:244.78AChE-IN-25
AChE-IN-25: selective, potent AChE inhibitor, non-competitive, IC50 = 2.95 μM, for Alzheimer's research.Fórmula:C20H15ClN4O4SForma y color:SolidPeso molecular:442.88AChE/BChE-IN-10
CAS:<p>AChE/BChE-IN-10 inhibits AChE/BChE (IC50: 0.176/0.47 μM), crosses the blood-brain barrier, and prevents Aβ-aggregation.</p>Fórmula:C26H30N2O2Pureza:99.55% - 99.88%Forma y color:SoildPeso molecular:402.53LY2979165
CAS:LY2979165 (mGlu2 agonist) is an orthosteric agonist of mGluR2 and can be used in studies about serving as an anti-depressant.Fórmula:C13H22N6O6SPureza:98.41%Forma y color:SolidPeso molecular:390.42Iclepertin
CAS:Iclepertin (BI-425809) is a GlyT1 inhibitor.Iclepertin is used for the treatment of Alzheimer;s disease and other CNS disorders.Fórmula:C20H18F6N2O5SPureza:98.89% - 98.93%Forma y color:SolidPeso molecular:512.42SB-224289 hydrochloride
CAS:SB-224289 hydrochloride (SB-224289A) is a selective antagonist of 5-HT1B receptor, with anxiolytic effect.Fórmula:C32H33ClN4O3Pureza:98.99% - 99.96%Forma y color:SolidPeso molecular:557.08AChE-IN-26
CAS:<p>AChE-IN-26 (compound 4a) is an AChE (acetylcholinesterase) inhibitor (IC50: 0.42 μM).</p>Fórmula:C21H21BrN2O3Pureza:99.24% - 99.85%Forma y color:SoildPeso molecular:429.31Umibecestat
CAS:Umibecestat inhibits human and mouse BACE-1 (IC50: 11 nM & 10 nM), potentially for Alzheimer's research.Fórmula:C19H15ClF7N5O2Pureza:99.88%Forma y color:SolidPeso molecular:513.8BDZ-g
CAS:BDZ-g: potent, selective AMPA receptor antagonist; useful for researching neurological disorders.Fórmula:C21H21N5O2SPureza:99.97%Forma y color:SolidPeso molecular:407.49BMS 299897
CAS:<p>BMS 299897, a sulfonamide γ-secretase inhibitor, inhibits Aβ production with an IC50 of 7 nM in HEK293 cells overexpressing APP.</p>Fórmula:C24H21ClF3NO4SPureza:99.82%Forma y color:SolidPeso molecular:511.94NB-360
CAS:NB-360: potent, brain-penetrant BACE1/2 inhibitor; IC50s: 5-6 nM; high selectivity vs pepsin, cathepsin E/D.Fórmula:C21H19F4N5O2Pureza:99.72%Forma y color:SolidPeso molecular:449.44-Amino-6-hydroxypyrazolo[3,4-d]pyrimidine
CAS:Fórmula:C5H5N5OPureza:>93.0%(HPLC)Forma y color:White to Light yellow to Light orange powder to crystallinePeso molecular:151.13(RS)-APICA
CAS:group II metabotropic glutamate receptor antagonistFórmula:C10H12NO5PForma y color:SolidPeso molecular:257.18


